BDBM741983 US20250163057, Compound I-159

SMILES C/C=C(C)/S(=O)(=O)NCc2nn(c1ccccc1)c5c2[C@H](c3ccc(F)cc3)[C@H](NC(=O)c4cccc(C(F)(F)F)c4)C(=O)N5CC

InChI Key InChIKey=ZEINUDXWKXSJPP-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 741983   

TargetDCN1-like protein 1(Human)
Cellarity

US Patent
LigandChemical structure of BindingDB Monomer ID 741983BDBM741983(US20250163057, Compound I-159)
Affinity DataIC50: 600nMAssay Description:The TR-FRET assay was designed following the Scott et al. protocol (Scott et al., Nat Chem Biol. 2017 August; 13(8): 850-857. Doi:10.1038/nchembio.23...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent

TargetDCN1-like protein 1(Human)
Cellarity

US Patent
LigandChemical structure of BindingDB Monomer ID 741983BDBM741983(US20250163057, Compound I-159)
Affinity DataIC50: 2.00E+3nMAssay Description:The TR-FRET assay was designed following the Scott et al. protocol (Scott et al., Nat Chem Biol. 2017 August; 13(8): 850-857. Doi:10.1038/nchembio.23...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent