BDBM774143 5-((1H-pyrazol-1- yl)methyl)-6- methoxy-N- ((2-methoxy-5-(3- methyloxetan-3- yl)phenyl)sulfonyl) picolinamide::US20250304535, Example C75

SMILES COc1ccc(C2(C)COC2)cc1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(OC)n1

InChI Key InChIKey=ONVISWMIHKYEBU-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 774143   

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774143BDBM774143(5-((1H-pyrazol-1- yl)methyl)-6- methoxy-N- ((2-met...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774143BDBM774143(5-((1H-pyrazol-1- yl)methyl)-6- methoxy-N- ((2-met...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent