Affinity DataIC50: 3nMAssay Description:Inhibition of EphA5 by [gamma33-P]ATP based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10.3nMAssay Description:Inhibition of human EPHA5 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21.5nMAssay Description:Inhibition of human EPHA5 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of N-terminal GST-tagged human EphA5 catalytic domain expressed in baculovirus preincubated for 5 mins measured after 10 mins in presence ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of ephrin-A1-Fc from EphA5 receptor Fc ectodomain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from rat EphA5 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human EphA5 (655 to 956 residues) using poly(Glu, Tyr) 4:1 as substrate measured after 40 mins in presence of [gamma33ATP] ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EPHA5 using poly[Glu:Tyr] (4:1) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of EPHA5More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 using Z-Leu-Arg-AMC as substrate compound treated for 30 min before substrate addition by...More data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 95nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Average Binding Constant for EPHA5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 95nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.90E+3nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 95nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Average Binding Constant for EPHA5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 360nMAssay Description:Average Binding Constant for EPHA5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Average Binding Constant for EPHA5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Average Binding Constant for EPHA5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:Average Binding Constant for EPHA5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 5.90E+3nMAssay Description:Average Binding Constant for EPHA5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Binding affinity to human EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHA5More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair