Report error Found 591 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-gamma'
Affinity DataKd: >0.00100nMAssay Description:Inhibition of [3H]-9-cis RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0800nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at full length human RXR gamma expressed in HEK293T cells measured after 16 hrs by Dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoid X receptor gamma using transactivation a...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Compound was tested for binding affinity against retinoid X receptor using 5 nM of [3H]-9-cis-RA as a radioligand in baculovirus expressed receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to baculovirus expressed retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity for Retinoic acid receptor RXR-gamma was determined by competing with 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity for Retinoic acid receptor RXR-gamma was determined by competing with 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity against RXR gamma receptor using [3H]9-cis-RA as radioligand in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity against RXR gamma receptor using [3H]9-cis-RA as radioligand in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-gamma was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Inhibition of RXRgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 3.80nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to baculovirus expressed retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Dissociation constant for binding to Retinoid X receptor gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at full length human RXR gamma expressed in HEK293T cells measured after 16 hrs by Dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]targretin binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity against retinoic Acid X gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity for retinoic acid receptor RXR gamma in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Transcriptional activation of Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4.30nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity for Retinoic acid receptor RXR-gamma was determined by competing with 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity for Retinoic acid receptor RXR-gamma was determined by competing with 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity towards recombinantly expressed Retinoic acid receptor RXR-gamma in baculoviral system, by using 5 nM [3H]targretin in a competitive...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]9-cis-RA binding to RXR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity against RXR gamma receptor using [3H]9-cis-RA as radioligand in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity against RXR gamma receptor using [3H]9-cis-RA as radioligand in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of [3H]9-cis-RA binding to RXR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity for Retinoic acid receptor RXR-gamma was determined by competing with 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding affinity for Retinoic acid receptor RXR-gamma was determined by competing with 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activation of Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of [3H]9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Binding affinity for Retinoic acid receptor RXR-gamma was determined by competing with 3[H]-9-cis-RAMore data for this Ligand-Target Pair











3D Structure (crystal)






















