1444 SMILES Strings for Cholesteryl ester transfer protein

Compound Name
SMILES String
COc1ccc(cc1-c1ccc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1cc(F)c(cc1-c1ccc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(CCC(O)=O)cc1-c1ccc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)C(F)(F)F |r|
COc1ccc(cc1-c1cnc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CCC1)N1CC(F)C1)-c1ccc(CO)cc1C |r|
COc1cc(F)c(cc1-c1cnc(nc1CN1C(=O)OC(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)N(C)C)C(C)C
COc1cc(F)c(cc1-c1cnc(nc1CN1C(=O)OC(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CCC1)N(C)C)C(C)C
COc1ccc(cc1-c1cnc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CCC1)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CCC1)N1CCOCC1)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CCC1)N(C)S(C)(=O)=O)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)N1CCOCC1)-c1ccc(cc1C)C(O)=O |r|
COC(=O)c1ccc(c(C)c1)-c1ccc(OC)c(c1)-c1cnc(SC)nc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1 |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)C(F)(F)F)C(C)C |r|
CC[C@@H]1C[C@@H](CN1C(=O)C1CCCCC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OC(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OCC(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OCC(C)(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OC1CCOCC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OCC1CCOCC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OCC1(C)COC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CCC(CC)OC(=O)N1C[C@H](C[C@H]1CC)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OCC(F)(F)F)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OC1CCCC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CCC(C)OC(=O)N1C[C@H](C[C@H]1CC)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OCC1(CC)COC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1C(=O)OC(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)N1CC[C@H](O)C1
CC[C@@H]1C[C@@H](CN1C(=O)OC(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cn[nH]c1
CC[C@@H]1C[C@@H](CN1C(=O)N1CCCC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1
CC[C@H]1C[C@H](CN1C(=O)N1CCCCC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1
CC[C@@H]1C[C@@H](CN1C(=O)N1CCOCC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1
CC[C@@H]1C[C@@H](CN1C(=O)N(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1
CC[C@@H]1C[C@@H](CN1c1nc(ncc1Cl)N1CCC(O)CC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)N1CCC(O)C1 |r|
CC[C@@H]1C[C@@H](CN1c1nc(ncc1Cl)N1CCC(O)CC1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1c1nc(ncc1Cl)N1CCC(CC1)C(O)=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r|
CC[C@@H]1C[C@@H](CN1c1nc(ncc1Cl)N1CCC(CC1)C(O)=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)N1CCOCC1 |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(C)cc(c1)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)-c1n[nH]c(=O)o1 |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(C)cc(c1)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)-c1nnc(N)o1 |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COC(=O)c1ccc(c(C)c1)-c1cc(c(OC)cc1F)-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)[C@H]1C[C@@H](C1)C(O)=O |r,wU:43.50,17.25,18.26,wD:41.45,14.15,(-4.15,6.78,;-2.82,7.55,;-1.49,6.78,;-.15,7.55,;1.18,6.78,;1.18,5.24,;-.15,4.47,;-1.49,5.24,;-2.82,4.47,;-4.15,5.24,;-5.49,4.47,;-5.49,2.93,;-4.15,2.16,;-2.82,2.93,;.05,1.27,;1.52,1.74,;2.42,.5,;1.52,-.75,;1.52,-2.29,;.05,-2.76,;-.85,-1.52,;-2.39,-1.52,;.05,-.27,;3,-2.69,;4.09,-1.6,;5.58,-2,;5.98,-3.48,;4.89,-4.57,;3.4,-4.17,;5.29,-6.06,;4.2,-7.15,;6.78,-6.46,;5.69,-7.55,;6.67,-.91,;8.16,-1.3,;6.27,.58,;7.76,.18,;-6.82,2.16,;-8.16,2.93,;-6.82,.62,;-8.16,1.39,;2.51,4.47,;2.91,2.98,;4.4,3.38,;4,4.87,;5.73,2.61,;7.07,3.38,;5.73,1.07,)|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C#N |r|
COc1ncc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
COc1ncc(Cl)cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
FC(F)(F)c1ccc(-c2cscc2C#N)c(c1)[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
COc1ccc(C)cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
COc1ccc(Cl)cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
FC(F)(F)c1ccc(c(c1)[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)-c1ccccc1Cl |r|
Cc1cocc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
FC(F)(F)c1ccc(C2=CCCCC2)c(c1)[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:8|
FC(F)(F)c1ccc(-c2ccsc2)c(c1)[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
COc1ccc(F)cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
FC(F)(F)c1ccc(-c2cccc(c2)C#N)c(c1)[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
COc1ncccc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
FC(F)(F)c1ccc(C2=CCCC2)c(c1)[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:8|
Fc1ccc(Cl)cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
Cc1cscc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
Fc1ccc(F)c(c1)-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
Cc1ccc(Cl)cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(C)cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(F)cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(C)cc(c1)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cccc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(Cl)cc(Cl)c1)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(Cl)cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1cnc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)C(C)C |r|
COc1ccc(cc1-c1ccc(F)cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1cc(F)c(cc1-c1ccc(F)cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1ccc(cc1-c1ccc(F)cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)-c1cnc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(nc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1cc(F)c(cc1-c1ccc(nc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)C(C)C |r|
COc1cc(F)c(cc1-c1cnc(nc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CCC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1CCC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(CCC(O)=O)cc1-c1ccc(cc1[C@@H]1CCC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
COc1ccc(cc1-c1ccc(nc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r,c:17|
COc1cc(F)c(cc1-c1cnc(nc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)C(C)C |r,c:18|
COc1cc(F)c(cc1-c1cnc(cc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)C(C)C |r,c:18|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r,c:18|
COc1cc(F)c(cc1-c1ccc(cc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r,c:18|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(C)cc(c1)C(F)(F)F)C(F)(F)F)C1CCC(CC1)C(O)=O |r,wU:17.25,18.26,wD:14.15,(-6.51,2,;-5.74,3.33,;-4.2,3.33,;-3.43,4.67,;-1.89,4.67,;-1.12,3.33,;-1.89,2,;-3.43,2,;-4.2,.67,;-5.74,.67,;-6.51,-.67,;-5.74,-2,;-4.2,-2,;-3.43,-.67,;-1.89,-.67,;-.99,.58,;.48,.1,;.48,-1.44,;1.38,-2.68,;.48,-3.93,;-.99,-3.45,;-2.32,-4.22,;-.99,-1.91,;2.72,-1.91,;2.72,-.37,;4.05,.4,;4.05,1.94,;5.38,-.37,;5.38,-1.91,;4.05,-2.68,;6.72,-2.68,;6.72,-4.22,;8.05,-1.91,;8.05,-3.45,;-6.51,-3.33,;-8.05,-3.33,;-5.74,-4.67,;-7.28,-4.67,;.42,3.33,;1.19,2,;2.73,2,;3.5,3.33,;2.73,4.67,;1.19,4.67,;5.04,3.33,;5.81,4.67,;5.81,2,)|
COc1cc(F)c(cc1-c1cnc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(C)cc(c1)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:17.25,18.26,44.52,wD:14.15,41.45,(-4,6.78,;-2.67,7.55,;-1.33,6.78,;,7.55,;1.33,6.78,;1.33,5.24,;,4.47,;-1.33,5.24,;-2.67,4.47,;-4,5.24,;-5.33,4.47,;-5.33,2.93,;-4,2.16,;-2.67,2.93,;-1.33,2.16,;.13,2.64,;1.04,1.39,;.13,.15,;.13,-1.39,;-1.33,-1.87,;-2.24,-.62,;-3.78,-.62,;-1.33,.62,;1.46,-2.16,;2.8,-1.39,;4.13,-2.16,;4.13,-3.7,;2.8,-4.47,;1.46,-3.7,;2.8,-6.01,;1.46,-6.78,;4.13,-6.78,;2.8,-7.55,;5.47,-1.39,;6.8,-2.16,;5.47,.15,;6.8,-.62,;-6.67,2.16,;-8,2.93,;-6.67,.62,;-8,1.39,;2.67,4.47,;2.67,2.93,;4,2.16,;5.33,2.93,;5.33,4.47,;4,5.24,;6.67,2.16,;8,2.93,;6.67,.62,)|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)[C@H]1C[C@H](O)[C@H](O)C1 |r|
COc1cc(F)c(cc1-c1cc(C)c(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cc(C)c(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1c(C)cc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r,wU:18.26,19.27,wD:15.16,(-2.67,8.32,;-2.67,6.78,;-1.33,6.01,;,6.78,;1.33,6.01,;1.33,4.47,;,3.7,;-1.33,4.47,;-2.67,3.7,;-4,4.47,;-4,6.01,;-5.33,3.7,;-5.33,2.16,;-4,1.39,;-2.67,2.16,;-1.33,1.39,;.13,1.87,;1.04,.62,;.13,-.62,;.13,-2.16,;-1.33,-2.64,;-2.24,-1.39,;-3.78,-1.39,;-1.33,-.15,;1.46,-2.93,;2.8,-2.16,;4.13,-2.93,;4.13,-4.47,;2.8,-5.24,;1.46,-4.47,;2.8,-6.78,;1.46,-7.55,;4.13,-7.55,;2.8,-8.32,;5.47,-2.16,;6.8,-2.93,;5.47,-.62,;6.8,-1.39,;-6.67,1.39,;-8,2.16,;-6.67,-.15,;-8,.62,;2.67,3.7,;2.67,2.16,;4,1.39,;5.33,2.16,;5.33,3.7,;4,4.47,;4,6.01,;6.67,1.39,;8,2.16,;6.67,-.15,)|
COc1ncc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(F)cc(c1)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(F)cc(c1)C(F)(F)F)C(F)(F)F)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1c(C)cc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r,wU:18.26,19.27,wD:15.16,(-2.67,8.32,;-2.67,6.78,;-1.33,6.01,;,6.78,;1.33,6.01,;1.33,4.47,;,3.7,;-1.33,4.47,;-2.67,3.7,;-4,4.47,;-4,6.01,;-5.33,3.7,;-5.33,2.16,;-4,1.39,;-2.67,2.16,;-1.33,1.39,;.13,1.87,;1.04,.62,;.13,-.62,;.13,-2.16,;-1.33,-2.64,;-2.24,-1.39,;-3.78,-1.39,;-1.33,-.15,;1.46,-2.93,;2.8,-2.16,;4.13,-2.93,;4.13,-4.47,;2.8,-5.24,;1.46,-4.47,;2.8,-6.78,;1.46,-7.55,;4.13,-7.55,;2.8,-8.32,;5.47,-2.16,;6.8,-2.93,;5.47,-.62,;6.8,-1.39,;-6.67,1.39,;-8,2.16,;-6.67,-.15,;-8,.62,;2.67,3.7,;2.67,2.16,;4,1.39,;5.33,2.16,;5.33,3.7,;4,4.47,;4,6.01,;6.67,1.39,;8,2.16,;6.67,-.15,)|
Cc1cc(ccc1-c1cnc(C)c(c1)-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r,c:17|
COc1ccc(cc1-c1ncc(cc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r,c:17|
COc1ncc(cc1-c1ncc(cc1[C@@H]1C=C[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r,c:17|
COc1ncc(cc1-c1ncc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C1CCC(=O)NC1C |r|
COc1ccc(cc1-c1ncc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ncc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)[C@H]1CNC(=O)OC1(C)C |r|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)[C@H]1OC(=O)N[C@H]1C |r|
COc1ccc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)[C@@H]1CC(=O)N[C@H]1C |r|
COc1ncc(cc1-c1ccc(nc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1[C@@H]1CC[C@H]2[C@H](OC(=O)N12)c1cccc(c1)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
O[C@H](CNCC(Cc1ccccc1)(c1cc(F)cc(OC(F)(F)C(F)F)c1)c1ccc(Cl)cn1)C(F)(F)F |r|
O[C@](C(=O)NCC(Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(F)cn1)(c1ccccc1)C(F)(F)F |r|
O[C@H](CNCC(Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(F)cn1)C(F)(F)F |r|
FC(F)(F)Oc1cccc(c1)C(CNC(=O)C1CC1(F)F)(Cc1ccccc1)c1cccc(OC(F)(F)F)c1
FC(F)(F)CNC(=O)NCC(Cc1ccccc1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
Cc1cc(CC(CNC[C@H](O)C(F)(F)F)(c2cccc(OC(F)(F)F)c2)c2cccc(OC(F)(F)F)c2)no1 |r|
O[C@H](CNCC(Cc1ccccn1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@@H](CN(C[C@H](O)C(F)(F)F)CC(Cc1ccccc1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CNCC(Cc1ccccc1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
Cc1ccc(CC(CNC[C@@H](O)C(F)(F)F)(c2cccc(OC(F)(F)F)c2)c2cccc(OC(F)(F)F)c2)cc1 |r|
FC(F)(F)CCNCC(Cc1ccccc1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
Oc1c(F)cccc1CNCC(Cc1ccccc1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
FC(F)(F)Oc1cccc(c1)C(CNc1ncc(cn1)N1CCOCC1)(Cc1ccccc1)c1cccc(OC(F)(F)F)c1
FC(F)(F)CS(=O)(=O)NCC(Cc1ccccc1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
CC(C)OC(=O)CCNCC(Cc1ccccc1)(c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
O[C@H](CN1[C@@H](CN(Cc2cc(F)cc(c2)C(F)(F)F)c2ccccc12)c1ccccc1)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(Cl)c2)c2ccccc12)c1ccccc1)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cc(Cl)cc(Cl)c2)c2ccccc12)c1ccccc1)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cc(Cl)cc(Cl)c2)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
Cc1ccccc1CN1C[C@H](N(C[C@@H](O)C(F)(F)F)c2ccccc12)c1cccc(c1)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(Cl)c2Cl)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2c(Cl)cccc2Cl)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
Cc1cc(CN2C[C@H](N(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(c2)C(F)(F)F)cc(Cl)n1 |r|
O[C@H](CN1[C@@H](CN(CC2CCCCC2)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2ccsc2)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2ccc(Cl)cc2)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(c2)C(F)(F)F)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cc(F)cc(c2)C(F)(F)F)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CCc1cc(CN2C[C@H](N(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(c2)C(F)(F)F)ccc1Cl |r|
Cc1ccc(cc1CN1C[C@H](N(C[C@@H](O)C(F)(F)F)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
Cc1cccc(CN2C[C@H](N(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(c2)C(F)(F)F)n1 |r|
CC(C)Oc1cccc(CN2C[C@H](N(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(c2)C(F)(F)F)n1 |r|
COc1cccnc1CN1C[C@H](N(C[C@@H](O)C(F)(F)F)c2ccccc12)c1cccc(c1)C(F)(F)F |r|
COc1cccc(CN2C[C@H](N(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(c2)C(F)(F)F)n1 |r|
CCOc1cccc(CN2C[C@H](N(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(c2)C(F)(F)F)n1 |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1ccc(Cl)cc1)C(F)(F)F |r|
COc1cc2ccc(cc2cc1OC)[C@@H]1CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc2N1C[C@@H](O)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1ccc2OCCOc2c1)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1ccc(F)cc1)C(F)(F)F |r|
Cc1ccc(cc1)[C@@H]1CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc2N1C[C@@H](O)C(F)(F)F |r|
COc1ccc(cc1)[C@@H]1CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc2N1C[C@@H](O)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1cccc2ccccc12)C(F)(F)F |r|
O[C@H](CN1C(CN(C2C=Cc3ccccc23)c2ccccc12)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r,c:8|
O[C@H](CN1C(CN(C2CCCc3ccccc23)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1C(CN(Cc2cccc(OC(F)(F)F)c2)c2cc(F)ccc12)c1cccc(OC(F)F)c1)C(F)(F)F |r|
CC(C)(O)c1ccc(cc1)C1CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc2N1C[C@@H](O)C(F)(F)F |r|
O[C@H](CN1C(CN(Cc2cccc(OC(F)F)c2)c2ccccc12)c1cccc(OC(F)F)c1)C(F)(F)F |r|
O[C@H](CN1C(CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1cccc(OC(F)F)c1)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2ccnc(c2)N2CCOCC2)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2ncccc2N2CCOCC2)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(OC(F)F)c2)c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1C(CN(Cc2cccc(OC(F)(F)F)c2)c2ccc(F)c(F)c12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(CC2=CCCCC2)c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r,t:8|
O[C@H](CN1[C@@H](CN(CC2CCOCC2)c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1C(CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1ccc(cc1)-c1ccccc1)C(F)(F)F |r|
O[C@H](CN1C(CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1cccc(c1)-c1ccccc1)C(F)(F)F |r|
CC(C)c1nc2CC3(CC3)C[C@H](O)c2c2c1[C@H](OC21CCOCC1)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2CC3(CC3)C[C@H](O)c2c2c1[C@H](OC21CCOCC1)c1ccc(c(c1)C#N)C(F)(F)F |r|
COc1cc(ccc1C(F)(F)F)[C@H]1OC2(CCOCC2)c2c1c(nc1CC3(CC3)C[C@H](O)c21)C(C)C |r|
CC(C)c1nc2CC3(CC3)C[C@H](O)c2c2c1[C@H](OC21CCOCC1)c1ccc(nc1)C(F)(F)F |r|
CC(C)c1nc2[C@H](O)C3(CC3)C[C@H](O)c2c2c1[C@H](OC21CCOCC1)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2[C@H](O)C3(CC3)C[C@H](O)c2c2c1[C@H](OC21CCOCC1)c1ccc(c(c1)C#N)C(F)(F)F |r|
COc1cc(ccc1C(F)(F)F)[C@H]1OC2(CCOCC2)c2c1c(nc1[C@H](O)C3(CC3)C[C@H](O)c21)C(C)C |r|
CC(C)c1nc2[C@H](O)C3(CC3)C[C@H](O)c2c2c1[C@H](OC21CCOCC1)c1ccc(nc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncccn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(Br)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
COc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(O)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)N1CCOCC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)N1CCCCC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CN1CCN(CC1)c1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)N1CCSCC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)N1CCS(=O)(=O)CC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)N1CCC(O)CC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC(C)c1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CCOc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC(C)Oc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OCCO)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CCCCCc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)C#N)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)C1=CCCCC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r,t:26|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)C1CC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(CO)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC(C)COc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC(C)CCOc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OCCCCC(O)=O)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC(C)Cc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(CCCCC(O)=O)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CCOCc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
COCc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC(C)OCc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC(C)COCc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CNC(=O)c1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CN(C)C(=O)c1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)C(=O)N1CCOCC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(CCCC(F)(F)F)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC(C)\C=C\c1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
Cc1noc(n1)-c1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CN(CCO)Cc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
C[C@H](O)COc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CN1CCC(CC1)Oc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OC[C@@H](O)CO)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OC[C@H](O)CO)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CN1CCC(C1)Oc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
C[C@@H](O)COc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC(C)(O)CCOc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC(C)(O)COc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OCCCS(C)(=O)=O)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OCCCO)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OCCC(F)(F)F)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OC(F)F)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(OCC(CO)CO)cn1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC(CO)(CO)COc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CN(Cc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F)S(C)(=O)=O |r|
CC(C)S(=O)(=O)N(C)Cc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CSc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)S(C)(=O)=O)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)-c1cccc(c1)C(O)=O)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
CN(CCO)c1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCN(CC1)c1ncc(cn1)N1CC[C@H](O)C1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCC(F)(F)CC1 |r|
COc1ncc(Cl)cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)C(C)C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1sc(C)nc1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1cnn(C)c1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)C1CC1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)nn(C)c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)noc1C |r|
COc1ncc(CCC(O)=O)cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)C(F)(F)F |r|
CCOc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)C(F)(F)F |r|
COc1ncc(Cl)cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)C1CC1 |r|
COc1ncc(Cl)cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(F)c1)N1CC(F)C1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(F)c1)N1CC(F)C1)C(C)C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)C(C)C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)C(C)(O)C(F)(F)F |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)n[nH]c1C |r|
CCCn1nc(C)c(c1C)-c1cnc(OC)c(c1)-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1 |r|
CCn1nc(C)c(c1C)-c1cnc(OC)c(c1)-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)nn(C(C)C)c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)nn(CC#N)c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)nn(CC(N)=O)c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)-c1c(C)n[nH]c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(O)C1)-c1c(C)n[nH]c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCCC1)-c1c(C)n[nH]c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1c(C)n[nH]c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCC1)-c1c(C)n[nH]c1C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)C(C)C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1[C@H](C)CC[C@H]1C)C(C)C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCC[C@@H]1C)C(C)C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCC1)C(C)C |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1c(C)cc(cc1C)-c1n[nH]c(=O)o1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1c(C)cc(cc1C)-c1n[nH]c(=O)o1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1ccc(cc1C)C(=O)Nc1nnn[nH]1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1ccc(cc1C)-c1n[nH]c(=O)o1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1ccc(cc1C)-c1n[nH]c(=O)o1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1ccc(cc1C)C(=O)Nc1nnn[nH]1 |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)-n1ccnc1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(F)c1)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cccc(OC(F)(F)F)c1)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(c1)C(F)(F)F)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(c1)C(F)(F)F)N1CC(F)(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(c1)C(F)(F)F)N1CC(F)C1)-c1c(C)cc(cc1C)C(O)=O |r|
C[C@H]1[C@H](OC(=O)N1Cc1nc(ncc1-c1sc(nc1C(C)(C)C)-c1ccc(cc1C)C(O)=O)N1CC(F)(F)C1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
C[C@H]1[C@H](OC(=O)N1Cc1nc(ncc1-c1sc(nc1C(C)(C)C)-c1ccc(cc1C)C(O)=O)N1CC(F)C1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
C[C@H]1[C@H](OC(=O)N1Cc1nc(ncc1-c1sc(nc1C)-c1ccc(cc1C)C(O)=O)N1CC(F)C1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
C[C@H]1[C@H](OC(=O)N1Cc1nc(ncc1-c1sc(nc1C)-c1ccc(cc1C)C(O)=O)N1CC(F)(F)C1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
C[C@H]1[C@H](OC(=O)N1Cc1nc(ncc1-c1sc(nc1C)-c1ccc(cc1C)C(O)=O)N1CCOCC1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
C[C@H]1[C@H](OC(=O)N1Cc1nc(ncc1-c1cc(cnc1C)-c1ccc(cc1C)C(O)=O)N1CC(F)C1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1ccc(cc1C)C(=O)OC(C)(C)C |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)-c1c(C)cc(cc1C)C(=O)OC(C)(C)C |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)-c1c(C)cc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)-c1ccc(cc1C)C(=O)OC(C)(C)C |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1ccc(cc1C)C(=O)OC(C)(C)C |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)(F)C1)-c1c(C)cc(cc1C)C(O)=O |r|
C[C@H]1[C@H](OC(=O)N1Cc1nc(ncc1-c1c(C)noc1C)N1CCC1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,wU:2.28,1.0,(2.48,.16,;1.14,-.61,;.67,-2.07,;-.87,-2.07,;-1.35,-.61,;-2.68,.16,;-.1,.3,;-.1,1.84,;-1.44,2.61,;-2.77,1.84,;-4.1,2.61,;-4.1,4.15,;-2.77,4.92,;-1.44,4.15,;-.1,4.92,;-.1,6.46,;-1.44,7.23,;1.36,6.93,;2.27,5.69,;1.36,4.44,;2.13,3.11,;-5.44,1.84,;-6.91,2.23,;-7.31,.75,;-5.82,.35,;1.76,-3.16,;3.24,-2.76,;4.43,-3.86,;3.93,-5.34,;2.45,-5.74,;1.36,-4.65,;2.05,-7.23,;.56,-7.62,;1.65,-8.71,;3.38,-8,;5.92,-3.48,;7.41,-3.1,;6.3,-4.97,;5.54,-1.99,)|
COc1ccc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C)C(O)=O |r,c:9|
COC(=O)c1ccc(c(C)c1)-c1cnc(OC)c(c1)C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1 |r,c:21|
COc1ncc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C)C(O)=O |r,c:9|
COc1ccc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1F)C(O)=O |r,c:9|
COC(=O)c1cccc(c1)-c1ccc(OC)c(c1)C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1 |r,c:20|
COC(=O)c1ccc(c(C)c1)-c1cc(C2=C(CN3[C@@H](C)[C@H](OC3=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)CC(C)(C)CC2)c(OC)cc1F |r,c:15|
COc1cc(F)c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C)C(O)=O |r,c:10|
COc1cc(F)c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1)C(O)=O |r,c:10|
COc1ncc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C(C)C)C(O)=O |r,c:9|
COc1ncc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1Cl)C(O)=O |r,c:9|
COc1ncc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1F)C(O)=O |r,c:9|
COc1ccc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(C(O)=O)c(F)c1F |r,c:9|
COc1ccc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1c(F)cc(cc1F)C(O)=O |r,c:9|
COc1ncc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(C(O)=O)c(F)c1F |r,c:9|
COc1ccc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1OC)C(O)=O |r,c:9|
COc1cc(c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1)C(O)=O)C(F)(F)F |r,c:9|
COc1cc(c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1F)C(O)=O)C(F)(F)F |r,c:9|
COc1cc(c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(C(O)=O)c(F)c1)C(F)(F)F |r,c:9|
COc1cc(c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1Cl)C(O)=O)C(F)(F)F |r,c:9|
COc1cc(c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C)C(O)=O)C(F)(F)F |r,c:9|
COc1ccc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C(F)(F)F)C(O)=O |r,c:9|
COc1cc(C)c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1)C(O)=O |r,c:10|
COc1cc(F)c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1Cl)C(O)=O |r,c:10|
COc1ccc(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1Cl)C(O)=O |r,c:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(F)cc(c1)-c1ccc(cc1C)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cccc(c1)-c1ccc(cc1C)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
COc1cc(F)c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1F)C(O)=O |r,c:10|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(F)cc(c1)-c1ccc(cc1C(F)(F)F)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1ccc(C)c(c1)-c1ccc(cc1C)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1ccc(F)c(c1)-c1ccc(cc1C)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
COc1cc(C)c(cc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C)C(O)=O |r,c:10|
COc1cc(cc(c1)-c1ccc(cc1C)C(O)=O)C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1 |r,c:20|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(ccc1F)-c1ccc(cc1C(F)(F)F)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1ccc(F)c(c1)-c1ccc(cc1C(F)(F)F)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(ccc1Cl)-c1ccc(cc1C)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(ccc1Cl)-c1ccc(cc1C(F)(F)F)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(ccc1F)-c1ccc(cc1Cl)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(cc(c1)C(F)(F)F)-c1ccc(cc1F)C(O)=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
CCNC(=O)c1ccc(-c2ccc(F)c(c2)C2=C(CN3[C@@H](C)[C@H](OC3=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)CC(C)(C)CC2)c(c1)C(F)(F)F |r,c:17|
C[C@H]1[C@H](OC(=O)N1CC1=C(CCC(C)(C)C1)c1cc(ccc1F)-c1ccc(cc1C(F)(F)F)C(=O)N1CCOCC1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r,t:9|
COc1ccc(nc1C1=C(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(C)(C)CC1)-c1ccc(cc1C(F)(F)F)C(O)=O |r,c:9|
CC[C@H]1C[C@H](C[C@@H](CC)N1C(=O)OC(C)(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)OC |r|
CC[C@@H]1C[C@@H](C[C@H](Cc2ccccc2)N1C(=O)OC(C)(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)N1CCOCC1 |r|
CC[C@@H]1C[C@@H](C[C@H](Cc2ccccc2)N1C(=O)OC(C)(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(Br)cn1 |r|
CC[C@@H]1C[C@@H](C[C@H](Cc2ccccc2)N1C(=O)OC(C)(C)C)N(Cc1cc(Cl)cc(c1)C(F)(F)F)c1ncc(Br)cn1 |r|
CCNC(=O)N1[C@H](CC)C[C@@H](C[C@@H]1Cc1ccccc1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(Br)cn1 |r|
CCCC(=O)N1[C@H](CC)C[C@@H](C[C@@H]1Cc1ccccc1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(Br)cn1 |r|
CC[C@@H]1C[C@@H](C[C@H](Cc2ccccc2)N1C(=O)OC(C)(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(OC)cn1 |r|
CC[C@H]1C[C@H](C[C@@H](CC)N1C(=O)O[C@H]1CC[C@@H](CC1)C(O)=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)N1CCOCC1 |r,wU:4.23,6.6,2.1,13.13,wD:16.20,(20.99,-12.46,;22.31,-13.23,;23.65,-12.46,;23.65,-10.92,;24.98,-10.15,;26.31,-10.92,;26.31,-12.46,;27.64,-13.23,;28.98,-12.46,;24.98,-13.22,;24.98,-14.76,;23.64,-15.53,;26.31,-15.53,;26.31,-17.07,;27.65,-17.84,;27.64,-19.38,;26.3,-20.15,;24.97,-19.37,;24.97,-17.84,;26.3,-21.69,;24.96,-22.46,;27.63,-22.46,;24.98,-8.61,;23.64,-7.83,;23.64,-6.29,;24.98,-5.53,;24.99,-3.99,;23.65,-3.22,;22.31,-4,;22.32,-5.54,;20.98,-3.23,;20.98,-1.69,;19.65,-4.01,;19.64,-2.46,;26.32,-3.22,;27.65,-3.99,;26.32,-1.68,;27.65,-2.45,;26.31,-7.84,;27.65,-8.61,;28.98,-7.84,;28.98,-6.3,;27.64,-5.53,;26.31,-6.3,;30.31,-5.53,;31.63,-6.3,;32.96,-5.54,;32.97,-4,;31.63,-3.22,;30.3,-3.99,)|
CC[C@H]1C[C@H](C[C@@H](CC)N1C(=O)O[C@H]1CC[C@@H](CC1)C(O)=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)-c1cnn(C)c1 |r,wU:4.23,6.6,2.1,13.13,wD:16.20,(37.57,-12.9,;38.91,-13.68,;40.24,-12.9,;40.24,-11.36,;41.57,-10.59,;42.9,-11.36,;42.9,-12.9,;44.24,-13.68,;45.57,-12.9,;41.57,-13.67,;41.57,-15.21,;40.24,-15.97,;42.91,-15.97,;42.91,-17.51,;44.24,-18.28,;44.23,-19.82,;42.89,-20.59,;41.56,-19.82,;41.57,-18.28,;42.89,-22.13,;41.55,-22.9,;44.22,-22.91,;41.57,-9.05,;40.24,-8.27,;40.24,-6.73,;41.58,-5.97,;41.58,-4.43,;40.24,-3.66,;38.9,-4.44,;38.91,-5.98,;37.57,-3.67,;37.56,-2.13,;36.23,-4.45,;36.23,-2.9,;42.91,-3.66,;44.25,-4.44,;42.91,-2.12,;44.24,-2.89,;42.9,-8.28,;44.24,-9.05,;45.57,-8.28,;45.57,-6.74,;44.23,-5.97,;42.9,-6.74,;46.9,-5.97,;48.3,-6.59,;49.34,-5.45,;48.56,-4.11,;49.19,-2.71,;47.05,-4.44,)|
CC[C@@H]1C[C@@H](c2cc(ccc2N1C(=O)OCC)C(F)(F)F)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)OC
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
Cc1cc(C)c2N(C[C@H]3CC[C@@H](CC3)C(O)=O)CCC[C@H](N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)c3nnn(C)n3)c2c1 |r,wU:20.21,11.14,wD:8.7,(-5.45,-18.22,;-4.12,-17.45,;-2.78,-18.22,;-1.45,-17.44,;-.11,-18.2,;-1.45,-15.91,;-.01,-15.34,;1.12,-16.38,;2.59,-15.92,;3.91,-16.71,;5.25,-15.96,;5.27,-14.42,;3.95,-13.63,;2.6,-14.38,;6.62,-13.68,;7.94,-14.47,;6.65,-12.14,;.44,-13.86,;-.45,-12.58,;-1.99,-12.47,;-3.03,-13.61,;-4.36,-12.84,;-4.37,-11.31,;-5.7,-10.54,;-5.7,-8.99,;-7.04,-8.22,;-8.37,-8.99,;-8.37,-10.54,;-7.04,-11.31,;-9.7,-11.31,;-11.04,-10.54,;-9.7,-12.85,;-11.05,-12.07,;-7.04,-6.69,;-5.71,-5.91,;-8.38,-5.92,;-7.06,-5.14,;-5.69,-13.62,;-7.1,-12.98,;-8.13,-14.13,;-7.35,-15.46,;-7.98,-16.87,;-5.85,-15.14,;-2.79,-15.14,;-4.12,-15.91,)|
CC[C@@H]1C[C@@H](C[C@H](Cc2ccccc2)N1C(=O)OC(C)(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)OC |r|
CC[C@@H]1C[C@@H](C[C@H](Cc2ccccc2)N1C(=O)OC(C)(C)C)N(Cc1cc(OC)cc(c1)C(F)(F)F)c1ncc(Br)cn1 |r|
CC[C@@H]1C[C@@H](C[C@H](Cc2ccccc2)N1C(=O)OC(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(Br)cn1 |r|
CC[C@H]1C[C@H](C[C@@H](CC)N1C(=O)OC(C)C)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ncc(cn1)N1CCOCC1 |r|
CCC(CC)CC1(CCCCC1)C(=O)Nc1ccccc1SC(=O)C(C)C
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCCCC(O)=O)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O |r,t:15|
[H][C@@]12CC[C@]3(C)[C@]([H])(CCC4=C5CC(C)(C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)CCCC(O)=O)C2(C)C |r,c:10|
C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)O)C)C)[C@@H]2[C@H]1C)C)C(=O)O
CC1(C)CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CC[C@H](OC(=O)c6ccccc6C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2C1)C(O)=O |r,c:10|
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCC(=O)NCCS(O)(=O)=O)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O |r,t:15|
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCN4CCOCC4)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O |r,t:15|
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCCC(O)=O)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O |r,t:15|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)CCCC(O)=O)C2(C)C |r,t:9|
[H][C@]12[C@@H](CC[C@@]1(CC[C@]1(C)[C@]2([H])CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCCC(O)=O)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O)C(C)=C |r|
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCCC(O)=O)C(C)(C)[C@]3([H])CC[C@@]12C)C(=O)OCC(O)=O |r,t:15|
CC1(C)CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CC[C@H](OC(=O)CCC(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2C1)C(O)=O |r,c:10|
CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CS)C(N)=O
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(cc1)N(Cc1cccc(c1)[N+]([O-])=O)Cc1cccc(c1)[N+]([O-])=O
Cc1ccc(cc1)S(=O)(=O)N(c1ccc(OCc2cccc(c2)C(F)(F)F)cc1)S(=O)(=O)c1ccc(C)cc1
Cc1ccc(cc1)S(=O)(=O)N(c1ccc(OCc2cccc(C)c2)cc1)S(=O)(=O)c1ccc(C)cc1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(cc1)N(Cc1cccc(Cl)c1)Cc1cccc(Cl)c1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(NCc2cccc(C)c2)cc1
COc1cccc(COc2ccc(cc2)N(S(=O)(=O)c2ccc(C)cc2)S(=O)(=O)c2ccc(C)cc2)c1
Cc1ccc(cc1)S(=O)(=O)N(c1ccc(OCc2cccc(Cl)c2)cc1)S(=O)(=O)c1ccc(C)cc1
Cc1ccc(cc1)S(=O)(=O)N(c1ccc(OCc2ccc(Cl)cc2)cc1)S(=O)(=O)c1ccc(C)cc1
CCc1cccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
COc1cccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
CCCOc1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1
CC(C)c1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1C
Cc1cc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)ccc1Cl
CC(C)c1cccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(Cl)cc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(F)c2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cc(F)cc(F)c2)c1)C(F)(F)F
CCCc1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(cc2)[N+]([O-])=O)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(Cc3ccccc3)cc2)c1)C(F)(F)F
Nc1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(cc2)C(F)(F)F)c1)C(F)(F)F
Cc1cccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
Cc1cc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)ccc1F
Cc1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1C
CCc1cc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)ccc1Cl
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(F)cc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(OC(F)(F)F)c2)c1)C(F)(F)F
Cc1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1
CCc1cc(C)cc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(Cl)c2Cl)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(F)c2[N+]([O-])=O)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(OC(F)(F)F)cc2)c1)C(F)(F)F
CN(C)c1cccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc3CCCCc3c2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccccc2Cl)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(cc2)-c2ccccc2)c1)C(F)(F)F
CC(C)(C)c1cccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
CCCCC(C)C1CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)O1
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC(=O)C(N)C(O)(C(F)(F)F)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
NC(C(=O)N[C@@](Cc1ccccc1)(c1cc(F)cc(OC(F)(F)C(F)F)c1)c1ccc(Cl)cn1)C(O)(C(F)(F)F)C(F)(F)F |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC(=O)C(N)C(O)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
OC(C(=O)N[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1)C(O)(C(F)(F)F)C(F)(F)F |r|
NC(C(=O)N[C@](Cc1ccccc1)(c1ccc(F)cc1)c1cc(F)cc(c1)C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F |r|
CC(C)NC(C(=O)N[C@](Cc1ccccc1)(c1ccc(F)cc1)c1cc(F)cc(c1)C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC(=O)C(O)C(O)(C(F)(F)F)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NCC(O)C(O)(C(F)(F)F)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
CC(C)(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC(=O)C(N)C(O)(C(F)(F)F)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
CN(C)C(C(=O)N[C@](Cc1ccccc1)(c1ccc(F)cc1)c1cc(F)cc(c1)C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NCC(N)C(O)(C(F)(F)F)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
NC(C(=O)N[C@](Cc1ccccc1)(c1ccc(F)c(OC2CC2)c1)c1cc(F)cc(OC(F)(F)C(F)F)c1)C(O)(C(F)(F)F)C(F)(F)F |r|
OC(CC(=O)N[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1)(C(F)(F)F)C(F)(F)F |r|
CNC(C(=O)N[C@](Cc1ccccc1)(c1ccc(F)cc1)c1cc(F)cc(c1)C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)c1ccccc1C(O)=O)C2(C)C |r,t:9|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)c1cccc(c1)C(O)=O)C2(C)C |r,t:9|
C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CC[C@H](OC(=O)CCC(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2[C@H]1C)C(O)=O |r,c:9|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)C1CC1C(O)=O)C2(C)C |r,t:9|
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(F)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)C(F)(F)F)c1cccc(F)c1)C(F)(F)F
O[C@@H](CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1ccc(Oc2ccccc2)cc1)C(F)(F)F
O[C@H](CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1ccc(OC(F)(F)F)cc1)c1cccc(F)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)C(F)(F)F)c1ccccc1)C(F)(F)F
OC(CN(Cc1ccc(OC(F)(F)F)cc1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1ccccc1C(F)(F)F)c1cccc(F)c1)C(F)(F)F
OC(CN(Cc1ccccc1)c1cccc(F)c1)C(F)(F)F
COc1cc(cc(OC)c1OC)N(C[C@@H](O)C(F)(F)F)Cc1cccc(SC(F)(F)F)c1
Cc1cccc(CN(CC(O)C(F)(F)F)c2cccc(F)c2)c1
OC(CN(Cc1ccc(F)c(c1)-c1ccco1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1ccccc1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1ccco1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1cccs1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1ccoc1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1ncccn1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1cccnc1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
CCOc1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
Cc1cccnc1-c1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
OC(CN(Cc1ccc(N2CCOCC2)c(c1)-c1ccco1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1ncccc1C(F)(F)F)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)-c1ccncc1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
Cn1cccc1-c1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
Cc1ccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)cc1-c1ccco1
OC(CN(Cc1cccc(c1)-c1ccccn1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](NC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1ncc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](NC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](NC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](NC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](NC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](N(C)C1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(cnc1OC)-c1ccc(cc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N(C)[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(cnc1OC)-c1ccc(cc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(cnc1OC)-c1c(C)cc(cc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(cnc1OC)-c1c(C)cc(cc1C)C(=O)NC1(CC1)C#N)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(ccc1OC)-c1ccc(cc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N(C)[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(ccc1OC)-c1ccc(cc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(CCC(O)=O)ccc1OC)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(ccc1OC)[C@H]1CC[C@@H](CC1)C(O)=O)C(F)(F)F |r,wU:9.11,41.49,wD:4.26,1.0,38.42,(47.22,-12.06,;46.14,-10.97,;47.47,-10.2,;47.16,-8.69,;45.63,-8.53,;44.99,-9.94,;43.67,-10.71,;42.26,-10.08,;43.99,-12.21,;45.51,-12.37,;46.28,-13.7,;45.51,-15.03,;46.27,-16.37,;47.82,-16.37,;48.59,-15.03,;47.81,-13.7,;50.13,-15.02,;50.52,-13.52,;51.62,-14.61,;50.9,-16.36,;45.5,-17.7,;46.59,-18.79,;45.1,-19.19,;43.96,-17.7,;44.85,-7.19,;43.32,-7.18,;42.57,-5.85,;43.33,-4.53,;44.85,-4.53,;45.62,-5.87,;47.17,-5.87,;47.93,-7.21,;49.47,-7.21,;50.25,-5.87,;49.47,-4.53,;47.93,-4.53,;47.16,-3.2,;47.92,-1.86,;50.24,-8.54,;49.45,-9.87,;50.21,-11.2,;51.75,-11.21,;52.53,-9.88,;51.76,-8.54,;52.51,-12.54,;54.05,-12.55,;51.74,-13.87,;41.02,-5.84,;41.02,-7.38,;39.68,-6.6,;40.25,-4.51,)|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(ccc1OC)-c1cccnc1C)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(ccc1OC)-c1ccc(nc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ncc1-c1cc(ccc1OC)-c1ccc(cc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1S(=O)(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(ccc1OC)-c1ccc(cc1C)C(O)=O)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1S(=O)(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1S(=O)(=O)N[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(ccc1OC)[C@H]1CC[C@@H](CC1)C(O)=O)C(F)(F)F |r,wU:10.12,42.50,wD:39.43,1.0,4.27,(14.26,-14.43,;13.17,-13.34,;14.51,-12.58,;14.2,-11.07,;12.66,-10.9,;12.03,-12.32,;10.7,-13.08,;9.18,-13.07,;9.95,-11.75,;11.03,-14.58,;12.55,-14.74,;13.32,-16.07,;14.85,-16.07,;15.63,-17.4,;14.85,-18.74,;13.31,-18.74,;12.54,-17.4,;12.54,-20.08,;12.13,-21.57,;11,-20.07,;13.62,-21.16,;17.17,-17.39,;17.56,-15.89,;18.66,-16.99,;17.94,-18.73,;11.89,-9.56,;10.36,-9.56,;9.6,-8.23,;10.36,-6.91,;11.89,-6.9,;12.66,-8.24,;14.2,-8.24,;14.97,-9.58,;16.51,-9.58,;17.28,-8.25,;16.5,-6.9,;14.97,-6.91,;14.2,-5.57,;14.96,-4.23,;17.27,-10.91,;16.49,-12.25,;17.25,-13.58,;18.79,-13.59,;19.57,-12.26,;18.8,-10.92,;19.55,-14.91,;21.07,-14.92,;18.78,-16.23,;8.06,-8.21,;6.72,-8.97,;7.29,-6.88,;8.05,-9.76,)|
OC(CN(Cc1cccc(c1)C(F)(F)F)c1cccc(Cl)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F
OC(CN(Cc1cccc(OCC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
CCCC(O)CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1
CC(=O)OC(CN(Cc1cccc(c1)C(F)(F)F)c1cccc(F)c1)C(F)(F)F
FC(F)C(F)(F)Oc1cccc(CN2CC(Oc3ccc(F)cc23)C(F)(F)F)c1
OC(CN(Cc1cccc(c1)C1CCCC1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)C(O)(C(F)(F)F)C(F)(F)F)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1)C=C
CC(C)(O)c1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
Cc1ccc(CN(CC(O)C(F)(F)F)c2cccc(F)c2)cc1
COc1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1)c1ccc(cc1)C(F)(F)F
OC(CN(Cc1cccc(SC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
CC(C)Oc1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
OC(CN(Cc1cccc(c1)C1CC1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1ccc(cc1)-c1ccccc1)c1cccc(F)c1)C(F)(F)F
OC(CN(Cc1cccc(c1)C(F)(F)F)c1cccc(c1)C(F)(F)F)C(F)(F)F
Cc1ccccc1N(CC(O)C(F)(F)F)Cc1cccc(c1)C(F)(F)F
OC(CN(Cc1cccc(Oc2ccccc2)c1)Cc1cccc(OC(F)(F)F)c1)C(F)(F)F
CC(C)(C)Oc1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
Cc1ccccc1CN(CC(O)C(F)(F)F)c1cccc(F)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(F)c1)C(F)(F)F
OC(COc1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1)C(F)(F)F
CC(C)Cc1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1)Cc1ccccc1
OC(CN(Cc1cccc(OC(F)(F)F)c1)Cc1cccc(OC(F)(F)F)c1)C(F)(F)F
OC(CN(Cc1cccc(Oc2ccccc2)c1)c1cccc(F)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1)c1ccccc1
OC(CN(Cc1cccc(Oc2ccccc2)c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
Cc1ccc(cc1)N(CC(O)C(F)(F)F)Cc1cccc(c1)C(F)(F)F
OC(CN(Cc1ccc2OC(F)(F)C(F)(F)Oc2c1)c1cccc(Oc2ccccc2)c1)C(F)(F)F
OC(CN(Cc1cccc(Oc2cccc(c2)C(F)(F)F)c1)c1cccc(F)c1)C(F)(F)F
Cc1cccc(c1)N(CC(O)C(F)(F)F)Cc1cccc(c1)C(F)(F)F
COC(=O)c1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1
Cc1ccc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1
CCc1cc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)ccc1Cl
CC(C)c1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1
Cc1cc(C)cc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OCc2cccc(c2)C(F)(F)F)c1)C(F)(F)F
CCc1cccc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OCc2ccccc2)c1)C(F)(F)F
CCc1cc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2cccc(c2)C(F)(F)C(F)(F)F)ccc1Cl
CCc1cc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2cc(ccc2F)C(F)(F)F)ccc1Cl
O[C@H](CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(OC(F)(F)F)c2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(S)cc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OC2CCCC2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(F)c2F)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(Cl)c(Cl)c2)c1)C(F)(F)F
CCc1cc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2cccc(OC(F)(F)F)c2)ccc1Cl
CCc1cc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2ccc(cc2F)C(F)(F)F)ccc1Cl
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OCc2ccc(OC(F)(F)F)cc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccccn2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccnc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(c2)C(F)(F)F)c1)C(F)(F)F
CC(C)c1cccc(Oc2cccc(c2)N(C[C@@H](O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(O)cc2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OC2CCCCC2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OCC2CCCCC2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OCc2cccc(OC(F)(F)F)c2)c1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccccc2[N+]([O-])=O)c1)C(F)(F)F
CC(C)Oc1cccc(c1)N(CC(O)C(F)(F)F)Cc1cccc(OC(F)(F)C(F)F)c1
CC(C)CCC1(CCCCC1)C(=O)Nc1cc(Cl)ccc1SC(=O)C(C)(C)C
COc1ccc(SC(=O)C(C)(C)C)c(NC(=O)C2(CCC(C)C)CCCCC2)c1
CC(C)CCC1(CCCCC1)C(=O)Nc1cc(C)ccc1SC(=O)C(C)(C)C
CC(C)(C)C(=O)Sc1ccccc1NC(=O)C1(C)CCCCC1
COc1ccc(SC(=O)C(C)(C)C)c(NC(=O)C2(C)CCCCC2)c1
CC(C)(C)C(=O)Sc1ccc(Cl)cc1NC(=O)C1(C)CCCCC1
CC(C)CCC1(CCCCC1)C(=O)Nc1ccccc1SC(=O)C(C)(C)C
CC(C)(C)C(=O)Sc1cc(F)ccc1NC(=O)C1(C)CCCCC1
CC(C)(C)C(=O)Sc1ccc(cc1NC(=O)C1(C)CCCCC1)C(F)(F)F
CC(C)CCC1(CCCCC1)C(=O)Nc1cc(F)ccc1SC(=O)C(C)(C)C
CC(C)CCC1(CCCCC1)C(=O)Nc1cc(ccc1SC(=O)C(C)(C)C)C(F)(F)F
CC(C)CCC1(CCCCC1)C(=O)Nc1cc(Cl)c(Cl)cc1SC(=O)C(C)(C)C
CC(C)(C)C(=O)Sc1cc(F)cc(F)c1NC(=O)C1(C)CCCCC1
CC(C)(C)C(=O)Sc1c(F)cccc1NC(=O)C1(C)CCCCC1
CC(C)(C)C(=O)Sc1ccc(cc1NC(=O)C1(C)CCCCC1)C#N
CC(C)CCC1(CCCCC1)C(=O)Nc1cc(ccc1SC(=O)C(C)(C)C)C#N
CC(C)(C)C(=O)Sc1ccc(F)cc1NC(=O)C1(C)CCCCC1
CC(C)CCC1(CCCCC1)C(=O)Nc1ccc(Cl)cc1SC(=O)C(C)(C)C
C[C@H]1[C@H](OC(=O)N1Cc1cc(ccc1-c1cc(ccc1Cl)-c1ccc(cc1C)C(O)=O)C(F)(F)F)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
COc1ccc(cc1-c1cnc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1ccc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cc(c(OC)nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCC1)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CC(F)C1)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCCC1)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N1CCOCC1)-c1ccc(cc1C)C(O)=O |r|
COc1ncc(c(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)n1)-c1cc(ccc1OC)-c1ccc(cc1C)C(O)=O |r|
CCc1ncc(c(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)n1)-c1cc(ccc1OC)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cccc(c1)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cccc(OC(F)(F)F)c1)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1ccc(OC(F)(F)F)cc1)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cccc(Cl)c1)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(Cl)cc(c1)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(c1)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(Cl)cc(Cl)c1)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cc(F)cc(F)c1)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cncc(c1)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1ccnc(c1)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
COc1ccc(cc1-c1cnc(nc1CN1[C@@H](C)[C@H](OC1=O)c1cccc(n1)C(F)(F)F)N(C)C)-c1ccc(cc1C)C(O)=O |r|
[H][C@@]12CC[C@H](N1C(=O)O[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1nc(Cl)ccc1-c1cc(C(C)C)c(F)cc1OC |r|
[H][C@@]12CC[C@H](N1C(=O)S[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)C[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F |r|
[H][C@@]12CC[C@H](N1C(=O)N(C)[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F |r|
[H][C@@]12CC[C@H](C1C(=O)O[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F |r|
[H][C@@]12CC[C@H](C1=NO[C@@H]2c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F |r,c:6|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1)C(O)=O |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccccc1C(O)=O |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccccc1C |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccccc1F |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccccc1 |r|
CC(C)c1cc(c(Cl)cc1F)-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)-c1ccc(cc1C)C(O)=O |r|
COc1c(ccc2Oc3c(OC(=O)N4CC5CCC5C4)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OC(=O)C4(C)C5CCC4CC5)c(C)c(C)c(Cl)c3OC(=O)c12)[C@@H](O)CC(C)(C)C |TLB:11:13:19.20:16.17,THB:14:13:19.20:16.17|
COc1c(ccc2Oc3c(O)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OC(=O)N4CCCC4)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OC(=O)C4(C)C5CCC4CC5)c(Br)c(C)c(Cl)c3OC(=O)c12)[C@@H](O)CC(C)(C)C |TLB:14:13:16.17:20.19,THB:11:13:16.17:20.19|
CCN(CC)C(=O)Oc1cc(C)cc2OC(=O)c3c(Oc12)ccc([C@@H](O)CC(C)C)c3OC
COc1c(ccc2Oc3c(OCCC(C)C)cc(C)cc3OC(=O)c12)C(O)CC(C)C
COc1c(ccc2Oc3c(OC(=O)C4CC5CC4C=C5)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C |c:19,TLB:11:13:18.19:16|
COc1c(ccc2Oc3c(OC(=O)[N+]45CCC(CC4)C5)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OCCC(C)C)cc(C)cc3OC(=O)c12)C(O)CC1CCCCC1
CCc1c(C)c(Cl)c2OC(=O)c3c(Oc2c1OC(=O)C1(C)C2CCC1CC2)ccc([C@@H](O)CC(C)(C)C)c3OC |TLB:17:19:25.26:22.23,THB:20:19:25.26:22.23|
COc1c(ccc2Oc3c(OC(=O)C4CCCC4)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OCCC(C)C)cc(C)cc3OC(=O)c12)C(O)CC1CC1
COc1c(ccc2Oc3c(OS(=O)(=O)c4c(F)cc(F)cc4F)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OCc4ccccc4)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OCCC(C)C)cc(C)cc3OC(=O)c12)C(O)C(C)C
COc1c(ccc2Oc3c(OC(=O)C(C)(C)C)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OS(=O)(=O)C(F)(F)F)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OC(=O)C4(C)C5CCC4CC5)c(Br)c(C)c(Cl)c3OC(=O)c12)[C@@H](O)CC(C)C |TLB:11:13:19.20:16.17,THB:14:13:19.20:16.17|
CCCCCS(=O)(=O)Oc1cc(C)cc2OC(=O)c3c(Oc12)ccc([C@@H](O)CC(C)C)c3OC
COc1c(ccc2Oc3c(OCCC(C)C)cc(C)cc3OC(=O)c12)C(O)CC(C)(C)C
COc1c(ccc2Oc3c(OCC4CCCC4)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OCCC(C)C)cc(C)cc3OC(=O)c12)C(O)CCC(C)C
COc1c(ccc2Oc3c(OC(=O)C4(C)CC5CC4C=C5)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C |c:20,TLB:11:13:19.20:17,THB:14:13:19.20:17|
COc1c(ccc2Oc3c(OS(=O)(=O)C(C)C)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
COc1c(ccc2Oc3c(OC(=O)C4(C)C5CCC4CC5)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C |TLB:11:13:16.17:20.19,THB:14:13:16.17:20.19|
COc1c(ccc2Oc3c(OC(=O)C4(C)C5CCC4CC5)c(C)c(C)c(Cl)c3OC(=O)c12)[C@@H](O)CC(C)C |TLB:11:13:16.17:20.19,THB:14:13:16.17:20.19|
COc1c(ccc2Oc3c(OC(=O)N(C(C)C)C(C)C)cc(C)cc3OC(=O)c12)[C@@H](O)CC(C)C
CCOC(=O)N1C(CC)CN(C(c2nnn(CC(N)=O)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(c2nnn(CC3CC3)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(C(=O)OC)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ccccc12 |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)OC)c2ccccc12 |w:6.6,11.11|
CCOC(=O)N1C(CC)CN(C(c2nnn(CCO)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCOC(=O)N1[C@H](CC)CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1C(=O)OCc1ccccc1)C(F)(F)F |w:5.4,2.1|
CCOC(=O)N1C(CC)CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(C(=O)OC)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(Cc2ccccc2)C(=O)OC)c2ccccc12 |w:6.6,11.11|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1CC1CCCCC1)C(F)(F)F |w:5.4,2.1|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1C(=O)N1CCCC1)C(F)(F)F |w:5.4,2.1|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1C[C@H]1CC[C@H](CC(O)=O)CC1)C(F)(F)F |w:5.4,2.1,wU:37.41,wD:34.37,(15.92,-9.74,;14.58,-10.51,;13.24,-9.74,;13.23,-8.21,;11.9,-7.44,;11.89,-5.9,;10.55,-5.13,;9.14,-5.76,;8.11,-4.61,;8.87,-3.27,;8.24,-1.87,;10.38,-3.59,;13.22,-5.12,;14.54,-5.9,;15.83,-5.14,;15.83,-3.65,;14.51,-2.88,;13.21,-3.64,;14.5,-1.31,;14.5,.24,;12.91,-1.32,;16,-1.3,;17.21,-5.93,;18.55,-6.7,;18,-4.55,;16.47,-7.23,;10.57,-8.22,;9.23,-7.45,;7.9,-8.23,;7.91,-9.77,;9.23,-10.53,;10.56,-9.76,;11.91,-10.52,;11.92,-12.07,;10.58,-12.84,;9.24,-12.08,;7.92,-12.85,;7.93,-14.38,;6.58,-15.17,;5.24,-14.4,;5.23,-12.84,;3.91,-15.17,;9.26,-15.15,;10.58,-14.38,;6.56,-7.47,;5.22,-6.7,;7.32,-6.13,;5.79,-8.81,)|
CCNC(=O)N1C(CC)CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(c2nnn(CCC(=O)OC)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1C(=O)N1CCOCC1)C(F)(F)F |w:5.4,2.1|
CCOC(=O)N1C(CC)CN(C(C(=O)OC)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(Br)ccc12 |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(C(=O)OC)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(Cl)c(Cl)cc12 |w:11.10,6.6|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1C(=O)NCCO)C(F)(F)F |w:5.4,2.1|
CCOC(=O)N1C(CC)CN(C(c2nnn(CCN(C)C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCCCC(CC)COC(=O)N1C(CC)CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:17.16,12.12,4.6|
CCCCOC(=O)N1C(CC)CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:13.12,8.8|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1C(=O)N(C)C)C(F)(F)F |w:5.4,2.1|
CCOC(=O)N1C(CC)CN(C(c2nnn(CC(=O)OC)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1C(=O)OCC(C)C)C(F)(F)F |w:5.4,2.1|
CCOC(=O)N1C(CC)CN(C(c2nnn(CCC#N)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCC1CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc2N1CC1CCCC1)C(F)(F)F |w:5.4,2.1|
CCOC(=O)N1[C@@H](CC)CN(C(c2nnn(C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10|
CCOC(=O)N1C(CC)CN(C(c2nnn(CC(=O)OC(C)(C)C)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
CCOC(=O)N1C(CC)CN(C(c2nnn(CC(O)=O)n2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(ccc12)C(F)(F)F |w:11.10,6.6|
Cc1cc(C)cc(Oc2cccc(CN(CC(O)C(F)(F)F)c3cccc(Oc4ccccc4)c3)c2)c1 |w:16.16|
OC(CN(Cc1cccc2OC(F)(F)C(F)(F)Oc12)c1cccc(Oc2ccccc2)c1)C(F)(F)F |w:1.0|
OC(CN(Cc1ccc(N2CCCCO2)c(c1)-c1ccco1)c1cccc(Oc2ccccc2)c1)C(F)(F)F |w:1.0|
CC(C)(O)c1cccc(c1)N(CC(O)C(F)(F)F)Cc1cccc(OC(F)(F)C(F)F)c1 |w:12.13|
CCCCC(O)CN(Cc1cccc(OC(F)(F)F)c1)c1cccc(Oc2ccccc2)c1 |w:4.4|
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OCc2ccccc2CC(F)(F)F)c1)C(F)(F)F |w:1.0|
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2ccc(F)c(F)c2)c1)C(F)(F)F |w:1.0|
CCCCc1ccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OC(F)(F)C(F)F)c2)cc1 |w:17.18|
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(OCc2ccccc2OC(F)(F)F)c1)C(F)(F)F |w:1.0|
OC(CN(Cc1cccc(c1)-c1cccc(n1)C(F)(F)F)c1cccc(Oc2ccccc2)c1)C(F)(F)F |w:1.0|
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(c1)-c1ccncc1)C(F)(F)F |w:1.0|
OC(CN(Cc1cccc(c1)-c1ccncn1)c1cccc(Oc2ccccc2)c1)C(F)(F)F |w:1.0|
Cc1cccc(n1)-c1cccc(CN(CC(O)C(F)(F)F)c2cccc(Oc3ccccc3)c2)c1 |w:15.16|
OC(CN(Cc1cccc(OC(F)(F)C(F)F)c1)c1cccc(Oc2cccc(CC(F)(F)F)c2)c1)C(F)(F)F |w:1.0|
CCc1cc(Oc2cccc3N(CC(O)C(F)(F)F)C(CCc23)c2cccc(OC(F)(F)C(F)F)c2)ccc1Cl
OC(CN1C(CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
O[C@@H](CN1[C@H](CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
OC(CN1C(CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(c1)C(F)(F)F)C(F)(F)F
OC(CN1C(CCc2c1cccc2-c1cccc(Cl)c1Cl)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
OC(CN1C(CCc2c1cccc2-c1cccc(Cl)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
OC(CN1C(CCc2c1cccc2-c1cccc(F)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
OC(CN1C(CCc2c1cccc2-c1cccc(c1)C(F)(F)F)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
COc1cccc(c1)-c1cccc2N(CC(O)C(F)(F)F)C(CCc12)c1cccc(OC(F)(F)C(F)F)c1
OC(CN1C(CCc2c1cccc2-c1cccc(c1)C#N)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
OC(CN1C(CCc2c1cccc2-c1ccc(OC(F)(F)F)cc1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
OC(CN1C(CCc2c1cccc2-c1cccnc1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
OC(CN1C(CCc2c1cccc2-c1cccs1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
CC(C)c1cccc(c1)-c1cccc2N(CC(O)C(F)(F)F)C(CCc12)c1cccc(OC(F)(F)C(F)F)c1
CC(C)Oc1cccc(c1)-c1cccc2N(CC(O)C(F)(F)F)C(CCc12)c1cccc(OC(F)(F)C(F)F)c1
OC(CN1C(CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F
OC(CF)CN1C(CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
OC(CCl)CN1C(CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
CC(C)C(O)CN1C(CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1
C[C@@H](O)CN1[C@H](CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1 |r|
O[C@@H](CN1[C@H](CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1[C@H](CCc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
COc1ccc(O)c(O)c1C1c2ccccc2CCc2ccccc12
COc1ccc(O)c(O)c1Cc1ccc2CCCCc2c1
COc1ccc(O)c(O)c1\C=C1/[C@@H](C)CC[C@H]2C(C)(C)CCC[C@]12C |r|
COc1ccc(O)c(OC)c1CC1=C(C)CCC2C(C)(C)CCC[C@]12C |c:13|
CC1=C(Cc2cccc(CO)c2O)[C@@]2(C)CCCC(C)(C)C2CC1 |c:1|
COc1ccc(O)c(O)c1Cc1cccc2ccccc12
COc1ccc(O)c(O)c1CC1=C(C)CCC2C(C)(C)CCC[C@]12C |c:12|
COc1c(O)ccc(O)c1CC1=C(C)CCC2C(C)(C)CCC[C@]12C |c:12|
CC1=C(Cc2ccc(O)c(O)c2O)[C@@]2(C)CCCC(C)(C)C2CC1 |c:1|
COc1ccc(O)c(O)c1CCC1[C@@H](C)CCC2C(C)(C)CCC[C@]12C
COc1c(O)cccc1CC1=C(C)CCC2C(C)(C)CCC[C@]12C |c:11|
CC1=C(Cc2cccc(O)c2O)[C@@]2(C)CCCC(C)(C)C2CC1 |c:1|
COc1ccc(O)c(O)c1Cc1ccc2ccccc2c1
Oc1ccc(Cc2ccccc2)cc1O
CCCCCCCCCCCCCc1n[nH]c(=S)n1-c1ccccc1
CCCCCCCCCCCCCCCP(O)(=O)OCc1ccccc1
CCCCCCCCCCCCCCCCCCP(O)(=O)OCc1ccccc1
CCCCCCCCCCCCCCCCCCP(O)(=O)CCc1ccccc1
CCCCCCCCCCCCCCP(O)(=O)Oc1ccc2ccccc2c1
CCCCCCCCCCCCCCP(O)(=O)OCc1cccc(Oc2ccccc2)c1
CCCCCCCCCCCCCCP(O)(=O)OCc1ccccc1
CCCCCCCCCCCCCCP(O)(=O)OCc1ccoc1
Clc1ccc(cc1)N1CCN(CC1)c1nc(nc(n1)-c1ccccc1)N1CCNCC1
Clc1ccc(cc1)N1CCN(CC1)c1nc(nc(n1)N1CCc2ccccc2C1)N1CCNCC1
Oc1ccc(CCNc2nc(nc(n2)N2CCN(CC2)c2ccc(Cl)cc2)N2CCNCC2)cc1O
Clc1ccc(cc1)N1CCN(CC1)c1nc(Cc2ccccc2)nc(n1)N1CCNCC1
Clc1ccc(cc1)N1CCN(CC1)c1nc(NCCc2ccccc2)nc(n1)N1CCNCC1
Clc1ccc(cc1)N1CCN(CC1)c1nc(nc(n1)N1CCNCC1)C#Cc1ccccc1
COc1ccc(CCNc2nc(nc(n2)N2CCN(CC2)c2ccc(Cl)cc2)N2CCNCC2)cc1O
CCCCc1nc(nc(n1)N1CCN(CC1)c1ccc(Cl)cc1)N1CCNCC1
CN(CCc1ccccc1)c1nc(nc(n1)N1CCN(CC1)c1ccc(Cl)cc1)N1CCNCC1
Clc1ccc(cc1)N1CCN(CC1)c1nc(Cc2ccc3ccccc3c2)nc(n1)N1CCNCC1
Clc1ccc(Cc2nc(nc(n2)N2CCN(CC2)c2ccc(Cl)cc2)N2CCNCC2)cc1
Clc1ccc(cc1)N1CCN(CC1)c1nc(N=NCc2ccccc2)nc(n1)N1CCNCC1 |w:17.19|
CC(C)C(O)CN1C(COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1
CC(C)(O)CN1C(COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1
CCCN1C(COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1
O[C@@H](CN1[C@H](COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
OC(CN1C(COc2c1cccc2-c1cccc(F)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F
O[C@@H](CN1[C@H](COc2c1cccc2-c1cc(F)cc(F)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1[C@H](COc2c1cccc2-c1cc(F)c(F)c(F)c1)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1[C@H](COc2c1cccc2-c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1[C@H](COc2c1cccc2-c1cc(F)cc(F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1[C@H](COc2c1cccc2-c1cc(F)c(F)c(F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1[C@H](COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
OC(CN1C(COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(Cl)c1)C(F)(F)F
CCOc1cccc(c1)C1COc2c(cccc2-c2cccc(OC(F)(F)F)c2)N1CC(O)C(F)(F)F
OC(CN1C(COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(SC(F)(F)F)c1)C(F)(F)F
OC(CN1C(COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1ccc2OC(F)(F)Oc2c1)C(F)(F)F
O[C@H](CF)CN1[C@H](COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1 |r|
O[C@@H](CF)CN1[C@H](COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1 |r|
C[C@H](O)CN1[C@H](COc2c1cccc2-c1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)C(F)F)c1 |r|
Clc1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)c1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2cccc(c2)C#N)cc1
Fc1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)c1
COc1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)c1
CC(OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N)(C(F)(F)F)C(F)(F)F
CC(OCCNc1ccc(cc1)-c1nc2cc(ccc2o1)C#N)(C(F)(F)F)C(F)(F)F
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2)cc1
CCc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
CCCc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
FC(F)(F)c1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2Cl)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C#N)cc1
Fc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
COc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
[O-][N+](=O)c1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
Cc1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)c1
FC(F)(F)c1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)c1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)OCc2ccccc2)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)NCc2ccccc2)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)CCc2ccccc2)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)CSc2ccccc2)cc1
Cc1ccccc1CNC(=O)c1ccc(cc1)-c1nc2cc(Cl)ccc2o1
Clc1ccc2oc(nc2c1)-c1ccc(NS(=O)(=O)Cc2ccccc2)cc1
CN(C(=O)COc1ccccc1C)c1ccc(cc1)-c1nc2cc(Cl)ccc2o1
CC(Oc1ccccc1)C(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
Cc1ccccc1COCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
FC(F)(F)c1ccccc1COCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
CCOCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
CC(C)OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
CC(C)(C)OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
FC(F)(F)C(OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N)C(F)(F)F
CC(C)(OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N)C(F)(F)F
FC(F)(F)C(OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N)(C(F)(F)F)C(F)(F)F
C(COc1ccccc1)Nc1ccc(cc1)-c1nc2ccccc2o1
CC(C)OCCNc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(c2o1)C(C)(C)O)C#N
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)ccc2o1
[O-][N+](=O)c1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)c1
Cc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)cc1
FC(F)(F)c1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)cc1
Clc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(cc2)C#N)cc1
Fc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)cc1
COc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)cc1
[O-][N+](=O)c1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(Cl)ccc3o2)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)CNc2ccccc2)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)COCc2ccccc2)cc1
Clc1ccc2oc(nc2c1)-c1ccc(NC(=O)CNCc2ccccc2)cc1
CC1(C)C[C@H](O)c2c(CCl)c(C(=O)c3ccc(cc3)C(F)(F)F)c(nc2C1)C1CCCC1 |r|
CCOC(=O)c1c2[C@@H](O)CC(C)(C)Cc2nc(C2CCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2C1CCN(CC1)C(=O)OCc1ccccc1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2C1CCNCC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2CN1CCCCC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2N1CCCC1 |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCCCC2)c1[C@@H](O)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c([C@@H](O)c1ccc(cc1)C(F)(F)F)c2C1CCCCC1 |r|
CC(C)c1nc2CC3(CCC3)C[C@H](O)c2c(C2CCCCC2)c1[C@@H](O)c1ccc(cc1)C(F)(F)F |r|
O[C@@H](c1ccc(cc1)C(F)(F)F)c1c(nc2CC3(CCC3)C[C@H](O)c2c1C1CCCCC1)C1CCCC1 |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCCCC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2C1CCCCC1 |r|
CC(C)c1nc2CC3(CCC3)C[C@H](O)c2c(C2CCCCC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
O[C@H]1CC2(CCC2)Cc2nc(C3CCCC3)c([C@@H](F)c3ccc(cc3)C(F)(F)F)c(C3CCCCC3)c12 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(Cc1ccc(cc1)C(F)(F)F)c2C1CCCCC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c([C@@H](F)c1ccc(cc1)C(F)(F)F)c2-c1ccc(F)cc1 |r|
CC(C)c1nc2CC3(CCC3)C[C@H](O)c2c(-c2ccc(F)cc2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F |r|
CCc1c2[C@@H](O)CC(C)(C)Cc2nc(C2CCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CCCc1c2[C@@H](O)CC3(CCC3)Cc2nc(C2CCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CCCCCc1c2[C@@H](O)CC(C)(C)Cc2nc(C2CCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1c2[C@@H](O)CC(C)(C)Cc2nc(C2CCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1c2[C@@H](O)CC3(CCC3)Cc2nc(C2CCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2C1CC1 |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2C1CCCC1 |r|
O[C@H]1CC2(CCC2)Cc2nc(C3CCCC3)c(C(=O)c3ccc(cc3)C(F)(F)F)c(C3CCCC3)c12 |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2CC3(CCC3)C[C@H](O)c2c(C2CCCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2C1CCCCC1 |r|
O[C@H]1CC2(CCC2)Cc2nc(C3CCCC3)c(C(=O)c3ccc(cc3)C(F)(F)F)c(C3CCCCC3)c12 |r|
CCC(C)c1c2[C@@H](O)CC(C)(C)Cc2nc(C2CCCC2)c1C(=O)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c(C1)nc(C1CCCC1)c(C(=O)c1ccc(cc1)C(F)(F)F)c2CC(F)(F)F |r|
CCCCCCCCOC(=O)c1ccc2Nc3cc4ccccc4cc3Nc2c1
Clc1ccc(SCc2ccc(NS(=O)(=O)c3ccccc3)cc2)cc1
CCN(CC)c1ccc(Nc2ccc(CC(=O)c3ccccc3)cc2)cc1
COc1ccc(cc1C(=O)NCCc2ccc(cc2)S(=O)(=O)NC(=O)NC3CCCCC3)Cl
COc1cccc(Oc2cccc(c2)N(CC(O)C(F)(F)F)Cc2cccc(OCC(O)C(F)(F)F)c2)c1
OC(CN(Cc1cccc(OC(F)(F)C(F)(F)F)c1)c1cccc(Oc2ccc(S)cc2)c1)C(F)(F)F
CCCC(O)CN(Cc1cccc(OC(F)(F)F)c1)c1ccccc1Oc1ccccc1
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1ccccc1Oc1ccccc1)c1ccc(cc1)C(F)(F)F
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1ccccc1Oc1ccccc1)c1ccccc1
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1ccccc1Oc1ccccc1)Cc1ccccc1
OC(CN(Cc1cccc(OC(F)(F)F)c1)c1ccccc1Oc1ccccc1)C=C
CC(C)c1ccc(Cc2cccc(c2)C(CC(C)C(C)(C)C)Cc2cccc(CC(C)(C)C(C)C)c2)cc1C
COc1ccc(cc1)-c1nc(NC(=O)c2ccc(OC)c(OC)c2)[se]c1Cc1ccccc1
COc1ccc(cc1)-c1nc(NC(=O)c2cc(OC)c(OC)c(OC)c2)[se]c1Cc1ccccc1
CCCCCC(=O)Nc1nc(c(Cc2ccccc2)[se]1)-c1ccc(O)cc1
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1ccccc1OC)C(F)(F)F
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(C)ccc1OC)C(F)(F)F
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(OC)ccc1OC)C(F)(F)F
CCOc1ccc(C)cc1-c1ccc(cc1CN(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)OC)C(F)(F)F
CCc1ccc(OC)c(c1)-c1ccc(cc1CN(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)OC)C(F)(F)F
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(ccc1OC)C(C)C)C(F)(F)F
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(C(C)C)c(F)cc1OC)C(F)(F)F
CCCc1ccc(OC)c(c1)-c1ccc(cc1CN(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)OC)C(F)(F)F
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(ccc1OC)C(C)(C)C)C(F)(F)F
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1ccccc1-c1cc(ccc1OC)C(C)C
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(ccc1OC)C(C)C)[N+]([O-])=O
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(N)ccc1-c1cc(ccc1OC)C(C)C
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(I)ccc1-c1cc(ccc1OC)C(C)C
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(ccc1OC)C(C)C)C#N
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(OC)ccc1-c1cc(ccc1OC)C(C)C
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(F)ccc1-c1cc(ccc1OC)C(C)C
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(Cl)ccc1-c1cc(ccc1OC)C(C)C
COC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cc1cc(ccc1-c1cc(ccc1OC)C(C)C)C(C)(C)C
CCOC(=O)c1ccc(cc1)N1CCN(CC(=O)Nc2ccc(cc2)-c2nc3cc(cc(C)c3o2)C#N)CC1
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2ccccc2C(F)(F)F)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2cccc(c2)C(F)(F)F)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2cccc(Cl)c2)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2ccc(Cl)cc2)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2cccc(c2)C(O)=O)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2ccc(cc2)C(F)(F)F)cc1)C#N
COC(=O)c1cccc(c1)N1CCN(CC(=O)Nc2ccc(cc2)-c2nc3cc(cc(C)c3o2)C#N)CC1
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CC2CCN(CC2)C(=O)OC(C)(C)C)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)C(=O)OC(C)(C)C)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)C(=O)OCC(C)(C)C)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)S(=O)(=O)Cc2ccccc2)cc1)C#N
CC(C)OC(=O)N1CCC(CC1)OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(C)c2o1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CCC2CCN(CC2)C(=O)OC(C)(C)C)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)C(=O)Oc2ccccc2)cc1)C#N
COc1cccc(c1)N1CCN(CC(=O)Nc2ccc(cc2)-c2nc3cc(cc(C)c3o2)C#N)CC1
CCC(C)(C)OC(=O)N1CCC(CC1)OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(C)c2o1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2ccccc2Cl)cc1)C#N
COc1ccc(cc1)N1CCN(CC(=O)Nc2ccc(cc2)-c2nc3cc(cc(C)c3o2)C#N)CC1
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)C(=O)NC(C)(C)C)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2ccccc2)cc1)C#N
CC(C)(C)OC(=O)N1CCC(CC1)OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)C(=O)OC(C)(C)C)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)C(=O)CC(C)(C)C)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CCC(C)(C)C)CC2)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC(=O)OC(C)(C)C)CC2)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)C(=O)OCc2ccccc2)cc1)C#N
O=C(COC1CCC1)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
O=C(COC1CCCC1)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
O=C(COC1CCCCC1)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
O=C(COC1CCCCCC1)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
CC12CCC(CC1)(CC2)OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
O=C(COC1CCC2CCCCC2C1)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
O=C(COC1CCOCC1)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
O=C(COC1CCNCC1)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
COC(=O)N1CCC(CC1)OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(C)c2o1)C#N
CCOC(=O)N1CCC(CC1)OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(C)c2o1)C#N
CCCCS(=O)(=O)N1CCC(CC1)OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(C)c2o1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)COC2CCN(CC2)S(=O)(=O)c2ccccc2)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCNCC2)cc1)C#N
COc1ccccc1N1CCN(CC(=O)Nc2ccc(cc2)-c2nc3cc(cc(C)c3o2)C#N)CC1
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2ccc(cc2)C(O)=O)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NC(=O)CN2CCN(CC2)c2ccc(cn2)C(F)(F)F)cc1)C#N
CC(C)Oc1ccc(F)cc1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
Cc1cc(cc2nc(oc12)-c1ccc(CCCN2CCN(CC2)c2ccc(cc2)C(F)(F)F)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(cc1)C#CCN1CCN(CC1)c1ccc(cc1)C(F)(F)F)C#N
Cc1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)CCN1CCN(CC1)c1ccc(cc1)C(F)(F)F)C#N
Cc1cc(cc2nc(oc12)-c1ccc(CC(=O)CN2CCN(CC2)c2ccc(cc2)C(F)(F)F)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F)C#N
Cc1cc(cc2nc(oc12)-c1ccc(OCN2CCN(CC2)c2ccc(cc2)C(F)(F)F)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(cc1)C(O)CCN1CCN(CC1)c1ccc(cc1)C(F)(F)F)C#N
Cc1cc(cc2nc(oc12)-c1ccc(CC(O)CN2CCN(CC2)c2ccc(cc2)C(F)(F)F)cc1)C#N
COC(CN1CCN(CC1)c1ccc(cc1)C(F)(F)F)Cc1ccc(cc1)-c1nc2cc(cc(C)c2o1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(NCC(O)CN2CCN(CC2)c2ccc(cc2)C(F)(F)F)cc1)C#N
Cc1cc(cc2nc(oc12)-c1ccc(cc1)N1CCC(N2CCN(CC2)c2ccc(cc2)C(F)(F)F)C1=O)C#N
Cc1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCCC1CCN(CC1)c1ccc(cc1)C(F)(F)F)C#N
Cc1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cc1)C(F)(F)F)C#N
CN(CC1CCN(CC1)c1ccc(cc1)C(F)(F)F)C(=O)c1ccc(cc1)-c1nc2cc(cc(C)c2o1)C#N
FC(F)(F)c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C4CC4)c3o2)C#N)CC1
FC(F)(F)c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(c3o2)C(F)(F)F)C#N)CC1
CC(C)(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)C(F)(F)F)C#N
CC(=C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)C(F)(F)F)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)C(F)(F)F)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1nccc(n1)C(F)(F)F)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccccn1)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1cccc(n1)C(F)(F)F)C#N
COc1cccc(n1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1cc(ccn1)C(F)(F)F)C#N
COC(=O)c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
COC(=O)c1cccc(n1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1cccc(n1)C(O)=O)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)[N+]([O-])=O)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(Br)cn1)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)C(C)=C)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)-c1ccccc1)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)-c1ccc(C)cc1)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)-c1cccc(C)c1)C#N
COc1cccc(Cl)c1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
COc1cc(F)c(cc1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1)C(C)C
CC(C)Oc1ccc(C)cc1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
CC(C)Oc1ccc(cc1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1)C(F)(F)F
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CCN(CC1)c1ccc(cn1)-c1cc(ccc1OCc1ccccc1)C(F)(F)F)C#N
CC(C)Oc1ccccc1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
CC(C)COc1ccccc1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
CC(C)c1ccccc1-c1ccc(nc1)N1CCC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)CC1
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CN(C(=O)O1)c1ccc(Cl)cn1)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@@H](CC1)c1ccc(Cl)cc1)C#N |r,wU:22.24,wD:25.31,(9.15,-44.24,;8.38,-45.58,;6.84,-45.58,;9.15,-46.91,;8.38,-48.24,;9.15,-49.58,;10.69,-49.57,;11.45,-48.25,;12.96,-47.93,;13.11,-46.4,;11.71,-45.77,;10.68,-46.91,;14.45,-45.63,;15.78,-46.4,;17.12,-45.63,;17.11,-44.08,;15.78,-43.31,;14.45,-44.08,;18.44,-43.3,;18.44,-41.76,;19.78,-44.07,;19.79,-45.61,;21.12,-46.37,;22.44,-45.59,;23.78,-46.37,;23.78,-47.91,;22.45,-48.68,;21.12,-47.91,;25.12,-48.68,;25.11,-50.22,;26.44,-50.99,;27.78,-50.22,;29.11,-50.98,;27.77,-48.67,;26.44,-47.9,;8.39,-50.92,;7.63,-52.26,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@@H](CC1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C#N |r,wU:22.24,wD:25.31,(22.07,-31.51,;21.3,-32.85,;19.76,-32.85,;22.07,-34.18,;21.3,-35.51,;22.08,-36.85,;23.62,-36.84,;24.38,-35.51,;25.89,-35.2,;26.04,-33.67,;24.64,-33.04,;23.61,-34.18,;27.37,-32.9,;28.71,-33.67,;30.04,-32.9,;30.04,-31.35,;28.7,-30.58,;27.38,-31.35,;31.37,-30.57,;31.36,-29.03,;32.71,-31.34,;32.71,-32.88,;34.05,-33.64,;35.37,-32.86,;36.71,-33.64,;36.71,-35.18,;35.37,-35.95,;34.04,-35.18,;38.04,-35.95,;39.37,-35.17,;40.7,-35.94,;40.7,-37.48,;39.37,-38.25,;38.04,-37.48,;39.37,-39.79,;38.03,-40.56,;40.7,-40.56,;39.36,-41.33,;42.03,-35.16,;43.37,-35.93,;42.02,-33.62,;43.11,-34.06,;21.32,-38.19,;20.55,-39.53,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@H](CC1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C#N |r,wU:22.24,25.31,(-6.91,-30.32,;-7.68,-31.66,;-9.22,-31.66,;-6.91,-32.99,;-7.68,-34.32,;-6.9,-35.66,;-5.36,-35.65,;-4.6,-34.32,;-3.09,-34.01,;-2.94,-32.48,;-4.34,-31.85,;-5.37,-32.99,;-1.61,-31.71,;-.27,-32.48,;1.06,-31.71,;1.06,-30.16,;-.28,-29.39,;-1.6,-30.16,;2.39,-29.38,;2.38,-27.84,;3.73,-30.15,;3.73,-31.69,;5.07,-32.45,;6.39,-31.67,;7.73,-32.45,;7.73,-33.99,;6.39,-34.76,;5.06,-33.99,;9.06,-34.76,;10.39,-33.98,;11.72,-34.75,;11.72,-36.29,;10.39,-37.06,;9.06,-36.29,;10.39,-38.6,;9.05,-39.37,;11.72,-39.37,;10.38,-40.14,;13.05,-33.97,;14.39,-34.74,;13.04,-32.43,;14.13,-32.87,;-7.66,-37,;-8.43,-38.34,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@@H](CC1)c1cccc(C)c1)C#N |r,wU:22.24,wD:25.31,(21.89,-21.76,;21.12,-23.09,;19.58,-23.09,;21.89,-24.43,;21.12,-25.76,;21.89,-27.1,;23.43,-27.09,;24.19,-25.76,;25.7,-25.44,;25.85,-23.91,;24.45,-23.28,;23.42,-24.43,;27.19,-23.14,;28.52,-23.91,;29.86,-23.14,;29.85,-21.59,;28.52,-20.83,;27.19,-21.6,;31.18,-20.82,;31.18,-19.28,;32.52,-21.58,;32.53,-23.12,;33.86,-23.89,;35.18,-23.11,;36.52,-23.88,;36.52,-25.42,;35.19,-26.19,;33.86,-25.43,;37.86,-26.19,;37.85,-27.73,;39.18,-28.5,;40.52,-27.73,;40.51,-26.18,;41.84,-25.41,;39.18,-25.42,;21.13,-28.44,;20.37,-29.77,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@H](CC1)c1cccc(C)c1)C#N |r,wU:22.24,25.31,(-7.19,-20.68,;-7.96,-22.01,;-9.5,-22.01,;-7.19,-23.34,;-7.96,-24.68,;-7.18,-26.01,;-5.64,-26.01,;-4.88,-24.68,;-3.37,-24.36,;-3.22,-22.83,;-4.62,-22.2,;-5.65,-23.35,;-1.89,-22.06,;-.55,-22.83,;.78,-22.06,;.78,-20.51,;-.56,-19.75,;-1.88,-20.52,;2.11,-19.74,;2.1,-18.2,;3.45,-20.5,;3.45,-22.04,;4.79,-22.81,;6.11,-22.03,;7.45,-22.8,;7.45,-24.34,;6.11,-25.11,;4.78,-24.35,;8.78,-25.11,;8.78,-26.65,;10.11,-27.42,;11.44,-26.65,;11.44,-25.1,;12.77,-24.33,;10.11,-24.34,;-7.94,-27.36,;-8.71,-28.69,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@@H](CC1)c1cccc(c1)C(F)(F)F)C#N |r,wU:22.24,wD:25.31,(20.88,-12.64,;20.11,-13.97,;18.57,-13.97,;20.88,-15.3,;20.11,-16.64,;20.88,-17.97,;22.42,-17.97,;23.18,-16.64,;24.69,-16.32,;24.84,-14.79,;23.44,-14.16,;22.41,-15.3,;26.18,-14.02,;27.51,-14.79,;28.85,-14.02,;28.84,-12.47,;27.51,-11.7,;26.18,-12.48,;30.17,-11.69,;30.17,-10.15,;31.51,-12.46,;31.51,-14,;32.85,-14.76,;34.17,-13.99,;35.51,-14.76,;35.51,-16.3,;34.18,-17.07,;32.85,-16.3,;36.85,-17.07,;36.84,-18.61,;38.17,-19.38,;39.51,-18.61,;39.5,-17.06,;38.17,-16.3,;40.83,-16.28,;42.17,-17.05,;40.83,-14.74,;41.91,-15.18,;20.12,-19.31,;19.36,-20.65,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@H](CC1)c1cccc(c1)C(F)(F)F)C#N |r,wU:22.24,25.31,(-8.51,-12.13,;-9.28,-13.46,;-10.82,-13.46,;-8.51,-14.8,;-9.28,-16.13,;-8.5,-17.47,;-6.97,-17.46,;-6.2,-16.13,;-4.7,-15.81,;-4.54,-14.28,;-5.94,-13.65,;-6.97,-14.8,;-3.21,-13.51,;-1.87,-14.29,;-.54,-13.51,;-.54,-11.96,;-1.88,-11.2,;-3.21,-11.97,;.79,-11.19,;.78,-9.65,;2.12,-11.95,;2.13,-13.49,;3.47,-14.26,;4.79,-13.48,;6.12,-14.25,;6.13,-15.79,;4.79,-16.56,;3.46,-15.8,;7.46,-16.56,;7.45,-18.1,;8.79,-18.87,;10.12,-18.1,;10.12,-16.55,;8.78,-15.79,;11.45,-15.78,;12.78,-16.54,;11.44,-14.24,;12.53,-14.68,;-9.26,-18.81,;-10.03,-20.14,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@@H](CC1)c1ccc(cc1)C(F)(F)F)C#N |r,wU:22.24,wD:25.31,(20.13,-4.03,;19.36,-5.36,;17.82,-5.36,;20.13,-6.69,;19.36,-8.03,;20.14,-9.36,;21.67,-9.36,;22.43,-8.03,;23.94,-7.71,;24.09,-6.18,;22.7,-5.55,;21.67,-6.69,;25.43,-5.41,;26.76,-6.18,;28.1,-5.41,;28.09,-3.86,;26.76,-3.09,;25.43,-3.87,;29.43,-3.08,;29.42,-1.54,;30.76,-3.85,;30.77,-5.39,;32.1,-6.15,;33.43,-5.38,;34.76,-6.15,;34.76,-7.69,;33.43,-8.46,;32.1,-7.69,;36.1,-8.46,;36.09,-10,;37.42,-10.77,;38.76,-10,;38.75,-8.45,;37.42,-7.69,;40.09,-10.76,;40.1,-12.3,;41.43,-9.99,;41.42,-11.53,;19.37,-10.7,;18.61,-12.04,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@H](CC1)c1ccc(cc1)C(F)(F)F)C#N |r,wU:22.24,25.31,(-7.64,-4.05,;-8.41,-5.38,;-9.95,-5.38,;-7.64,-6.72,;-8.41,-8.05,;-7.63,-9.39,;-6.1,-9.38,;-5.33,-8.05,;-3.83,-7.73,;-3.67,-6.2,;-5.07,-5.57,;-6.1,-6.72,;-2.34,-5.43,;-1,-6.2,;.33,-5.43,;.33,-3.88,;-1.01,-3.12,;-2.34,-3.89,;1.66,-3.11,;1.65,-1.57,;3,-3.87,;3,-5.41,;4.34,-6.18,;5.66,-5.4,;7,-6.17,;7,-7.71,;5.66,-8.48,;4.33,-7.72,;8.33,-8.48,;8.32,-10.02,;9.66,-10.79,;10.99,-10.02,;10.99,-8.47,;9.65,-7.71,;12.33,-10.79,;12.33,-12.33,;13.66,-10.02,;13.65,-11.56,;-8.39,-10.73,;-9.16,-12.06,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@@H](CC1)c1ccc(cc1)C(C)(C)C)C#N |r,wU:22.24,wD:25.31,(19.49,4.45,;18.72,3.12,;17.18,3.12,;19.49,1.79,;18.72,.45,;19.5,-.88,;21.03,-.88,;21.8,.45,;23.3,.77,;23.46,2.3,;22.06,2.93,;21.03,1.78,;24.79,3.07,;26.13,2.3,;27.46,3.07,;27.46,4.62,;26.12,5.38,;24.79,4.61,;28.79,5.39,;28.78,6.93,;30.12,4.63,;30.13,3.09,;31.47,2.32,;32.79,3.1,;34.12,2.33,;34.13,.79,;32.79,.02,;31.46,.78,;35.46,.02,;35.45,-1.52,;36.79,-2.29,;38.12,-1.52,;38.12,.03,;36.78,.79,;39.46,-2.29,;39.46,-3.83,;40.79,-1.51,;40.78,-3.06,;18.74,-2.23,;17.97,-3.56,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CC[C@H](CC1)c1ccc(cc1)C(C)(C)C)C#N |r,wU:22.24,25.31,(-7.37,5.12,;-8.14,3.79,;-9.68,3.79,;-7.37,2.45,;-8.14,1.12,;-7.37,-.22,;-5.83,-.21,;-5.07,1.12,;-3.56,1.44,;-3.41,2.97,;-4.81,3.6,;-5.84,2.45,;-2.07,3.74,;-.74,2.97,;.6,3.74,;.59,5.29,;-.74,6.05,;-2.07,5.28,;1.92,6.06,;1.92,7.61,;3.26,5.3,;3.27,3.76,;4.6,2.99,;5.92,3.77,;7.26,3,;7.26,1.46,;5.93,.69,;4.6,1.45,;8.6,.69,;8.59,-.85,;9.92,-1.62,;11.26,-.85,;11.25,.7,;9.92,1.46,;12.59,-1.62,;12.59,-3.16,;13.92,-.85,;13.91,-2.39,;-8.13,-1.56,;-8.89,-2.89,)|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CN(C(=O)O1)c1ccc(cn1)C(C)=C)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CN(C(=O)O1)c1ccc(cn1)-c1ccccc1C#N)C#N
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CN(C(=O)O1)c1ccc(cn1)-c1ccc(C)s1)C#N
CC(C)Oc1ccc(C)cc1-c1ccc(nc1)N1CC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)OC1=O
CC(C)Oc1ccc(F)cc1-c1ccc(nc1)N1CC(CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)OC1=O
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NCC1CN(C(=O)O1)c1ccc(cn1)-c1ccccc1OC(F)(F)F)C#N
CC(C)Oc1ccc(F)cc1-c1ccc(nc1)N1C[C@@H](CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)OC1=O |r|
CC(C)Oc1ccc(F)cc1-c1ccc(nc1)N1C[C@H](CNC(=O)c2ccc(cc2)-c2nc3cc(cc(C(C)C)c3o2)C#N)OC1=O |r|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@@H]1CN(C(=O)O1)c1ccc(cn1)-c1ccccc1OC(F)(F)F)C#N |r|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@H]1CN(C(=O)O1)c1ccc(cn1)-c1ccccc1OC(F)(F)F)C#N |r|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@]1(C)CN(C(=O)O1)c1ccc(cn1)-c1ccccc1OC(F)(F)F)C#N |r|
CC(C)c1cc(cc2nc(oc12)-c1ccc(cc1)C(=O)NC[C@@]1(C)CN(C(=O)O1)c1ccc(cn1)-c1ccccc1OC(F)(F)F)C#N |r|
COc1ccc(cc1-c1ccc(cc1CN1C[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1ccccc1)C(F)(F)F)C(C)C |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@H](C)[C@@H](OC1=O)c1ccccc1)C(F)(F)F)C(C)C |r|
COc1ccc(cc1-c1ccc(cc1CN1[C@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
CC[C@H]1[C@H](OC(=O)N1Cc1cc(ccc1-c1cc(ccc1OC)C(C)C)C(F)(F)F)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1C[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1C(=O)O[C@H](c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C1(C)C)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccccc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(F)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(Cl)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(Br)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(I)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C#N)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)[N+]([O-])=O)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(N)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(C)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)(C)C)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(SC)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
CCCSc1ccc(c(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c1)-c1cc(C(C)C)c(F)cc1OC |r|
COc1cc(F)c(cc1-c1ccc(SC(C)C)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(SC(F)(F)F)cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C1=CCCC1)C(C)C |r,t:41|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)(C)F)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)(C)O)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C1CC1)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)S(C)(=O)=O)C(C)C |r|
CCCS(=O)(=O)c1ccc(c(CN2[C@@H](C)[C@H](OC2=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c1)-c1cc(C(C)C)c(F)cc1OC |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)S(=O)(=O)C(C)C)C(C)C |r|
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)S(=O)(=O)C(F)(F)F)C(C)C |r|
COc1ccc(cc1-c1ccc(cc1CN1C(COC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C
COc1ccc(cc1-c1ccc(cc1CN1C[C@@H](OC1=O)c1ccccc1)C(F)(F)F)C(C)C |r|
COc1ccc(cc1-c1ccc(cc1CN1C[C@H](OC1=O)c1ccccc1)C(F)(F)F)C(C)C |r|
COC(=O)N(Cc1ccccc1)Cc1cc(ccc1-c1cc(ccc1OC)C(C)C)C(F)(F)F
CC1(C)CCC[C@]2(C)C3C=C4C(Cl)C(=O)C(=O)C=C4OC3CC[C@@]12C |c:17,t:9|
C[C@]1(CO)[C@H](O)C(=O)C[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2CCc2cocc12 |r|
C[C@H](CCCc1ccoc1)[C@H](C[C@H]1C(C)=CC[C@H]2C(C)(C)CCC[C@]12C)OS([O-])(=O)=O |c:15|
CC(=O)C1C=C2OC3CC[C@@]4(C)C(C)(C)CCC[C@]4(C)C3C=C2C(C(C)=O)=C1C(C)=O |c:23,29,t:4|
COc1ccc(O)c2O[C@@]34CCCC(C)(C)C3CC[C@H](C)[C@@]4(C)Cc12
COC1=CC(=O)C(=O)C(C[C@]2(C)[C@@H](C)CC[C@@]3(C)[C@H]2CCCC3=C)C1=O |r,t:2|
C[C@H]1CCC2C(C)(C)CCC[C@]22Oc3ccc(O)cc3C[C@]12C
CC1(C)CCC[C@@]2(C)[C@H]1CC[C@]1(C)OC3=CC(=O)C(=O)CC3=C[C@H]21 |r,c:23,t:15|
C[C@H]1CC[C@@]2(C)[C@@H](CCC=C2C)[C@]1(C)Cc1cc(O)ccc1O |r,c:9|
CCCCCCCCCCCCC\C=C\C(O)C(N)CO[C@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O |r|
CCCCCCCCCCCCC/C=C/[C@H]([C@H](CO)N)O
CCCCCCCCCCCCCCCC(=O)N[C@@H](CO)[C@H](O)\C=C\CC\C=C\CCCCCCCCC
CCCCCCCCCCCCCCC[C@@H](O)[C@@H](N)CO |r|
CCCCCCCCCCCCC\C=C\[C@@H](O)[C@H](CO)N(C)C |r|
CCCCCCCCCCCCC\C=C\[C@@H](O)[C@@H](N)COP([O-])(=O)OCC[N+](C)(C)C
CCCCCCCCCCCCCCCC(=O)N[C@@H](CO)[C@H](O)\C=C\CCCCCCCCCCCCC |r|
CCCCCCCCCCCCCCCC(=O)N[C@@H](CO)[C@H](O)\C=C\CC\C=C\C=C\CCCCCCC
CCCCCCCCCCCCCCCC(=O)N[C@@H](CO)[C@H](O)\C=C\CC\C=C\CCCCCCCC(C)C
CC(C)CNC(=O)\C=C\[C@@H]1C[C@H]1[C@@H]1C[C@H]1[C@@H]1C[C@H]1[C@@H]1C[C@H]1[C@@H]1C[C@H]1\C=C\[C@@H]1C[C@H]1C |r|
CCC(CC)CC1(CCCCC1)C(=O)Nc1ccccc1SC
CCCCCCC1(CCCCC1)C(=O)Nc1ccccc1S
CCC1(CCCCC1)C(=O)Nc1ccccc1S
CCC(CC)CC1(CCCCC1)C(=O)Nc1ccccc1SC(C)=O
O=C(Nc1ccccc1SSc1ccccc1NC(=O)C1CCCCC1)C1CCCCC1
CC(C)(C)C(=O)Nc1ccc(SSc2ccc(NC(=O)C(C)(C)C)cc2)cc1
CCC(CC)CC1(CCCCC1)C(=O)Nc1ccccc1S
CCCCC(=O)Nc1ccccc1SSc1ccccc1NC(=O)CCCC
CC1(CCCCC1)C(=O)Nc1ccccc1S
CCCCCCCC(=O)Nc1ccccc1SSc1ccccc1NC(=O)CCCCCCC
CC(C)(C)C(=O)Nc1ccccc1SSc1ccccc1NC(=O)C(C)(C)C
CCC(CC)CC1(CCCCC1)C(=O)Nc1ccccc1SC(=O)C(C)(C)C
O=C(Nc1ccccc1SSc1ccccc1NC(=O)c1ccccc1)c1ccccc1
CCCC1(CCCCC1)C(=O)Nc1ccccc1S
CC1(CCCCC1)C(=O)Nc1ccccc1OC(=O)Cc1ccccc1
CCC(=O)Nc1ccccc1SSc1ccccc1NC(=O)CC
CCCCCCCC1(CCCCC1)C(=O)Nc1ccccc1S
CC1(CCCCC1)C(=O)Nc1ccccc1SC(=O)Cc1ccccc1
CN(C(=O)C(C)(C)C)c1ccccc1SSc1ccccc1N(C)C(=O)C(C)(C)C
CC(C)(C)NC(=O)c1ccccc1SSc1ccccc1C(=O)NC(C)(C)C
CCCCC1(CCCCC1)C(=O)Nc1ccccc1S
CC1(CCCCC1)C(=O)Nc1ccccc1SSc1ccccc1NC(=O)C1(C)CCCCC1
CC(C)C(=O)Nc1ccccc1SSc1ccccc1NC(=O)C(C)C
CC(C)(C)C(=O)Nc1cccc(SSc2cccc(NC(=O)C(C)(C)C)c2)c1
CCCCCC1(CCCCC1)C(=O)Nc1ccccc1S
CC(=O)Nc1ccccc1SSc1ccccc1NC(C)=O
CC(C)CCCC1(CCCCC1)C(=O)Nc1ccccc1S
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)cc(Cl)c2o1
CC(=O)c1cc(C)cc2nc(oc12)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
COC(=O)c1cccc2nc(oc12)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)[N+]([O-])=O
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C(F)(F)F
CC(=O)c1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(OC(F)(F)F)ccc2o1
Cc1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2c(C)cccc2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cccc(C(O)=O)c2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2ccc(cc2o1)N1CCCC1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2ccc(F)cc2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2ccc(cc2o1)[N+]([O-])=O
COc1ccc2nc(oc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C(C)(C)C
COc1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(F)ccc2o1
COC(=O)c1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2c(cccc2o1)[N+]([O-])=O
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(F)cc2)cc1
Cc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)cc1
Cc1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c1
COC(=O)c1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(C)cc(C)c2o1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(Cl)cc2)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2cccc(Cl)c2)cc1
CC(C)c1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2cccc(F)c2)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2F)cc1
CC(C)c1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(C)cc(C)c2o1
COC(=O)c1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2Cl)cc1
COc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)cc1
COc1cccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(cc2)C#N)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2cccc(c2)C#N)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C#N)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(F)cc2C)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(Br)cc2C)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(Cl)cc2C)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(Cl)c(c2)C(F)(F)F)cc1
Cc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c(C)c1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(Cl)c(Cl)c2)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2cccc(OC(F)(F)F)c2)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2OC(F)(F)F)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2cccc(c2)-c2ccccc2)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2-c2ccccc2)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C(F)(F)F)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2cccc(c2)C(F)(F)F)cc1
Cc1cc(C)cc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2c(Cl)cccc2Cl)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2cc(Cl)ccc2Cl)cc1
Cc1ccc(C)c(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(OC(F)(F)F)cc2)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(cc2)C(F)(F)F)cc1
COC(=O)c1c(Cl)ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(ccc3o2)C#N)c1C
Cc1cc(Br)ccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
Clc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(ccc3o2)C#N)c2CCCc12
Cc1cc(Cl)ccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C#N
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(Cl)c(C)c2C)cc1
COC(=O)c1c(Cl)ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(C)cc(C)c3o2)c1C
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(C)c3CCCc23)cc1
Cc1c(Cl)ccc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(ccc3o2)C#N)c1C
FC(F)(F)c1cc(OCC(=O)Nc2ccc(cc2)-c2nc3cc(ccc3o2)C#N)ccc1Cl
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(Cl)c3CCCc23)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(Cl)c2o1)C#N
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(cc(c2o1)C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2oc(nc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)cc([N+]([O-])=O)c2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Cl)cc(Br)c2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cccc(C)c2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(Br)ccc2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(CO)ccc2o1
COC(=O)c1ccc2nc(oc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2ccc(Cl)cc2o1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)C(O)=O
COc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(C)cc(C)c2o1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2c(C)cccc2Cl)cc1
Cc1cc(C)c2oc(nc2c1)-c1ccc(NC(=O)COc2ccc(cc2)-c2ccccc2)cc1
Cc1ccc2nc(oc2c1)-c1ccc(NC(=O)COc2ccccc2C)cc1
Cc1ccccc1OCC(=O)Nc1ccc(cc1)-c1nc2cc(ccc2o1)-c1ccccc1
CCOC(=O)N1[C@H](CC)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(cc(C)c12)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(Cl)cc(c2)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(Cl)cc(c2)C(F)(F)F)c2nnn(C)n2)c2nc(C)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C#N)c2nnn(C)n2)c2nc(C)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(F)cc(c2)C(F)(F)F)c2nnn(C)n2)c2nc(C)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(Cl)cc(Cc3cncc(c3)C(F)(F)F)c2)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC)C(F)(F)F |r|
CCOC(=O)N1[C@H](CC)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc12)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OCCO)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OCC(C)(C)C(O)=O)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OCCN(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC1CCOCC1)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC1CCN(C)CC1)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OCCc1nnn[nH]1)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OCCN1CCOCC1)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OCCN1CCN(C)CC1)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)C(C)C)C(F)(F)F |r|
CCCC(=O)N1[C@H](CC)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc12)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)c1c(C)cnn1C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1CC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1CCC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2nc(OC)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2nc(C)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2nc(ccc2N1C(=O)OC(C)C)N(C)C |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2nc(ccc12)C(F)(F)F |r|
CC(C)OC(=O)N1[C@@H](C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2nc(ccc12)C(F)(F)F)C1CC1 |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)N1CCCC1 |r|
CC[C@@H]1C[C@H](N(Cc2cc(Cl)cc(Cl)c2)c2nnn(C)n2)c2nc(C)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2nc(Br)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(C)n[nH]2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(C)no2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn[nH]2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnnn2C)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(OC)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(Br)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(C)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCN)n2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCO)n2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)N(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(N)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(NC)ccc2N1C(=O)OC(C)C |r|
CCNc1ccc2N([C@H](CC)C[C@H](N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)c3nnn(C)n3)c2n1)C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)N1CCOCC1 |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)N1CCNCC1 |r|
CC[C@H]1C[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@H]1C[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(C)ccc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(OC)c(C)cc2N1C(=O)OC(C)C |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2nc(N)c(C)cc2N1C(=O)OC(C)C |r|
CCC1CC(N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2sccc2N1C(=O)OC(C)C
CCC1CC(N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2ccc(C)nc2N1C(=O)OC(C)C
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C#N)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2noc(C)n2)c2nc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(n2)C2CNC2)c2cc(ccc12)C(F)(F)F |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(n2)C2CCNCC2)c2cc(ccc12)C(F)(F)F |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCN3CCCC3)n2)c2cc(ccc12)C(F)(F)F |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCN3CC3)n2)c2cc(ccc12)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCCN(C)C)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCCN)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCCO)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CC(=O)N(C)C)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CC(N)=O)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CC(=O)OC)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CC(O)=O)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCN)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCO)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCCl)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCC#N)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CC3CC3)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CC(C)C)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(n2)C(C)(C)C)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(n2)C(C)C)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CCCCn1nnc(n1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)[C@H]1C[C@@H](CC)N(C(=O)OC(C)C)c2ccc(cc12)C(F)(F)F |r|
CC(C)OC(=O)N1[C@@H](C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCN)n2)c2cc(ccc12)C(F)(F)F)C1CC1 |r|
CC(C)OC(=O)N1[C@@H](C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCN)n2)c2cc(ccc12)C(F)(F)F)C(C)C |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCN)n2)c2cc(ccc12)C(F)(F)F |r|
CC(C)OC(=O)N1[C@@H](C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCCO)n2)c2cc(ccc12)C(F)(F)F)C(C)C |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CCCO)n2)c2cc(ccc12)C(F)(F)F |r|
CC(C)OC(=O)N1[C@@H](C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2cc(ccc12)C(F)(F)F)C1CC1 |r|
CC(C)OC(=O)N1[C@@H](C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2cc(ccc12)C(F)(F)F)C(C)C |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(n2)C2CCN(C)CC2)c2cc(ccc12)C(F)(F)F |r|
CCCn1nnc(n1)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)[C@H]1C[C@@H](CC)N(C(=O)OC(C)C)c2ccc(cc12)C(F)(F)F |r|
CCC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC(C)OC(=O)N1[C@H](C)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2cc(ccc12)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(C)no2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(C)n[nH]2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(C)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn[nH]2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
CCOC(=O)N1[C@H](CC)C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)=O)c2cc(ccc12)C(F)(F)F |r|
CC[C@@H]1C[C@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2nnn(CC#N)n2)c2cc(ccc2N1C(=O)OC(C)C)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@@](Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)N[C@@H]1CCOC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)N[C@@H]1CCOC1=O)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@@](Cc1ccccc1)(NC(=O)N[C@@H]1CCOC1=O)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCC(F)(F)C1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@@](Cc1ccccc1)(NC(=O)NC1CCC(F)(F)C1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCCCC1(F)F)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCCC(F)(F)C1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCC(F)(F)CC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@@](Cc1ccccc1)(NC(=O)N[C@@H]1CCOC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@@](Cc1ccccc1)(NC(=O)NC1CCCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCC(F)(F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N[C@@H]1CCC(F)(F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N[C@H]1CCC(F)(F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CC1(F)F)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CC(F)(F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CCCC1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CCC(F)(F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CC[C@H](F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CC[C@@H](F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CC(F)(F)C(F)(F)C1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CCC(C1)C(F)(F)F)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CCC[C@H]1C(F)(F)F)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)N1CCC[C@@H]1C(F)(F)F)c1ccc(Cl)cn1 |r|
CCCNC(=O)N[C@@](Cc1ccccc1)(c1cc(F)cc(OC(F)(F)C(F)F)c1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)NCCC(F)(F)F)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)NCC(F)(F)C(F)(F)F)c1ccc(Cl)cn1 |r|
CCNC(=O)N[C@@](Cc1ccccc1)(c1cc(F)cc(OC(F)(F)C(F)F)c1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)NCC(F)(F)F)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@](Cc1ccccc1)(NC(=O)c1ccc(F)c(c1)C(F)(F)F)c1ccc(Cl)cn1 |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1F)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Cc1ccc(C[C@](NC(=O)NC2CCCC2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)cc1 |r|
Fc1cc(cc(c1)[C@](CC=C)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1ccc(C[C@](NC(=O)NC2CCCC2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)cc1 |r|
Cc1nc(C[C@](NC(=O)NC2CCCC2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)no1 |r|
Cc1csc(C[C@](NC(=O)NC2CCCC2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)n1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@@](Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cccc(c1)C(Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1
FC(F)(F)Oc1cccc(c1)C(Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1
COc1ccc(cn1)[C@@](Cc1ccccc1)(NC(=O)NC1CCCC1)c1cc(F)cc(c1)C(F)(F)F |r|
Fc1cc(cc(c1)C(Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)nc1)C(F)(F)F
Fc1ccc(nc1)[C@@](Cc1ccccc1)(NC(=O)NC1CCCC1)c1cc(F)cc(c1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(cn1)C#N)C(F)(F)F |r|
FC(F)(F)c1cccc(c1)C(Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1
Fc1ccc(nc1)C(Cc1ccccc1)(NC(=O)NC1CCCC1)c1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(c1)C(Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccccn1
Fc1ccc(cc1C(F)(F)F)C(=O)NC(Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccccn1
CC(C)(C)NC(=O)NC(Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccccn1
CC(C)(C)CC(=O)OC(Cc1ccccc1)(c1cccc(OC(F)(F)C(F)F)c1)c1ccccn1
CC(C)(C)CC(=O)OC(Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccc(Cl)cn1
CC(C)(C)CC(=O)O[C@](Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccccn1 |r|
CC(C)(C)CC(=O)O[C@@](Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccccn1 |r|
COC(=O)C[C@](NC(=O)NC1CCCC1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1 |r|
Fc1cc(cc(c1)[C@](Cc1ccccn1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1nnc[nH]1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1ccc(cc1)C(=O)NC(Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccccn1
FC(F)(F)c1cccc(c1)C(=O)NC(Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccccn1
CC(C)(C)CC(=O)NC(Cc1ccccc1)(c1cccc(c1)C(F)(F)F)c1ccccn1
FC(F)(F)c1cccc(c1)C(Cc1ccccc1)(NC(=O)c1ccccc1)c1ccccn1
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@@](Cc1ccccc1)(Nc1nc2ccc(F)cc2[nH]1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@@](Cc1ccccc1)(Nc1nc2ccccc2[nH]1)c1ccc(Cl)cn1 |r|
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1nc2ccccc2[nH]1)c1ccc(Cl)cn1)C(F)(F)F
Fc1cc(cc(c1)C(Cc1ccccc1)(NC(=O)NC1CCCC1)c1ccc(Cl)cn1)C(F)(F)F
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1nc2ccccc2s1)c1ccc(Cl)cn1)C(F)(F)F
Cc1sc(N[C@](Cc2ccccc2)(c2cc(F)cc(OC(F)(F)C(F)F)c2)c2ccc(Cl)cn2)nc1C(F)(F)F |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@@](Cc1ccccc1)(Nc1nc(cs1)C(F)(F)F)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@@](Cc1ccccc1)(Nc1nc2CCCCc2s1)c1ccc(Cl)cn1 |r|
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@@](Cc1ccccc1)(Nc1nc(c(Br)s1)C(F)(F)F)c1ccc(Cl)cn1 |r|
Cc1nc(N[C@](Cc2ccccc2)(c2cc(F)cc(OC(F)(F)C(F)F)c2)c2ccc(Cl)cn2)sc1C |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(Nc1nc2CCCCc2s1)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@@](Cc1ccccc1)(Nc1nc2CCCc2s1)c1ccc(Cl)cn1)C(F)(F)F |r|
Cc1nc(N[C@@](Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)sc1C |r|
Cc1nc(N[C@](Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)sc1C |r|
COC(=O)c1sc(NC(Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)nc1C
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1nc(c(Br)s1)C(F)(F)F)c1ccc(Cl)cn1)C(F)(F)F
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1nc(cs1)C(F)(F)F)c1ccc(Cl)cn1)C(F)(F)F
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1nc2CCCCc2s1)c1ccc(Cl)cn1)C(F)(F)F
CC(C)(C)c1csc(NC(Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)n1
CCc1csc(NC(Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)n1
Cc1cnc(NC(Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)s1
Cc1nc(NC(Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)sc1C
FC(F)C(F)(F)Oc1cc(F)cc(c1)[C@@](Cc1ccccc1)(Nc1nc2c(F)cc(F)cc2[nH]1)c1ccc(Cl)cn1 |r|
Cn1nnc(NC(Cc2ccccc2)(c2cc(F)cc(c2)C(F)(F)F)c2ccc(Cl)cn2)n1
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1ncc(o1)-c1ccccc1)c1ccc(Cl)cn1)C(F)(F)F
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1nc2ccccc2o1)c1ccc(Cl)cn1)C(F)(F)F
Fc1cc(cc(c1)C(Cc1ccccc1)(Nc1nnc([nH]1)-c1ccccc1)c1ccc(Cl)cn1)C(F)(F)F
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@@H](OC21CCCC1)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccccc1 |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(F)cc1 |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(cc1)C#N |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(cc1)C(C)(C)C#N |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(cc1)C(C)(C)C |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1cccc(c1)C(F)(F)F |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(OC(F)(F)F)cc1 |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(cn1)C(F)(F)F |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(nc1)C(F)(F)F |r|
CCc1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCC1)c1ccc(cc1)C(F)(F)F |r|
CC1(C)C[C@H](O)c2c3c([C@H](OC33CCCC3)c3ccc(cc3)C(F)(F)F)c(nc2C1)C1CCCC1 |r|
CC1(C)C[C@H](O)c2c3c([C@H](OC33CCCC3)c3ccc(cc3)C(F)(F)F)c(nc2C1)C1CCOCC1 |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC2(C)C)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCCCC1)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2CC(C)(C)C[C@H](O)c2c2c1[C@H](OC21CCOCC1)c1ccc(cc1)C(F)(F)F |r|
CC(C)c1nc2CC(C)(C)C[C@@H](O)c2c2c1[C@@H](OC21CCOCC1)c1ccc(cc1)C(F)(F)F |r|
NCC(O)C(F)(F)F
CC(=O)Oc1ccc2c(c1)occ(-c1ccc(NC(=O)COc3ccccc3)cc1)c2=O
CC(=O)Oc1ccc2c(c1)occ(-c1ccc(NC(=O)COc3ccccc3C)cc1)c2=O
CCOC(=O)c1ccc(NC(=O)CCN(Cc2ccc(F)cc2)c2cccc(Oc3ccccc3)c2)cc1
CCOC(=O)c1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1ccc(Cl)c(Cl)c1
CCOC(=O)c1ccc(NC(=O)CCN(c2cccc(Oc3ccccc3)c2)S(=O)(=O)c2ccc(F)cc2)cc1
CCOC(=O)c1ccc(NC(=O)CCN(Cc2ccc(F)cc2)c2ccc(cc2)-c2ccccc2)cc1
CCOC(=O)c1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1cccc(Oc2ccccc2)c1
OC(=O)c1ccc(NC(=O)CCN(Cc2ccc(F)cc2)c2ccc(Cl)c(Cl)c2)cc1
CCOC(=O)c1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1ccc(Cl)c(c1)-c1ccccc1
CCOC(=O)c1ccc(NC(=O)CCN(Cc2ccc(F)cc2)c2ccc(Cl)c(c2)-c2ccccc2)cc1
CCOC(=O)c1ccc(NC(=O)CCN(Cc2ccc(F)cc2)c2cc(Cl)cc(c2)-c2ccccc2)cc1
CCOC(=O)c1ccc(NC(=O)CCN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ccc(Cl)c(Cl)c2)cc1
CCOC(=O)c1ccc(NC(=O)CCN(c2ccc(Cl)c(c2)-c2ccccc2)S(=O)(=O)c2ccc(F)cc2)cc1
COc1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1ccc(Oc2ccccc2)cc1
CCOC(=O)c1ccc(NC(=O)CCN(Cc2ccc(F)cc2)c2ccc(Cl)c(Cl)c2)cc1
CCOC(=O)c1ccc(NC(=O)CCN(c2cc(Cl)cc(c2)-c2ccccc2)S(=O)(=O)c2ccc(F)cc2)cc1
CCOC(=O)c1ccc(NC(=O)CCN(Cc2ccc(cc2)C(F)(F)F)c2ccc(Cl)c(Cl)c2)cc1
CCOC(=O)c1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(cc1)C(F)(F)F)c1ccc(Cl)c(Cl)c1
CCOC(=O)c1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1ccc(Oc2ccccc2)cc1
COc1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1ccc(Cl)c(Cl)c1
CC(C)(C)NC(=O)CCN(Cc1ccc(F)cc1)c1ccc(Cl)c(Cl)c1
Fc1ccc(CN(CCC(=O)NC2CCCCC2)c2ccc(Cl)c(Cl)c2)cc1
Fc1ccc(CN(CCC(=O)NC2CC2)c2ccc(Cl)c(Cl)c2)cc1
CCCCN(CC1CC1)C(=O)CCN(Cc1ccc(F)cc1)c1ccc(Cl)c(Cl)c1
COc1ccc(cc1OC)C(CC(=O)c1ccccc1)Nc1ccc(Cl)cc1
Fc1ccc(CN(CCC(=O)N2CCN(CC2)c2ccccc2)c2ccc(Cl)c(c2)C(F)(F)F)cc1
COc1cc(F)c(cc1-c1ccc(cc1CN1[C@H](C)[C@@H](OC1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(C)C |r|
COc1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1cccc(Oc2ccccc2)c1
CCOC(=O)c1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1cccc(c1)-c1ccccc1
COc1ccc(cc1)N1CCN(CC1)C(=O)CCN(Cc1ccc(F)cc1)c1cccc(c1)-c1ccccc1
CCc1cc(ccc1Cl)N(CCC(=O)N1CCN(CC1)c1ccccc1)Cc1ccc(F)cc1
Cc1cc(ccc1Br)N(CCC(=O)N1CCN(CC1)c1ccccc1)Cc1ccc(F)cc1
Fc1ccc(CN(CCC(=O)N2CCN(CC2)c2ccccc2)c2cccc(c2)-c2ccccc2)cc1
Fc1ccc(CN(CCC(=O)N2CCN(CC2)c2ccccc2)c2ccc(Cl)c(Cl)c2)cc1
Fc1ccc(CN(CCC(=O)N2CCN(CC2)c2ncccn2)c2ccc(Cl)c(Cl)c2)cc1
Fc1ccc(CN(CCC(=O)N2CCOCC2)c2ccc(Cl)c(Cl)c2)cc1
O[C@@H](CN1C[C@](Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1[C@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1[C@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1[C@@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
CC1(Cc2cccc(OC(F)(F)F)c2)CN(C[C@@H](O)C(F)(F)F)c2ccccc12 |r|
CC1(CN(C[C@@H](O)C(F)(F)F)c2ccccc12)c1cccc(OC(F)(F)F)c1 |r|
O[C@H](CN1CC(Cc2ccccc2)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1CC(Cc2ccccc2OC(F)(F)F)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
COc1ccc(CC2(CN(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(OC(F)(F)F)c2)cc1 |r|
O[C@H](CN1CC(Cc2cccc(c2)C#N)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
COC(=O)c1cccc(CC2(CN(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(OC(F)(F)F)c2)c1 |r|
O[C@H](CN1CC(Cc2cccc(c2)C(O)=O)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
CS(=O)(=O)c1cccc(CC2(CN(C[C@@H](O)C(F)(F)F)c3ccccc23)c2cccc(OC(F)(F)F)c2)c1 |r|
O[C@H](CN1CC(Cc2cccc(Br)c2)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
Cc1csc(CC2(CN(C[C@@H](O)C(F)(F)F)c3c2cccc3F)c2cccc(OC(F)(F)F)c2)n1 |r|
O[C@H](CN1CC(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(Cl)c1)C(F)(F)F |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1ccc(OC(F)(F)F)cc1)C(F)(F)F |r|
CC(C)Oc1cc(ccn1)C1(Cc2cccc(OC(F)(F)F)c2)CN(C[C@@H](O)C(F)(F)F)c2ccccc12 |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1ccnc(c1)C(F)(F)F)C(F)(F)F |r|
Cc1cccc2N(C[C@@H](O)C(F)(F)F)CC(Cc3cccc(OC(F)(F)F)c3)(c12)c1cccc(OC(F)(F)F)c1 |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2cc(F)ccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1CC(Cc2ccccc2)(c2cc(OC(F)(F)F)ccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2cc(OC(F)(F)F)ccc12)c1ccccc1)C(F)(F)F |r|
C[C@H](O)CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2ccc(cc12)C(F)(F)F)c1cccc(OC(F)(F)F)c1 |r|
Cc1cccc2c1N(C[C@@H](O)C(F)(F)F)CC2(Cc1cccc(OC(F)(F)F)c1)c1cccc(OC(F)(F)F)c1 |r|
O[C@H](CN1CC(Cc2cccc(OC(F)(F)F)c2)(c2cccc(F)c12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1[C@@H](CN(Cc2cccc(OC(F)(F)F)c2)c2ccccc12)c1cccc(OC(F)(F)C(F)F)c1)C(F)(F)F |r|
C[C@@H](N1C[C@H](N(C[C@@H](O)C(F)(F)F)c2ccccc12)c1cccc(c1)C(F)(F)F)c1cccc(c1)C(F)(F)F |r|
O[C@H](CN1C[C@@](Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@H](CN1C[C@](Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
O[C@@H](CN1C[C@@](Cc2cccc(OC(F)(F)F)c2)(c2ccccc12)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
C[C@H](O)CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1 |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NCC(=O)CC(F)(F)F)c1ccc(Cl)cn1)C(F)(F)F |r|
CO[C@H](CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1)C(F)(F)F |r|
CC(=O)O[C@H](CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1)C(F)(F)F |r|
OC(CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1)CC(F)(F)F |r|
O[C@H](CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1)C(F)(F)F |r|
Fc1cc(cc(c1)[C@](Cc1ccccc1)(NC(=O)c1ccc(F)c(c1)C(F)(F)F)c1ccc(Cl)cn1)C(F)(F)F |r|
C[C@@H](O)CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1 |r|
OC[C@H](O)CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1 |r|
OC[C@@H](O)CN[C@@](Cc1ccccc1)(c1cc(F)cc(c1)C(F)(F)F)c1ccc(Cl)cn1 |r|
O[C@H](CN[C@@](Cc1ccccc1)(c1cc(F)cc(OC(F)(F)C(F)F)c1)c1ccc(Cl)cn1)C(F)(F)F |r|
OC(CN[C@@](Cc1ccccc1)(c1cc(F)cc(OC(F)(F)C(F)F)c1)c1ccc(Cl)cn1)CC(F)(F)F |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC[C@@H](O)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC[C@H](O)C(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC[C@H](O)CC(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
CC(C)Oc1cc(ccc1F)[C@@](Cc1ccccc1)(NC[C@@H](O)CC(F)(F)F)c1cc(F)cc(OC(F)(F)C(F)F)c1 |r|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)N2CCNCC2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)N2CCN(C)CC2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(OCCCC(O)=O)cn2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)CCC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)c2ccccc2CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)CCc2ccccc12)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)CC(CC1)C(C)(C)C)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2ccnn2C)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)CCCCC1)C(C)C |c:9|
CCC1CCC(=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)C1)c1cc(ccc1OC)C(C)C |t:5|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(OCCO)cn2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)CC(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2c(C)noc2C)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)OCc2ccccc2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)N2CCC(CC2)C(O)=O)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)N2CCC(CC2)NC(C)=O)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)N2CCC(N)CC2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)OCC(C)C)CC(C)(C)CC1)C(C)C |c:9|
COC(=O)N(CC1=C(CCC(C)(C)C1)c1cc(ccc1OC)C(C)C)Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F |t:6|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cccs2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)N2CCOCC2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(OCC(O)=O)cn2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(cn2)-c2cnn(C)c2)CCCC1)C(C)C |c:9|
COC(=O)COc1cnc(nc1)N(CC1=C(CCC(C)(C)C1)c1cc(ccc1OC)C(C)C)Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F |t:15|
COCCOc1cnc(nc1)N(CC1=C(CCC(C)(C)C1)c1cc(ccc1OC)C(C)C)Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F |t:14|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(Br)cn2)CC(C)(C)CC1)C(C)C |c:9|
COc1ccc(cc1C1=C(CN(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ncc(O)cn2)CC(C)(C)CC1)C(C)C |c:9|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)CC(=O)N[C@H]1C[C@@H](CC)N(C(=O)OCC)c3ccc(cc13)C(F)(F)F)C2(C)C |r,t:9|
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCCC(=O)N[C@H]4C[C@@H](CC)N(C(=O)OCC)c5ccc(cc45)C(F)(F)F)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O |r,t:15|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)CCC(=O)N[C@H]1C[C@@H](CC)N(C(=O)OCC)c3ccc(cc13)C(F)(F)F)C2(C)C |r,t:9|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(O)=O)[C@@]1(C)CC[C@H](OC(=O)CCCC(=O)N[C@H]1C[C@@H](CC)N(C(=O)OCC)c3ccc(cc13)C(F)(F)F)C2(C)C |r,t:9|
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CCC(=O)N[C@H]4C[C@@H](CC)N(C(=O)OCC)c5ccc(cc45)C(F)(F)F)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O |r,t:15|
[H][C@@]12CC(C)(C)CC[C@@]1(CC[C@]1(C)C2=CC[C@]2([H])[C@@]3(C)CC[C@H](OC(=O)CC(=O)N[C@H]4C[C@@H](CC)N(C(=O)OCC)c5ccc(cc45)C(F)(F)F)C(C)(C)[C@]3([H])CC[C@@]12C)C(O)=O |r,t:15|