Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'NEDD8-conjugating enzyme Ubc12'
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  108nMAssay Description:Binding affinity to human UBE2M incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50245225(CHEMBL4099097 | US11116757, No. A15)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to N-terminally acetylated human UBE2MMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50311743(CHEMBL487992 | GARTANIN)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of Ubc12 (unknown origin)-neddylation incubated for 30 mins in presence of ATP by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
LigandPNGBDBM50478216(CHEBI:600520 | Micafungin | Mycamine)
Affinity DataIC50: 3.99E+4nMAssay Description:Inhibition of UBE2M neddylation in human AGS cells incubated for 3 days by immunoblot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed