1308 SMILES Strings for A disintegrin and metalloproteinase with thrombospondin motifs 5

Compound Name
SMILES String
CC(=O)N1CC(=CC1c1ccccc1)c1cc(F)ccc1F |c:5|
CC(=O)N1N=C(CC1c1ccccc1)c1cc(F)ccc1F |c:4|
CC(C)(C)C(=O)N1CC(=CC1c1ccccc1)c1cc(F)ccc1F |c:8|
CC(C)(C)C(=O)N1N=C(CC1c1ccccc1)c1cc(F)ccc1F |c:7|
CN(C)C(=O)N1CC(=C[C@H]1c1ccccc1)c1cc(F)ccc1F |c:7|
CN(C)C(=O)N1N=C(CC1c1ccccc1)c1cc(F)ccc1F |c:6|
CN(C1CCNCC1)C(=O)N1CC(=C[C@H]1c1ccccc1)c1cc(F)ccc1F |c:13|
[H][C@]1(C=C(CN1C(=O)N(C)C1CCN(CC1)C(C)=O)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
[H][C@]1(C=C(CN1C(=O)N(C)CCCN)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
[H][C@]1(C=C(CN1C(=O)C(C)(C)CN)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
[H][C@]1(C=C(CN1C(=O)[C@@H](N)C(C)C)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
[H][C@]1(C=C(CN1C(=O)[C@H](N)C(C)C)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
N[C@@H](C1CC1)C(=O)N1CC(=C[C@H]1c1ccccc1)c1cc(F)ccc1F |c:10|
[H][C@]1(C=C(CN1C(=O)[C@@H](N)C(C)(C)C)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
[H][C@]1(C=C(CN1C(=O)[C@@H](NC(=O)OCCO)C(C)(C)C)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
[H][C@]1(C=C(CN1C(=O)[C@@H](O)C1CC1)c1cc(F)ccc1F)c1ccccc1 |r,c:2|
CC(=O)N1N=C(C[C@H]1c1cccc(O)c1)c1cc(F)ccc1F |r,c:4|
CC(=O)N1[C@@H](CC(=N1)c2ccccc2Cl)c3cccc(c3)O
CNC(=O)N1N=C(CC1c1ccccc1)c1cc(F)ccc1F |c:5|
CNC(=O)N1N=C(CC1(C)c1ccccc1)c1cc(F)ccc1F |c:5|
CNC(=O)N1N=C(CC1(CO)c1ccccc1)c1cc(F)ccc1F |c:5|
CCNC(=O)N1N=C(CC1(CCO)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCO)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCO)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCN)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1[C@](CC(=N1)c2cc(ccc2F)F)(CCCN)c3ccccc3
CCNC(=O)N1N=C(CC1(CCCCN)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCNCc1ccccc1)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCN(C)C)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCN1CC2CC1C=C2)c1ccccc1)c1cc(F)ccc1F |c:6,21|
CCNC(=O)N1N=C(CC1(CCCC[N+](C)(C)[O-])c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCNC(=O)c1ccccc1)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCNC(=O)c1ccccn1)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCNC(=O)c1ncc[nH]1)c1ccccc1)c1cc(F)ccc1F |c:6|
CCNC(=O)N1N=C(CC1(CCCCNC(=O)c1cnc[nH]1)c1ccccc1)c1cc(F)ccc1F |c:6|
CN(C)C(=O)N1N=C(CC1(CCCN)c1ccccc1)c1cc(F)ccc1F |c:6|
NCCCC1(CC(=NN1C(=O)N1CCC1)c1cc(F)ccc1F)c1ccccc1 |c:6|
NCCCC1(CC(=NN1C(=O)N1CCCC1)c1cc(F)ccc1F)c1ccccc1 |c:6|
NCCCC1(CC(=NN1C(=O)N1CCCCC1)c1cc(F)ccc1F)c1ccccc1 |c:6|
NCCCC1(CC(=NN1C(=O)N1CCOCC1)c1cc(F)ccc1F)c1ccccc1 |c:6|
CN(C)C(=O)N1N=C(C[C@@]1(CCCN)c1ccccc1)c1cc(F)ccc1F |r,c:6|
CC(=O)N1CCN(CCCC2(CN(N=C2C(C)=O)c2cc(F)ccc2F)c2ccccc2)CC1 |c:13|
CN(CCCC1(CN(N=C1C(C)=O)c1cc(F)ccc1F)c1ccccc1)Cc1cc(C)no1 |c:8|
CC(=O)C1=NN(CC1(CCCN1CCS(=O)(=O)CC1)c1ccccc1)c1cc(F)ccc1F |t:3|
CC(=O)C1=NN(CC1(CCCN1CCOCC1)c1ccccc1)c1cc(F)ccc1F |t:3|
CC(=O)C1=NN(CC1(CCCN1CC(F)C1)c1ccccc1)c1cc(F)ccc1F |t:3|
CC(=O)C1=NN(CC1(CCCN1CCCC1)c1ccccc1)c1cc(F)ccc1F |t:3|
CC(=O)C1=NN(CC1(CCCN1C[C@@H]2C[C@H]1CO2)c1ccccc1)c1cc(F)ccc1F |r,t:3|
CN(C)CCCC1(CN(N=C1C(C)=O)c1cc(F)ccc1F)c1ccccc1 |c:9|
CC(=O)N1CCN(CCCC2(CN(N=C2C(C)=O)c2cc(Cl)ccc2F)c2ccccc2)CC1 |c:13|
CC(=O)N1CCN(CCCC2(CN(N=C2C(C)=O)c2cc(Br)ccc2F)c2ccccc2)CC1 |c:13|
CC(=O)N1CCN(CCCC2(CN(N=C2C(C)=O)c2ccccc2F)c2ccccc2)CC1 |c:13|
CC(=O)N1CCN(CCCC2(CN(N=C2C(C)=O)c2cc(ccc2F)C(F)(F)F)c2ccccc2)CC1 |c:13|
Cc1ccc(c(c1)N2C[C@@](C(=N2)C(=O)C)(CCCN3CCN(CC3)C(=O)C)c4ccccc4)F
CN(C)CCC[C@]1(CN(N=C1C(C)=O)c1cc(C)ccc1F)c1ccccc1 |r,c:9|
CC(=O)N1CCN(CCC[C@]2([C@@H]3COc4ccc(F)cc4N3N=C2C(C)=O)c2ccccc2)CC1 |r,c:24|
NC(=O)[C@H](CCC(O)=O)NC(=O)CCc1ccc(cc1)-c1cc(cs1)-c1ccccc1 |r|
NC(=O)[C@H](CCC(O)=O)NC(=O)c1ccc(cc1)-c1cc(cs1)-c1ccccc1 |r|
Cc1ccc(s1)-c1ccc(CCC(=O)N[C@@H](CCC(O)=O)C(N)=O)cc1 |r|
NC(=O)[C@H](CCC(O)=O)NC(=O)CCc1ccc(cc1)-c1ccc(cc1)-c1ccccc1 |r|
NC(=O)[C@H](CCC(O)=O)NC(=O)CCc1ccc(cc1)-c1ccc(s1)-c1ccccc1 |r|
C[C@H](Cc1ccc(cc1)C(F)(F)F)C(=O)NC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC[C@H](Cc1ccc(cc1)C(F)(F)F)C(=O)NC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)c1ccc(C[C@@H](C2CC2)C(=O)NC[C@]2(NC(=O)NC2=O)C2CC2)cc1 |r|
CC(C)[C@H](Cc1ccc(cc1)C(F)(F)F)C(=O)NC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC(C)(Cc1ccc(cc1)C(F)(F)F)C(=O)NC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1(CCC(=O)N2CCN(CC2)c2ccccc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccc(Cl)cc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCN(CC1)c1ccccc1
Clc1ccc(cc1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Cc1ccccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Cc1cccc(N2CCN(CC2)C(=O)CCC2(NC(=O)NC2=O)c2ccccc2)c1C
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCN(CC1)c1ccc2ccccc2c1
Fc1cc(ccc1Cl)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Cc1cccc(N2CCN(CC2)C(=O)CCC2(C)NC(=O)NC2=O)c1C
Cc1ccccc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1cc(Cl)ccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCN(CC1)c1ccc2cnccc2c1
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCN(CC1)c1ccc2ccccc2n1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1cc(Cl)ccc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1c(Cl)cccc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccccc2Cl)NC(=O)NC1=O
Clc1ccccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Cc1c(Cl)cccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Cc1cccc(C)c1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Cc1cc(ccc1[N+]([O-])=O)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCN(CC1)c1ccc2occc2c1
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCN(CC1)c1ccc2scnc2c1
Cc1ccccc1N1CCN(CC1)C(=O)CC[C@]1(NC(=O)NC1=O)c1ccccc1 |r|
CC1(CCC(=O)N2CCN(CC2)c2ccc(Br)cc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccccc2C#N)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccccc2F)NC(=O)NC1=O
Cc1ccc(N2CCN(CC2)C(=O)CCC2(NC(=O)NC2=O)c2ccccc2)c(C)c1
CC(C)C1(CCC(=O)N2CCN(CC2)c2ccccc2C)NC(=O)NC1=O
CC(C)C1(CCC(=O)N2CCN(CC2)c2cc(Cl)ccc2C)NC(=O)NC1=O
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Cc1ccccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
CC1(CCC(=O)N2CCN(CC2)c2ccc(F)c(F)c2)NC(=O)NC1=O
Cc1ccc(N2CCN(CC2)C(=O)CCC2(C)NC(=O)NC2=O)c(C)c1
Cc1ccc(C)c(c1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2Cl)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccccn2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cccnc2)NC(=O)NC1=O
CN(C)CCC1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCN(CC1)c1cccnc1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
CC1(CCC(=O)N2CCN(CC2)c2cccc(F)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cccc(Br)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccc(Cl)c(F)c2)NC(=O)NC1=O
CN(C)c1ccccc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1ccc(F)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccc(F)c(Cl)c2)NC(=O)NC1=O
CC(C)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
CC(C)C1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
Clc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Cc1cccc(N2CCN(CC2)C(=O)CCC2(NC(=O)NC2=O)C2CC2)c1C
CN(C)CCC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2nccs2)NC(=O)NC1=O
Cc1c(F)cccc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1cc(F)ccc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
CC1CN(CCN1c1ccccc1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1ccccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
CC1(CCC(=O)N2CCN(CC2)c2ccc(F)cc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccc(Cl)c(Cl)c2)NC(=O)NC1=O
O=C(CCC1(NC(=O)NC1=O)c1cccnc1)N1CCN(CC1)c1ccccc1
Cc1cccc(N2CCN(CC2)C(=O)CCC2(NC(=O)NC2=O)c2cccnc2)c1C
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CCC1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CCC1
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CCCCC1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CCCCC1
Clc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(Cl)cc1
Cc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
Cc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cc(Cl)ccc2C)NC(=O)NC1=O
COc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
COc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cc(Cl)ccc2C)NC(=O)NC1=O
CN(C)CCOc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
CN(C)CCOc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2ccccc2C)NC(=O)NC1=O
CN(C)Cc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2ccccc2C)NC(=O)NC1=O
CN(C)Cc1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cncc(F)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cncc(Cl)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cncc(Br)c2)NC(=O)NC1=O
Cc1ccc(C)c(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Cc1ccc(C)c(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Cc1ccc(C)c(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Fc1ccc(cc1F)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Fc1ccc(cc1Cl)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Cc1ccc(F)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Cc1cc(Cl)c(F)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1cc(F)c(F)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Fc1ccc(cc1F)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Fc1ccc(cc1Cl)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Cc1c(F)cccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Cc1c(Cl)cccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Cc1c(F)cccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Cc1c(F)cccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Cc1cccc(N2CCN(CC2)C(=O)CCC2(NC(=O)NC2=O)c2ccccn2)c1C
Cc1c(Cl)cccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Fc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Cc1ccc(F)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
CC1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
CC1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
CC(C)(C)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C(C)(C)C
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CCCC1
Cc1ccc(Cl)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CCCC1
Clc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Fc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
Fc1ccc(cc1F)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Fc1ccc(cc1Cl)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Fc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Cc1ccc(F)cc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
CC1(CCC(=O)N2CCN(CC2)c2cc(F)cc(Cl)c2)NC(=O)NC1=O
CN(C)CC1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
CN(C)CC1(CCC(=O)N2CCN(CC2)c2ccccc2C)NC(=O)NC1=O
CN(C)CC1(CCC(=O)N2CCN(CC2)c2cc(Cl)ccc2C)NC(=O)NC1=O
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN(CC1)c1cccc(Cl)c1
CCC1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
COc1cccc(c1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
CS(=O)(=O)c1ccc(cc1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(cc1)C#N
CC1CN(CCN1c1ccc(Cl)cc1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
CC1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
C[C@@H]1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC1CN(CCN1c1cc(F)ccc1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1
CC1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
C[C@@H]1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1 |r|
COc1ccc(Cl)cc1C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
COc1ccc(Cl)cc1C1(CCC(=O)N2CCN(CC2)c2cc(Cl)ccc2C)NC(=O)NC1=O
C[C@@H]1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
C[C@H]1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
C[C@H]1CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1 |r|
O=C(CCC1(NC(=O)NC1=O)C1CC1)N1CCN(CC1)c1ccccc1
Cc1c(Cl)cc(Cl)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2cc(F)cc(F)c2)NC(=O)NC1=O
Cc1cccc(c1)C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)cc1)C(=O)CCC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(F)ccc1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1ccccc1C1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1ccc(Cl)cc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)ccc1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC1CN(CCN1c1cccc(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
CC1CN(CCN1c1cccc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccc2NC(=O)Cc2c1
COCCN(C)CC1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cccc(Cl)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
C[C@]1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
Clc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(CNCc2ccccc2)NC(=O)NC1=O
CNc1ccccc1N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
COCC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
COCCNC(=O)CC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC(C)(C)OC(=O)CC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
OCCNC(=O)CC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cccc(F)c1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(Cl)cc1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cc(F)cc(Cl)c1 |r|
O=C(CCC1(NC(=O)NC1=O)C1CC1)N1CCN(CC1)c1cccc(c1)C#N
CC(CC1(NC(=O)NC1=O)C1CNC1)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
CSCCC1(CC(C)C(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC(CC1(CC2CCN(CC2)C(=O)OC(C)(C)C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
CC(CC1(NC(=O)NC1=O)C1CCOCC1)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
CC(CC1NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
OC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1(CN2CCOCC2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1cc(F)c(Cl)cc1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(F)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(CC2CCNCC2)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1ccc(Cl)c(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CN(C)c1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(CCN)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1ccc(F)c(F)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1ccc(F)c(F)c1
C[C@@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(F)cc(F)c1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cccc(Cl)c1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cccc(F)c1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(F)ccc1C |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(C)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccccc1 |r|
NCC1(CCC(=O)N2CCN(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
CC(CC1(CCS(C)(=O)=O)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
Clc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1(CC(CO)C(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN(CC1)c1cc(F)ccc1C
COCCOCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(F)ccc1C
COCC1(CC(C)C(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN(CC1)c1cccc(Cl)c1C
CC(=O)NCC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
COCC1(CC(C)C(=O)N2CCN(CC2)c2ccc(F)c(F)c2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)cc(F)c2)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cccc(Cl)c1C
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2ccc(F)c(F)c2)NC(=O)NC1=O |r|
NCC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(Cl)cc(Cl)c2C)NC(=O)NC1=O |r|
Clc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CCC1(CNCc2ccccc2)NC(=O)NC1=O
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)ccc2C)NC(=O)NC1=O |r|
COC(=O)CC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cccc(F)c2)NC(=O)NC1=O |r|
OC(=O)CC1(CCC(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
COCC1(CC(C)C(=O)N2CCN(CC2)c2cc(F)ccc2C)NC(=O)NC1=O
CC(CC1(NC(=O)NC1=O)c1ccccn1)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
O=C(CCC1(NC(=O)NC1=O)C1CC1)N1CCN(CC1)c1ccncc1
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cccc(Cl)c2C)NC(=O)NC1=O |r|
COCC1(CC(C)C(=O)N2CCN(CC2)c2cc(F)c(Cl)c(F)c2)NC(=O)NC1=O
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cccc(Cl)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cccc2ccoc12)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(NC(=O)NC1=O)C1CN(C1)C(=O)OC(C)(C)C)C(=O)N1CCN(CC1)c1ccc(F)c(F)c1
C[C@H]1CN(CCN1c1cccc(c1)-c1ccncc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(CCNC(=O)OC(C)(C)C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1ccc(F)c(F)c1
C[C@H]1CN(CCN1c1cccc(c1)-c1cn[nH]c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CCC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1cccc(c1)-c1cnn(C)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cccc(Cl)c1C |r|
C[C@H]1CN(CCN1c1nccc(Cl)n1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
Cc1cc(CC(CC2(C)NC(=O)NC2=O)C(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)n(C)n1
C[C@H]1CN(CCN1c1ccc(Cl)nn1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(NC(=O)NC1=O)C1CN(C1)C(=O)OC(C)(C)C)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
C[C@H]1CN(CCN1c1cnccn1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(NC(=O)NC1=O)C1CNC1)C(=O)N1CCN(CC1)c1ccc(F)c(F)c1
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(C)nc1 |r|
CC(CC1(CCN)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1ccc(F)c(F)c1
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccncc1 |r|
CC(CC1(CN2CCOCC2)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1cnc2ccccc2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1C[C@H](C)N([C@H](C)C1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H]1CN(CCN1c1ccc2n(C)ccc2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
COCC1(CC(C)C(=O)N2C[C@H](C)N([C@H](C)C2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc2ccn(C)c2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(NC(=O)NC1=O)c1ccccn1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
COCC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cccc(F)c1 |r|
CC(CC1(CN2CCOCC2)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(Cl)cc(Cl)c1 |r|
Cc1c(Cl)cc(F)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC(CC1(NC(=O)NC1=O)C1CNC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
COC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cccc(F)c1 |r|
CC(CC1(NC(=O)NC1=O)C1CN(C1)C(C)=O)C(=O)N1CCN(CC1)c1ccc(F)c(F)c1
COC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(F)cc(Cl)c1 |r|
CC(CC1(NC(=O)NC1=O)C1CN(C1)C(C)=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
C[C@H]1CN(CCN1c1ccc2[nH]ncc2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
Cc1cc(Cl)c(Cl)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
C[C@H]1CN(CCN1c1ccc2n(C)ncc2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(C)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(CN2CCC(F)(F)C2)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1ccc(C)c(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(CN2CCC(F)(F)C2)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
C[C@H]1CN(CCN1c1ccc(F)cc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC1(CC(CC#N)C(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1ccnc(Cl)n1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c2cc(cc(c2)F)F)C(=O)CC[C@@]3(C(=O)NC(=O)N3)C4CC4
C[C@H]1CN(CCN1c1cccnn1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(Cl)ncn1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cncc(C)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)n1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cncnc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(Cl)nc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1ccc2ncsc2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccnc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1ccc(C)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cncc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
C[C@H]1CN(CCN1c1cncc(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
C[C@H]1CN(CCN1c1cc(Cl)c(Cl)cc1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
CC(CC1(NC(=O)NC1=O)c1ccccn1)C(=O)N1CCN([C@@H](C)C1)c1cccc(F)c1 |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
CC(CC1(NC(=O)NC1=O)c1ccccn1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
C[C@H]1CN(CCN1c1cccc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)cc1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
CCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cccc(F)c2)NC(=O)NC1=O |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cncc(F)c1 |r|
Cc1cc(N2CCN(CC2)C(=O)CCC2(C)NC(=O)NC2=O)c(F)cc1Cl
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cncc(Cl)c1 |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)C(CO)CC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
CC(CC1(NC(=O)NC1=O)c1ccccn1)C(=O)N1CCN([C@@H](C)C1)c1cccc(Cl)c1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
C[C@H]1CN(CCN1c1cccc(Br)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1C[C@H](C)N([C@@H](C)C1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1cccnc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
C[C@H]1CN(CCN1c1ccc2[nH]ccc2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(ccn1)-c1cccc(c1)N1CCN(C[C@@H]1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cccnc1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1cncc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cncc(Cl)c1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1cccnc1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cncc(F)c1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1ccc(C)nc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(Cl)ccn1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1cnccn1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cnccn1 |r|
C[C@H]1CN(CCN1c1cnnc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cnccn1 |r|
C[C@H]1CN(CCN1c1ccn(C)n1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc2n(C)ccc12)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(F)cc(c1)-c1cn[nH]c1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1ccnc(C)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
COC[C@]1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)cc(c2)-c2cn[nH]c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cncc(c1)C#N)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1cncnc1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
COC[C@]1(C[C@H](C)C(=O)N2CCN([C@@H](C)C2)c2ccc(F)c(Cl)c2)NC(=O)NC1=O |r|
C[C@@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(c1)-c1cn[nH]c1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cncnc1 |r|
C[C@@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cc(F)cc(c1)-c1cn[nH]c1 |r|
C[C@H]1CN(CCN1c1cccc2n(C)ncc12)C(=O)CCC1(CNC(=O)N1)C1CC1 |r|
COC[C@]1(C[C@H](C)C(=O)N2CCN([C@@H](C)C2)c2cccc(c2)-c2cn[nH]c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(F)cc(c1)C#N)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1ccc(Cl)nn1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
Fc1cc(F)cc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(nc1)C(F)(F)F
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1ncccn1 |r|
COc1cccc(n1)C1(CCC(=O)N2CCN([C@@H](C)C2)c2cc(F)cc(F)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(C)nc1 |r|
C[C@H]1CN(CCN1c1cnc2ccn(C)c2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(C)nc1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(c1)-c1cn[nH]c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(C)nc1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cccc(c1)-c1cn[nH]c1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(C)nc1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(c1)-c1cn[nH]c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cc(C)on1 |r|
C[C@H]1CN(CCN1c1ccc2cnn(C)c2c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cocn1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cncc(C)c1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cn(C)cn1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)cc1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(c1)N(C)C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1noc(C)n1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CNc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccn(C)n1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1coc(C)n1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1nc(C)oc1C |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cnn(C)c1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cnccn1 |r|
CC(CC1(NC(=O)NC1=O)C1CN(C)C1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
C[C@H]1CN(CCN1c1cccc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cnccn1 |r|
C[C@H]1CN(CCN1c1cc(C)c(Cl)c(C)c1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1cccnc1 |r|
Cc1cc(cc(C)c1Cl)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1nc(C)no1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
Cc1cc(ccc1Cl)N1CCN(CC1)C(=O)CCC1(CC(=O)NCCO)NC(=O)NC1=O
C[C@H]1CN(CCN1c1cccc(c1)-c1c(C)n[nH]c1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1c[nH]c(C)n1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(F)c(Cl)c(F)c1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1c[nH]nc1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
COc1ccc(cn1)C1(CCC(=O)N2CCN([C@@H](C)C2)c2cc(F)cc(F)c2)NC(=O)NC1=O |r|
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2ccc(F)c(Cl)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(F)cc(c1)-c1cn[nH]c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1cc[nH]n1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cncc(Cl)c2)NC(=O)NC1=O |r|
CCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cncc(F)c2)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cn(C)cn1 |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cocn1 |r|
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cncc(Cl)c2)NC(=O)NC1=O |r|
COCC1(CCC(=O)N2CCN([C@@H](C)C2)c2cncc(F)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)cc1 |r|
CC(CC1(COCc2ccccc2)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2ccc(F)cc2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccnc(C)c1 |r|
CC(CC1(CO)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1cccc(c1)-c1ccnn1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(F)cc(Cl)c1 |r|
C[C@H]1CN(CCN1c1cccc(c1)-c1c(C)noc1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(Cl)c(Cl)c1 |r|
CC(C)n1cc(cn1)-c1cccc(c1)N1CCN(C[C@@H]1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(Cl)cc(Cl)c1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cccc(c1)-c1cn[nH]c1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(F)c1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
CC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(Cl)cc(Cl)c1C |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1 |r|
CC1(CC(COCc2ccccc2)C(=O)N2CCN(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
C[C@H]1CN(CCN1c1ccc(Cl)c(F)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
CC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(C)c1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1 |r|
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cnccn1 |r|
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)cc(Cl)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cnccn1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ncccn1 |r|
COCC1(CC(C)C(=O)N2CCN(CC2)c2cccc(Cl)c2C)NC(=O)NC1=O
C[C@H]1CN(CCN1c1cc(F)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ncccn1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1ccc(C)nc1 |r|
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cocn1 |r|
COCC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1cc(Cl)cc(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cn(C)cn1 |r|
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cn(C)cn1 |r|
CC(C)C(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
CC(C)c1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN(CC1)c1cc(Cl)cc(Cl)c1
C[C@H]1CN(CCN1c1ccc(Cl)c(C)c1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CC(CC1NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
CCc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CCC1(CC(O)=O)NC(=O)NC1=O |r|
CC(CC1(NC(=O)NC1=O)c1ccccn1)C(=O)N1CCN([C@@H](C)C1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(c1)C(F)(F)F)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)C(CO)CC1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(c1)C(F)F)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2ccc(F)c(Cl)c2)NC(=O)NC1=O |r|
CCc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CCC1(CCC(=O)OC(C)(C)C)NC(=O)NC1=O |r|
CCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)cc(Cl)c2)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(CF)c1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CCC1(CCC(O)=O)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc(F)c(Cl)c1)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2ccc(Cl)c(c2)C(F)(F)F)NC(=O)NC1=O |r|
COCC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
COCC1(CC(C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)c(Cl)c(F)c2)NC(=O)NC1=O |r|
COC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1ccc(F)c(Cl)c1 |r|
CCc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)C(C)CC1(COC)NC(=O)NC1=O |r|
COCC(CC1(C)NC(=O)NC1=O)C(=O)N1CCN([C@@H](C)C1)c1cc(F)cc(Cl)c1 |r|
COC(=O)c1cn(CCN([C@@]2(C[C@H]2c2ccccc2)C(O)=O)S(=O)(=O)c2ccc(cc2)-c2ccc(Cl)cc2)cn1 |r|
OC(=O)[C@]1(C[C@H]1c1ccccc1)NS(=O)(=O)c1ccc(cc1)-c1ccc(Cl)cc1 |r|
OC(=O)[C@@]1(C[C@@H]1c1ccccc1)NS(=O)(=O)c1ccc(cc1)-c1ccc(Cl)cc1 |r|
OC(=O)[C@@]1(C[C@@H]1c1ccccc1)NS(=O)(=O)c1ccc(s1)-c1ccc(Cl)cc1 |r|
OC(=O)[C@@]1(C[C@@H]1c1ccccc1)NS(=O)(=O)c1ccc(s1)-c1cccc(Cl)c1 |r|
OC(=O)[C@@]1(C[C@@H]1c1ccccc1)NS(=O)(=O)c1ccc(s1)-c1ccc(Cl)cn1 |r|
OC(=O)[C@@]1(C[C@@H]1c1ccccc1)NS(=O)(=O)c1ccc(s1)-n1cc(Cl)cn1 |r|
O=C(CC[C@@H]1NC(=O)NC1=O)N1CCC(CC1)c1ccccc1 |r|
O=C(CCC1NC(=O)NC1=O)N1CCC(CC1)c1ccccc1
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCC(CC1)c1ccccc1
CC1(CCC(=O)N2CCC(CC2)c2ccccc2)NC(=O)NC1=O
CC(C)C1(CCC(=O)N2CCC(CC2)c2ccccc2)NC(=O)NC1=O
COc1ccccc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
O=C(CCC1(NC(=O)NC1=O)C1CC1)N1CCC(CC1)c1ccccc1
Cc1ccc(cc1)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC1(CCC(=O)N2CCC(CC2)c2cc(Cl)cc(Cl)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCC(CC2)c2ccc(F)cc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCC(CC2)c2cccc(Cl)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCC(CC2)c2ccc(Cl)cc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCC(CC2)c2cccc(F)c2)NC(=O)NC1=O
CC1(CCC(=O)N2CCC(CC2)c2ccccc2F)NC(=O)NC1=O
Cc1cccc(c1)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
O=C(CCC1(NC(=O)NC1=O)c1cccnc1)N1CCC(CC1)c1ccccc1
Clc1cc(Cl)cc(c1)C1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Clc1cccc(c1)C1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
Fc1cccc(c1)C1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
C[C@@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1CCC(CC1)c1ccccc1 |r|
COc1cc(cc(OC)c1Cl)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(OC)c1Cl)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCC(CC1)c1ccccc1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCC(CC1)c1ccc(Cl)cc1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCC(CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCC(CC1)c1ccc(F)cc1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCC(CC1)c1cccc(C)c1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCC(CC1)c1cccc(F)c1 |r|
C[C@@H](C[C@@]1(C)NC(=O)NC1=O)C(=O)N1CCC(CC1)c1cccc(Cl)c1 |r|
COc1ccc(cc1)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1ccc(cc1)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(ccc1Cl)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(C2CCN(CC2)C(=O)CC[C@H]2NC(=O)NC2=O)c(C)cc1Cl |r|
COc1cc(OC)cc(c1)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1ccc(OC)c(c1)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(ccc1Cl)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(C2CCN(CC2)C(=O)CCC2(C)NC(=O)NC2=O)c(C)cc1Cl
COc1cc(OC)cc(c1)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1ccc(OC)c(c1)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1ccc(Cl)cc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1ccc(Cl)cc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(Cl)ccc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(Cl)ccc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(F)c1F)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(F)c1Cl)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1Cl)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1c(Cl)cc(Cl)cc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
Cc1c(Cl)cc(Cl)cc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(F)cc(c1)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Fc1cc(ccc1Cl)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(ccc1F)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
Fc1ccc(cc1F)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
CC1(CCC(=O)N2CCC(CC2)c2ccc(Cl)c(F)c2)NC(=O)NC1=O
COc1cc(ccc1F)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
CC1(CCC(=O)N2CCC(CC2)c2ccc(F)c(F)c2)NC(=O)NC1=O
Cc1ccccc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1ccccc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
Cc1cc(Cl)ccc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(Cl)c(Cl)cc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(Cl)c(Cl)cc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
Cc1cc(Cl)c(F)cc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
Cc1cc(Cl)c(F)cc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1c(Cl)cc(Cl)cc1C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)cc(c1)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)cc(c1)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1Cl)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1c(Cl)cc(Cl)cc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
Cc1cc(Cl)c(Cl)cc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(OC)c1F)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(Cl)c1F)C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1c(Cl)cccc1C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1c(Cl)cccc1C1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
C[C@H]1CN(CC[C@H]1c1ccc(F)c(F)c1)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CC[C@@H]1c1ccc(F)c(F)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CC[C@H]1c1ccc(F)c(F)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(Cl)ccc1C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1F)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1F)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1F)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(ccc1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1c(Cl)cccc1C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCOc1cc(cc(OC)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCOc1cc(cc(OC)c1Cl)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(Cl)c(C)cc1C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(N(C)C)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
Cc1cc(cc(C)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)c(Cl)cc1C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)ccc1C1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(C)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CC[C@H]1c1ccc(F)c(F)c1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)c(F)cc1C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(F)c(Cl)cc1C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1Cl)C1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCC(CC2)c2cc(F)c(Cl)c(OC)c2)NC(=O)NC1=O |r|
CCc1cc(cc(OC)c1Cl)C1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(COC)NC(=O)NC1=O |r|
CCc1cc(cc(OC)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cc(cc(OC)c1Cl)C1CCN(CC1)C(=O)CC[C@@]1(COC)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCC(CC2)c2cc(Cl)c(F)cc2OC)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCC(CC2)c2ccc(Cl)cc2OC)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCC(CC2)c2cc(F)c(Cl)cc2OC)NC(=O)NC1=O |r|
COc1cc(F)c(Cl)cc1C1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
CC1(CCC(=O)N2CCC(CC2)c2ccc(s2)-c2ccccc2F)NC(=O)NC1=O
COc1cc(cc(C)c1Cl)C1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCC(CC2)c2cc(C)c(Cl)c(OC)c2)NC(=O)NC1=O |r|
COc1cc(cc(C)c1Cl)C1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cccc(c1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
CC1(CCC(=O)N2CCN(CC2)c2ccc(OC(F)(F)F)cc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCN(CC2)c2ccccc2OC(F)(F)F)NC(=O)NC1=O
COc1ccc(cc1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
COc1ccccc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cccc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
COc1cc(ccc1F)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(ccc1Cl)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(OC)cc(c1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
CCOc1cccc(c1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(ccc1F)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
COc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1cc(OC)cc(c1)N1CCN(C[C@@H]1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)[C@@H](C)C[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)c1cccnc1
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1Cl)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1ccc(C)c(c1)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cccc(N2CCN(CC2)C(=O)CCC2(C)NC(=O)NC2=O)c1C
COc1cc(N2CCN(CC2)C(=O)CCC2(C)NC(=O)NC2=O)c(C)cc1Cl
COc1ccc(C)c(c1)N1CCN(C[C@@H]1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1cc(N2CCN(C[C@@H]2C)C(=O)CCC2(C)NC(=O)NC2=O)c(C)cc1Cl |r|
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(cc(F)c1Cl)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(F)c1Cl)N1CCN(C[C@@H]1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1Cl)N1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(N2CCN(C[C@@H]2C)C(=O)[C@@H](C)C[C@@]2(C)NC(=O)NC2=O)c(C)cc1Cl |r|
COC[C@]1(C[C@H](C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)c(F)c(OC)c2)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCN([C@@H](C)C2)c2ccc(Cl)c(OC)c2)NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1Cl)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@]1(NC(=O)NC1=O)c1ccccn1 |r|
COc1cc(cc(Cl)c1F)N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)[C@@H](C)C[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(CN2CCC(F)(F)C2)NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1F)N1CCN(C[C@@H]1C)C(=O)CCC1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)[C@@H](C)C[C@]1(NC(=O)NC1=O)c1ccccn1 |r|
COc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)[C@@H](CO)C[C@@]1(C)NC(=O)NC1=O |r|
CC[C@]1(C[C@H](C)C(=O)N2CCN(CC2)c2cc(F)c(F)c(OC)c2)NC(=O)NC1=O |r|
COc1cc(Cl)c(C)cc1N1CCN(CC1)C(=O)CCC1(C)NC(=O)NC1=O
COC[C@]1(C[C@H](C)C(=O)N2CCN(CC2)c2cc(F)c(F)c(OC)c2)NC(=O)NC1=O |r|
COc1cncc(c1)N1CCN(C[C@@H]1C)C(=O)CCC1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)CCC1(NC(=O)NC1=O)c1cccc(C)n1 |r|
COc1cc(cc(Cl)c1F)N1CCN(C[C@@H]1C)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(cc(Cl)c1F)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cncc(c1)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(cc(F)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(N2CCN(C[C@@H]2C)C(=O)CC[C@@]2(C)NC(=O)NC2=O)c(C)cc1F |r|
COc1c(Cl)cccc1N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cccc(c1)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cc(ccc1Cl)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)ccc1N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1F)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)ccc1N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(F)ccc1N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCOc1cc(cc(OC)c1Cl)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCOc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
C[C@H]1CN(CCN1c1ccc(Cl)c(OC(F)(F)F)c1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1F)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1ccc(Cl)cc1N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(ccc1F)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)c(Cl)cc1N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)c(C)cc1N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(Cl)cc(c1)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(N(C)C)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(C)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CC[C@H]1CN(CCN1c1ccc(Cl)c(OC)c1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(ccc1Cl)N1CCN(C[C@@H]1C(C)C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCOc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(C)c1Cl)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(F)c(F)cc1N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cc(cc(OC)c1Cl)N1CCN(CC1)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
CCc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@@]1(COC)NC(=O)NC1=O |r|
COc1cc(ccc1Cl)N1CCN(CC1C(F)(F)F)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(F)c1Cl)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCN([C@@H](C)C2)c2cc(F)c(Cl)c(OC)c2)NC(=O)NC1=O |r|
COc1cc(cc(F)c1Cl)N1CCN(CC1)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCN(CC2)c2cc(F)c(Cl)c(OC)c2)NC(=O)NC1=O |r|
CCc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@@]1(COC)NC(=O)NC1=O |r|
COc1cc(cc(C)c1Cl)N1CCN(C[C@@H]1C)C(=O)[C@@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COC[C@]1(C[C@H](C)C(=O)N2CCN([C@@H](C)C2)c2cc(C)c(Cl)c(OC)c2)NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(C[C@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)[C@H](C)C[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(F)cc(c1)N1CCN(CC1)C(=O)[C@H](C)C[C@@]1(C)NC(=O)NC1=O |r|
COc1cc(OC)cc(c1)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1F)N1CCN(C[C@@H]1C)C(=O)[C@H](C)C[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc(cc(OC)c1Cl)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1ccc(C)c(c1)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cccc(N2CCN(CC2)C(=O)CC[C@H]2NC(=O)NC2=O)c1C |r|
COc1cc(N2CCN(CC2)C(=O)CC[C@H]2NC(=O)NC2=O)c(C)cc1Cl |r|
COc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1ccc(C)c(c1)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(N2CCN(C[C@@H]2C)C(=O)CC[C@H]2NC(=O)NC2=O)c(C)cc1Cl |r|
COc1cc(cc(F)c1Cl)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(F)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1Cl)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(ccc1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@]1(C)NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1F)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(Cl)c1F)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
CCOc1cc(cc(OC)c1Cl)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
CCOc1cc(cc(OC)c1Cl)N1CCN(C[C@@H]1C)C(=O)CC[C@H]1NC(=O)NC1=O |r|
COc1cc(cc(OC)c1F)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
FC(F)(F)c1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Clc1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)Oc1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1ccc2CCN(CCc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)c1ccc2CN(CCc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1CN(CCc2ccc(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
O=C(CC[C@]1(NC(=O)NC1=O)C1CC1)N1CCc2ccccc2CC1 |r|
FC(F)Oc1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
O=C(CC[C@]1(NC(=O)NC1=O)C1CC1)N1Cc2ccccc2C1 |r|
O=C(CC[C@]1(NC(=O)NC1=O)C1CC1)N1Cc2cccnc2C1 |r|
O=C(CC[C@]1(NC(=O)NC1=O)C1CC1)N1Cc2ccncc2C1 |r|
C[C@H]1N(Cc2ccccc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Fc1cccc2CN(Cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Fc1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Fc1cc2CN(Cc2cc1F)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Clc1cc2CN(Cc2cc1Cl)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCc2ccc(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1CN(CCc2ccc(F)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cccc2CCN(CCc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1(C)CN(CCc2ccccc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCc2ccc(F)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1CN(CCc2ccc(F)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC(C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
C[C@@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
C[C@H](C[C@@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
CC[C@@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
CC(C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2cc(Cl)c(Cl)cc2C1 |r|
C[C@@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2cc(Cl)c(Cl)cc2C1 |r|
COc1cc2CN(Cc2cc1Cl)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
COc1cc2CN(Cc2cc1Cl)C(=O)C(C)C[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1CN(CCc2cc(Cl)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1CN(CCc2cc(Cl)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCc2cc(Cl)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1CN(CCc2ccc(Cl)c(Cl)c12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1CN(CCc2ccc(Cl)c(Cl)c12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCc2ccc(Cl)c(Cl)c12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Fc1cc2CN(Cc2cc1C(F)(F)F)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)c1cc2CN(Cc2cc1Cl)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC1N(Cc2cc(Cl)c(cc12)C(F)(F)F)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1N(Cc2cc(Cl)c(cc12)C(F)(F)F)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
OCC(CC1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2cc(Cl)c(Cl)cc2C1
FC(F)(F)c1ccc2CN(Cc2c1)C(=O)CCC1(NC(=O)NC1=O)c1nccs1
Fc1ccc2CCN(CCc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)c1ccc2CCN(CCc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC(C)C(C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
CC(C)[C@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
[O-][N+](=O)c1cc2CN(Cc2cc1Cl)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)c1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Clc1cc2CN(Cc2cc1I)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Nc1cc2CN(Cc2cc1Cl)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Cc1cc2CN(Cc2cc1Cl)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)c1cc2CN(Cc2cc1Br)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)c1ccc2CN(Cc2c1)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Clc1cc2CN(Cc2cc1Cl)C(=O)CCC1(NC(=O)NC1=O)c1ccccn1
Cn1ccnc1C1(CCC(=O)N2Cc3ccc(cc3C2)C(F)(F)F)NC(=O)NC1=O
Cn1ccnc1[C@]1(CCC(=O)N2Cc3ccc(cc3C2)C(F)(F)F)NC(=O)NC1=O |r|
CC1(CC1)[C@@]1(CCC(=O)N2Cc3ccc(cc3C2)C(F)(F)F)NC(=O)NC1=O |r|
FC(F)(F)c1ccc2CN(Cc2c1)C(=O)C(COCc1ccccc1)CC1(NC(=O)NC1=O)C1CC1
CC1N(Cc2cc(Cl)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1N(Cc2cc(Cl)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCc2ccc(Cl)c(F)c12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1CN(CCc2ccc(Cl)c(F)c12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1CN(CCc2cc(F)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@H]1CN(CCc2cc(F)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
C[C@@H]1N(Cc2cc(Cl)c(Cl)cc12)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CC(C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2cc(Cl)c(Cl)cc2C1C |r|
C[C@H]1N(Cc2cc(Cl)c(cc12)C(F)(F)F)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
FC(F)(F)Cc1ccc2CN(Cc2c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Cn1ccnc1C1(CCC(=O)N2Cc3cc(Cl)c(cc3C2)C(F)(F)F)NC(=O)NC1=O
Cn1ccnc1[C@]1(CCC(=O)N2Cc3cc(Cl)c(cc3C2)C(F)(F)F)NC(=O)NC1=O |r|
FC(F)c1cc2CN(Cc2cc1F)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |r|
Cc1cc(no1)C1(CCC(=O)N2Cc3cc(Cl)c(cc3C2)C(F)(F)F)NC(=O)NC1=O
Cn1ccc(n1)C1(CCC(=O)N2Cc3cc(Cl)c(cc3C2)C(F)(F)F)NC(=O)NC1=O
Cc1cc(n[nH]1)C1(CCC(=O)N2Cc3cc(Cl)c(cc3C2)C(F)(F)F)NC(=O)NC1=O
FC(F)(F)c1cc2CN(Cc2cc1Cl)C(=O)CCC1(NC(=O)NC1=O)c1ncccn1
Cc1nc(co1)C1(CCC(=O)N2Cc3cc(Cl)c(cc3C2)C(F)(F)F)NC(=O)NC1=O
CCn1ccnc1C1(CCC(=O)N2Cc3cc(Cl)c(cc3C2)C(F)(F)F)NC(=O)NC1=O
FC(F)(F)c1cc2CN(Cc2cc1Cl)C(=O)CC[C@@]1(NC(=O)NC1=O)c1nccs1 |r|
FC(F)(F)c1cc2CN(Cc2cc1Cl)C(=O)CC[C@@]1(NC(=O)NC1=O)c1ccccn1 |r|
FC(F)(F)c1cc2CN(Cc2cc1Cl)C(=O)CC[C@@]1(NC(=O)NC1=O)c1cnccn1 |r|
OC[C@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2cc(Cl)c(cc2C1)C(F)(F)F |r|
CCC(C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
CC[C@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2ccc(cc2C1)C(F)(F)F |r|
C[C@H](C[C@]1(NC(=O)NC1=O)C1CC1)C(=O)N1Cc2cc(Cl)c(Cl)cc2C1 |r|
Cc1cc(COc2ccc(cc2)C(=O)NC2(CC(=O)NO)CCNCC2)c2ccccc2n1
Cc1cc(COc2ccc(cc2)C(=O)NC2(CC(=O)NO)CCOCC2)c2ccccc2n1
SC1=NC(=O)C(S1)=Cc1cccc(Oc2ccccc2)c1 |w:7.8,t:1|
OC(=O)CCN1C(=S)S\C(=C\c2ccc(OCc3ccccc3)c(OCc3ccccc3)c2)C1=O
OC(=O)C(N1C(=S)S\C(=C\c2ccc(OCc3ccccc3)c(OCc3ccccc3)c2)C1=O)c1ccccc1 |w:3.3|
SC1=NC(=O)C(S1)=Cc1cccc(Oc2ccc(Cl)cc2)c1 |w:7.8,t:1|
COc1ccc(Oc2cccc(C=C3SC(S)=NC3=O)c2)cc1 |w:12.11,c:16|
Cc1ccc(Oc2cccc(C=C3SC(S)=NC3=O)c2)cc1 |w:11.10,c:15|
O=C1N(C(=S)S\C1=C\c1ccc(OCc2ccccc2)c(OCc2ccccc2)c1)c1ccccc1
SC1=NC(=O)C(S1)=Cc1cc(OCc2ccccc2)cc(OCc2ccccc2)c1 |w:7.8,t:1|
COc1cc(C=C2SC(S)=NC2=O)ccc1OCc1ccccc1 |w:5.4,c:9|
O=C1N(Cc2ccccc2)C(=S)S\C1=C\c1ccc(OCc2ccccc2)c(OCc2ccccc2)c1
COc1cc(C=C2SC(=S)NC2=O)ccc1OCc1ccc(Cl)cc1 |w:5.4|
O=C1N(CCc2ccccc2)C(=S)S\C1=C\c1ccc(OCc2ccccc2)c(OCc2ccccc2)c1
COc1ccc(COc2ccc(C=C3SC(=S)NC3=O)cc2OC)cc1 |w:12.11|
OC(=O)CN1C(=S)S\C(=C\c2ccc(OCc3ccccc3)c(OCc3ccccc3)c2)C1=O
OC(=O)[C@@H](Cc1ccccc1)N1C(=S)S\C(=C\c2ccc(OCc3ccccc3)c(OCc3ccccc3)c2)C1=O
CC(C)(C)c1ccc(Oc2cccc(C=C3SC(S)=NC3=O)c2)cc1 |w:14.13,c:18|
OC(=O)CN1C(=S)S\C(=C\c2cccc(Oc3ccc(Cl)c(Cl)c3)c2)C1=O
OC(=O)C(N1C(=S)S\C(=C\c2cccc(Oc3ccc(Cl)c(Cl)c3)c2)C1=O)c1ccccc1 |w:3.3|
SC1=NC(=O)C(S1)=Cc1cccc(Oc2ccc(Cl)c(Cl)c2)c1 |w:7.8,t:1|
SC1=NC(=O)C(S1)=Cc1cccc(Oc2cc(Cl)cc(Cl)c2)c1 |w:7.8,t:1|
OC(=O)[C@@H](Cc1ccccc1)N1C(=S)S\C(=C\c2cccc(Oc3ccc(Cl)c(Cl)c3)c2)C1=O
CC(C)[C@@H](N1C(=S)S\C(=C\c2ccc(OCc3ccccc3)c(OCc3ccccc3)c2)C1=O)C(O)=O
CC(C)(C)c1ccc(Oc2cccc(C=C3SC(O)=NC3=O)c2)cc1 |w:14.13,c:18|
Clc1ccc(Oc2cccc(\C=C3\NC(=O)NC3=O)c2)cc1
Clc1cc(Cl)cc(Oc2cccc(\C=C3\NC(=O)NC3=O)c2)c1
FC(F)(F)c1ccc(Oc2cccc(C=C3SC(S)=NC3=O)c2)cc1 |w:14.13,c:18|
CC(C)[C@@H](N1C(=S)S\C(=C\c2cccc(Oc3ccc(Cl)c(Cl)c3)c2)C1=O)C(O)=O
OC1=NC(=O)C(S1)=Cc1cccc(Oc2ccc(Cl)cc2)c1 |w:7.8,t:1|
OC1=NC(=O)C(S1)=Cc1cccc(Oc2ccc(Cl)c(Cl)c2)c1 |w:7.8,t:1|
OC1=NC(=O)C(S1)=Cc1cccc(Oc2cc(Cl)cc(Cl)c2)c1 |w:7.8,t:1|
CC(C)(C)c1ccc(Oc2cccc(\C=C3\NC(=O)NC3=O)c2)cc1
CN1C(=O)NC(=O)\C1=C/c1cccc(Oc2ccc(Cl)cc2)c1
SC1=NC(=O)C(S1)=Cc1cccc(OCc2ccccc2)c1 |w:7.8,t:1|
CN1C(=S)S\C(=C\c2ccc(OCc3ccccc3)c(OCc3ccccc3)c2)C1=O
SC1=NC(=O)C(S1)=Cc1ccc(OCc2ccccc2)c(OCc2ccccc2)c1 |w:7.8,t:1|
CCN1C(=S)S\C(=C\c2ccc(OCc3ccccc3)c(OCc3ccccc3)c2)C1=O
Cn1nc(c(C=C2SC(=S)NC2=O)c1SCc1ccccc1Cl)C(F)(F)F |w:5.4|
FC(F)(F)c1nn(c(N2CCN(CC2)c2ccc(Cl)cc2)c1C=C1SC(=S)NC1=O)-c1ccccc1 |w:22.24|
SC1=NC(=O)C(S1)=Cc1c(SCc2cccs2)n(nc1-c1ccccc1)-c1ccccc1 |w:7.8,t:1|
SC1=NC(=O)C(S1)=Cc1c(SCc2ccco2)n(nc1-c1ccccc1)-c1ccccc1 |w:7.8,t:1|
Oc1nc(S)sc1Cc1c(SCc2ccc(Cl)cc2)n(nc1C(F)(F)F)-c1ccccc1
SC1=NC(=O)C(S1)=Cc1c(SCc2ccco2)n(nc1-c1ccccc1)C1CCCCC1 |w:7.8,t:1|
Cn1nc(c(C=C2SC(S)=NC2=O)c1SCc1ccc(Cl)cc1)C(F)(F)F |w:5.4,c:9|
SC1=NC(=O)C(S1)=Cc1c(nn(C2CCCCC2)c1N1CCN(CC1)c1ncccn1)-c1ccccc1 |w:7.8,t:1|
FC(F)(F)c1nn(c(SCc2ccc(Cl)cc2)c1C=C1SC(S)=NC1=O)-c1ccccc1 |w:18.19,c:24|
FC(F)(F)c1nn(c(OCCc2cccs2)c1C=C1SC(S)=NC1=O)-c1ccccc1 |w:17.18,c:23|
FC(F)(F)c1nn(C2CCCCC2)c(N2CCN(CC2)c2ncccn2)c1C=C1SC(S)=NC1=O |w:27.30,c:35|
CN1CCN(CC1)c1c(C=C2SC(S)=NC2=O)c(nn1-c1ccccc1)-c1ccccc1 |w:9.9,c:14|
FC(F)(F)c1nn(C2CCCCC2)c(SCc2ccc(Cl)cc2)c1C=C1SC(S)=NC1=O |w:24.26,c:31|
Cn1nc(c(C=C2SC(=S)NC2=O)c1N1CCN(CC1)c1ccc(Cl)cc1)C(F)(F)F |w:5.4|
FC(F)(F)c1nn(c(OCCc2ccc(Cl)cc2)c1C=C1SC(S)=NC1=O)-c1ccccc1 |w:19.20,c:25|
FC(F)(F)c1nn(c(SCc2ccccc2)c1C=C1SC(S)=NC1=O)-c1ccccc1 |w:17.18,c:23|
Cn1nc(c(C=C2SC(=S)NC2=O)c1SCc1ccc(cc1)C(C)(C)C)C(F)(F)F |w:5.4|
Cn1nc(c(C=C2SC(=S)NC2=O)c1SCc1ccco1)-c1ccccc1 |w:5.4|
Fc1ccc(CCOc2c(C=C3SC(S)=NC3=O)c(nn2-c2ccccc2)C(F)(F)F)cc1 |w:10.9,c:14|
Cc1ccc(Sc2c(C=C3SC(=S)NC3=O)c(nn2C)-c2ccccc2)cc1 |w:8.7|
CN1c2ccc(cc2C(=O)N(C1=O)Cc3ccc(cc3)C(=O)O)C#CCc4ccccc4
CCCCOc1ccc(Nc2c(N(C)O)c(=O)c2=O)cc1
CCCCOc1ccc(Nc2c(N(O)Cc3ccccc3)c(=O)c2=O)cc1
CCCCOc1ccc(Nc2c(N(O)C(C)C)c(=O)c2=O)cc1
ONC(=O)[C@H]1COCC[C@H]1NC(=O)c1ccc(Cn2c(nc3ccccc23)C(F)(F)F)cc1 |r|
COc1ccc(cc1)C1=NNC2(S1)C(=O)N(Cc1ccccc1)c1ccc(C)cc21 |t:9|
C[C@H]1C[C@](CC(=O)NO)(C[C@@H](C)N1)NC(=O)c1ccc(OCc2cc(C)nc3ccccc23)cc1 |r|
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1Cl
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1[N+]([O-])=O
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1C#N
Cc1ccc(cc1)C(NC(=O)CNCc1ccccc1)c1cc(Cl)c2cccnc2c1O
Oc1c(cc(Br)c2cccnc12)C(NC(=O)COc1ccccc1)c1cccc(c1)[N+]([O-])=O
CN(CC(=O)NC(c1ccc(C)cc1)c1cc(Cl)c2cccnc2c1O)c1ccccc1
CN(CC(=O)NC(c1ccc(C)cc1)c1cc(Cl)c2cccnc2c1O)Cc1ccccc1
CC(=O)c1ccc(NCC(=O)NC(c2cccc(c2)[N+]([O-])=O)c2cc(Cl)c3cccnc3c2O)cc1
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1
Cc1cc(NCC(=O)NC(c2ccccc2Cl)c2cc(Cl)c3cccnc3c2O)ccc1Cl
Cc1cc(NCC(=O)NC(c2cccc(F)c2)c2cc(Cl)c3cccnc3c2O)ccc1Cl
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)CNCc1ccccc1)c1ccccc1Cl
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)CNCc1ccccc1)c1cccc(F)c1
CN(CC(=O)NC(c1ccccc1Cl)c1cc(Cl)c2cccnc2c1O)c1ccccc1
CN(CC(=O)NC(c1cccc(F)c1)c1cc(Cl)c2cccnc2c1O)c1ccccc1
CN(CC(=O)NC(c1ccccc1Cl)c1cc(Cl)c2cccnc2c1O)Cc1ccccc1
CC(=O)Nc1ccc(NCC(=O)NC(c2cccc(c2)[N+]([O-])=O)c2cc(Cl)c3cccnc3c2O)cc1
CN(CC(=O)NC(c1cccc(F)c1)c1cc(Cl)c2cccnc2c1O)Cc1ccccc1
CN(CC(=O)NC(c1cccc(c1)[N+]([O-])=O)c1cc(Cl)c2cccnc2c1O)c1ccccc1
CN(CC(=O)NC(c1cccc(c1)[N+]([O-])=O)c1cc(Cl)c2cccnc2c1O)Cc1ccccc1
Oc1c(cc(Br)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1Cl
Oc1c(cc([N+]([O-])=O)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1Cl
Cc1cc(C(NC(=O)COc2ccccc2)c2cccc(c2)[N+]([O-])=O)c(O)c2ncccc12
Cc1cc(C(NC(=O)COc2ccccc2)c2ccccc2Cl)c(O)c2ncccc12
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccc(Cl)cc1)c1ccccc1
CN(C)c1cccc(OCC(=O)NC(c2cccc(F)c2)c2cc(Cl)c3cccnc3c2O)c1
Cc1ccc(cc1)C(NC(=O)COc1ccccc1)c1cc(Cl)c2cccnc2c1O
CC(=O)Nc1ccc(OCC(=O)NC(c2cccc(F)c2)c2cc(Cl)c3cccnc3c2O)cc1
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1cccnc1)c1cccc(F)c1
COc1ccc(cc1)C(NC(=O)COc1cccnc1)c1cc(Cl)c2cccnc2c1O
COc1ccc(cc1)C(NC(=O)COc1ccc(C)cc1)c1cc(Cl)c2cccnc2c1O
COc1ccc(OCC(=O)NC(c2ccc(OC)cc2)c2cc(Cl)c3cccnc3c2O)cc1
COc1ccc(cc1)C(NC(=O)COc1cccc(c1)N(C)C)c1cc(Cl)c2cccnc2c1O
COc1ccc(cc1)C(NC(=O)COc1ccc(Oc2ccccc2)cc1)c1cc(Cl)c2cccnc2c1O
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1cccnc1)c1cccc(c1)[N+]([O-])=O
Oc1c(ccc2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1
Oc1c(cc(F)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1
Oc1c(cc([N+]([O-])=O)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1
Cc1ccc(cc1)C(NC(=O)COCc1ccccc1)c1cc(Cl)c2cccnc2c1O
Cc1cc(NCC(=O)NC(c2cccc(c2)[N+]([O-])=O)c2cc(Cl)c3cccnc3c2O)ccc1Cl
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1cccc(F)c1
CC(=O)Nc1ccc(OCC(=O)NC(c2ccccc2Cl)c2cc(Cl)c3cccnc3c2O)cc1
CN(C)c1cccc(NCC(=O)NC(c2ccc(C)cc2)c2cc(Cl)c3cccnc3c2O)c1
CC(=O)c1ccc(OCC(=O)NC(c2cccc(c2)[N+]([O-])=O)c2cc(Cl)c3cccnc3c2O)cc1
Cc1cc(OCC(=O)NC(c2ccccc2Cl)c2cc(Cl)c3cccnc3c2O)ccc1Cl
Cc1ccc(cc1)C(NC(=O)CNc1ccc(Cl)c(C)c1)c1cc(Cl)c2cccnc2c1O
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COCc1ccccc1)c1cccc(F)c1
Cc1cc(OCC(=O)NC(c2cccc(c2)[N+]([O-])=O)c2cc(Cl)c3cccnc3c2O)ccc1Cl
CC(C)(C)c1ccc(OCC(=O)NC(c2ccccc2Cl)c2cc(Cl)c3cccnc3c2O)cc1
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1cc(Cl)cc(Cl)c1)c1cccc(c1)[N+]([O-])=O
COc1ccc(cc1)C(NC(=O)COc1ccc(NC(C)=O)cc1)c1cc(Cl)c2cccnc2c1O
Cc1ccc(OCC(=O)NC(c2ccccc2)c2cc(Cl)c3cccnc3c2O)cc1
COc1ccc(cc1)C(NC(=O)COc1ccc(Cl)c(C)c1)c1cc(Cl)c2cccnc2c1O
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1cccc(c1)[N+]([O-])=O
COc1ccc(cc1)C(NC(=O)COc1ccccc1)c1cc(Cl)c2cccnc2c1O
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1F
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccc(Cl)cc1
Cc1ccccc1C(NC(=O)COc1ccccc1)c1cc(Cl)c2cccnc2c1O
CC(=O)c1ccc(NCC(=O)NC(c2ccc(C)cc2)c2cc(Cl)c3cccnc3c2O)cc1
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccc(cc1)[N+]([O-])=O
Oc1c(cc(Cl)c2cccnc12)C(NC(=O)COc1ccccc1)c1ccccc1C(F)(F)F
CN(C)c1cccc(OCC(=O)NC(c2ccccc2Cl)c2cc(Cl)c3cccnc3c2O)c1
Cc1ccc(cc1)C(NC(=O)CNc1ccc(cc1)C#N)c1cc(Cl)c2cccnc2c1O
CC(C)[C@@H](NS(=O)(=O)c1ccc(cc1)-c1ccc(COc2ccc(cc2)C(=O)C2CCCCC2)cc1)C(O)=O |r|
CC(C)[C@@H](NS(=O)(=O)c1ccc(cc1)-c1ccc(COc2ccc3C(=O)CCCc3c2)cc1)C(O)=O |r|
CC(C)[C@@H](NS(=O)(=O)c1ccc(cc1)-c1ccc(COc2ccc(cc2)C(=O)C(C)C)cc1)C(O)=O |r|
CC(C)[C@H](NS(=O)(=O)c1ccc2c(c1)oc1ccc(cc21)N1CCOC1=O)C(O)=O |r|
Cc1cc(cc(n1)C(=O)NCc1ccc(F)cc1)-c1nnn(C[C@H]2CC[C@@H](CC2)C(O)=O)n1 |r,wU:26.31,wD:23.24,(30.11,-12.24,;29.32,-10.92,;30.07,-9.57,;29.28,-8.26,;27.74,-8.27,;26.98,-9.62,;27.77,-10.94,;25.44,-9.64,;24.69,-10.98,;24.66,-8.31,;23.12,-8.33,;22.33,-7.01,;23.08,-5.67,;22.3,-4.34,;20.75,-4.36,;19.97,-3.04,;20,-5.72,;20.79,-7.03,;30.03,-6.91,;29.39,-5.51,;30.52,-4.46,;31.87,-5.21,;33.27,-4.57,;34.61,-5.32,;34.63,-6.85,;35.98,-7.6,;37.3,-6.81,;37.27,-5.26,;35.93,-4.52,;38.65,-7.56,;38.68,-9.1,;39.97,-6.77,;31.57,-6.73,)|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1ccc(s1)-n1cc(Cl)cn1)C(O)=O |r|
C[C@@]1(C[C@@]1(NS(=O)(=O)c1ccc(s1)-n1cc(Cl)cn1)C(O)=O)c1ccccc1 |r|
C[C@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1ccc(s1)-c1ccc(Cl)cc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1ccc(s1)-c1ccc(Cl)cc1)C(O)=O |r|
C[C@@]1(C[C@@]1(NS(=O)(=O)c1ccc(s1)-c1ccc(Cl)cc1)C(O)=O)c1ccccc1 |r|
OC(=O)[C@@]1(C[C@@H]1C1CCCCC1)NS(=O)(=O)c1ccc(s1)-n1cc(Cl)cn1 |r|
CC(C)[C@H]1C[C@@]1(NS(=O)(=O)c1ccc(s1)-n1cc(Cl)cn1)C(O)=O |r|
C[C@H]1[C@@H](C)[C@@]1(NS(=O)(=O)c1ccc(s1)-n1cc(Cl)cn1)C(O)=O |r|
Clc1ccc(OCc2n[n-]c(=S)n2Cc2ccc(cc2)-c2ccccc2)cc1
Clc1ccc(OCc2n[n-]c(=S)n2Cc2ccccc2-c2ccccc2)cc1
S=c1[n-]nc(Cc2ccc(cc2)-c2ccccc2)n1Cc1ccccc1-c1ccccc1
S=c1[n-]nc(CCc2nc(no2)-c2ccccc2)n1CCCn1ccnc1
Clc1ccc2OC(CNc2c1)c1n[n-]c(=S)n1Cc1ccc(cc1)-c1ccccc1
S=c1[n-]nc(Cc2nc(no2)-c2ccccc2)n1CCCn1ccnc1
CSc1nnc(Cc2nc(no2)-c2ccccc2)n1CCCn1ccnc1
Clc1ccc(OCc2n[n-]c(=S)n2Cc2cccc(c2)-c2ccccc2)cc1
Clc1ccc(OCc2n[n-]c(=S)n2Cc2ccccc2)cc1
Fc1ccc(OCc2n[n-]c(=S)n2Cc2ccc(cc2)-c2ccccc2)cc1
S=c1[n-]nc(Cc2ccc(cc2)-c2ccccc2)n1CCCc1ccccc1
CSc1nnc(COc2ccc(Cl)cc2)n1Cc1ccccc1-c1ccccc1
Clc1ccc(OCc2n[n-]c(=S)n2CCCn2ccnc2)cc1
S=c1[n-]nc(Cc2nc(no2)-c2ccccc2)n1CCCc1ccccc1
S=c1[n-]nc(Cc2nc(no2)-c2cnccn2)n1CCCc1ccccc1
CSc1nnc(COc2ccc(Cl)cc2)n1Cc1ccc(cc1)-c1ccccc1
Clc1ccc(OCc2n[n-]c(=S)n2CCCc2ccccc2)cc1
Clc1ccc(OCc2n[n-]c(=S)n2CCc2ccccc2)cc1
S=c1[n-]nc(Cc2nc(no2)-c2ccccc2)n1Cc1ccccc1-c1ccccc1
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCc2c(C1)nc1cc(F)ccn21)C(O)=O |r|
COc1ccc2n3CCN(Cc3nc2c1)S(=O)(=O)N[C@]1([C@H](C)[C@@H]1c1ccccc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)nc1cc(C)ccc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)nc1cc(ccc21)C#N)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)nc1ccc(F)cc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)nc1cc(F)ccc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)nc1ccccc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1Cc2nc3cc(Cl)ccn3c2C1)C(O)=O |r|
CC1(C)C[C@@H](O)CN([C@H]1C(=O)NO)S(=O)(=O)c1ccc(OCc2ccc(Cl)cc2Cl)cc1
C[C@@H]1[C@](C)(c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1cc(on1)C(F)F)C(O)=O |r|
C[C@@H]1[C@](C)(c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1ccc(s1)C#N)C(O)=O |r|
C[C@@H]1[C@](C)(c2ccccc2)[C@]1(NS(=O)(=O)N1CCc2c(C1)nn1cc(F)ccc21)C(O)=O |r|
C[C@@H]1[C@](C)(c2ccccc2)[C@]1(NS(=O)(=O)N1CCc2c(C1)nc1cc(F)ccn21)C(O)=O |r|
C[C@@H]1[C@](C)(c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)nc1cc(F)ccc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCc2c(C1)[nH]c1cc(F)ccc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCc2c(C1)nn1cc(F)ccc21)C(O)=O |r|
ONC(=O)[C@@H](NCC1CC1)[C@@H](Cc1cccc(O)c1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12 |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1cc2nn3cc(Cl)ccc3c2s1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1cc2nc3cc(Cl)ccn3c2s1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1ccc(s1)-n1cc(C)cn1)C(O)=O |r|
COc1cnn(c1)-c1ccc(s1)S(=O)(=O)N[C@]1([C@H](C)[C@@H]1c1ccccc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1cc(C)c(s1)-n1cc(Cl)cn1)C(O)=O |r|
CC(C)(NC(=O)[C@H](CCC(O)=O)NC(=O)c1ccc(cc1)-c1ccccc1)c1ccccc1 |r|
ONC(=O)c1nc2ccccc2c2C(=O)N(Cc12)c1ccc(OCc2ccccc2)cc1
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1ccc(F)cc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1ccc(cc1)C1CC1)C(O)=O
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN(C(CO)C1)c1ccc(Cl)cc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN(c2ccc(Cl)cc2)C(C)(C)C1)C(O)=O |r|
CCC1CN(CCN1c1ccc(Cl)cc1)S(=O)(=O)N[C@]1([C@H](C)[C@@H]1c1ccccc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@@H](C)C1)c1ccc(Cl)cc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1ccc(Cl)cc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCC(=CC1)c1ccc(Cl)cc1)C(O)=O |r,c:19|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN(CC1)c1ccc(Cl)cc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1cc2[nH]c3ccc(F)cc3c2s1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1cc2[nH]c3cc(F)ccc3c2s1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)c1cc2[nH]c3cc(Cl)ccc3c2s1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)cc1cc(Cl)sc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCc2c(C1)nc1cc(Cl)ccn21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)nc1cc(Cl)ccc21)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCn2c(C1)cc1cc(Cl)ccc21)C(O)=O |r|
COCc1cc(no1)N1CCN(C[C@H]1C)S(=O)(=O)N[C@]1([C@H](C)[C@@H]1c1ccccc1)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1cc(on1)C(C)(F)F)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1cc(on1)C(F)F)C(O)=O |r|
C[C@@H]1[C@H](c2ccccc2)[C@]1(NS(=O)(=O)N1CCN([C@H](C)C1)c1ccc(s1)C#N)C(O)=O |r|
C[C@@H](C[C@@](C)(CS(=O)(=O)N1CCC(CCc2c(C)noc2C)CC1)N(O)C=O)c1ncc(F)cn1 |r|
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCCCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCOC(C)(C)C1)N(O)C=O
CN1CCC(CS(=O)(=O)N2CCC(CCc3c(C)noc3C)CC2)(CC1)N(O)C=O
CS(=O)(=O)c1ccc(CCC2CCN(CC2)S(=O)(=O)CC2(CCOCC2)N(O)C=O)c(c1)C1CC1
Cc1cc(ccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O)S(C)(=O)=O
Cc1cc(Cl)ccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
Cc1ccccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
Cc1ccncc1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
ON(C=O)C1(CS(=O)(=O)N2CCC(CCc3ccccc3)CC2)CCOCC1
ON(C=O)C1(CS(=O)(=O)N2CCC(CCc3ccc(F)cc3C(F)(F)F)CC2)CCN(CC1)C(=O)C1CCC1
Cc1cc(ccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCN(CC1)C(=O)C1CCC1)N(O)C=O)C(F)(F)F
Cc1cc(Cl)ccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCN(CC1)C(=O)C1CCC1)N(O)C=O
Cc1nsc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
Cc1cnc(C)c(CCC2CCN(CC2)S(=O)(=O)CC2(CCOCC2)N(O)C=O)c1
Cc1cccnc1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
Cc1cc(C)c(CCC2CCN(CC2)S(=O)(=O)CC2(CCOCC2)N(O)C=O)cn1
Cc1ccccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCN(CC1)C(=O)C1CCC1)N(O)C=O
Cc1cc(CCC2CCN(CC2)S(=O)(=O)CC2(CCOCC2)N(O)C=O)c(C)cn1
Cc1cc(F)ccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCN(CC1)C(=O)C1CCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCN(CC1)C(=O)N1CCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCN(CC1)S(C)(=O)=O)N(O)C=O
Cc1cc(F)ccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
CC(=O)N1CCC(CS(=O)(=O)N2CCC(CCc3c(C)noc3C)CC2)(CC1)N(O)C=O
Cc1ncccc1CCC1CCN(CC1)S(=O)(=O)CC1(CCOCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCC(F)(F)CC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCS(=O)(=O)CC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCCCCC1)N(O)C=O
Cc1noc(C)c1CCC1CCN(CC1)S(=O)(=O)CC1(CCN(CC1)C(=O)C1CCC1)N(O)C=O
OC(=O)CC[C@H](NC(=O)c1ccc(cc1)-c1ccccc1)c1nnc(CCc2ccccc2)o1 |r|
COc1cc(CCc2nnc(o2)[C@H](CCC(O)=O)NC(=O)c2ccc(cc2)-c2ccccc2)cc(OC)c1OC |r|
COc1cc(Cc2nnc(o2)[C@H](CCC(O)=O)NC(=O)c2ccc(cc2)-c2ccccc2)cc(OC)c1OC |r|
COc1ccc(CCc2nnc(o2)[C@H](CCC(O)=O)NC(=O)c2ccc(cc2)-c2ccccc2)cc1 |r|
CC(C)[C@@H](NS(=O)(=O)c1ccc(cc1)-c1ccc(OCc2oc3ccccc3c2C)cc1)C(O)=O |r|
CC(C)[C@@H](NS(=O)(=O)c1ccc(cc1)-c1ccc(OCc2cccc(c2)C(F)(F)F)cc1)C(O)=O |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC#N)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCc2csc(n2)-c2ccccc2)nc(NC2CCCC2)n1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCOC)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCO)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCC(C)C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CCCN(C)c1nc(NCc2csc(n2)-c2ccccc2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCc2csc(n2)-c2ccccc2)nc(NC2CC2)n1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC2CC2)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CCCNc1nc(NCc2csc(n2)-c2ccccc2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1ncnc(NCc2csc(n2)-c2cccs2)n1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(F)cc1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1cccc(c1)C#N |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1cccc(O)c1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(cc1)-c1ccccc1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(C)c(C)c1 |r|
Cc1ccc(cc1F)S(=O)(=O)N[C@@H]1CCN(C1)c1nc(NCCc2cccc3ccccc23)nc(N[C@H]2CCCCNC2=O)n1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(cc1)C#N |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(cc1)S(C)(=O)=O |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2csc(n2)-c2cccs2)n1 |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2cccc(c2)-c2ccccc2)n1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1cccc(Cl)c1 |r|
C=CCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc2ccccc2c1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2csc(n2)-c2cccs2)n1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCC2CCOCC2)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2ccc(cc2)-c2ccccc2)n1 |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CCCCNc1nc(NCc2ccc(CCCC)cc2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCNc1nc(NCc2cn(C)cn2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCCNc1nc(NCc2cc(cs2)C#N)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCCNc1nc(NCc2cc(C)cs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCCNc1nc(NCc2cccc(C)c2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCCNc1nc(NCc2cccc(C)n2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
Cc1nc(CNc2nc(NCCC=C)nc(n2)N2CCC[C@@H]2CNS(=O)(=O)c2ccc(cc2)C(F)(F)F)cs1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(O)cc1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(Cl)cc1 |r|
CCCCNc1nc(NCc2ccsc2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCCNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(cc1)C(F)(F)F |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2ccccc2)n1 |r|
Cc1ccc(cc1F)S(=O)(=O)N[C@@H]1CCN(C1)c1nc(NCc2ccccc2)nc(N[C@H]2CCCCNC2=O)n1 |r|
COc1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
FC(F)(F)c1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
C=CCCNc1nc(NCc2csc(n2)-c2ccccc2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)C1CC1 |r|
C=CCCNc1nc(NCc2csc(n2)-c2ccccc2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccccc1 |r|
C[C@@]1(O)CCCN([C@H]1C(=O)NO)S(=O)(=O)c1ccc(OCc2ccc(F)cc2Cl)cc1
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCc2csc(n2)-c2cccs2)[nH]c(=O)n1 |r|
FC(F)(F)c1cccc(c1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCCC=C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@@H]1CCN(C1)c1nc(NCCC=C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CNc1nc(NCc2csc(n2)-c2cccs2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(cc1)C(F)(F)F |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCCN1c1nc(NCC2CC2)nc(NCc2csc(n2)-c2cccs2)n1 |r|
CCCCNc1nc(NC(C)C)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
CCCCNc1nc(NCC2CC2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@H]1CCN(C1)c1nc(NCCC=C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
FC(F)(F)c1ccc(cc1)S(=O)(=O)NC[C@@H]1CCCN1c1nc(NCCC=C)nc(NCc2csc(n2)-c2ccccc2)n1 |r|
CCCCNc1nc(NC2CCCC2)nc(n1)N1CCC[C@@H]1CNS(=O)(=O)c1ccc(CCC)cc1 |r|
ONC(=O)CNS(=O)(=O)c1ccc(Oc2ccccc2)cc1
ONC(=O)CNS(=O)(=O)c1ccc(OCc2ccccc2)cc1
ONC(=O)CNS(=O)(=O)c1ccc(Oc2ccccc2)nc1
ONC(=O)CCNS(=O)(=O)c1ccc(Oc2ccccc2)cc1
ONC(=O)CNS(=O)(=O)c1ccc(OCc2ccc(F)cc2Cl)cc1
CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CC(C)C)CC(=O)NO |r|
CC(C)CN(CC(=O)NO)S(=O)(=O)c1ccc(OCc2ccccc2)cc1
CCCCOc1ccc(cc1)S(=O)(=O)NCC(=O)NO
C[C@]1(C(=O)NC(=O)N1)CNC(=O)COc2ccc(cc2)Cl
C[C@]1(CNC(=O)c2cc3cc(Cl)ccc3o2)NC(=O)NC1=O |r|
Clc1ccc2oc(cc2c1)C(=O)NC[C@]1(NC(=O)NC1=O)c1ccccc1 |r|
Cc1cccnc1[C@]1(CNC(=O)c2cc3cc(Cl)ccc3o2)NC(=O)NC1=O |r|
c1cc2c(cc1Cl)cc(o2)C(=O)NC[C@@]3(C(=O)NC(=O)N3)c4nccs4
Cn1ccnc1[C@]2(C(=O)NC(=O)N2)CNC(=O)c3cc4cc(ccc4o3)Cl
Cn1nccc1[C@]1(CNC(=O)c2cc3cc(Cl)ccc3o2)NC(=O)NC1=O |r|
Cn1ccnc1[C@]1(CNC(=O)c2cc3cc(ccc3o2)C(F)(F)F)NC(=O)NC1=O |r|
CCN(C(=O)c1ccc(CNc2nc(NCCN3CCN(C)CC3)nc(n2)N2CCc3cc(OC)c(OC)cc3C2)cc1)c1cccc(C)c1
CC(C)C[C@H]([C@@H](C(=O)NO)O)C(=O)N[C@H](C(=O)NC)C(C)(C)C
FC(F)(F)c1ccc(CCC(=O)NC[C@]2(NC(=O)NC2=O)C2CC2)cc1 |r|
C[C@@H](Cc1ccc(cc1)C(F)(F)F)C(=O)NC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CN(C)C(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
CCCc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
CC(C)c1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
CCc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
O=C1CS\C(N1)=C\c1nc(cs1)-c1ccccc1
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccc(Br)cn1
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccn1
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1sccc1Br
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccc(Br)s1
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1cccs1
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccc(cc1)-c1ccccc1
COc1ccc(cc1)-c1nc(\C=C2/NC(=O)CS2)sc1CC(O)=O
Cc1ccc(cc1)-c1nc(\C=C2/NC(=O)CS2)sc1CC(O)=O
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1O
Cc1csc(Cc2nc(c(CC(O)=O)s2)-c2ccccc2)n1
Cn1c(Cc2nc(c(CC(O)=O)s2)-c2ccccc2)nc2ccccc12
OC(=O)Cc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
OC(=O)CCCc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
OC(=O)CCc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
CC(C(O)=O)c1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
OC(=O)c1sc(\C=C2/NC(=O)CS2)nc1-c1ccccc1
OC(=O)CCc1sc(\C=C2/NC(=O)CS2)nc1-c1ccccn1
ONC(=O)C1(CCN(Cc2ccccc2)CC1)S(=O)(=O)c1ccc(Oc2ccc(Cl)cc2)cc1
OC(=O)CCc1sc(\C=C2/NC(=O)CS2)nc1-c1ccc(Br)cn1
OC(=O)CCc1sc(\C=C2/NC(=O)CS2)nc1-c1sccc1Br
OC(=O)CCc1sc(\C=C2/NC(=O)CS2)nc1-c1ccc(cc1)-c1ccccc1
Clc1ccc(OCC(=O)NNC(=S)NCc2cccnc2)cc1
Clc1ccc(OCC(=O)Nn2ccn(Cc3ccc(cc3)-c3ccccc3)c2=S)cc1
Clc1ccc(OCC(=O)NCC(=S)NCc2ccc(cc2)-c2ccccc2)cc1
CN(NC(=S)NCCCCC1CCCCC1)C(=O)COc1ccc(Cl)cc1
CN(NC(=S)NCc1ccc(cc1)-c1ccccc1)C(=O)COc1ccc(Cl)cc1
CC(=O)NNC(=S)NCCCCC1CCCCC1
COc1ccc(OCC(=O)NNC(=S)NCCCCC2CCCCC2)cc1
O=C(COc1ccccc1)NNC(=S)NCCCCC1CCCCC1
Fc1ccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)cc1
O=C(COc1ccc(cc1)-c1ccccc1)NNC(=S)NCc1ccc(cc1)-c1ccccc1
SC(CNC(=O)COc1ccc(Cl)cc1)C(=O)NCCc1ccccc1
Clc1ccc(CCNC(=S)NNC(=O)Cc2ccc(cc2)-c2ccccc2)cc1
Clc1ccc(OCC(=O)NNC(=S)N2CCC(Cc3ccccc3)CC2)cc1
CN(CCCCc1ccccc1)C(=S)NNC(=O)COc1ccc(Cl)cc1
Clc1ccc(cc1)C(=O)NNC(=S)NCCCCC1CCCCC1
O=C(Cc1nc(no1)-c1cnccn1)NNC(=S)NCCCCC1CCCCC1
O=C(Cc1nc(no1)-c1ccccc1)NNC(=S)NCCCCC1CCCCC1
O=C(Cc1ccc(cc1)-c1ccccc1)NNC(=S)NCCCCC1CCCCC1
Clc1ccc2OC(CNc2c1)C(=O)NNC(=S)NCCCCC1CCCCC1
O=C(COc1cccc2ccccc12)NNC(=S)NCCCCC1CCCCC1
[O-][N+](=O)c1ccc(OCC(=O)NNC(=S)NCCCCC2CCCCC2)cc1
FC(F)(F)c1ccc(OCC(=O)NNC(=S)NCCCCC2CCCCC2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCCCCC2CCCCC2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCCCCc2ccccc2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCCCc2ccccc2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCCCn2ccnc2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCCc2ccccc2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCc2ccccc2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCc2ccccc2-c2ccccc2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCc2cccc(c2)-c2ccccc2)cc1
Clc1ccc(NCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)cc1
Clc1ccc(cc1)C(=O)NNC(=S)NCc1ccc(cc1)-c1ccccc1
Clc1ccc2OC(CNc2c1)C(=O)NNC(=S)NCc1ccc(cc1)-c1ccccc1
CC(C)(Oc1ccc(Cl)cc1)C(=O)NNC(=S)NCc1ccc(cc1)-c1ccccc1
[O-][N+](=O)c1ccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)cc1
O=C(COc1cccc2ccccc12)NNC(=S)NCc1ccc(cc1)-c1ccccc1
O=C(COc1ccc2ccccc2c1)NNC(=S)NCc1ccc(cc1)-c1ccccc1
O=C(COc1ccc(OCc2ccccc2)cc1)NNC(=S)NCc1ccc(cc1)-c1ccccc1
COc1ccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)cc1
Clc1ccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)cc1Cl
Clc1ccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)c(Cl)c1
Clc1cccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)c1
Clc1ccccc1OCC(=O)NNC(=S)NCc1ccc(cc1)-c1ccccc1
FC(F)(F)c1ccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)cc1
O=C(COc1ccccc1)NNC(=S)NCc1ccc(cc1)-c1ccccc1
Clc1ccc(OCC(=O)NNC(=S)NCc2ccc(cc2)-c2ccccc2)cc1
CCCC1SC(NC1=O)=Cc1nc2ccc(F)cc2[nH]1 |w:9.10|
CCCC1SC(NC1=O)=Cc1nc2ccc(cc2[nH]1)C(F)(F)F |w:9.10|
CCCC1S\C(NC1=O)=C\c1nc2cc(C)c(C)cc2[nH]1
CCCC1SC(NC1=O)=Cc1nc2ccc(C)cc2[nH]1 |w:9.10|
CCCC1SC(NC1=O)=Cc1nc2c(C)cccc2[nH]1 |w:9.10|
OCCC1S\C(NC1=O)=C\c1nc2ccccc2[nH]1
OC(=O)CC1S\C(NC1=O)=C\c1nc2ccccc2[nH]1
CCCCC1S\C(NC1=O)=C\c1nc2ccccc2[nH]1
CCCC1S\C(NC1=O)=C\c1nc2ccccc2[nH]1
CCC1S\C(NC1=O)=C\c1nc2ccccc2[nH]1
Cc1ccc2nc(C=C3NC(=O)CS3)[nH]c2c1C |w:7.6|
Cc1cc2nc(\C=C3/NC(=O)CS3)[nH]c2cc1C
Cc1ccc2nc(C=C3NC(=O)CS3)[nH]c2c1 |w:7.6|
Cc1cccc2[nH]c(C=C3NC(=O)CS3)nc12 |w:8.7|
Cn1c(\C=C2/NC(=O)CS2)nc2ccccc12
CC1S\C(NC1=O)=C\c1nc2ccccc2[nH]1
O=C1CS\C(N1)=C\c1nc-2c(CSc3ccccc-23)s1
O=C1CS\C(N1)=C\c1nc-2c(CCc3ccccc-23)s1
O=C1CS\C(N1)=C\c1nc-2c(Cc3ccccc-23)s1
O=C1CS\C(N1)=C\c1nc2cc3ccccc3cc2[nH]1
O=C1CS\C(N1)=C\c1nc2ccccc2[nH]1
O=C1CS\C(N1)=C\c1nc2ccccc2s1
O=C1CS\C(N1)=C\c1nc2ccccc2o1
O=C1CSC(N1)=Cc1cnc[nH]1 |w:6.7|
O=C1CS\C(N1)=C\c1cccs1
Oc1csc(\C=C2/NC(=O)CS2)n1
O=C1CS\C(N1)=C\c1nc(cs1)-c1ccccn1
Cc1cnc(n1C)[C@]1(CNC(=O)c2cc3cc(Cl)ccc3o2)NC(=O)NC1=O |r|
CCn1ccnc1[C@]1(CNC(=O)c2cc3cc(ccc3o2)C(F)(F)F)NC(=O)NC1=O |r|
FC(F)(F)c1ccc2oc(cc2c1)C(=O)NC[C@]1(NC(=O)NC1=O)C1CC1 |r|
CCn1ccnc1[C@]1(CNC(=O)c2cc3cc(Cl)ccc3o2)NC(=O)NC1=O |r|
Cc1cnc(n1C)[C@]1(CNC(=O)c2cc3cc(ccc3o2)C(F)(F)F)NC(=O)NC1=O |r|
O=C(CCC1NC(=O)NC1=O)N1CCN(CC1)c1ccccc1
Fc1ccc(cc1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
Clc1ccc(cc1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
COc1ccc(cc1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
FC(F)(F)c1ccc(cc1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
O=C(CCC1NC(=O)NC1=O)N1CCN(CC1)c1ccc(cc1)-c1ccccc1
Fc1cccc(c1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
Clc1cccc(c1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
COc1cccc(c1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
O=C(CCC1NC(=O)NC1=O)N1CCN(CC1)c1cccc(c1)-c1ccccc1
Clc1ccccc1N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
COc1ccccc1N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
O=C(CCC1NC(=O)NC1=O)N1CCN(CC1)c1ccccn1
O=C(CCC1NC(=O)NC1=O)N1CCN(CC1)c1cccnc1
O=C(CCC1NC(=O)NC1=O)N1CCN(CC1)c1ccncc1
O=C(CCC1NC(=O)NC1=O)N1CCN(CC1)C1CCCCC1
Clc1ccc(cc1Cl)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
Clc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CCC1NC(=O)NC1=O
O=C(CC1NC(=O)NC1=O)N1CCN(CC1)c1ccccc1
O=C(CCCC1NC(=O)NC1=O)N1CCN(CC1)c1ccccc1
CC1CN(CCN1C(=O)CCC1(C)NC(=O)NC1=O)c1ccccc1
CC1(CCC(=O)N2CC3CC2CN3c2ccccc2)NC(=O)NC1=O
CC1(CCC(=O)N2CCc3ccccc3C2)NC(=O)NC1=O
CC1(C)CN(CCN1c1ccccc1)C(=O)CCC1(NC(=O)NC1=O)c1ccccc1
O=C(CCC1(NC(=O)NC1=O)c1ccccc1)N1CCCN(CC1)c1ccccc1
CC1(CCN(CC1)C(=O)CCC1(NC(=O)NC1=O)C1CC1)c1ccccc1
O=C(CCC1(NC(=O)NC1=O)C1CC1)N1CC2CCC(C1)N2c1ccccc1
Cc1ccccc1N1CCN(CC1)C(=O)CC[C@@]1(NC(=O)NC1=O)c1ccccc1 |r|
Clc1cccc(c1)N1CCN(CCCC2(NC(=O)NC2=O)c2ccccc2)CC1
Clc1cc(Cl)cc(c1)N1CCN(CC1)C(=O)CC[C@H]1NC(=O)NC1=O |r|
CC(C)(Cc1ccc(F)cc1)NC(=O)[C@H](CCC(O)=O)NC(=O)c1ccc(cc1)-c1ccccc1 |r|
CC1[C@](C)(c2ccccc2)[C@]1(NS(=O)(=O)N1CCc2c(C1)nc1cc(F)ccn21)C(O)=O |r|
CCCNc1nc(NCc2nccn2C)nc(n1)N1CCCC1CNS(=O)(=O)c1ccc(CCC)cc1
ONC(=O)C[C@@H](Cc1cccc(O)c1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12
c1cc(c(cc1C2=CC(=O)c3c(cc(cc3O2)O)O)O)O
CC(C)[C@@H](N(Cc1cn(CCCO[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2NC(C)=O)nn1)S(=O)(=O)c1ccc(cc1)-c1ccccc1)C(O)=O |r|
CCC(C)N(Cc1cn(CCCO[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2NC(C)=O)nn1)S(=O)(=O)c1ccc(cc1)-c1ccccc1 |r|
c1c(cc(c(c1O)O)O)[C@@H]2[C@@H](Cc3c(cc(cc3O2)O)O)OC(=O)c4cc(c(c(c4)O)O)O
Oc1cc(O)c2C[C@@H](OC(=O)c3cc(O)c(O)c(O)c3)[C@H](Oc2c1)c1ccc(O)c(O)c1 |r|
c1cc(c(cc1\C=C\c2cc(cc(c2)O)O)O)O
c1cc(c(c(c1)O)O)O