BDBM755951 3-(5-(4-(((2S,5S)-2,5- dimethylpyrrolidin-1-yl)methyl)-1- methyl-1H-pyrrolo[2,3-b]pyridin- 6-yl)-1-oxoisoindolin-2- yl)piperidine-2,6-dione::US20250214991, Compound 108

SMILES C[C@H]1CC[C@H](C)N1Cc1cc(-c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)nc2c1ccn2C

InChI Key InChIKey=SQXRXDMFVNECNV-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 755951   

TargetDNA damage-binding protein 1/Protein cereblon(Human)
Oncopia Therapeutics, Inc. D/B/A/ Sk Life Science Labs

US Patent
LigandChemical structure of BindingDB Monomer ID 755951BDBM755951(3-(5-(4-(((2S,5S)-2,5- dimethylpyrrolidin-1-yl)met...)
Affinity DataIC50: 65nMAssay Description:The binding potency was determined using HTRF assay technology (Perkin Elmer). Compounds were serially diluted in DMSO and 0.2 μL volume was transfer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent