Report error Found 324 Enz. Inhib. hit(s) with Target = 'Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A'
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Mus musculus)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Inhibition of PDE11A4 in mouse HT-22 cells assessed as reduction in cAMP hydrolytic activity using [3H]-cAMP as substrate pretreated with compound fo...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Mus musculus)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Inhibition of PDE11A4 in mouse HT-22 cells assessed as reduction in cAMP hydrolytic activity using [3H]-cAMP as substrate pretreated with compound fo...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Mus musculus)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Inhibition of PDE11A4 in mouse HT-22 cells assessed as reduction in cAMP hydrolytic activity using [3H]-cAMP as substrate pretreated with compound fo...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Mus musculus)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataEC50: 2.20E+4nMAssay Description:Inhibition of PDE11A4 in mouse HT-22 cells assessed as reduction in cGMP hydrolytic activity using [3H]-cGMP as substrate pretreated with compound fo...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Mus musculus)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Inhibition of PDE11A4 in mouse HT-22 cells assessed as reduction in cGMP hydrolytic activity using [3H]-cGMP as substrate pretreated with compound fo...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Mus musculus)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataEC50: 2.20E+4nMAssay Description:Inhibition of PDE11A4 in mouse HT-22 cells assessed as reduction in cGMP hydrolytic activity using [3H]-cGMP as substrate pretreated with compound fo...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of PDE11A (unknown origin)More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of N-terminal GST-tagged full length recombinant human PDE11A expressed in Baculovirus infected Sf9 insect cells using FAM-cAMP as substra...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PDE11A4 expressed in baculovirus infected sf9 cells using FAM-cyclic-3',5-AMP as su...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Inhibition of N-terminal GST-tagged full length recombinant human PDE11A expressed in Baculovirus infected Sf9 insect cells using FAM-cAMP as substra...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant PDE11A-mediated hydrolysis of cGMP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 11.8nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PDE11A4 (1 to 943 residues) expressed in Sf9 insect cells using cAMP as substrateMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PDE11A4 (1 to 943 residues) expressed in Sf9 insect cells using cAMP as substrateMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of N-terminal GST-tagged human PDE11A4 expressed in baculovirus infected sf9 cells using [3H]cGMP as substrate measured after 30 mins by s...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PDE11A4 (1 to 943 residues) expressed in Sf9 insect cells using cAMP as substrateMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human phosphodiesterase 11More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of full length recombinant human PDE11A4 using 3',5'-[3H]cGMP as substrate after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of PDE11A catalytic domain (588 to 911 residues) (unknown origin) expressed in Escherichia coli BL21 using 3H-cAMP as substrate after 15 m...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PDE11A4 expressed in baculovirus infected sf9 cells using FAM-cyclic-3',5-AMP as su...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:In vitro enzyme assays were conducted via the Ba(OH)2 precipitation method of Wang et al. (32) using recombinant human PDE11A4, PDE10A1, PDE5A1, PDE6...More data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant PDE11A-mediated hydrolysis of cGMP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PDE11A4 (1 to 943 residues) expressed in Sf9 insect cells using cAMP as substrateMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibitory activity against phosphodiesterase 11 (PDE11) obtained from recombinant Sf9 expressionMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PDE11A4 (1 to 943 residues) expressed in Sf9 insect cells using cAMP as substrateMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PDE11A4 (1 to 943 residues) expressed in Sf9 insect cells using cAMP as substrateMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PDE11A4 (1 to 943 residues) expressed in Sf9 insect cells using cAMP as substrateMore data for this Ligand-Target Pair
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL
TargetDual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A(Human)
Montclair State University
Curated by ChEMBL
Montclair State University
Curated by ChEMBL


































