Report error Found 214 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor'
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 4.90nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 6.90nMAssay Description:Agonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as increase Ca2+ mobilization after 3 mins by Fluo-4 AM-based ...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 10.4nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 30.2nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 37.5nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]QRFP43 from human GPR103 receptor expressed in HEK cells after 90 mins incubation by scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 43.2nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Agonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as increase Ca2+ mobilization after 3 mins by Fluo-4 AM-based ...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 66nMAssay Description:Agonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as increase Ca2+ mobilization after 3 mins by Fluo-4 AM-based ...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]QRFP43 from human GPR103 receptor expressed in HEK cells after 90 mins incubation by scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 94nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 95.3nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 136nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 164nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 166nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 185nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 233nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 233nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 237nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research and Innovation In Biomedicine (Irib)
Curated by ChEMBL




































