Compile Data Set for Download or QSAR
maximum 50k data
Found 3895 Enz. Inhib. hit(s) with Target = 'Casein kinase II subunit alpha'
TargetCasein kinase II subunit alpha'/beta(Homo sapiens (Human))
Cylene Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataKi:  0.220nMAssay Description:Inhibition of human recombinant CK2alpha/CK2beta using RRRDDDSDDD peptide as substrate by radiometric assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214466(CHEMBL398149 | N-(3-(8-cyano-4-(cyclopropylamino)p...)
Affinity DataKi:  0.260nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214473(CHEMBL230354 | N-(3-(8-CYANO-4-(PHENYLAMINO)PYRAZO...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataKi:  0.380nMAssay Description:Inhibition of CK2alpha (unknown origin) using RRRADDSDDDDD as substrate in presence of [gamma33P]-ATP by autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataKi:  0.380nMAssay Description:Inhibition of CK2 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50566496(CHEMBL4846181)
Affinity DataKi:  0.420nMAssay Description:Inhibition of CK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374656(CHEMBL401544)
Affinity DataKi:  0.800nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374653(CHEMBL271020)
Affinity DataKi:  1.30nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374654(CHEMBL271645)
Affinity DataKi:  1.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374662(CHEMBL256401)
Affinity DataKi:  1.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214454(CHEMBL230462 | N-(3-(8-cyano-4-(cyclobutylamino)py...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374658(CHEMBL401614)
Affinity DataKi:  2nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374651(CHEMBL257219)
Affinity DataKi:  2.20nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374655(CHEMBL401945)
Affinity DataKi:  2.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374657(CHEMBL257736)
Affinity DataKi:  3.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374660(CHEMBL256189)
Affinity DataKi:  3.60nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374659(CHEMBL402246)
Affinity DataKi:  4nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214444(2-(p-toluidino)-4-(phenylamino)pyrazolo[1,5-a][1,3...)
Affinity DataKi:  5nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214465(2-(4-chlorobenzylamino)-4-(phenylamino)pyrazolo[1,...)
Affinity DataKi:  5nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374661(CHEMBL402306)
Affinity DataKi:  5.20nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508987(CHEMBL4465651)
Affinity DataKi:  7nMAssay Description:Inhibition of CK2alpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214477(4-(phenylamino)-2-(4-(pyridin-2-yl)piperazin-1-yl)...)
Affinity DataKi:  7nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374652(CHEMBL271848)
Affinity DataKi:  7.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214474(CHEMBL230353 | N-(3-(8-cyano-4-(phenethylamino)pyr...)
Affinity DataKi:  8nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214460(2-(CYCLOHEXYLMETHYLAMINO)-4-(PHENYLAMINO)PYRAZOLO[...)
Affinity DataKi:  8nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214448(2-(3,4-dimethoxyphenylamino)-4-(phenylamino)pyrazo...)
Affinity DataKi:  9nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214464(CHEMBL230568 | N-(3-(8-methyl-4-(phenylamino)pyraz...)
Affinity DataKi:  11nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214450(2-(3,4-dihydroisoquinolin-2(1H)-yl)-4-(phenylamino...)
Affinity DataKi:  11nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214457(2-(2,3-dihydro-1H-inden-2-ylamino)-4-(phenylamino)...)
Affinity DataKi:  12nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214453(2-(isopentylamino)-4-(phenylamino)pyrazolo[1,5-a][...)
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214468(4-(phenylamino)-2-(pyrrolidin-1-yl)pyrazolo[1,5-a]...)
Affinity DataKi:  14nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214446(2,4-bis(phenylamino)pyrazolo[1,5-a][1,3,5]triazine...)
Affinity DataKi:  15nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214443(CHEMBL230673 | N-(3-(8-bromo-4-(cyclopropylamino)p...)
Affinity DataKi:  17nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University Of Padova

LigandPNGBDBM34046(iodinated benzimidazole, 9a)
Affinity DataKi:  19nM ΔG°:  -45.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM4078(6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0...)
Affinity DataKi:  20nMAssay Description:Inhibition of CK2alpha (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University Of Padova

LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  23nM ΔG°:  -45.4kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214471(2-(4-(diethylamino)phenylamino)-4-(phenylamino)pyr...)
Affinity DataKi:  23nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214452(2-(4-ETHYLPIPERAZIN-1-YL)-4-(PHENYLAMINO)PYRAZOLO[...)
Affinity DataKi:  24nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)
Affinity DataKi:  24nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374663(CHEMBL404508)
Affinity DataKi:  24nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214446(2,4-bis(phenylamino)pyrazolo[1,5-a][1,3,5]triazine...)
Affinity DataKi:  24nMAssay Description:Inhibition of corn CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University Of Padova

LigandPNGBDBM34044(iodinated benzimidazole, 7a)
Affinity DataKi:  24nM ΔG°:  -45.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University Of Padova

LigandPNGBDBM34051(iodinated benzimidazole, 14)
Affinity DataKi:  27nM ΔG°:  -44.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)
Affinity DataKi:  31nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50420549(CHEMBL2087008)
Affinity DataKi:  32nMAssay Description:Inhibition of CK2alpha (unknown origin) using RRRADDSDDDDD as substrate in presence of [gamma33P]-ATP by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214451(CHEMBL230463 | N-(3-(4-(cyclopropylamino)-8-methyl...)
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul Ii Catholic University Of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 3895 total ) | Next | Last >>
Jump to: