BDBM741341 US20250162989, Compound I-93

SMILES COc1cc(NC(=O)[C@H](CC2CCN(C)CC2)NC(=O)c2ccc(F)cc2)ccc1S(=O)(=O)NC(C)(C)CO

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 741341   

LigandPNGBDBM741341(US20250162989, Compound I-93)
Affinity DataIC50: 525nMAssay Description:USP30 (25 ng/μl) tested against K48-linked diubiquitin (5.6 μM). USP30 was diluted in a buffer containing 40 mM Tris, 0.01% BSA, 1 mM DTT and K48 in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
LigandPNGBDBM741341(US20250162989, Compound I-93)
Affinity DataIC50: 525nMAssay Description:In vitro biochemical assay to establish the potency of compounds for USP30 inhibition: a 384-well plate assay using a fluorophore tagged substrate of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details