Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Synaptic vesicle membrane protein VAT-1 homolog'
TargetSynaptic vesicle membrane protein VAT-1 homolog(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50459706(CHEMBL4214264)
Affinity DataIC50: 4.48E+3nMAssay Description:Covalent binding affinity to VAT1 at Cys residue in human NCI-H358 cells assessed as reduction of log2 H/L ratio for tryptic peptide ACGLNFADLMAR inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetSynaptic vesicle membrane protein VAT-1 homolog(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50459706(CHEMBL4214264)
Affinity DataIC50: 4.54E+3nMAssay Description:Covalent binding affinity to VAT1 at Cys residue in human NCI-H358 cells assessed as reduction of log2 H/L ratio for tryptic peptide CLVLTGFGGYDK inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetSynaptic vesicle membrane protein VAT-1 homolog(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  7.96E+3nMAssay Description:Binding affinity to human VAT1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSynaptic vesicle membrane protein VAT-1 homolog(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  1.45E+5nMAssay Description:Binding affinity to human VAT1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed