BDBM758699 N-(5-(N-(tert-butyl)sulfamoyl)-5,6- dihydro-4H-pyrrolo[3,4-d]thiazol-2-yl)- 4-(5-cyano-2-methoxyphenyl)-6- methylnicotinamide::US20250230171, Compound 275

SMILES COc1ccc(C#N)cc1-c1cc(C)ncc1C(=O)Nc1nc2c(s1)CN(S(=O)(=O)NC(C)(C)C)C2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 758699   

LigandPNGBDBM758699(N-(5-(N-(tert-butyl)sulfamoyl)-5,6- dihydro-4H-pyr...)
Affinity DataIC50: 8nMAssay Description:POLθ-mediated ATP hydrolysis was measured using the ADP-Glo Kinase Assay (Promega Corporation, Madison, WI). Reactions were performed in white 384-we...More data for this Ligand-Target Pair
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Date in BDB:
TBA
Entry Details