1493 SMILES Strings for DCN1-like protein 1

Compound Name
SMILES String
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)C=C)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)\C=C\CN(C)C)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)CC1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)C1CCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2s1)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)C1=CCCN(C)C1)Cc1ccccc1 |r,t:27|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)CCl)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN(C)C)C1CCCCC1 |r|
CCN(CC)CC(=C)C(=O)NC[C@@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)CC)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCCCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)Cn1ccnc1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CC(F)(F)C1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCN(C)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCS(=O)(=O)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCN(CCO)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCC(F)(F)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C=C)Cc1ccncc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C=C)Cc1cccnc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNS(=O)(=O)C=C)Cc1cccnc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)Cc1cccnc1 |r|
CCC(=O)N[C@@H](Cc1cn2cc(Cl)ccc2n1)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C(=C)CN1CCOCC1)Cc1ccc(F)cc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C=C)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)CCl)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)/C=C/CN3CCOCC3)C4CCCCC4
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC1CCCCC1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)Nc1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NCc1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccc(Cl)cc1)c1ccc(Cl)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCc2ccccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CCc2ccccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCCc2ccccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CCCc2ccccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CCOc2ccccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2n1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1cc2ccccc2cn1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccn1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1cccnc1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1cccc(C)n1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc(C)cn1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccccc2n1C)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](CC(F)(F)F)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](Cc1cccs1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CN(C)C)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN1CCOCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@@H](N)Cc1ccc2ccccc2c1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCNC1CCN(C)CC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CCC(=O)N[C@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCNC1CCN(C)CC1)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](CN)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CN)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2cc(F)ccc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccccc2s1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2cc(Cl)ccc2s1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccccc2o1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2cc(Cl)ccc2o1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(Cl)cc2o1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(OC)cc2o1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2cc(Cl)ccc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2c(F)cccc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(F)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccccc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CNCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CNCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](c1cn(CCN)nn1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CNCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CNCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)N[C@@H]1CN(C)Cc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2cccc(Cl)c12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccc(Cl)cc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2cc(Cl)ccc12 |r|
CCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2c(Cl)cccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)[C@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)NC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)OC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2cc(Cl)ccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2cccc(Cl)c2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)NCCc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CNCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](CC1CCNCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](Cc1ccccn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCNCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12)C(C)(C)O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](Cc1cccnc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](Cc1ccncc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C[C@H]1CC[C@H](CN)CC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r,wU:20.21,25.27,wD:5.4,33.35,42.44,22.23,(-8.19,.95,;-6.86,1.72,;-5.53,.95,;-4.19,1.72,;-5.53,-.59,;-4.19,-1.36,;-4.19,-2.9,;-5.53,-3.67,;-5.69,-5.21,;-7.19,-5.53,;-7.96,-6.86,;-9.5,-6.86,;-10.27,-5.53,;-11.81,-5.53,;-9.5,-4.19,;-7.96,-4.19,;-6.93,-3.05,;-2.86,-.59,;-2.86,.95,;-1.52,-1.36,;-.19,-.59,;-.19,.95,;-.96,2.28,;-.19,3.61,;-.96,4.95,;-2.5,4.95,;-3.59,6.04,;-3.19,7.52,;-3.27,3.61,;-2.5,2.28,;1.14,-1.36,;1.14,-2.9,;2.48,-.59,;3.81,-1.36,;3.81,-2.9,;5.14,-3.67,;5.14,-5.21,;6.48,-5.98,;6.48,-7.52,;5.14,-.59,;5.14,.95,;6.48,-1.36,;7.81,-.59,;7.81,.95,;9.15,1.72,;10.48,.95,;10.48,-.59,;11.81,-1.36,;11.81,-2.9,;10.48,-3.67,;9.15,-2.9,;9.15,-1.36,)|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)C(C)C)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](C[C@H]1CC[C@H](CN)CC1)C(=O)N[C@@H]1CCOc2ccccc12 |r,wU:20.21,35.38,wD:5.4,30.32,43.46,32.34,(-9.38,3.51,;-7.84,3.51,;-7.07,2.18,;-7.84,.85,;-5.53,2.18,;-4.19,1.41,;-4.19,-.13,;-5.53,-.9,;-5.69,-2.43,;-7.19,-2.75,;-7.96,-4.09,;-9.5,-4.09,;-10.27,-2.75,;-11.81,-2.75,;-9.5,-1.42,;-7.96,-1.42,;-6.93,-.27,;-2.86,2.18,;-2.86,3.72,;-1.52,1.41,;-.19,2.18,;-.19,3.72,;1.14,4.49,;1.14,6.03,;-.19,6.8,;-1.52,6.03,;-1.52,4.49,;1.14,1.41,;1.14,-.13,;2.48,2.18,;3.81,1.41,;3.81,-.13,;4.58,-1.46,;3.81,-2.8,;4.58,-4.13,;6.12,-4.13,;6.89,-5.47,;6.12,-6.8,;6.89,-2.8,;6.12,-1.46,;5.14,2.18,;5.14,3.72,;6.48,1.41,;7.81,2.18,;7.81,3.72,;9.15,4.49,;10.48,3.72,;10.48,2.18,;11.81,1.41,;11.81,-.13,;10.48,-.9,;9.15,-.13,;9.15,1.41,)|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](C1CCNCC1)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CC1CCNCC1)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CC1CCNCC1)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CC1CCNCC1)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CC1CCN(C)CC1)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CC1CCN(C)CC1)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(C)cc2o1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2o1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(CC)cc2o1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2o1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCNCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C[C@H]1CC[C@H](CN)CC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r,wU:20.21,25.27,wD:5.4,33.35,42.44,22.23,(-8.19,.95,;-6.86,1.72,;-5.53,.95,;-4.19,1.72,;-5.53,-.59,;-4.19,-1.36,;-4.19,-2.9,;-5.53,-3.67,;-5.69,-5.21,;-7.19,-5.53,;-7.96,-6.86,;-9.5,-6.86,;-10.27,-5.53,;-11.81,-5.53,;-9.5,-4.19,;-7.96,-4.19,;-6.93,-3.05,;-2.86,-.59,;-2.86,.95,;-1.52,-1.36,;-.19,-.59,;-.19,.95,;-.96,2.28,;-.19,3.61,;-.96,4.95,;-2.5,4.95,;-3.59,6.04,;-3.19,7.52,;-3.27,3.61,;-2.5,2.28,;1.14,-1.36,;1.14,-2.9,;2.48,-.59,;3.81,-1.36,;3.81,-2.9,;5.14,-3.67,;5.14,-5.21,;6.48,-5.98,;6.48,-7.52,;5.14,-.59,;5.14,.95,;6.48,-1.36,;7.81,-.59,;7.81,.95,;9.15,1.72,;10.48,.95,;10.48,-.59,;11.81,-1.36,;11.81,-2.9,;10.48,-3.67,;9.15,-2.9,;9.15,-1.36,)|
CCC(=O)N[C@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C[C@H]1CC[C@H](CN)CC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r,wU:20.21,5.4,25.27,wD:33.35,42.44,22.23,(-9.38,1.11,;-7.84,1.11,;-7.07,-.23,;-7.84,-1.56,;-5.53,-.23,;-4.19,-1,;-4.19,-2.54,;-5.53,-3.31,;-5.69,-4.84,;-7.19,-5.16,;-7.96,-6.49,;-9.5,-6.49,;-10.27,-5.16,;-11.81,-5.16,;-9.5,-3.82,;-7.96,-3.82,;-6.93,-2.68,;-2.86,-.23,;-2.86,1.31,;-1.52,-1,;-.19,-.23,;-.19,1.31,;-1.28,2.4,;-.88,3.89,;-1.97,4.98,;-3.46,4.58,;-4.55,5.67,;-4.15,7.16,;-3.86,3.09,;-2.77,2,;1.14,-1,;1.14,-2.54,;2.48,-.23,;3.81,-1,;3.81,-2.54,;5.14,-3.31,;5.14,-4.85,;6.48,-5.62,;6.48,-7.16,;5.14,-.23,;5.14,1.31,;6.48,-1,;7.81,-.23,;7.81,1.31,;9.15,2.08,;10.48,1.31,;10.48,-.23,;11.81,-1,;11.81,-2.54,;10.48,-3.31,;9.15,-2.54,;9.15,-1,)|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](Cc1ccccn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](Cc1ccncc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](C1CCOCC1)C(=O)N[C@H](CCCCN)C(=O)N[C@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C[C@H]1CC[C@H](CN)CC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)N[C@@H]1CCOc2ccccc12 |r,wU:20.21,25.27,wD:33.35,44.46,5.4,22.23,(-9.38,1.75,;-7.84,1.75,;-7.07,.41,;-7.84,-.92,;-5.53,.41,;-4.19,-.36,;-4.19,-1.9,;-5.53,-2.67,;-5.69,-4.2,;-7.19,-4.52,;-7.96,-5.85,;-9.5,-5.85,;-10.27,-4.52,;-11.81,-4.52,;-9.5,-3.19,;-7.96,-3.19,;-6.93,-2.04,;-2.86,.41,;-2.86,1.95,;-1.52,-.36,;-.19,.41,;-.19,1.95,;-.96,3.29,;-.19,4.62,;-.96,5.95,;-2.5,5.95,;-3.27,7.29,;-4.81,7.29,;-3.27,4.62,;-2.5,3.29,;1.14,-.36,;1.14,-1.9,;2.48,.41,;3.81,-.36,;3.81,-1.9,;5.14,-2.67,;5.14,-4.21,;6.48,-4.98,;6.48,-6.52,;5.14,-7.29,;7.81,-7.29,;5.14,.41,;5.14,1.95,;6.48,-.36,;7.81,.41,;7.81,1.95,;9.15,2.72,;10.48,1.95,;10.48,.41,;11.81,-.36,;11.81,-1.9,;10.48,-2.67,;9.15,-1.9,;9.15,-.36,)|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C[C@H]1CC[C@H](CNC(=O)COCCOCCOCCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)CC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)N[C@@H]1CCOc2ccccc12 |r,wU:25.27,20.21,wD:22.23,5.4,61.65,72.76,47.48,55.56,50.52,(-9.38,-12.24,;-7.83,-12.24,;-7.07,-13.57,;-7.83,-14.9,;-5.53,-13.57,;-4.19,-14.34,;-4.19,-15.88,;-5.53,-16.65,;-5.69,-18.18,;-7.19,-18.5,;-7.96,-19.83,;-9.5,-19.83,;-10.27,-18.5,;-11.81,-18.5,;-9.5,-17.17,;-7.96,-17.17,;-6.93,-16.02,;-2.86,-13.57,;-2.86,-12.03,;-1.52,-14.34,;-.19,-13.57,;-.19,-12.03,;-.96,-10.7,;-.19,-9.36,;-.96,-8.03,;-2.5,-8.03,;-3.27,-6.69,;-4.81,-6.69,;-5.58,-5.36,;-7.12,-5.36,;-4.81,-4.03,;-5.58,-2.69,;-4.81,-1.36,;-5.58,-.03,;-4.81,1.31,;-5.58,2.64,;-4.81,3.97,;-5.58,5.31,;-4.81,6.64,;-5.58,7.98,;-4.81,9.31,;-5.58,10.64,;-7.12,10.64,;-4.81,11.98,;-5.58,13.31,;-4.81,14.64,;-5.58,15.98,;-6.91,16.75,;-8.42,17.07,;-8.58,18.6,;-7.17,19.23,;-6.4,20.56,;-4.9,20.24,;-3.75,21.27,;-4.74,18.71,;-6.14,18.08,;-3.27,-9.36,;-2.5,-10.7,;1.14,-14.34,;1.14,-15.88,;2.48,-13.57,;3.81,-14.34,;3.81,-15.88,;5.14,-16.65,;5.14,-18.19,;6.48,-18.96,;6.48,-20.5,;7.81,-21.27,;5.14,-21.27,;5.14,-13.57,;5.14,-12.03,;6.48,-14.34,;7.81,-13.57,;7.81,-12.03,;9.14,-11.26,;10.48,-12.03,;10.48,-13.57,;11.81,-14.34,;11.81,-15.88,;10.48,-16.65,;9.14,-15.88,;9.14,-14.34,)|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CNCc2ccccc12 |r|
CCC(=O)N[C@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CNCc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN(C)C)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CN(C)CCCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1nc2ccc(Cl)cc2s1)C1CCCC1)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccc(Cl)c1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1cn2cc(Cl)ccc2n1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CNC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1cn2cc(ccc2n1)C(C)C)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CCC(=O)N[C@@H](Cc1cn2cc(Cl)ccc2n1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CCOc2ccccc12 |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(Cl)cc2s1)NC(=O)CC |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(C)cc2s1)NC(=O)CC |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(CC)cc2s1)NC(=O)CC |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CN)C1CCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CN)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CN)CC1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CN)C1CCOCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C)CN |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)c(Cl)c2s1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Br)cc2s1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)(C)C)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCCC1)C(=O)NCCCCCN(C)C |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)C(C)C)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccc(F)cc1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)n(n1)-c1ccccc1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)n(n1)C(C)C)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccccc1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccc(Cl)cc1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(CC)c(s1)-c1ccccc1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)[C@H](C)CN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)[C@@H](C)CN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@H](CNC(=O)CCN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccc(Cl)c1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccccc1Cl)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccc(cc1)C#N)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccc(cc1)[N+]([O-])=O)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccccn1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccnc1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1ccncc1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccc(c1)C#N)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccc(Br)c1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccc(c1)C(F)(F)F)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccc(F)c1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)NCCN |r|
COCCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)NCCN |r|
NCCNC(=O)[C@H](Cc1nc2ccc(Cl)cc2s1)NC(=O)CCOc1ccccc1 |r|
NCCNC(=O)[C@H](Cc1nc2ccc(Cl)cc2s1)NC(=O)CCOCc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1cn(cn1)-c1cccc(Cl)c1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)CCN1CCOCC1)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)NCc1ccccn1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)NCc1cccnc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)NCc1ccncc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)NC(c1ccccn1)c1ccccn1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C1=CN(CCN)NN1)c1ccccc1 |r,t:43|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](c1cn(CCO)nn1)c1ccccc1 |r|
CCC(=O)N[C@@H](Cc1cn2cc(Cl)ccc2n1)C(=O)N[C@H](CN)Cc1ccccc1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CN)C1CCCCC1 |r|
CCC(=O)N[C@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CN)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)CCN3CCOCC3)C4CCCCC4
CCC(=O)N[C@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CNC(=O)CCN1CCOCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(Cl)cc2s1)C(=O)NCc1ccccn1 |r|
CCC(=O)N[C@H](CNC(=O)c1ccccc1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)Cc1ccccc1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)C1CCCCC1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)CC1CCCC1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)c1ccccn1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)Cc1ccccn1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)Nc1ccccc1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CN(Cc1ccccc1)Cc1ccccc1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)[C@@H](N)C1CCCC1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)[C@H](N)C1CCCC1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCCCC1)Cc1nc2ccc(Cl)cc2s1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CN1CCOCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CO)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CN(C)C)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)CN1CCOCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)CCCN1CCOCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(C)CC1)C1CCCCC1 |r|
CCC(=O)N[C@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CNC(=O)C1CCN(C)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)c1ccncc1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNc1ccncn1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](COCCN1CCOCC1)C1CCCCC1 |r|
CC(C)c1ccc2nc(C[C@H](NC(=O)C3CC3)C(=O)N[C@H](CN)C3CCCCC3)sc2c1 |r|
CC(C)C(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CN)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc(C)c(s1)-c1cccc(Cl)c1)C(=O)N[C@H](CN)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)NCCN |r|
CC(C)C(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)NCCN |r|
CC(C)c1ccc2nc(C[C@H](NC(=O)C3CC3)C(=O)NCCN)sc2c1 |r|
CC(C)CC(C)C(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)NCCN |r,w:4.4|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCN(CC1)C(=O)OC(C)(C)C)C(=O)NCCN1CCOCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCNCC1)C(=O)NCCN1CCOCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCNCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)NC1CCNCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(CC1)C1COC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)NC(CSc1nncn1C)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C12CCN(CC1)CC2)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)c1nnc[nH]1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)c1ncc[nH]1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)c1cn(C)cn1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)c1c[nH]cn1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CNC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CN(C)C1)C1CCCCC1 |r|
CCN1CCC(CC1)C(=O)NC[C@@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)CC)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(CC1)C(C)C)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(CCO)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](Cn1cc(CN)nn1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](Cn1cc(CO)nn1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNS(=O)(=O)C1CCNCC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(CCF)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(CCOCCOCCOCCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(CCOCCOCCOCCNC(=O)c2ccc3c(c2)C(=O)OC32c3ccc(O)cc3Oc3cc(O)ccc23)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)NC1CCN(C)CC1)C1CCCCC1 |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNS(=O)(=O)C1CCN(C)CC1)C1CCCCC1 |r|
CCC(=O)N[C@H](CN)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCCCC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCC(C)(C)CC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCC(F)(F)CC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCOCC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCCC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCCCCC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(N)CCCCCCC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1(CN)CCCCC1)Cc1nc2ccc(cc2s1)C(C)C |r|
CCC(=O)N[C@H](CNC(=O)C1CCCCN1)Cc1nc2ccc(cc2s1)C(C)C |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccccc2s1)NC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(Cl)cc2s1)NC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@@H](N)Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)C1CC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)NC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)OC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CC(F)(F)F)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCOCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCNCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C1CCCCC1)C(=O)N[C@@H](CCCCN)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(C)=O)C(=O)N[C@@H](CCCCN)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(C)=O)C(N)=O |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(C)=O |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)CC |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1nc2cc(Cl)ccc2s1)NC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](C)CN |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC=O |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@@H](N)Cc1nc2ccc(cc2s1)C(C)C |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)C(C)C |r|
CCCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CN)[C@@H](C)CC |r|
CC[C@H](C)[C@@H](CN)NC(=O)[C@H](Cc1nc2ccc(cc2s1)C(C)C)NC(=O)NC |r|
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@H](CNC(=O)C1CCN(CC1)C1CCOCC1)C1CCCCC1 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
C=CS(=O)(=O)N(C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CN1CCC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C=C/C(=O)OC)nn(-c3ccccc3)c21
C=C(CC(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](CC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC)C(=O)OC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(C)CC#N)nn(-c3ccccc3)c21
C/C=C/S(=O)(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C(C)(C)C#N)nn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)N[C@H](C)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@H](O)CNC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CCNC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)C#CCN3CCOCC3)nn(-c3ccccc3)c21
C=C(CN1C[C@@H]2C[C@H]1CO2)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c([C@@H](C)NC#N)nn(-c3ccccc3)c21
C/C=C(CN1CCOCC1)/C(=O)NCc3nn(c2ccccc2)c6c3[C@H](c4ccc(F)cc4)[C@H](NC(=O)c5cccc(C(F)(F)F)c5)C(=O)N6CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C=C/C(=O)NCCO)nn(-c3ccccc3)c21
C=C(C)C(=O)N[C@@H](C)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CC(=O)OC)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CN(C)C)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C#CCN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(CN(C)C#N)nn(-c3ccccc3)c21
C=C(Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC)C(=O)O
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C3(C#N)CCOCC3)nn(-c3ccccc3)c21
C/C=C/C(=O)N[C@@H](C)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)NCCCO)nn(-c3ccccc3)c21
C=C(CN1CCC(C)(O)C1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(C)C(=O)Nc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C/C=C(CN1CCOCC1)/C(=O)NCc3nn(c2ccccc2)c6c3[C@@H](c4ccc(F)cc4)[C@H](NC(=O)c5cccc(C(F)(F)F)c5)C(=O)N6CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C3=CCCN(C)C3)nn(-c3ccccc3)c21
C=CC(=O)N(C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C(=O)[C@H](C)Cl)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)NC(C)(C)C#N)nn(-c3ccccc3)c21
C=C(CN1CCC(F)(F)C1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C(=O)[C@H](C)Cl)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)C(c2ccc(F)cc2)c2c(C(=O)N3CCC[C@H]3C#N)nn(-c3ccccc3)c21
C=C(C(=O)OCC)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)NCCO)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C3(C#N)CC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)NC)nn(-c3ccccc3)c21
CCN6C(=O)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)[C@@H](c2ccc(F)cc2)c5c(/C=C/3CCC(=O)N3)nn(c4ccccc4)c56
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)N(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(C)(C)N(C)C#N)nn(-c3ccccc3)c21
CCN5C(=O)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)[C@@H](c2ccc(F)cc2)c4c(CC/C=C/C(=O)NC)nn(c3ccccc3)c45
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@@H](C)N(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C=C/C(=O)OC(C)(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(N)=O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)C3(C#N)CC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CC/C=C/C(=O)N(C)C)nn(-c3ccccc3)c21
C=C(CN1CCC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CN1CC2CCC(C1)O2)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CC#CC(=O)Nc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C3(N(C)C#N)CC3)nn(-c3ccccc3)c21
C=C(C(=O)O)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(C)S(=O)(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C(=O)/C=C/CN3CCOCC3)nn(-c3ccccc3)c21
C=C(CN1CC2CC(C1)O2)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CN1CCOCC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C=C/C(=O)O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CC[C@@H](C#N)C3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C#N)CCF)nn(-c3ccccc3)c21
C/C=C/C(=O)Nc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)C(C)(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C=C/C(N)=O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)C3=CCCC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)C3(C#N)CCOCC3)nn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C#CCN3CCOCC3)nn(-c3ccccc3)c21
CCN5C(=O)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)[C@@H](c2ccc(F)cc2)c4c(CC/C=C/C(=O)N(C)C)nn(c3ccccc3)c45
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(/C=C3/CCC(=O)N3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(CNC(=O)C3=C(C(=O)OC)CCC3)nn(-c3ccccc3)c21
C=C(CN1CCC(F)(F)C1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@@H](C)NC#N)nn(-c3ccccc3)c21
C=CS(=O)(=O)N[C@H](C)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CN1CCOCC1)C(=O)Nc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(C3(N(C)C#N)CC3)nn(-c3ccccc3)c21
C=C(C(=O)O)c1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC)C(=O)OC(C)(C)C
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c([C@@H](C)N(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)CC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)NCCC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(C3(NC#N)CC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)[C@H](C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(CNC(=O)C3=CCN(C)C3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C3(NC#N)CC3)nn(-c3ccccc3)c21
C=C(C(=O)NCc1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC)C(C)N1CCOCC1
C=C(C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC)C(C)N1CCOCC1
CC#CC(=O)N(C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CC/C=C/C(=O)NC)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)C#CCN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCC[C@@H]3C#N)nn(-c3ccccc3)c21
C=C(CN1CC(F)(F)C1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNCC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(CNC(=O)C3=C(C(=O)OC)CC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(CNC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)NCCCN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C3(C#N)COC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)[C@@H](C)Cl)nn(-c3ccccc3)c21
C=C(CN(C)C1COC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CC(=O)OC)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN5C(=O)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)[C@H](c2ccc(F)cc2)c4c(CNC(=O)/C=C(C)/C(=O)OC)nn(c3ccccc3)c45
C=C(Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC)C(N)=O
C=C(CO)C(=O)NCc1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C(=O)/C=C/C(=O)OC)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C(C)=C/C(=O)OC)nn(-c3ccccc3)c21
C=C(COC)C(=O)NCc1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN3CC=CS3(=O)=O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(CN(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)NC3(C#N)CC3)nn(-c3ccccc3)c21
C=C(COC)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C34CC3C4)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C#N)nn(-c3ccccc3)c21
C=C(CO)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C(=O)/C=C/CN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)NCCN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C3=C(C(=O)OC)CC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)[C@@H](F)Cl)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCCC[C@@H]3C#N)nn(-c3ccccc3)c21
C=CC(=O)Nc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C/C=C/C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CC/C=C/C(N)=O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)/C=C/C(F)(F)F)nn(-c3ccccc3)c21
CCN5C(=O)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)[C@@H](c2ccc(F)cc2)c4c(CC/C=C/C(=O)O)nn(c3ccccc3)c45
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC/C=C/C(=O)OC)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CC/C=C/C(=O)OC)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@@H](O)CNC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C/C=C/C(=O)OC)nn(-c3ccccc3)c21
C=C(CC(=O)NCc1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC)C(=O)OC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(CN(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CC/C=C/C(=O)O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)C3=C(C(=O)OC)CCC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)/C=C/C(=O)OC)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CC[C@H](C#N)C3)nn(-c3ccccc3)c21
C=C(CN1CC2(COC2)C1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
C=C(CN1CCC1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(CN(C)C(=O)/C=C/C(=O)OC)nn(-c3ccccc3)c21
CCN5C(=O)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)[C@@H](c2ccc(F)cc2)c4c(CC/C=C/C(N)=O)nn(c3ccccc3)c45
C=CC(=O)N[C@@H](C)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(C)(C)NC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C(=O)[C@H](F)Cl)nn(-c3ccccc3)c21
C=C(C(=O)OC(C)(C)C)[C@@H](O)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)CC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)NCC#N)nn(-c3ccccc3)c21
C=C(CN1CC2(COC2)C1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN5C(=O)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)[C@@H](c2ccc(F)cc2)c4c(CNC(=O)/C=C(C)/C(=O)OC)nn(c3ccccc3)c45
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CCN(C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)C3=CCC3)nn(-c3ccccc3)c21
C=C(C(=O)O)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C=C/C(=O)NCCN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)/C(C)=C/C(=O)OC)nn(-c3ccccc3)c21
C=C(C)C(=O)N(C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N[C@H](C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CNC(=O)[C@@H](C)C#N)nn(-c3ccccc3)c21
C/C=C(C)/S(=O)(=O)NCc2nn(c1ccccc1)c5c2[C@H](c3ccc(F)cc3)[C@H](NC(=O)c4cccc(C(F)(F)F)c4)C(=O)N5CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@@H](C)N(C#N)COP(=O)(O)O)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NC(=O)CCl)nn(-c3ccccc3)c21
C[C@@H](NC#N)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CCOP(=O)(O)O
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(NS(=O)(=O)CCl)nn(-c3ccccc3)c21
N#CN(CCCCN(C)C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@@H](C)N(C#N)CCCN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CC(F)(F)C[C@H]3C#N)nn(-c3ccccc3)c21
N#CN(CCCN(C)C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
N#CN(CCCO)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
N#CN(CCO)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)NCC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(C(=O)N[C@@H](C)C#N)nn(-c3ccccc3)c21
N#CN(CCCCN(C)C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(CN(C)C/C=C/C(=O)OC)nn(-c3ccccc3)c21
COC(=O)/C=C/CN(C)Cc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC(C)C
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCCC[C@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(CC#N)CCCN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@@H](CN(C)C)NC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3C[C@H](F)C[C@H]3C#N)nn(-c3ccccc3)c21
C[C@@H](NC#N)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CCO
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CC[C@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCOC[C@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCC[C@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c([C@@H](CF)NC#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCNC[C@@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCNC[C@@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(C)CC#N)nn(-c3ccccc3)c21
CCN(CC#N)C(=O)c1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(CC#N)C3CC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)C(c2ccc(F)cc2)c2c(C(=O)N(CC#N)C3COC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(CC#N)CCO)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(CC#N)CC(=O)OC)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(CC#N)CCC(=O)OC)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(C)[C@H](C)C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(C)[C@@H](C#N)CCO)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(C)[C@@H](C#N)C3COC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCC[C@H]3C#N)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCC[C@H]3C#N)nn(-c3cccc(OCCCN4CC5(COC5)C4)c3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(C)[C@@H](C#N)C3COC3)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCOC[C@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(C(=O)N3CCOCC3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CCOC[C@@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(CC(=O)NCC#N)nn(-c3ccccc3)c21
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C=C(CN1CC(O)C1)C(=O)NCc1nn(-c2ccccc2)c2c1[C@H](c1ccc(F)cc1)[C@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CC
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CCN1C(=O)[C@@H](NC(=O)C2CCC(F)(F)CC2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2ccc(C3CCN(C)CC3)cc2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N(C)[C@@H](C#N)CCN(C)C3COC3)nn(C3CCOCC3)c21
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CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(C(=O)N3CCS(=O)(=O)C[C@H]3C#N)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(C(=O)N3CC[C@H]3C#N)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CS(=O)(=O)C[C@H]3C#N)nn(C3CCOCC3)c21
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CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)cc2)c2c(C(=O)N3CC[C@H](F)[C@H]3C#N)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2ccc3c(c2)OCCO3)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCC(=O)N[C@@H]1C(=O)N(CC)c2c(c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn2C2CCOCC2)[C@@H]1C1CC1
CCN1C(=O)[C@@H](NC(=O)c2c(Cl)ccc(OC)c2F)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C#N)c2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)C(C2CC2)C2CC2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)CC[C@@H]3C)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)C23CC(C(F)(F)F)(C2)C3)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(C(=O)N(CC#N)C3CC3)nn(C3CC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](C2CC2)c2c(C(=O)N3[C@@H](C#N)C[C@@H]4C[C@@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)cc2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn([C@@H]3CCOC3)c21
CCN1C(=O)[C@@H](NC(=O)c2ccc3nn[nH]c3c2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2ccc3snnc3c2)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc3ccoc23)[C@@H](C2CC2)c2c(C(=O)N3[C@H](C#N)C[C@H]4C[C@H]43)nn(C3CCOCC3)c21
C=C(CN1CCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN(C)C1COC1)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=CS(=O)(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2(COC2)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2CC1CO2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1C2COCC1C2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCC(C)(O)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC(F)(F)C1)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2(CCOC2)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2CC1C2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC(F)(F)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)Nc1ccccc1[C@H]1c2cnn(-c3ccccc3)c2N(CC)C(=O)[C@@H]1NC(=O)c1cccc(C(F)(F)F)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)[C@H](C)Cl)c2)c2c(C)nn(-c3ccccc3)c21
C=C(C)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)[C@H](F)Cl)c2)c2c(C)nn(-c3ccccc3)c21
CC#CC(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C3=CCCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2N2CC=CC2=O)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC#N)c2)c2c(C)nn(-c3ccccc3)c21
C/C=C/C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C3=CCCC3)c2)c2c(C)nn(-c3ccccc3)c21
C=CC(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2NC(C)=O)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C=C/C(F)(F)F)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(N3CC=CC3=O)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC#N)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CN(C)C#N)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CNC#N)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccc(F)c(NC(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C3=CCCN(C)C3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)C3=C(C(=O)OC)CC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C#CCN3CCOCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cncc(NC(=O)C3=CCC3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)C3=CCN(C)C3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C=C/CN(C)C)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(N(C)C(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CN(C)C#N)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CC(=O)OC)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C(Cl)Cl)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCC(F)(F)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2NC(=O)C23CC2C3)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C(C#N)=C/C(C)C)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C=C/CN3CCOCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)[C@H](C)Cl)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CN(C)C#N)c2cnn(-c3ccccc3)c21
C=C(CC(=O)OC)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2NC(=O)CCl)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C3=CCN(C)C3)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CCO)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)/C=C/CN(C)C)c2F)c2cnn(-c3ccccc3)c21
C=C(CC(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1)C(=O)OC
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)C3=CCCN(C)C3)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCC1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCC(F)(F)C1)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN(C)CC1COC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2(CCO2)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2(COC2)C1)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CNC(=O)/C=C/C(=O)OC)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C(C#N)=C/C3CC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C(C#N)=C/C(C)(C)C)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)C3=CCC3)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CO)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2NC(=O)[C@H](C)Br)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)/C=C(C)C(=O)OC)c2)c2cnn(-c3ccccc3)c21
C=CC(=O)N(C)c1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C=C/C(F)(F)F)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CO)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=CC(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C3=CCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cc(NC(=O)/C=C/CN(C)C)ccc2F)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C34CC3C4)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCOCC1)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)N(C)c1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cc(F)cc(NC(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccnn2C(F)(F)F)c1
C=C(CO)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(C)S(=O)(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2-n2sccc2=O)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2N(C)C#N)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(N(C)C(=O)C3=CCC3)c2)c2cnn(-c3ccccc3)c21
Cc1nn(-c2ccccc2)c2c1[C@H](c1cccc(NC(=O)C3=CCC3)c1)[C@@H](NC(=O)c1cccc(C(F)(F)F)c1)C(=O)N2CCO
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C3=CCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)/C(C)=C/C(=O)OC)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CC(F)(F)C1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=CC(=O)N(C)c1ccccc1[C@H]1c2cnn(-c3ccccc3)c2N(CC)C(=O)[C@@H]1NC(=O)c1cccc(C(F)(F)F)c1
CC#CC(=O)N(C)c1ccccc1[C@H]1c2cnn(-c3ccccc3)c2N(CC)C(=O)[C@@H]1NC(=O)c1cccc(C(F)(F)F)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(N(C)C(=O)/C=C/C(F)(F)F)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C(F)Cl)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CNC(=O)C2=CCC2)c2cnn(-c3ccccc3)c21
C=C(CN1CCC(F)(F)C1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)CC#N)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CN(C)C#N)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CNC(=O)C(F)Cl)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(CNC(=O)C3=CCCN(C)C3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cc(NC(=O)/C=C/CN(C)C)ccc2F)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C3=C(C(=O)OC)CCC3)c2)c2cnn(-c3ccccc3)c21
C=C(CC(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1)C(=O)OC
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2NC(=O)CCl)c2c(C)nn(-c3ccccc3)c21
C=CC(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C(C)Cl)c2)c2cnn(-c3ccccc3)c21
C=CC(=O)NCc1ccccc1[C@@H]1c2cnn(-c3ccccc3)c2N(CC)C(=O)[C@H]1NC(=O)c1cccc(C(F)(F)F)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CNC(=O)C(C)Cl)c2cnn(-c3ccccc3)c21
C/C=C(CN1CCOCC1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(CNC(=O)/C=C(C)C(=O)OC)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)C3=C(C(=O)OC)CCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(CNC(=O)C3=C(C(=O)OC)CC3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(CNC(=O)C3=C(C(=O)OC)CCC3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CNC(=O)/C=C/CN(C)C)c2cnn(-c3ccccc3)c21
C=C(CC(=O)OC)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccccc2NC#N)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C3CCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(C)=O)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(CNC(=O)/C(C)=C/C(=O)OC)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C3=CCC3)c2)c2cnn(-c3ccccc3)c21
C/C=C(/C)S(=O)(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(CNC(=O)C3=CCN(C)C3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2ccc(F)c(NC(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(N3CC=CS3(=O)=O)c2)c2c(C)nn(-c3ccccc3)c21
C/C=C/S(=O)(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C#CCN(C)C)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C#CCN(C)C)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(CN1CC2CCC(C1)O2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCC1)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC#N)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C#CCN3CCOCC3)c2)c2c(C)nn(-c3ccccc3)c21
C=C(F)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C=C/C(=O)OC)c2)c2c(C)nn(-c3ccccc3)c21
C/C=C(CN1CCOCC1)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)/C=C/C(=O)OC)c2)c2cnn(-c3ccccc3)c21
C=C(CN1C[C@@H]2C[C@H]1CO2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)/C(C)=C/C(=O)OC)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CN(C)C)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CCO)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)C3=CCN(C)C3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2ccccc2CNC#N)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)[C@H](F)Cl)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cc(F)cc(NC(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
C/C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)NCc1ccccc1[C@@H]1c2cnn(-c3ccccc3)c2N(CC)C(=O)[C@H]1NC(=O)c1cccc(C(F)(F)F)c1
C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C3=C(C(=O)OC)CC3)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CC2(COC2)C1)C(=O)NCc1cccc([C@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)/C=C(C)C(=O)OC)c2)c2c(C)nn(-c3ccccc3)c21
C=C(COC)C(=O)Nc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CC#CC(=O)Nc1ccccc1[C@H]1c2cnn(-c3ccccc3)c2N(CC)C(=O)[C@@H]1NC(=O)c1cccc(C(F)(F)F)c1
C=C(CN1C[C@@H]2C[C@H]1CO2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2(COC2)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C=C/CN(C)C)c2)c2c(CO)nn(-c3ccccc3)c21
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(NC(=O)/C=C/CN(C)C)c2)c2c(CN(C)C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(NC(=O)/C=C/CN(C)C)n2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)n1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)C(C)N(C)C1COC1
C=C(CN1CCN(C2COC2)CC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2(COC2)C1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)C(C)N1CC2(COC2)C1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)C3=CCN(C)C3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1CC=C(C(=O)Nc2cccc([C@@H]3c4c(C)nn(-c5ccccc5)c4N(CC)C(=O)[C@H]3NC(=O)c3nccc(C(F)(F)F)n3)c2)C1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)C3=CCN(C4COC4)C3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1CC=C(C(=O)Nc2cccc([C@@H]3c4c(C)nn(-c5ccccc5)c4N(CC)C(=O)[C@H]3NC(=O)c3ccn(C(F)(F)F)n3)c2)C1
C=C(CN1CCC(F)(F)C1)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)Nc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(CNC(=O)C(COC)CN3CCC(F)(F)C3)c2)c2cnn(-c3ccccc3)c21
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1)C(C)(C)N(C)C1COC1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1
C/C=C(CN1CC2(COC2)C1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2CC1CO2)C(=O)NCc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CN(C)C/C=C/C(=O)OC(C)(C)C)c2)c2cnn(-c3ccccc3)c21
C=C(CN(C)C1COC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1)C(C)N1CC2CC(C1)O2
C/C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(CN1CC2(COC2)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C3=CCN(C)C3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)/C=C/C(=O)N(C)C)c2)c2c(C)nn(-c3ccccc3)c21
C=C(CN1CCC12COC2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCC12COC2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C/C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(C(=O)N3CCC[C@H]3C#N)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(C(=O)N3CCC[C@@H]3C#N)c2)c2cnn(-c3ccccc3)c21
C/C=C(CN1CCC12COC2)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2CC(C1)O2)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(CN(C)C1COC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CN(C)C/C=C/C(=O)N3CCCC3)c2)c2cnn(-c3ccccc3)c21
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)C(C)N1CCC12COC2
C/C=C(/CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2CC(C1)O2)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2ccccc2/C=C/C#N)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2ccccc2/C=CC#N)c2cnn(-c3ccccc3)c21
C=C(CN1CC(F)(F)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)/C=C/C(=O)N3CCCC3)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(CN3CC=CS3(=O)=O)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)/C=C/CN(C)C)n2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccnn2C)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)F)c2)c1)C(C)N(C)C1COC1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C)n2)c1)C(C)N(C)C1COC1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)C3=CCC3)n2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C=C(CN1CCOCC1)C(=O)N[C@H](C)c1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc3c2CN(C#N)C3)c2cnn(-c3ccccc3)c21
C=C(CN1CC2(COC2)C1)C(=O)NCc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C/C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1)C(C)N1CC2CC(C1)O2
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1)C(C)N1CC2CC(C1)O2
C/C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C=C(CN1C2CCC1COC2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2CC(C1)O2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC(O)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2CCC(C1)O2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2CCC1CO2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2CC1CO2)C(=O)NCc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCOCC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1)C(C)N1CCOCC1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(CC(F)(F)F)n2)c1
C=C(CN1CCOCC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCOCC1)C(=O)N[C@@H](C)c1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)[C@@H](C)N(C)C1COC1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)N(C)c1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1
C/C=C(CN1CC2(COC2)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(CN1CCC1)C(=O)NCc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2(COC2)C1)C(=O)NCc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1)C(C)N(C)C1COC1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC/C=C/C(=O)OC(C)(C)C)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC/C=C/C(=O)N3CCCC3)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)F)n2)c1
C/C=C(CN1CCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)C(C)N1CCN(C2COC2)CC1
C=C(Cn1ccnc1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1)C(C)N(C)C1COC1
C/C=C(CN1CCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2CC(C1)O2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1)C(C)N1CCN(C2COC2)CC1
C=C(CN(C)C1COC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cncc(NC(=O)C3=CCC3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cncc(NC(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
C/C=C(CN1CC2(COC2)C1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C/C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2ccn(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)C3=CCN(C)C3)c2)c2cnn(-c3ccccc3)c21
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)C(C)N1CC2CC(C1)O2
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1)C(C)N1CCC12COC2
C/C=C(CN1CCOCC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1)C(C)N(C)C1COC1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(CNC(=O)C(C)C(C)N3CCC3)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cncc(NC(=O)/C=C/CN(C)C)c2)c2cnn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(C(=O)N3C[C@@H](F)C[C@H]3C#N)c2)c2cnn(-c3ccccc3)c21
C=C(Cn1cc(F)cn1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCC12COC2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)n1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(CCF)n2)c1)C(C)N(C)C1COC1
CCC(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C/C=C(CN1CC2CC(C1)O2)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CN(C)C/C=C/C(=O)N(C)C)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(CC#N)n2)c1
C/C=C(CN1CCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1)C(C)N(C)C1COC1
C=C(C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1)C(C)N1CCC12COC2
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1)C(C)N1CCC12COC2
C=C(CN(C)C1COC1)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2CC(C1)O2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CC2CCC(C1)O2)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC(=O)C3=CCN(C)C3)n2)c2cnn(-c3ccccc3)c21
C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(C(=O)N3C[C@H](F)C[C@H]3C#N)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(CC)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1)C(C(C)C)N(C)C1COC1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)n1
C=C(C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1)C(C)N(C)C1COC1
C=C(CN1CCN(C2COC2)CC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(CCF)n2)c1
CCC(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)/C=C/C(=O)OC(C)(C)C)c2)c2c(C)nn(-c3ccccc3)c21
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(CNC(=O)C(COC)CN3CCC(F)(F)C3)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CC(C)(O)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@@H](c2cccc(CNC(=O)C3=CCN(C)C3)c2)c2c(C)nn(-c3ccccc3)c21
C/C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C=C(CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(CC(F)F)n2)c1
C/C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1
C=C(CN1CCN(C2COC2)CC1)C(=O)N[C@H](C)c1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(CN1CCC1)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(CN1CCC(F)(F)C1)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(/CN1CCN(C2COC2)CC1)C(=O)N(C)c1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2csc(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(C(=O)N(C)CC#N)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCC12COC2)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2cccc(C(F)(F)F)c2)[C@H](c2cccc(CNC/C=C/C(=O)N(C)C)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCC12COC2)C(=O)N(C)Cc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C=C(CN1CCC1)C(=O)NCc1cccc([C@H]2c3c(C)nn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
C=C(CN1CC2(CCC2O)C1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2cccc(C(F)(F)F)c2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(NC(=O)C3=CCN(C)C3)n2)c2cnn(-c3ccccc3)c21
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)C(C)N1CC2(COC2)C1
C=C(CN(C)C1COC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
CCN1C(=O)[C@@H](NC(=O)c2nccc(C(F)(F)F)n2)[C@H](c2cccc(C(=O)N3CC(F)(F)C[C@H]3C#N)c2)c2cnn(-c3ccccc3)c21
C=C(CN1CCN(C2COC2)CC1)C(=O)N[C@@H](C)c1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(/CN1CCOCC1)C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C3CC3)n2)c1
C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)[C@H](C)N(C)C1COC1
C/C=C(CN1CCN(C2COC2)CC1)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1
C/C=C(CN(C)C1COC1)C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1
C/C=C(/C(=O)Nc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2nccc(C(F)(F)F)n2)c1)C(C)N1CCC1
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(C)c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(F)c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(Cl)c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(cc1)C(F)(F)F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(Cl)cc1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(Br)cc1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(C)cc1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(cc1)C(C)C
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(cc1)C(C)(C)C
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(Cl)c(c1)[N+]([O-])=O
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(F)c(F)c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(C#N)c(c1)C(F)(F)F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(F)c(c1)C(F)(F)F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(c1)C(F)(F)F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(ccc1F)C(F)(F)F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(Cl)ccc1F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(Br)cc1C
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc2ncsc2c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc2CCCc2c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc2ccccc2c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc2ncccc2c1
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(c1)C(F)(F)F
Fc1cc(NC(=O)N(Cc2ccccc2)C2CCN(CCCc3ccccc3)CC2)cc(c1)C(F)(F)F
Cn1cncc1CN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(c1)C(F)(F)F
Cc1ccc(CN2CCC(CC2)N(Cc2ccccc2)C(=O)Nc2cc(F)cc(c2)C(F)(F)F)o1
Fc1cc(NC(=O)N(Cc2ccccc2)C2CCN(CC3CCOC3)CC2)cc(c1)C(F)(F)F
COc1cccc(CN2CCC(CC2)N(Cc2ccccc2)C(=O)Nc2cc(F)cc(c2)C(F)(F)F)c1
Fc1cc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3ccncc3)CC2)cc(c1)C(F)(F)F
Fc1cc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3nc4ccccc4s3)CC2)cc(c1)C(F)(F)F
Fc1cc(NC(=O)N(Cc2ccccc2)C2CCN(C\C=C\c3ccccc3)CC2)cc(c1)C(F)(F)F
Fc1cc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3ccc(Cc4ccccc4)cc3)CC2)cc(c1)C(F)(F)F
Cn1ccc2cc(CN3CCC(CC3)N(Cc3ccccc3)C(=O)Nc3cc(F)cc(c3)C(F)(F)F)ccc12
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(Cl)c1
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)[N+]([O-])=O
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C#N
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(F)c1
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1F)C(F)(F)F
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(F)c(c1)C(F)(F)F
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(F)c(Cl)c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(C)C
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(I)cc1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(C)c(F)c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(Cl)c1
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(nc1C)C(F)(F)F
CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc2OCOc2c1
CSC(C)CCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(c1)C(F)(F)F
Cn1ccnc1CN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(c1)C(F)(F)F
COc1ccccc1CN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cc(F)cc(c1)C(F)(F)F
Fc1cc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3cccc(Oc4ccccc4)c3)CC2)cc(c1)C(F)(F)F
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(F)c1
CCCCN1CCC(CC1)N(Cc2ccccc2)C(=O)Nc3ccc(c(c3)Cl)Cl
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1ccc(C)c(Cl)c1
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)C1CC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CCCC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CCSC)NC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CCSC)NC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
c1ccc(cc1)CN2CCC(CC2)NC(=O)Nc3cccc(c3)C(F)(F)F
Fc1ccc(CN2CCC(CC2)NC(=O)Nc2cccc(c2)C(F)(F)F)cc1
CCCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3cc[nH]n3)CC2)c1
FC(F)(F)CCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCCS(=O)(=O)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3ccc4OCOc4c3)CC2)c1
Cc1cccc(CN2CCC(CC2)NC(=O)Nc2cccc(c2)C(F)(F)F)c1
Cc1ccccc1CN1CCC(CC1)NC(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)NC2CCN(Cc3cccc(Cl)c3)CC2)c1
Fc1cccc(CN2CCC(CC2)NC(=O)Nc2cccc(c2)C(F)(F)F)c1
FC(F)(F)c1cccc(NC(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1
FC(F)(F)c1cccc(NC(=O)NC2CCN(CC2)C(=O)c2ccccc2)c1
O=C(NC1CCN(Cc2ccccc2)CC1)Nc1ccccc1
COc1cccc(NC(=O)NC2CCN(Cc3ccccc3)CC2)c1
Ic1cccc(NC(=O)NC2CCN(Cc3ccccc3)CC2)c1
CSc1cccc(NC(=O)NC2CCN(Cc3ccccc3)CC2)c1
O=C(NC1CCN(Cc2ccccc2)CC1)Nc1cccc(c1)-n1cccc1
O=C(NC1CCN(Cc2ccccc2)CC1)Nc1cccc(CN2CCOCC2)c1
CCCN1CCC(CC1)N(CCC(C)C)C(=O)Nc1cccc(c1)C(F)(F)F
CCCN1CCC(CC1)N(CCOC)C(=O)Nc1cccc(c1)C(F)(F)F
CCCN1CCC(CC1)N(CC1CCCCC1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCN1CCC(CC1)N(Cc1cccnc1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCN1CCC(CC1)N(Cc1ccncc1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCN1CCC(CC1)N(Cc1cc(F)cc(c1)C(F)(F)F)C(=O)Nc1cccc(c1)C(F)(F)F
CCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCCCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(CC3CC3)CC2)c1
CC(C)(C)CN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
CC(C)(C)CCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(CC2)C(=O)C=C)c1
CCCS(=O)(=O)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3c[nH]cn3)CC2)c1
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3ccccc3)CC2)c1
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3cccnc3)CC2)c1
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3ccc4OCCOc4c3)CC2)c1
CCCCN1CCC(CC1)N(Cc1ccc2OCOc2c1)C(=O)Nc1cccc(c1)C(F)(F)F
CC(C)(C)N1CCC(CC1)N(Cc1ccc2OCOc2c1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
CCCN1CCC(CC1)N(Cc2ccc3c(c2)OCO3)C(=O)Nc4cccc(c4)C(F)(F)F
Cc1ccc(NC(=O)NC2CCN(Cc3ccccc3)CC2)cc1Cl
Cn1nccc1-c1cccc(NC(=O)NC2CCN(Cc3ccccc3)CC2)c1
CCCN1CCC(CC1)N(Cc1ccco1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)NC2CCN(Cc3ccccc3Cl)CC2)c1
Cc1ccc(CN2CCC(CC2)NC(=O)Nc2cccc(c2)C(F)(F)F)cc1
FS(F)(F)(F)(F)c1cccc(NC(=O)NC2CCN(Cc3ccccc3)CC2)c1
O=C(NC1CCN(Cc2ccccc2)CC1)Nc1ccc2OCOc2c1
CCCCN(C1CCN(CCC)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(CC3CCCC3)CC2)c1
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(Cc3nccs3)CC2)c1
Fc1ccc(CN2CCC(CC2)N(Cc2ccccc2)C(=O)Nc2cccc(c2)C(F)(F)F)cc1
CC(=O)O[C@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1cccc(c1)C(F)(F)F |r|
CCCN(C1CCN(CCC)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCNCC2)c1
CC(C)CCN1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
Fc1ccccc1CN1CCC(CC1)NC(=O)Nc1cccc(c1)C(F)(F)F
Cc1cccc(NC(=O)NC2CCN(Cc3ccccc3)CC2)c1
CCCN1CCC(CC1)N(CC(C)C)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)N(Cc2ccccc2)C2CCN(CC3CCCCC3)CC2)c1
CCOc1cc(CN2CCC(CC2)N(Cc2ccccc2)C(=O)Nc2cccc(c2)C(F)(F)F)cc(Cl)c1O
CCCC(=O)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(c1)C(F)(F)F
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nccn2C)c1C#N
Clc1cccc(c1)-c1nc(SCC#C)nc(Sc2nccs2)c1C#N
CN(C)CCn1nnnc1Sc1nc(SCC#C)nc(-c2ccc(C)cc2)c1C#N
CN(C)CCn1nnnc1Sc1nc(SCC#C)nc(-c2cccc(Cl)c2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nnnn2C)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2ccccc2)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2cccc(Cl)c2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(N2CCSCC2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2ccccn2)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2ccc3oc(=O)ccc3c2)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2c[nH]c3ccccc23)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2ccc[nH]2)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2ccc(Cl)cc2)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2ccc(Br)cc2)c1C#N
Cc1ccc(cc1)-c1nc(SCC#C)nc(Sc2nnnn2C)c1C#N
COc1cccc(c1)-c1nc(SCC#C)nc(Sc2nnnn2C)c1C#N
Cn1nnnc1Sc1nc(SCC#C)nc(-c2ccc(Cl)c(Cl)c2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(N2CCNCC2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(N2CCOCC2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Nc2cccc(c2)C(F)(F)F)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nnnn2CCN(C)C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nc[nH]n2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2ccc(N)s2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nnc(C)s2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nncs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nc(C)c(C)s2)c1C#N
Clc1ccc(cc1)-c1nc(SCC#C)nc(Sc2nccs2)c1C#N
Brc1ccc(cc1)-c1nc(SCC#C)nc(Sc2nccs2)c1C#N
Clc1ccc(cc1Cl)-c1nc(SCC#C)nc(Sc2nccs2)c1C#N
O=c1ccc2cc(ccc2o1)-c1nc(SCC#C)nc(Sc2nccs2)c1C#N
C#CCSc1nc(Sc2nccs2)c(C#N)c(n1)-c1ccncc1
CN(C)CCn1nnnc1Sc1nc(SCC#C)nc(-c2ccc(Cl)c(Cl)c2)c1C#N
CN(C)CCn1nnnc1Sc1nc(SCC#C)nc(-c2ccc3oc(=O)ccc3c2)c1C#N
Clc1ccc(cc1)-c1nc(SCC=C)nc(Sc2nccs2)c1C#N
Clc1ccc(cc1)-c1nc(SCc2cn(Cc3ccccc3)nn2)nc(Sc2nccs2)c1C#N
CCCC(C)N1CCC(CC1)N(Cc1ccccc1NC(=O)C=C)C(=O)Nc1cccc(c1)C(F)(F)F
CC(C)c1ccc(cc1)-c1nc(SCC#C)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Nc2nnnn2C)c1C#N
COc1ccc(Nc2nc(SCC#C)nc(-c3cc(OC)c(OC)c(OC)c3)c2C#N)cc1
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nnc(N)s2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nc(C)cs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(Sc2nc3ccccc3s2)c1C#N
Cc1ccc(cc1)-c1nc(SCC#C)nc(Sc2nccs2)c1C#N
C#CCSc1nc(Sc2nccs2)c(C#N)c(n1)-c1ccc[nH]1
CN(C)CCn1nnnc1Sc1nc(SCC#C)nc(-c2ccc(Cl)cc2)c1C#N
CCCSc1nc(Sc2nccs2)c(C#N)c(n1)-c1ccc(Cl)cc1
Cn1nnnc1Sc1nc(SCC#C)nc(-c2cccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC#C)nc(N2CCCCC2)c1C#N
Sc1n[nH]c(n1)-c1ccccc1
Cc1ccccc1-c1nnc(S)[nH]1
Fc1ccccc1-c1nnc(S)[nH]1
Sc1n[nH]c(n1)-c1ccccc1Cl
Sc1n[nH]c(n1)-c1ccccc1Br
COc1ccccc1-c1nnc(S)[nH]1
Oc1ccccc1-c1nnc(S)[nH]1
Nc1ccccc1-c1nnc(S)[nH]1
Sc1nnc([nH]1)-c1ccccc1-c1ccccc1
Sc1n[nH]c(n1)-c1cccc(Br)c1
COc1cccc(c1)-c1nnc(S)[nH]1
Nc1cccc(c1)-c1nnc(S)[nH]1
Sc1nnc([nH]1)-c1cccc(c1)S(=O)(=O)N1CCOCC1
Sc1nnc([nH]1)-c1ccc2OCOc2c1
Cc1ccc(cc1)-c1nnc(S)[nH]1
Sc1n[nH]c(n1)-c1ccc(Cl)cc1
COc1ccc(cc1)-c1n[nH]c(S)n1
CCC(=O)N[C@@H](Cc1nc2ccc(cc2s1)C(C)C)C(=O)N[C@@H](CNC(=O)CCN1CCOCC1)C1CCCCC1 |r|
CSc1nc(n[nH]1)-c1ccccc1
C#CCSc1nnc([nH]1)-c1ccccc1
C=CCSc1n[nH]c(n1)-c1ccccc1
C(Sc1nnc([nH]1)-c1ccccc1)c1ccccc1
O=C(CSc1nnc([nH]1)-c1ccccc1)Nc1ccccc1
O=C(CSc1n[nH]c(n1)-c1ccccc1)NC1CCCCC1
O=C(CSc1n[nH]c(n1)-c1ccccc1)c1ccccc1
COc1cccc(c1)C(=O)CSc1nnc([nH]1)-c1ccccc1
S(Sc1nnc([nH]1)-c1ccccc1)c1nnc([nH]1)-c1ccccc1
Cc1ccccc1-c1nnc(SSc2nnc([nH]2)-c2ccccc2C)[nH]1
Fc1ccccc1-c1nnc(SSc2nnc([nH]2)-c2ccccc2F)[nH]1
Clc1ccccc1-c1nnc(SSc2nnc([nH]2)-c2ccccc2Cl)[nH]1
Brc1ccccc1-c1nnc(SSc2nnc([nH]2)-c2ccccc2Br)[nH]1
COc1ccccc1-c1nnc(SSc2nnc([nH]2)-c2ccccc2OC)[nH]1
Oc1ccccc1-c1nnc(SSc2nnc([nH]2)-c2ccccc2O)[nH]1
S(Sc1nnc([nH]1)-c1ccccc1-c1ccccc1)c1nnc([nH]1)-c1ccccc1-c1ccccc1
Brc1cccc(c1)-c1nnc(SSc2nnc([nH]2)-c2cccc(Br)c2)[nH]1
COc1cccc(c1)-c1nnc(SSc2nnc([nH]2)-c2cccc(OC)c2)[nH]1
O=S(=O)(N1CCOCC1)c1cccc(c1)-c1nnc(SSc2nnc([nH]2)-c2cccc(c2)S(=O)(=O)N2CCOCC2)[nH]1
C1Oc2ccc(cc2O1)-c1nnc(SSc2nnc([nH]2)-c2ccc3OCOc3c2)[nH]1
Cc1ccc(cc1)-c1nnc(SSc2nnc([nH]2)-c2ccc(C)cc2)[nH]1
Clc1ccc(cc1)-c1nnc(SSc2nnc([nH]2)-c2ccc(Cl)cc2)[nH]1
CCN1c2c([C@@H]([C@H](NC(=O)c3cccc(c3)C(F)(F)F)C1=O)c1ccc(F)cc1)c(CN)nn2-c1ccccc1 |r|
CCCSc1nc(Sc2nccs2)c(C#N)c(n1)-c1cc(OC)c(OC)c(OC)c1
COc1cc(cc(OC)c1OC)-c1nc(SCC=C)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC2CCCCC2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccncc2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccoc2C(F)(F)F)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2nc3ccccc3[nH]2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2c(C)noc2C)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCCc2ccccc2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC(=O)Nc2ccccc2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCC(=O)NC(=O)Nc2ccccc2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Sc2nnnn2CCN(C)C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Sc2nc(C)cs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Sc2nc(C)c(C)s2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(NCc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Nc2ccc(Cl)cc2)c1C#N
COc1ccc(Nc2nc(SCc3ccccc3)nc(-c3cc(OC)c(OC)c(OC)c3)c2C#N)cc1
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(NC(C)(C)N2CCOCC2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Nc2ccc(O)c(Cl)c2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2)nc(Nc2cccc(Cl)c2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2cccc(c2)C(F)(F)F)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(cc2)C(F)(F)F)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2cccc(C)c2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(C)cc2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccccc2C)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(cc2)C(C)(C)C)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(Cl)cc2)nc(Sc2nccs2)c1C#N
COc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2cc(OC)c(OC)c(OC)c2)cc1
COC(=O)c1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2cc(OC)c(OC)c(OC)c2)cc1
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc3ccccc3c2)nc(Sc2nccs2)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2cccc(c2)C(F)(F)F)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(cc2)C(F)(F)F)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(Cl)cc2)nc(Sc2nnnn2C)c1C#N
COc1ccc(CSc2nc(Sc3nnnn3C)c(C#N)c(n2)-c2cc(OC)c(OC)c(OC)c2)cc1
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc3ccccc3c2)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2cccc(C)c2)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(cc2)C(C)(C)C)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(C)cc2)nc(Sc2nnnn2C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2cccc(c2)C(F)(F)F)nc(Sc2nnnn2CCN(C)C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(cc2)C(F)(F)F)nc(Sc2nnnn2CCN(C)C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(Cl)cc2)nc(Sc2nnnn2CCN(C)C)c1C#N
COc1ccc(CSc2nc(Sc3nnnn3CCN(C)C)c(C#N)c(n2)-c2cc(OC)c(OC)c(OC)c2)cc1
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc3ccccc3c2)nc(Sc2nnnn2CCN(C)C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2cccc(C)c2)nc(Sc2nnnn2CCN(C)C)c1C#N
COc1cc(cc(OC)c1OC)-c1nc(SCc2ccc(C)cc2)nc(Sc2nnnn2CCN(C)C)c1C#N
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2ccccc2)cc1
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2ccccc2C)cc1
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2cccc(C)c2)cc1
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2ccc(C)cc2)cc1
COc1ccc(cc1)-c1nc(SCc2ccc(C)cc2)nc(Sc2nccs2)c1C#N
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2ccc(Cl)cc2)cc1
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2ccc(Br)cc2)cc1
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2ccc(Oc3ccccc3)cc2)cc1
COc1ccc(cc1OC)-c1nc(SCc2ccc(C)cc2)nc(Sc2nccs2)c1C#N
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2c[nH]c3ccccc23)cc1
Cc1ccc(CSc2nc(Sc3nccs3)c(C#N)c(n2)-c2cccs2)cc1
COc1cc(cc(OC)c1OC)-c1cc(Sc2nnnn2C)nc(SCc2ccc(Cl)cc2)n1
COc1ccc(CNc2nc(Sc3nnnn3C)cc(n2)-c2cc(OC)c(OC)c(OC)c2)cc1
Cn1nnnc1Sc1cc(-c2ccccc2)nc2ncnn12
CN(C)CCn1nnnc1Sc1cc(C)nc2nc(SCc3ccc(Cl)cc3)nn12
CN(C)CCn1nnnc1Sc1ccnc2nc(SCc3ccc(Br)cc3)nn12