Report error Found 3519 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A'
Affinity DataAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataKd: 1.90nM EC50: 28nMAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 3.5nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 1.40nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.900nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.5nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 104nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 4nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 37nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.700nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 6.90nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 1.30nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.990nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 3.70nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.640nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.100nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.320nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 3.70nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 280nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.00900nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Human)
Hadassah-University Hospital
Curated by ChEMBL
Hadassah-University Hospital
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type CCKA receptor expressed in CHO-K1 cells assessed as calcium level by FDSS assayMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type CCKA receptor expressed in CHO-K1 cells assessed as calcium level by FDSS assayMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type CCKA receptor expressed in CHO-K1 cells assessed as calcium level by FDSS assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Displacement of [125I]CCK-8s from recombinant human CCK1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.447nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.166nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0251nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 269nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.107nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at human CCK1R expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair








































