BDBM747568 US12325697, Compound AGX-8

SMILES CCNc1cc(-c2nn(CC(C)C)cc2-c2nncn2C)cc(N2Cc3c(cccc3C(F)(F)F)C2=O)n1

InChI Key InChIKey=LFHJZBFJLHRBCR-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 747568   

TargetIsoform Truncated 1 of E3 ubiquitin-protein ligase CBL-B [36-427] (Human)
Nimbus Clio

US Patent

LigandBDBM747568(US12325697, Compound AGX-8)Copy SMILESCopy InChI

Affinity DataIC50: 3.00E+4nMAssay Description:Fluorescein-BODIPY labeled UBED2D(C85K)-Ub was prepared by conjugating ubiquitin (Ub) labeled at its N-terminus with Fluorescein-BODIPY maleimide (Th...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
10/4/2025
Entry Details
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