BDBM736532 US20250136553, Compound 243a

SMILES COc1cccc(OC)c1S(=N)(=O)NC(=O)c1ccc(Cn2cccn2)c(OC)n1

InChI Key InChIKey=VCKDIJJAYULYBZ-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736532   

TargetHistone acetyltransferase KAT6A(Human)
Olema Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 736532BDBM736532(US20250136553, Compound 243a)
Affinity DataIC50: 17nMAssay Description:TR-FRET based methods were used for assaying compounds of the present invention for KAT6A enzyme inhibitory activity. TR-FRET is a homogeneous proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2025
Entry Details
US Patent