BDBM773584 5-(1,3-dimethyl-1H-pyrazol-5-yl)-N-((5-fluoro-2,3-dihydrobenzofuran-4-yl)methyl)-4-methoxypyrido[3,4-d]pyrimidin-8-amine::US12421228, Example 57

SMILES COc1ncnc2c(NCc3c(F)ccc4c3CCO4)ncc(-c3cc(C)nn3C)c12

InChI Key InChIKey=BSADBCJLAGZTDC-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 773584   

TargetHistone-binding protein RBBP4/Histone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12/Zinc finger protein AEBP2(Human)
Mirati Therapeutics

US Patent

LigandBDBM773584(5-(1,3-dimethyl-1H-pyrazol-5-yl)-N-((5-fluoro-2,3-...)Copy SMILESCopy InChI

Affinity DataIC50: 250nMMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
1/7/2026
Entry Details
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