Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform'
TargetSerine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform(Homo sapiens)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to human PPP2R1A incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
LigandPNGBDBM50090505((1R,7S)-2,6-Dimethyl-4,10-dioxa-tricyclo[5.2.1.0*2...)
Affinity DataIC50: 8.00E+3nMAssay Description:Compound was tested for inhibitory concentration of Protein Phosphatase 2A (PP2A).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetSerine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform(Homo sapiens)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PPP2R1A (unknown origin) incubated for 1 hr by colloidal coomassie staining based LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
LigandPNGBDBM50289212(4,10-Dioxa-tricyclo[5.2.1.0*2,6*]dec-8-ene-3,5-dio...)
Affinity DataIC50: 4.00E+4nMAssay Description:Compound was tested for inhibitory concentration of Protein Phosphatase 2A (PP2A).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandPNGBDBM50366474(NORCANTHARIDIN)
Affinity DataIC50: 7.00E+4nMAssay Description:Compound was tested for inhibitory concentration of Protein Phosphatase 2A (PP2A).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetSerine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform(Homo sapiens)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  2.03E+5nMAssay Description:Binding affinity to human PPP2R1A incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
LigandPNGBDBM50289213(7-Oxa-bicyclo[2.2.1]hept-5-ene-2,3-dicarboxylic ac...)
Affinity DataIC50: 3.00E+5nMAssay Description:Compound was tested for inhibitory concentration of Protein Phosphatase 2A (PP2A).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article