Report error Found 60 Enz. Inhib. hit(s) with Target = 'N-acetylated-alpha-linked acidic dipeptidase 2'
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 1.5nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 1.70nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 4.30nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 4.5nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 4.80nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 6.30nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 6.40nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 7nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 8nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 14.4nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 14.9nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 23nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 24nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 30nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 41nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 53nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 67nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 87nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 95.3nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 106nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 169nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: >300nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: >300nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 300nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: >300nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 335nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 338nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 392nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: >500nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: >500nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: >500nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: >500nMAssay Description:Binding affinity to human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 505nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 939nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.11E+3nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.29E+3nMAssay Description:In vitro inhibitory activity against human Glutamate carboxypeptidase II by using fluorescent assayMore data for this Ligand-Target Pair
TargetN-acetylated-alpha-linked acidic dipeptidase 2(Human)
University of Illinois At Chicago
Curated by ChEMBL
University of Illinois At Chicago
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Displacement of [177Lu]LU-PSMA-617 from human recombinant GCPIII assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair

















































