BDBM769507 (3R)-6-chloro-3,11-dimethyl-10-oxa-2,13,17,18,21-pentaazapentacyclo[13.5.2.18,11.04,9.011,22]tricosa-1(21),4,6,8,15::US12410191, Example 22

SMILES C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC2(C)Cc3cc(Cl)cc1c3O2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 769507   

LigandPNGBDBM769507((3R)-6-chloro-3,11-dimethyl-10-oxa-2,13,17,18,21-p...)
Affinity DataIC50: 0.360nMAssay Description:Table 1: The experimental methods were operated according to the steps in the kit instruction, and were briefly described as follows: a test compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
LigandPNGBDBM769507((3R)-6-chloro-3,11-dimethyl-10-oxa-2,13,17,18,21-p...)
Affinity DataIC50: 0.520nMAssay Description:Table 1: The experimental methods were operated according to the steps in the kit instruction, and were briefly described as follows: a test compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
LigandPNGBDBM769507((3R)-6-chloro-3,11-dimethyl-10-oxa-2,13,17,18,21-p...)
Affinity DataIC50: 0.980nMAssay Description:Table 1: The experimental methods were operated according to the steps in the kit instruction, and were briefly described as follows: a test compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
LigandPNGBDBM769507((3R)-6-chloro-3,11-dimethyl-10-oxa-2,13,17,18,21-p...)
Affinity DataIC50: 4.60nMAssay Description:Table 1: The experimental methods were operated according to the steps in the kit instruction, and were briefly described as follows: a test compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
LigandPNGBDBM769507((3R)-6-chloro-3,11-dimethyl-10-oxa-2,13,17,18,21-p...)
Affinity DataIC50: 4.97nMAssay Description:Table 1: The experimental methods were operated according to the steps in the kit instruction, and were briefly described as follows: a test compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetNT-3 growth factor receptor [G623R](Homo sapiens (Human))TBA
LigandPNGBDBM769507((3R)-6-chloro-3,11-dimethyl-10-oxa-2,13,17,18,21-p...)
Affinity DataIC50: 7.40nMAssay Description:Table 1: The experimental methods were operated according to the steps in the kit instruction, and were briefly described as follows: a test compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details