BDBM757579 5-Bromo-6-(dimethylamino)-N-(2-ethoxybenzene-1-sulfonyl)-1-benzofuran-2-carboxamide::US12357603, Example 218

SMILES CCOc1ccccc1S(=O)(=O)NC(=O)c1cc2cc(Br)c(N(C)C)cc2o1

InChI Key InChIKey=JXJVTSAAGCCYEE-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 757579   

TargetHistone Acetyltransferase KAT6A [194-810]/Zinc Finger Protein Neuro-d4 (DPF1)/ Histone Acetyltransferase Type B Catalytic Subunit (HAT1)(Homo sapiens (Human))
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US Patent

LigandBDBM757579(5-Bromo-6-(dimethylamino)-N-(2-ethoxybenzene-1-sul...)Copy SMILESCopy InChI

Affinity DataIC50: 4.73E+3nMAssay Description:Recombinant human His-tagged Kat6a protein (amino acids 194-810), was purified in-house from Baculovirus-infected insect cells (Sf9). Histone H4 pept...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
10/28/2025
Entry Details
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