Compile Data Set for Download or QSAR
Report error Found 256 Enz. Inhib. hit(s) with Target = 'Homeodomain-interacting protein kinase 1'
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50400734BDBM50400734(CHEMBL1591531)
Affinity DataIC50: 0.367nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110183BDBM50110183(Abemaciclib | LY-2835219 | US10696678, Example LY2...)
Affinity DataKi: <10nMAssay Description:Inhibition of wild-type human partial length HIPK1 (M146 to I555 residues) expressed in mammalian expression system assessed as residual activity at ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563555BDBM50563555(CHEMBL4750420)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563556BDBM50563556(CHEMBL4743939)
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 124970BDBM124970(US8765747, 2)
Affinity DataKd:  34nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172243BDBM50172243(CHEMBL3103192)
Affinity DataIC50: 40nMAssay Description:Inhibition of Hipk1 (unknown origin) by quantitative PCRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563541BDBM50563541(CHEMBL4743730)
Affinity DataIC50: 51nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4814BDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  55nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563554BDBM50563554(CHEMBL4790030)
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50242737BDBM50242737((R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimet...)
Affinity DataKd:  93nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399540BDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17055BDBM17055((9S)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydr...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809279BDBM809279((Z)-2-(benzo[d]thiazol-6-ylamino)-5-((1-methyl-1H-...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 16673BDBM16673(BAY439006 | CHEMBL1336 | BAY 43-9006 | 4-[4-({[4-c...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50242737BDBM50242737((R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimet...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809267BDBM809267((Z)-5-(benzo[d]thiazol-5-ylmethylene)-2-(benzo[d]t...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563539BDBM50563539(CHEMBL4762964)
Affinity DataIC50: 125nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50248614BDBM50248614(CHEMBL4066819)
Affinity DataKd:  160nMAssay Description:Binding affinity to partial length human HIPK1 (M146 to I555 residues) expressed in mammalian expression system by kinome scan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2019
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31085BDBM31085(cid_11409972 | 1-[4-[(4-ethylpiperazin-1-yl)methyl...)
Affinity DataKd:  170nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563537BDBM50563537(CHEMBL4789951)
Affinity DataIC50: 177nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50560704BDBM50560704(CHEMBL4754195)
Affinity DataIC50: 187nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50560704BDBM50560704(CHEMBL4754195)
Affinity DataIC50: 187nMAssay Description:Inhibition of human HIPK1 by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563538BDBM50563538(CHEMBL4797457)
Affinity DataIC50: 209nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563540BDBM50563540(CHEMBL4740998)
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 15138BDBM15138(Biochemistry 469551 Compound 11 | 5-indazolyl pyri...)
Affinity DataKd:  230nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17055BDBM17055((9S)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydr...)
Affinity DataKd:  230nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563557BDBM50563557(CHEMBL4790791)
Affinity DataIC50: 235nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563533BDBM50563533(CHEMBL4777288)
Affinity DataIC50: 248nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563535BDBM50563535(CHEMBL4791451)
Affinity DataIC50: 264nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563544BDBM50563544(CHEMBL4778370)
Affinity DataIC50: 278nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563534BDBM50563534(CHEMBL4778153)
Affinity DataIC50: 285nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36409BDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataKd:  300nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347750BDBM50347750(CHEMBL1802358)
Affinity DataKd:  320nMAssay Description:Binding affinity to HIPK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563536BDBM50563536(CHEMBL4741919)
Affinity DataIC50: 354nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50355504BDBM50355504(CHEMBL1908393)
Affinity DataKd:  420nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50355496BDBM50355496(CHEMBL1908397)
Affinity DataKd:  430nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25013BDBM25013(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Affinity DataKd:  510nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4552BDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataKd:  520nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50563551BDBM50563551(CHEMBL4777533)
Affinity DataIC50: 545nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50627498BDBM50627498(CHEMBL5405969 | US12643887, Example 31)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809235BDBM809235((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((4-methox...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50627541BDBM50627541(CHEMBL5418020 | US12643887, Example 6)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809273BDBM809273((Z)-2-((1H-indol-5-yl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809256BDBM809256((Z)-5-((1-methyl-1H-benzo[d]imidazol-6-yl)methylen...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809297BDBM809297((Z)-5-(benzo[d]thiazol-6-ylmethylene)-24(1-methyl-...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809280BDBM809280((Z)-5-((1H-benzo[d]imidazol-6-yl)methylene)-2-(ben...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809295BDBM809295(N-(1,3-benzothiazol-6-yl)-N-[(4Z)-4-[(1,3-benzothi...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809215BDBM809215((Z)—N-(4-(benzo[d][1,3]dioxol-5-ylmethylene)-5-oxo...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809302BDBM809302((Z)-2-((4-aminophenyl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Korea Institute of Science & Technology (Kist)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 809296BDBM809296((Z)-2-(benzo[d]thiazol-6-ylamino)-5-(thiazol-5-ylm...)
Affinity DataIC50: 550nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

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