BDBM747267 US20250179094, Compound 6::US20250215017, Compound 6

SMILES Cc1cccc(-c2nc[nH]c2-c2ccnc(-c3nc4c([nH]3)CN(C(=O)N3CCCC3)C4)c2)n1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 747267   

TargetTGF-beta receptor type-1(Human)TBA
LigandPNGBDBM747267(US20250179094, Compound 6 | US20250215017, Compoun...)
Affinity DataIC50: 22nMAssay Description:The principle of the activity assay was that TGFβR1 phosphorylates the substrate TGFβR1tide, consuming ATP in the process. This experiment employed t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetTGF-beta receptor type-1(Human)TBA
LigandPNGBDBM747267(US20250179094, Compound 6 | US20250215017, Compoun...)
Affinity DataIC50: 22nMAssay Description:The principle of the activity assay was that TGFβR1 phosphorylates the substrate TGFβR1tide, consuming ATP in the process. This experiment employed t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details