BDBM774142 5-((1H-pyrazol-1- yl)methyl)- 6-methoxy-N- ((2-methoxy-5- (6-methyl- 2-oxaspiro[3.3] heptan-6- yl)phenyl)sulfonyl) picolinamide::US20250304535, Example C74

SMILES COc1ccc(C2(C)CC3(COC3)C2)cc1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(OC)n1

InChI Key InChIKey=LPESTQFXXIZGQB-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 774142   

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774142BDBM774142(5-((1H-pyrazol-1- yl)methyl)- 6-methoxy-N- ((2-met...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774142BDBM774142(5-((1H-pyrazol-1- yl)methyl)- 6-methoxy-N- ((2-met...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent