Report error Found 6003 Enz. Inhib. hit(s) with Target = '72 kDa type IV collagenase'
Displayed 1 to 50 (of 6003 total ) | Next | Last >>
Affinity DataIC50: 0.00400nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of recombinant human AMPA-activated MMP2 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate measured after 40 mins by spectrofluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of human recombinant MMP2 using fluorescence peptide Cy3-PLGLK(Cy5Q)AR-NH2 substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of human recombinant MMP2 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetryMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of APMA-activated recombinant human MMP-2 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0340nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-N2 as substrate preincubated for 10 to 15 mins followed by sub...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0340nMAssay Description:Inhibition of human recombinant MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-N2 as substrate preincubated for 5 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Lys-Pro- Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2 as substrate incubated for 2 hrs prior to substrate addition...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0440nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataKi: 0.0440nMAssay Description:Inhibition of MMP2 (unknown origin) using Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate incubated for 5 min followed by substrate addition and...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0449nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0460nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0480nMAssay Description:Inhibitory concentration against Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 0.0480nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0480nMAssay Description:In vitro selective inhibition against matrix metalloprotease-2 (MMP-2) using fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibition of human MMP-2 assessed as inhibition constant using MCA-Pro-Leu-Gly-Leu-DPA-Ala-Arg-NH2 substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0510nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0550nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0550nMAssay Description:Inhibition of recombinant human MMP2 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 as a substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Inhibitory activity against matrix metalloprotease-2 (MMP2)More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibitory constant against matrix metalloprotease-2More data for this Ligand-Target Pair


























3D Structure (crystal)















