Report error Found 247 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a/V1b receptor'
Affinity DataKd: 0.650nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 3.80nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataKd: 17.8nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 42nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 50nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataKd: 53nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
Affinity DataKd: 82nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibition of [3H]arginine vasopressin binding to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 280nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair































