Compile Data Set for Download or QSAR
Report error Found 144 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A/B'
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 0.700nMAssay Description:In vitro Inhibitory activity of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT (serotonin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138499(2-Phenethyl-4,5-dihydro-1H-imidazole | CHEMBL14210)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50224952(CHEMBL441014)
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
LigandPNGBDBM50225462(CHEMBL554775)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138435(N-(12-Guanidino-dodecyl)-N-(1-phenethyl-piperidin-...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50225466(CHEMBL544509)
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
LigandPNGBDBM50225455(CHEMBL555332)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
LigandPNGBDBM50225456(CHEMBL545207)
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
LigandPNGBDBM50225453(CHEMBL541803)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473129(Phenamazoline)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50224950(CHEMBL8877)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50228339(CHEMBL58177)
Affinity DataIC50: 42nMAssay Description:In vitro inhibitory activity against Monoamine oxidase in baboon brain was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2019
Entry Details Article
PubMed
LigandPNGBDBM50225463(CHEMBL538992)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Bovine)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50121457(1-[3-(2,4-Dihydroxy-phenyl)-5-m-tolyl-4,5-dihydro-...)
Affinity DataKi:  50nMAssay Description:Inhibitory activity against Monoamine oxidase from Bovine brain mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50225449(CHEMBL543328)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Bovine)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50121456(1-[3-(2,4-Dihydroxy-phenyl)-5-o-tolyl-4,5-dihydro-...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against Monoamine oxidase from Bovine brain mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50225452(CHEMBL553995)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50474215(CHEMBL2092860)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179394(CHEMBL68608)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138436(N-(8-Guanidino-octyl)-N-(1-phenethyl-piperidin-4-y...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224947(CHEMBL8848)
Affinity DataIC50: 140nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50224967(CHEMBL275108)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
LigandPNGBDBM50225464(CHEMBL545677)
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
LigandPNGBDBM50224970(CHEMBL8695)
Affinity DataIC50: 170nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473618(CHEMBL337945)
Affinity DataKi:  182nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473198(CHEMBL13925)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50025082(2-(4-Chloro-2,3-dihydro-1H-indol-5-yl)-1-methyl-et...)
Affinity DataIC50: 200nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50003138(CHEMBL542711 | Methyl-(1-methyl-nonyl)-prop-2-ynyl...)
Affinity DataIC50: 210nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50224948(CHEMBL8712)
Affinity DataIC50: 240nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
LigandPNGBDBM50224950(CHEMBL8877)
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473621(CHEMBL131775)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 280nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50003149(CHEMBL542465 | Methyl-(1-methyl-undecyl)-prop-2-yn...)
Affinity DataIC50: 280nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50421578(CHEMBL13789)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50003140(CHEMBL541325 | Methyl-(1-methyl-hexyl)-prop-2-ynyl...)
Affinity DataIC50: 320nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50025084(2-(1-Ethyl-6-methyl-2,3-dihydro-1H-indol-5-yl)-1-m...)
Affinity DataIC50: 330nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224966(CHEMBL8467)
Affinity DataIC50: 360nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
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