Compile Data Set for Download or QSAR
Report error Found 213 Enz. Inhib. hit(s) with Target = 'Heat shock protein 75 kDa, mitochondrial'
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718142(US20250042884, Compound I-8)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718139(US20250042884, Compound I-4)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718140(US20250042884, Compound I-5)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718138(US20250042884, Compound I-3)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718136(US20250042884, Compound I-1)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50439624(CHEMBL1910764)
Affinity DataKd:  5.80nMAssay Description:Binding affinity to recombinant human Trap-1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50439623(CHEMBL2419342)
Affinity DataKd:  5.90nMAssay Description:Binding affinity to recombinant human Trap-1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718143(US20250042884, Compound I-9)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718144(US20250042884, Compound I-11)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718141(US20250042884, Compound I-6)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718137(US20250042884, Compound I-2)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataKd:  10nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) expressed in Escherichia coli BL21-Cod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718145(US20250042884, Comparative Compound 2)
Affinity DataIC50: 15.5nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataKi:  16nMAssay Description:Binding affinity to human recombinant TRAP1 after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50136674((R)-duloxetine | LY248685 | (3R)-N-methyl-3-(1-nap...)
Affinity DataIC50: 35.5nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50439621(STA-9090 | GANETESPIB)
Affinity DataIC50: 38nMAssay Description:Inhibition of TRAP1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataIC50: 38nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50650777(CHEMBL5633816)
Affinity DataKd:  40nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50650766(CHEMBL5633903)
Affinity DataKd:  40nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50439621(STA-9090 | GANETESPIB)
Affinity DataIC50: 51nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50439625(CHEMBL2419341)
Affinity DataKd:  52nMAssay Description:Binding affinity to recombinant human Trap-1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571897(CHEMBL4866705)
Affinity DataIC50: 58nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571903(CHEMBL4863672)
Affinity DataIC50: 62nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM20800(CHEMBL467399 | 6-chloro-9-[(4-methoxy-3,5-dimethyl...)
Affinity DataKi:  62nMAssay Description:Binding affinity to human recombinant TRAP1 after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571908(CHEMBL4864922)
Affinity DataIC50: 64nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571896(CHEMBL4869481)
Affinity DataIC50: 66nMAssay Description:Inhibition of TRAP1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571896(CHEMBL4869481)
Affinity DataIC50: 66nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718146(US20250042884, Compound of formula A)
Affinity DataIC50: 75.5nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571901(CHEMBL4879021)
Affinity DataIC50: 77nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50240873(CHEMBL4068596)
Affinity DataIC50: 79nMAssay Description:Inhibition of FITC3-labeled PU-H71 binding to recombinant human N-terminal His6-tagged TRAP1 (60 to 561 residues) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50650767(CHEMBL5633571)
Affinity DataKd:  80nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571921(CHEMBL4866958)
Affinity DataIC50: 82nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571910(CHEMBL4876871)
Affinity DataIC50: 83nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50650774(CHEMBL5633012)
Affinity DataKd:  90nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571923(CHEMBL4863988)
Affinity DataIC50: 90nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM20800(CHEMBL467399 | 6-chloro-9-[(4-methoxy-3,5-dimethyl...)
Affinity DataIC50: 90nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50650771(CHEMBL5632075)
Affinity DataKd:  90nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571918(CHEMBL4871630)
Affinity DataIC50: 100nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50240875(CHEMBL4080323)
Affinity DataIC50: 138nMAssay Description:Inhibition of FITC3-labeled PU-H71 binding to recombinant human N-terminal His6-tagged TRAP1 (60 to 561 residues) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50240873(CHEMBL4068596)
Affinity DataIC50: 143nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50650776(CHEMBL5631806)
Affinity DataKd:  160nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571900(CHEMBL4857569)
Affinity DataIC50: 170nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571909(CHEMBL4860652)
Affinity DataIC50: 178nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataIC50: 192nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50031735(CHEMBL3360305)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataIC50: 205nMAssay Description:Displacement of PU-FITC3 from recombinant TRAP-1 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataIC50: 205nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50571922(CHEMBL4850126)
Affinity DataIC50: 230nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50650763(CHEMBL5633174)
Affinity DataKd:  230nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataKd:  240nMAssay Description:Binding affinity to TRAP1 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
Displayed 1 to 50 (of 213 total ) | Next | Last >>
Jump to: