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Report error Found 1450 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 1'
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476140(CHEMBL373632)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50474230(CHEMBL3349516)
Affinity DataKi:  0.158nMAssay Description:Binding affinity towards human Somatostatin receptor type 1 (sst1) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50294254((4R,7S,10S,13R,16S,19R)-19-((R)-2-amino-3-(4-hydro...)
Affinity DataIC50: 0.190nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst1 receptor by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50474219(CHEMBL3349522)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards human Somatostatin receptor type 1 (sst1) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2018
Entry Details

TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476134(CHEMBL437296)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50019568(CHEMBL411836 | SRIF-14 | Somatostatin receptor lig...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423465(ERGOLINE)
Affinity DataKd:  0.204nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423299(CHEMBL401290)
Affinity DataKd:  0.214nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423475(CHEMBL252032)
Affinity DataKd:  0.240nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50474221(CHEMBL3349521)
Affinity DataKi:  0.251nMAssay Description:Binding affinity towards human Somatostatin receptor type 1 (sst1) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423480(CHEMBL254505)
Affinity DataKd:  0.282nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.290nMAssay Description:Displacement of [125I]somatostatin from human SSTR1 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50495074(CHEMBL3098601)
Affinity DataKi:  0.310nMAssay Description:Displacement of [125I]-somatostatin from human SSTR1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Mouse)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM392076(US10301272, Example 7/9)
Affinity DataIC50: 0.310nMAssay Description:Displacement of [125I]Tyr11-somatostatin-14 from mouse SST receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82547(SRIF-D-Trp8)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-somatostatin from human SSTR1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476138(CHEMBL376485)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.360nMAssay Description:Inhibition of human sst1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50294254((4R,7S,10S,13R,16S,19R)-19-((R)-2-amino-3-(4-hydro...)
Affinity DataEC50:  0.370nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423478(CHEMBL252033)
Affinity DataKd:  0.372nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  0.372nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423472(CHEMBL401309)
Affinity DataKd:  0.380nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50064772(Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity towards human sst1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423481(CHEMBL254499)
Affinity DataKd:  0.389nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423483(CHEMBL398526)
Affinity DataKd:  0.389nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423314(CHEMBL251754)
Affinity DataKd:  0.398nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476137(CHEMBL222751)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423317(CHEMBL440236)
Affinity DataKd:  0.407nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2018
Entry Details

TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [125I]-somatostatin from human SSTR1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214421(SOMATOSTATIN RECEPTOR LIGAND)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2018
Entry Details

TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50212467(Sandostatinm)
Affinity DataIC50: 0.460nMAssay Description:Compound was tested for free energy of binding against somatostatin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2018
Entry Details

TargetSomatostatin receptor type 1(Rat)
Tulane University

Curated by PDSP Ki Database
LigandPNGBDBM50423477(CHEMBL252618)
Affinity DataKd:  0.490nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2012
Entry Details Article
PubMed
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