Compile Data Set for Download or QSAR
Report error Found 332 Enz. Inhib. hit(s) with Target = 'ATP-binding cassette sub-family C member 9'
LigandPNGBDBM50476002(CHEMBL217511)
Affinity DataEC50:  0.676nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475970(CHEMBL426334)
Affinity DataEC50:  0.912nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475995(CHEMBL218564)
Affinity DataEC50:  1nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475999(CHEMBL214561)
Affinity DataEC50:  1.20nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475981(CHEMBL413532)
Affinity DataEC50:  1.80nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50473998(CHEMBL11983)
Affinity DataKd:  2.80nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50475993(CHEMBL217810)
Affinity DataEC50:  2.80nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475995(CHEMBL218564)
Affinity DataEC50:  3.70nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475995(CHEMBL218564)
Affinity DataEC50:  3.72nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475953(CHEMBL384564)
Affinity DataEC50:  3.89nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50476020(CHEMBL217847)
Affinity DataEC50:  6nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474006(Rilmakalim)
Affinity DataKd:  7.10nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50473999(CHEMBL275679)
Affinity DataKd:  7.40nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474017(CHEMBL12339)
Affinity DataKd:  8.90nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474024(CHEMBL269681)
Affinity DataKd:  9.80nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50475971(CHEMBL386363)
Affinity DataEC50:  9.80nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474004(Bimakalim)
Affinity DataKd:  10nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474007(CHEMBL11714)
Affinity DataKd:  11nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474001(CHEMBL12305)
Affinity DataKd:  13nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50475973(CHEMBL265269)
Affinity DataEC50:  14nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474017(CHEMBL12339)
Affinity DataKd:  15nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474011(CHEMBL276151)
Affinity DataKd:  15nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474024(CHEMBL269681)
Affinity DataKd:  15nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50473998(CHEMBL11983)
Affinity DataKd:  17nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50475983(CHEMBL216766)
Affinity DataEC50:  17nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50476011(CHEMBL216284)
Affinity DataEC50:  18nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475982(CHEMBL215375)
Affinity DataEC50:  19nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50473999(CHEMBL275679)
Affinity DataKd:  19nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50475997(CHEMBL386119)
Affinity DataEC50:  20nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475997(CHEMBL386119)
Affinity DataEC50:  20nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474001(CHEMBL12305)
Affinity DataKd:  20nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50062397(N''-cyano-N-(1,1-dimethylpropyl)-N'-pyridin-3-ylgu...)
Affinity DataEC50:  22nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475972(CHEMBL216546)
Affinity DataEC50:  22.9nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475972(CHEMBL216546)
Affinity DataEC50:  23nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474002(CHEMBL267301)
Affinity DataKd:  23nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474007(CHEMBL11714)
Affinity DataKd:  23nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50475972(CHEMBL216546)
Affinity DataEC50:  23nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50476003(CHEMBL426160)
Affinity DataEC50:  26.9nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475977(CHEMBL386582)
Affinity DataEC50:  26.9nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50062397(N''-cyano-N-(1,1-dimethylpropyl)-N'-pyridin-3-ylgu...)
Affinity DataKi:  27nMAssay Description:Binding affinity was determined by displacement of [3H]P1075 from its binding sites in canine cardiac membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 9(Rat)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50474006(Rilmakalim)
Affinity DataKd:  27nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50476003(CHEMBL426160)
Affinity DataEC50:  27nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50476013(CHEMBL261996)
Affinity DataEC50:  27nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475961(CHEMBL214841)
Affinity DataEC50:  27.5nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475991(CHEMBL320983)
Affinity DataEC50:  28nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475961(CHEMBL214841)
Affinity DataEC50:  28nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475966(CHEMBL384576)
Affinity DataEC50:  28nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475961(CHEMBL214841)
Affinity DataEC50:  29nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50476004(CHEMBL386323)
Affinity DataEC50:  30nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50044253(CHEMBL11684 | (3S,4R)-3-hydroxy-2,2-dimethyl-4-(2-...)
Affinity DataEC50:  35nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
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