Report error Found 551 Enz. Inhib. hit(s) with Target = 'Methionine--tRNA ligase'
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 0.452nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of 1 mM A...More data for this Ligand-Target Pair
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 0.493nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of 50 uM ...More data for this Ligand-Target Pair
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 0.593nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of 500 uM...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory concentration against Methionyl-tRNA synthetase in a pyrophosphate exchange assayMore data for this Ligand-Target Pair
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 1.20nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of 50 uM ...More data for this Ligand-Target Pair
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 1.40nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of 20 uM ...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 3.10nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of 20 uM ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 4.90nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Binding affinity to Enterococcus faecalis type 1 MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant by ITC analysi...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
TargetMethionine--tRNA ligase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Sun Yat-sen University
Curated by ChEMBL
Sun Yat-sen University
Curated by ChEMBL
Affinity DataKd: 6nMAssay Description:Binding affinity to Staphylococcus aureus MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of 1 mM A...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS(methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Compound tested for inhibition of Staphylococcus aureus MRS (methionyl tRNA synthetase) in aminoacylation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against Staphylococcus aureus methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against Escherichia coli Methionyl-tRNA synthetase was determinedMore data for this Ligand-Target Pair

3D Structure (crystal)








































