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Report error Found 84 Enz. Inhib. hit(s) with Target = 'Ectonucleoside triphosphate diphosphohydrolase 1'
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50546288(CHEMBL4743437)
Affinity DataIC50: 10nMAssay Description:Inhibition of CD39 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50546280(CHEMBL4761506)
Affinity DataIC50: 10nMAssay Description:Inhibition of CD39 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50527134(CHEMBL4471306 | US20230295213, Compound a)
Affinity DataIC50: 10nMAssay Description:Inhibition of CD39 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50615669(CHEMBL5277365)
Affinity DataIC50: 50nMAssay Description:Inhibition of human NTPDase1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50378649(CHEMBL597197)
Affinity DataKi:  328nMAssay Description:Inhibition of rat CD39 expressed in CHO cells using ATP as substrate incubated for 10 mins by UV absorbance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50615668(CHEMBL5283491)
Affinity DataIC50: 500nMAssay Description:Inhibition of human NTPDase1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Mouse)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 500nMAssay Description:Inhibition of mouse CD39More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50010311(CHEMBL2364580)
Affinity DataKi:  800nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Cheng-Prus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50552127(CHEMBL4750781)
Affinity DataKi:  800nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Dixon and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50552126(CHEMBL4797422)
Affinity DataKi:  900nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Dixon and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468622(CHEMBL4285649)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468632(CHEMBL4293491)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Mouse)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50241052(1,2,3,4,6-pentakis-O-(3,4,5-trihydroxybenzoyl)-bet...)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of mouse CD39More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468637(CHEMBL4295005)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50307836(Sodium 1-Amino-4-(2-anthracenylamino)-9,10-dioxo-9...)
Affinity DataKi:  2.59E+3nMAssay Description:Inhibition of human NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50552128(CHEMBL4787368)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human CD39 expressed in green monkey Cos-7 cells using ATP as substrate preincubated for 3 mins followed by substrate addition by malac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50010311(CHEMBL2364580)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Malachite ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468623(CHEMBL4290501)
Affinity DataIC50: 6.21E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468631(CHEMBL4291645)
Affinity DataIC50: 9.02E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM511076(2-(((2R,3S,4R,5R)-5-(6-amino-2-chloro-9H-purin-9-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length human CD39 expressed in human K562 cells incubated for 40 mins in presence of ATP by Kinase Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Bovine)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50369522(CHEMBL610358)
Affinity DataKi:  1.00E+4nMAssay Description:Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50561221(CHEMBL4745473 | US11377469, Example 95)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CD39 expressed in CHO cells incubated for 4 hrs before addition of AMP and further incubated for 60 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468629(CHEMBL4279910)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50268725(sodium 1-amino-4-(4-hydroxyphenylamino)-9,10-dioxo...)
Affinity DataKi:  1.07E+4nMAssay Description:Inhibition of human NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50179358(CHEMBL1206141)
Affinity DataKi:  1.10E+4nMAssay Description:Competitive inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 15 mins by Dixo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50227019(sodium 1-amino-4-(4-chlorophenylamino)-9,10-dioxo-...)
Affinity DataKi:  1.57E+4nMAssay Description:Inhibition of rat CD39 expressed in CHO cells using ATP as substrate incubated for 10 mins by UV absorbance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Bovine)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50369524(CHEMBL607720)
Affinity DataKi:  1.60E+4nMAssay Description:Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human CD39 expressed in green monkey Cos-7 cells using ATP as substrate preincubated for 3 mins followed by substrate addition by malac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of human NTPDase1 expressed in African green monkey COS7 cell membrane fraction using ATP as substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50527649(CHEMBL4467828)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CD39 expressed in CHO cells using ATP as substrate preincubated for 1 hr followed by substrate addition and measured after 50 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50552129(CHEMBL4744335)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of rat CD39 expressed in CHO cells using ATP as substrate incubated for 10 mins by UV absorbance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50029031(CHEMBL223344 | 1-Amino-4-{4-[4-chloro-6-(3-sulfo-p...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50187685(CHEMBL597418)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human NTPDase1 expressed in CHO cells using ADP as substrate incubated for 10 mins by capillary electrophoresis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50029031(CHEMBL223344 | 1-Amino-4-{4-[4-chloro-6-(3-sulfo-p...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of rat recombinant NTPDase1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50029031(CHEMBL223344 | 1-Amino-4-{4-[4-chloro-6-(3-sulfo-p...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of rat NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM23722(4-chloro-1-[(4-chlorophenyl)carbonyl]-3,5-dimethyl...)
Affinity DataIC50: 2.24E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50195359(ARL-67156 | CHEMBL223145)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of rat recombinant NTPDase1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50195359(ARL-67156 | CHEMBL223145)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50552126(CHEMBL4797422)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Malachite ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Bovine)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50369523(CHEMBL612159)
Affinity DataKi:  3.10E+4nMAssay Description:Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50552127(CHEMBL4750781)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Malachite ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468627(CHEMBL390695)
Affinity DataIC50: 3.61E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468626(CHEMBL4280275)
Affinity DataIC50: 3.65E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468634(CHEMBL4283075)
Affinity DataIC50: 3.72E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468639(CHEMBL4291589)
Affinity DataIC50: 3.85E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Human)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50307835(Sodium 1-amino-4-[4-fluoro-2-carboxyphenylamino]-9...)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of human NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468628(CHEMBL4286443)
Affinity DataIC50: 4.15E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468636(CHEMBL4288181)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468633(CHEMBL4283728)
Affinity DataIC50: 4.42E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rat)
Arcus Biosciences

Curated by ChEMBL
LigandPNGBDBM50468624(CHEMBL4284994)
Affinity DataIC50: 4.45E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
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