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Report error Found 171 Enz. Inhib. hit(s) with Target = 'Leukotriene B4 receptor 2'
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50013889(5,12-Dihete | CHEMBL65061 | LTB4 | 5,12-Hete | (S-...)
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50013889(5,12-Dihete | CHEMBL65061 | LTB4 | 5,12-Hete | (S-...)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81801(CAS_5283121 | NSC_5283121 | LTC4)
Affinity DataKi:  3.35nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50292408(5S-hydroxy-6R-(S-cysteinylglycinyl)-7E,9E,11E,14Z-...)
Affinity DataKi:  3.48nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM85081(CAS_5280876 | NSC_5280876 | 12-oxo-LTB4)
Affinity DataKi:  7.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81521(NSC_1589 | CAS_1589 | 20-OH-LTB4)
Affinity DataKi:  7.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81522(CGS 23130)
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM85702(NSC_5283125 | CAS_5283125 | LTB5)
Affinity DataKi:  9.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81521(NSC_1589 | CAS_1589 | 20-OH-LTB4)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50001611((Z)-3-{3-(2-Carboxy-ethyl)-4-[6-(4-methoxy-phenyl)...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50544639(CHEMBL4637519)
Affinity DataKd:  15nMAssay Description:Displacement of [3H]LTB4 from HA-epitope tagged human BLT2 expressed in CHOK1 cells incubated for 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561399(CHEMBL4761937)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561396(CHEMBL4789730)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81522(CGS 23130)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561401(CHEMBL4777675)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561373(CHEMBL4754213)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561372(CHEMBL4793225)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50544639(CHEMBL4637519)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50001611((Z)-3-{3-(2-Carboxy-ethyl)-4-[6-(4-methoxy-phenyl)...)
Affinity DataKi:  35nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561382(CHEMBL4759277)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561384(CHEMBL4742371)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50472434(CHEMBL2112887)
Affinity DataIC50: 40nMAssay Description:Inhibition of binding of [3H]LTB4 (1 nM) to intact human polymorphonuclear leukocytes (PMNs)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM85696(LTB4-20-hydroxy)
Affinity DataKi:  41nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561389(CHEMBL4753057)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561394(CHEMBL4781057)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561365(CHEMBL4785658)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561376(CHEMBL4752602)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561370(CHEMBL4755616)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561381(CHEMBL4753841)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561371(CHEMBL4778464)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561363(CHEMBL4745083)
Affinity DataEC50:  61nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81519(LY 255283 | CHEMBL15766 | CAS_117690-79-6 | CGS 23...)
Affinity DataKi:  66nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50577226(CHEMBL4872989)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human BLT2 overexpressed in CHO-K1 cells assessed as accumulation of inositol monophosphate measured after 90 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561367(CHEMBL4748248)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50472441(CHEMBL153555)
Affinity DataIC50: 80nMAssay Description:Inhibition of binding of [3H]LTB4 (1 nM) to intact human polymorphonuclear leukocytes (PMNs)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50013889(5,12-Dihete | CHEMBL65061 | LTB4 | 5,12-Hete | (S-...)
Affinity DataKi:  93nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561366(CHEMBL4746259)
Affinity DataEC50:  96nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561385(CHEMBL4755611)
Affinity DataEC50:  103nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81519(LY 255283 | CHEMBL15766 | CAS_117690-79-6 | CGS 23...)
Affinity DataKi:  116nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM79408((5R)-6-[6-[(1E,3S,5Z)-3-hydroxyundeca-1,5-dienyl]p...)
Affinity DataKi:  120nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM81520(CGS 23113)
Affinity DataKi:  124nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50001610(CHEMBL14823 | CGS 24115 | 7-[3-(4-Acetyl-3-methoxy...)
Affinity DataKi:  131nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50652323(CHEMBL5641746)
Affinity DataKi:  132nMAssay Description:Displacement of 3H-LTB4 from human BLT2 expressed in CHO cell membrane assessed as inhibition constant incubated for 60 mins by liquid scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561369(CHEMBL4757022)
Affinity DataEC50:  134nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50001610(CHEMBL14823 | CGS 24115 | 7-[3-(4-Acetyl-3-methoxy...)
Affinity DataKi:  137nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2011
Entry Details
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50317628(4-{2-(2-Carboxy-ethyl)-3-[6-(3,5-di-pyridin-4-yl-p...)
Affinity DataIC50: 143nMAssay Description:Antagonist activity at FLAG-tagged human BLT2 receptor expressed in HEK293 cells assessed as inhibition of LTB4-stimulated calcium mobilization prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50212626(LY-255283)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]LTB4 from HA-epitope tagged human BLT2 expressed in CHOK1 cells incubated for 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM85703(NSC_5283162 | CAS_5283162 | ETE-12-Oxo)
Affinity DataKi:  155nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50317626(4-{3-[6-(3-5-Benzo[1,3]dioxolyl-5-thiophen-3-ylphe...)
Affinity DataIC50: 164nMAssay Description:Antagonist activity at FLAG-tagged human BLT2 receptor expressed in HEK293 cells assessed as inhibition of LTB4-stimulated calcium mobilization prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 2(Human)
Ciba-Geigy

Curated by PDSP Ki Database
LigandPNGBDBM50561368(CHEMBL4788291)
Affinity DataEC50:  167nMAssay Description:Agonist activity at human BLT2 isoform 2 expressed in CHO-K1 cells over-expressing GNA14 assessed as stimulation of IP-1 accumulation incubated for 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
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