BDBM85150 CCK-A Agonist 25

SMILES COc1ccc(cc1)N(C(C)C)C(=O)CN1c2ccccc2N(c2ccccc2)C(=O)C(Cc2nn(C)c3ccccc23)C1=O

InChI Key InChIKey=VQXCMRAQZMSGPR-UHFFFAOYSA-N

Data  2 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 85150   

TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85150(CCK-A Agonist 25)
Affinity DataKi:  42.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Glaxo Wellcome Research and Development

Curated by ChEMBL
LigandPNGBDBM85150(CCK-A Agonist 25)
Affinity DataIC50: 43nMAssay Description:Binding affinity against human Cholecystokinin type A receptor by displacement of [125I]CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85150(CCK-A Agonist 25)
Affinity DataKi:  2.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85150(CCK-A Agonist 25)
Affinity DataIC50: 2.40E+3nMAssay Description:Binding affinity against human Cholecystokinin type B receptor by displacement of [125I]CCK-8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed