BDBM757551 6-(Dimethylamino)-7-fluoro-N-((2-methylquinolin-8-yl)sulfonyl)benzofuran-2-carboxamide::US12357603, Example 190

SMILES Cc1ccc2cccc(S(=O)(=O)NC(=O)c3cc4ccc(N(C)C)c(F)c4o3)c2n1

InChI Key InChIKey=UGHPGDQCGXLVBW-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 757551   

TargetHistone Acetyltransferase KAT6A [194-810]/Zinc Finger Protein Neuro-d4 (DPF1)/ Histone Acetyltransferase Type B Catalytic Subunit (HAT1)(Homo sapiens (Human))
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US Patent

LigandBDBM757551(6-(Dimethylamino)-7-fluoro-N-((2-methylquinolin-8-...)Copy SMILESCopy InChI

Affinity DataIC50: 1.40E+3nMAssay Description:Recombinant human His-tagged Kat6a protein (amino acids 194-810), was purified in-house from Baculovirus-infected insect cells (Sf9). Histone H4 pept...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
10/28/2025
Entry Details
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