BDBM736544 5-((1H-pyrazol-1-yl)methyl)-N-((2,6-dimethoxy-4-(pyridin-3- ylethynyl)phenyl)sulfonyl)-6-methoxypicolinamide::US20250136553, Compound 269

SMILES COc1cc(C#Cc2cccnc2)cc(OC)c1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(OC)n1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736544   

LigandPNGBDBM736544(5-((1H-pyrazol-1-yl)methyl)-N-((2,6-dimethoxy-4-(p...)
Affinity DataIC50: 12nMAssay Description:TR-FRET based methods were used for assaying compounds of the present invention for KAT6A enzyme inhibitory activity. TR-FRET is a homogeneous proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
TBA
Entry Details