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Report error Found 95 Enz. Inhib. hit(s) with Target = 'Threonine--tRNA ligase'
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426188(CHEMBL2311920)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426188(CHEMBL2311920)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426182(CHEMBL2311926)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426183(CHEMBL2311925)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426182(CHEMBL2311926)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426184(CHEMBL2311924)
Affinity DataKi:  2nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426190(CHEMBL2311918)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426194(CHEMBL2316966)
Affinity DataKi:  2.70nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426184(CHEMBL2311924)
Affinity DataKi:  3nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426190(CHEMBL2311918)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426180(CHEMBL2311928)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426183(CHEMBL2311925)
Affinity DataKi:  4.10nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426181(CHEMBL2311927)
Affinity DataKi:  5.20nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  5.30nMAssay Description:Binding affinity to human TARS incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426181(CHEMBL2311927)
Affinity DataKi:  5.70nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase, mitochondrial(Homo sapiens)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  5.90nMAssay Description:Binding affinity to human TARS2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426189(CHEMBL2311919)
Affinity DataKi:  8.20nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426187(CHEMBL2311921)
Affinity DataKi:  9.30nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426200(CHEMBL2311917)
Affinity DataKi:  9.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426189(CHEMBL2311919)
Affinity DataKi:  10nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426200(CHEMBL2311917)
Affinity DataKi:  13nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50366646(CHEMBL1163068)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against cognate Staphylococcus aureus threonyl tRNA synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604793(CHEMBL5169990)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426193(CHEMBL2316967)
Affinity DataKi:  23nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426186(CHEMBL2311922)
Affinity DataKi:  25nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426194(CHEMBL2316966)
Affinity DataKi:  32nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604793(CHEMBL5169990)
Affinity DataKd:  35nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604793(CHEMBL5169990)
Affinity DataKd:  37nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of tRNA Leucin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426179(CHEMBL2311929)
Affinity DataKi:  39nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50129555(CHEMBL70590 | cid_310900 | 2-((1S,8R,9S,11R,13S,15...)
Affinity DataIC50: 43nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604793(CHEMBL5169990)
Affinity DataKd:  44nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of glycine by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625969(CHEMBL5405159)
Affinity DataKd:  49nMAssay Description:Inhibition of human cytosolic ThrRS assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50426183(CHEMBL2311925)
Affinity DataIC50: 57nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  58nMAssay Description:Binding affinity to human TARS incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426197(CHEMBL2316963)
Affinity DataKi:  70nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426187(CHEMBL2311921)
Affinity DataKi:  72nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604793(CHEMBL5169990)
Affinity DataKd:  75nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of ATP by isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426178(CHEMBL2316960)
Affinity DataKi:  83nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426180(CHEMBL2311928)
Affinity DataKi:  91nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50625969(CHEMBL5405159)
Affinity DataIC50: 100nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604786(CHEMBL5204569)
Affinity DataIC50: 103nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426185(CHEMBL2311923)
Affinity DataKi:  115nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625967(CHEMBL5430875)
Affinity DataKd:  115nMAssay Description:Inhibition of human cytosolic ThrRS assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetThreonine--tRNA ligase 1, cytoplasmic(Human)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625968(CHEMBL5424310)
Affinity DataKd:  126nMAssay Description:Inhibition of human cytosolic ThrRS assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetThreonine--tRNA ligase(Yersinia pestis)
Trius Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426177(CHEMBL2316961)
Affinity DataKi:  132nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50366646(CHEMBL1163068)
Affinity DataIC50: 160nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50129555(CHEMBL70590 | cid_310900 | 2-((1S,8R,9S,11R,13S,15...)
Affinity DataKi:  160nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetase expressed in Escherichia coli Rossetta 2 (DE3) assessed as apparent inhibition constant ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604793(CHEMBL5169990)
Affinity DataKd:  166nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of tRNA Threon...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50426177(CHEMBL2316961)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetThreonine--tRNA ligase(Salmonella enterica)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50604788(CHEMBL5176566)
Affinity DataIC50: 194nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
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