980 SMILES Strings for Epidermal growth factor receptor [T790M,L858R]

Compound Name
SMILES String
Nc1ncnc2n(nc(-c3ccc(Oc4ccc(F)cc4)cc3)c12)[C@@H]1CCCN(C1)C(=O)C=C |r|
Nc1ncnc2n(nc(-c3ccc(Oc4ccccc4)c(Cl)c3)c12)[C@@H]1CCCN(C1)C(=O)C=C |r|
COc1ccc(Nc2ncc3ncc(=O)n(-c4ccc(N)cc4)c3n2)cc1
COc1ccc(Nc2ncc3ncc(=O)n(-c4ccc(NC(=O)C=C)cc4)c3n2)cc1
C=CC(=O)Nc1ccc(cc1)-n1c2nc(Nc3ccc(cc3)N3CCOCC3)ncc2ncc1=O
COc1ccc(Nc2ncc3nc(C)c(=O)n(-c4ccc(NC(=O)C=C)cc4)c3n2)cc1
COc1ccc(Nc2ncc3ncc(=O)n(-c4cccc(N)c4)c3n2)cc1
COc1ccc(Nc2ncc3ncc(=O)n(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CCC(=O)Nc1cccc(c1)-n1c2nc(Nc3ccc(OC)cc3)ncc2ncc1=O
CCC(=O)Nc1ccc(cc1)-n1c2nc(Nc3ccc(OC)cc3)ncc2ncc1=O
COc1ccc(Nc2ncc3ncc(=O)n(-c4ccc(NC(=O)\C=C\CN(C)C)cc4)c3n2)cc1
COc1ccc(Nc2ncc3ncc(=O)n(-c4cccc(NC(=O)\C=C\CN(C)C)c4)c3n2)cc1
COc1ccc(Nc2ncc3ncc(=O)n(-c4ccc(OC(=O)C=C)cc4)c3n2)cc1
CN(C)C\C=C\C(=O)Nc1ccc(cc1)-n1c2nc(Nc3ccccc3)ncc2ncc1=O
CN(C)C\C=C\C(=O)Nc1cccc(c1)-n1c2nc(Nc3ccccc3)ncc2ncc1=O
C=CC(=O)Nc1ccc(cc1)-n1c2nc(Nc3ccccc3)ncc2ncc1=O
C=CC(=O)Nc1cccc(c1)-n1c2nc(Nc3ccccc3)ncc2ncc1=O
Clc1ccc(Nc2ncc3ncc(=O)n(-c4ccc(NC(=O)C=C)cc4)c3n2)cc1
Clc1ccc(Nc2ncc3ncc(=O)n(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
C=CC(=O)Nc1cccc(c1)-n1c2nc(Nc3ccc(cc3)N3CCOCC3)ncc2ncc1=O
CN1CCN(CC1)c1ccc(Nc2ncc3ncc(=O)n(-c4ccc(NC(=O)C=C)cc4)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3ncc(=O)n(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
C=CC(=O)Nc1cccc(c1)-n1c2nc(Nc3ccc(cc3)N3CCCCC3)ncc2ncc1=O
C=CC(=O)Nc1cccc(c1)-n1c2nc(Nc3ccc(cc3)N3CCCC3)ncc2ncc1=O
CCN(CC)c1ccc(Nc2ncc3ncc(=O)n(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CC(=O)Nc1ccc(Nc2ncc3ncc(=O)n(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
NC(=O)c1ccc(Nc2ncc3ncc(=O)n(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
COc1ccc(Nc2ncc3nc(C)c(=O)n(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
COc1ccc(cc1)-n1c2nc(Nc3cccc(NC(=O)C=C)c3)ncc2ncc1=O
COc1ccc(cc1)-n1c2nc(Nc3cccc(N)c3)ncc2ncc1=O
COc1ccc(cc1)-n1c2nc(Nc3ccc(NC(=O)C=C)cc3)ncc2ncc1=O
COc1ccc(cc1)-n1c2nc(Nc3ccc(N)cc3)ncc2ncc1=O
COc1cc(ccc1Nc1ncc2ncc(=O)n(-c3ccc(NC(=O)C=C)cc3)c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2ncc(=O)n(-c3cccc(NC(=O)C=C)c3)c2n1)N1CCN(C)CC1
CN1CCN(CC1)c2ccc(c(c2)OC)Nc3ncc(c(n3)Oc4cccc(c4)NC(=O)C=C)Cl
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2cc(cc(c2)C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2cc(F)cc(c2)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)c1cc(ccc1CN1CCOCC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cc(ccc1CN1CCCCC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN(C)[C@H]1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
CN(C)[C@@H]1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
CN1CCN(Cc2ccc(cc2)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)c1cc(ccc1CN1CCN2CCC[C@@H]2C1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
C[C@H]1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C[C@@H](C)O1 |r|
FC(F)(F)c1nnc2CN(Cc3ccc(cc3C(F)(F)F)C(=O)N[C@@H]3[C@H]4Oc5ccc(Oc6ccnc7NC(=O)CCc67)cc5[C@@H]34)CCn12 |r|
O[C@H]1CCCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
O[C@@H]1CCCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
OCCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2Cl)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2Br)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN(C)C1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2Cl)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2Br)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN(C)Cc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CC(C)(N)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
NC1(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cc(ccc1CN1CCNCC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCCCCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
C[C@H]1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CCN1 |r|
C[C@@H]1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CCN1 |r|
CN(C)[C@@H]1CCCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
CN(C)[C@@H]1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CCN1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@H]2[C@@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@H]23)CC1 |r|
FC(F)(F)c1cccc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1ccc(cc1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Cc1cccc(F)c1C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1ccccc1C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1cccc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1ccc(cc1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1ccc(cc1F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1cc(ccc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CC(C)(C#N)c1cccc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1ccccc1C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1ccnc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
O=C(N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12)c1cccc(c1)C1(CC1)C#N |r|
CN(C)[C@H]1CCCN(C1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN(C)[C@@H]1CCCN(C1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1CCN(CC1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCN1CCN(CC1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1CCC(CC1)Oc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1CCN(CCOc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)c1cccc(\C=C\C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)c1 |r|
O=C(N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12)c1ccc(o1)-c1ccccc1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)NC2C3Oc4c(cc(Oc5ccnc6NC(=O)CCc56)cc4C)C23)CC1
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)NC2C3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4C23)CC1
CCN1CCN(Cc2ccc(cc2C)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
Cc1cc(ccc1CO)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cccc(CC(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)c1 |r|
FC(F)(F)c1cc(ccn1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cncc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cccc(n1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CC1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC(C)N1C(=O)OC(C)(C)C |r|
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN(C)C1CCN(CC1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
COc1cc(ccc1CN1CCN(C)CC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCN1CCN(Cc2ccc(cc2OC)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCC(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
[#6]-[#6]-[#7]-1-[#6]-[#6]\[#6](-[#6]-[#6]-1)=[#6]/c1ccc(cc1C(F)(F)F)-[#6](=O)-[#7]-[#6@@H]-1-[#6@H]-2-[#8]-c3ccc(-[#8]-c4ccnc5-[#7]-[#6](=O)-[#6]-[#6]-c45)cc3-[#6@@H]-1-2 |r|
OCc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1C(C)(C)CC(CC1(C)C)Oc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCN1CCN(Cc2ccc(cc2OC(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)OCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)OCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc(c5)C(=O)NC)cc4[C@@H]23)CC1 |r|
CNC(=O)c1cc(Oc2ccc3O[C@@H]4[C@@H](NC(=O)c5ccc(CN6CCN(C)CC6)c(c5)C(F)(F)F)[C@@H]4c3c2)ccn1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc(N)c5)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)NCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)NCc56)cc4[C@@H]23)CC1 |r|
C#Cc1cccc(c1)Nc2c3cc4c(cc3ncn2)OCCOCCOCCO4
CC(=O)N1CCN(CC1)c2ccc(c(c2)OC)Nc3ncc(c(n3)Nc4cccc(c4)NC(=O)C=C)C(F)(F)F
COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2C(=O)C(N)=O)n1)N1CCC(CC1)N(C)C
COc1cc(Nc2ncc(Cl)c(Nc3ccccc3C(=O)C(=O)N(C)C)n2)ccc1N1CCN(C)CC1
COc1ccc(NC(=O)C=C)cc1Nc1ncc(Cl)c(Nc2ccccc2C(=O)C(=O)N(C)C)n1
CN(C)C(=O)C(=O)c1ccccc1Nc1cc(Cl)ccc1Cl
CN(C)C(=O)C(=O)c1ccccc1Nc1nc(Nc2ccc3OCCN(C(=O)C=C)c3c2)ncc1Cl
CN(C)CCOc1ccc(Nc2ncc(Cl)c(Nc3ccccc3C(=O)C(=O)N(C)C)n2)cc1NC(=O)C=C
COc1cc(Nc2ncc(Cl)c(Nc3ccccc3C(=O)C(=O)N(C)C)n2)ccc1N1CCC(CC1)N(C)C
COc1ccccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F
COc1ccccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F
COc1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
COc1ccc(Nc2ncc(Cl)c(Nc3cccc(NC(=O)C=C)c3)n2)c(OC)c1OC
COc1ccc(Nc2ncc(Br)c(Nc3cccc(NC(=O)C=C)c3)n2)c(OC)c1OC
COc1cccc(Nc2ncc(Br)c(Oc3cccc(NC(=O)C=C)c3)n2)c1OC
COc1ccc(Nc2ncc(Cl)c(Oc3cccc(NC(=O)C=C)c3)n2)c(OC)c1OC
COc1ccc(Nc2ncc(Br)c(Oc3cccc(NC(=O)C=C)c3)n2)c(OC)c1OC
COc1ccc(Nc2ncc(c(Oc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
COc1ccc(Nc2ncc(c(Oc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1OC
COc1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1OC
COc1ccccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1
COc1ccc(Nc2ncc(Br)c(Oc3cccc(NC(=O)C=C)c3)n2)c(OC)c1
COc1cccc(Nc2ncc(Br)c(Nc3cccc(NC(=O)C=C)c3)n2)c1OC
COc1ccc(Nc2ncc(Cl)c(Oc3cccc(NC(=O)C=C)c3)n2)c(OC)c1
COc1cccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c1OC
COc1cccc(Nc2ncc(Cl)c(Oc3cccc(NC(=O)C=C)c3)n2)c1OC
COc1ccccc1Nc1ncc(Cl)c(Nc2cccc(NC(=O)C=C)c2)n1
COc1ccccc1Nc1ncc(F)c(Oc2cccc(NC(=O)C=C)c2)n1
COc1ccc(Nc2ncc(Br)c(Nc3cccc(NC(=O)C=C)c3)n2)c(OC)c1
COc1ccc(Nc2ncc(Cl)c(Nc3cccc(NC(=O)C=C)c3)n2)c(OC)c1
COc1ccccc1Nc1ncc(Br)c(Nc2cccc(NC(=O)C=C)c2)n1
COc1cccc(Nc2ncc(c(Oc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c1OC
CC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
Cc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(COC)c23)c1F
CC(C)CS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)CC(C)C)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OC)c23)c1F
CCOc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OC)c23)c1F
CC(C)c1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(C)C)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CC3)c12
Oc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CCOCC3)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(CC(C)C)c23)c1F
CC(C)Cc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(Cl)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(N3CCOCC3)c12
COc1ccc(cn1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OC)c23)c1F
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
CC(C)CNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(OC3CCOCC3)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(O)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(C#N)c12
CCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4cc(C)cc(C)c4)c3F)c12
CNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Cc1cc(C)cc(c1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
CC(C)COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CC(C)c1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(O)c23)c1F
Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(Cl)c23)c1F
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(Cl)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CCCC3)c12
COc1ccc(cc1F)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(Nc3ccccc3)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OCC)c23)c1F
CC(C)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CC4)c23)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CC4)c23)c1F
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC(C)C)c23)c1F
OCCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CC(C)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(C)C)c3F)c12
CC(C)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4cc(C)cc(C)c4)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CCOCC4)c23)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CCOCC4)c23)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(Nc4ccccc4)c23)c1F
CN(C)c1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3COC3)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC(C)C)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NCC3CC3)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(OCC3CC3)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CCOC3)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC(C)C)c23)c1F
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4COC4)c23)c1F
CN1CCC(CC1)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
COCCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CN(C)CCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4COC4)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(N3CCCC3)c12
Cn1cc(Nc2ncnc3[nH]cc(C(=O)c4c(F)ccc(NS(=O)(=O)c5ccc(cc5)C(F)(F)F)c4F)c23)cn1
CCn1cc(Nc2ncnc3[nH]cc(C(=O)c4c(F)ccc(NS(=O)(=O)c5ccc(cc5)C(F)(F)F)c4F)c23)cn1
CCCS(=O)(=O)Nc1ccc(F)c(C=O)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C=O
Fc1ccc(NS(=O)(=O)c2ccccc2)c(F)c1C=O
C=CC(=O)Nc1cccc(c1)-c1cccc2cnc(Nc3ccc(cc3)N3CCOCC3)nc12
COc1cc(ccc1Nc1ncc2cccc(-c3cccc(NC(=O)C=C)c3)c2n1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CC(=O)N1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3ccc(C)c(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cncc(NC(=O)C=C)c4)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cn1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)c(F)c1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4F)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4F)c3n2)cn1
CC(=O)N1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4F)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4Cl)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4ccnc(NC(=O)C=C)c4)c3n2)cc1
OCCN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
FCCN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4F)c3n2)cc1
COc1c(NC(=O)C=C)cccc1-c1cccc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cc(NC(=O)C=C)ccc4F)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4C#N)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1Cl
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1C#N
COc1cc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)ccc1N1CCN(C)CC1
CN1CCN(CC1CO)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
FCCN1CC(C1)Oc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CCC(Oc2ccc(Nc3ncc4cccc(-c5cccc(NC(=O)C=C)c5)c4n3)cc2)C(F)C1
CN1CCC(Oc2ccc(Nc3ncc4cccc(-c5cccc(NC(=O)C=C)c5F)c4n3)cc2)C(F)C1
CN1CCN(CC1)c1ncc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1Cl
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1C(N)=O
CN1CCN(CC1)c1ccc(Nc2ncc3ccc(F)c(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
FCCN1CCN(CC1)c1ccc(Nc2ncc3ccc(F)c(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
OCCN1CC(C1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
FCCN1CC(C1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CCC(Nc2ccc(Nc3ncc4cccc(-c5cccc(NC(=O)C=C)c5)c4n3)cc2)C(F)C1
CN1CCN(C(=O)C1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
COCCOc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
OCCOc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
C=CC(=O)Nc1cccc(c1)-c1cccc2cnc(Nc3ccc(OCCN4CCC4)cc3)nc12
CN(C)CCOc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CCC(CC1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CC[C@@H](C1)Oc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CC[C@H](C1)Oc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CCC(CC1)Oc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CC[C@@H](C1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CC[C@H](C1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
OCCN1CCC(CC1)Oc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
FCCN1CCC(CC1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
OCCN1CCC(CC1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
CN1CCC(CC1)Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)c(F)c1
CN1CCC(CC1)Oc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)c(F)c1
CC(C)(O)CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
OCCN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)c(F)c1
OCCN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)c(F)c1F
CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)c(F)c1F
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC1CN(C1)C(=O)C=C
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC1CCN(CC1)C(=O)C=C
Fc1ccc(Nc2ncnc3cc(O[C@H]4CCOC4)c(NC4CN(C4)C(=O)C=C)cc23)cc1Cl
Fc1ccc(Nc2ncnc3cc(O[C@H]4CCOC4)c(NC4CCN(CC4)C(=O)C=C)cc23)cc1Cl
Fc1ccc(Nc2ncnc3cc(O[C@H]4CCOC4)c(NC4CCN(C4)C(=O)C=C)cc23)cc1Cl
COc1cc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC1CCN(CC1)C(=O)C=C
COc1cc2ncnc(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC1CCN(CC1)C(=O)C=C
COc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1NC1CCN(CC1)C(=O)C=C
COc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1NC1CN(C1)C(=O)C=C
COc1cc2ncnc(Nc3cccc(c3)C(C)=O)c2cc1NC1CCN(CC1)C(=O)C=C
COc1cc2ncnc(Nc3cccc(c3)C(C)=O)c2cc1NC1CN(C1)C(=O)C=C
COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC1CN(C1)C(=O)C=C
COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC1CCN(CC1)C(=O)C=C
COCCOc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC1CN(C1)C(=O)C=C
COCCOc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC1CCN(CC1)C(=O)C=C
Fc1ccc(Nc2ncnc3cc(OCCN4CCOCC4)c(NC4CN(C4)C(=O)C=C)cc23)cc1Cl
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1SC1CN(C1)C(=O)C=C
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1SC1CCN(C1)C(=O)C=C
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1SC1CCN(CC1)C(=O)C=C
Fc1ccc(Nc2ncnc3ccc(NC4CCN(CC4)C(=O)C=C)cc23)cc1Cl
COc1cc2c(cc1OCCCN3CCOCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
COc1cc(N2CCN(C)CC2)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(Nc2ccccc2C(=O)C(=O)N(C)C)n1
COOc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1c(-c2ccc(OCc3ccccn3)c(Cl)c2)n(C)c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1c(-c2ccccc2)n(C)c2ccccc12
CCOC(=O)c1cnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)nc1-c1cn(C)c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1cn(C)c2ccccc12
COc1cc(N(C)CC2CCCN2C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1cn(C)c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(C)c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1c[nH]c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1cn(C)c2ncccc12
COc1cc(N(C)C[C@@H]2CCCN2C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1cn(C)c2ccccc12 |r|
COc1cc(N(C)C[C@H]2CCCN2C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1cn(C)c2ccccc12 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1c[nH]c2ccccc12
CNCCN(C)c1cc(OC)c(Nc2nccc(n2)-c2cn(C)c3ccccc23)cc1NC(=O)C=C
CNCCN(C)c1cc(OC)c(Nc2ncc(C(=O)OC(C)C)c(n2)-c2cn(C)c3ccccc23)cc1NC(=O)C=C
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1c[nH]c2ncccc12
COc1cc(OCCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1cn(C)c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(CC(N)=O)c2ccccc12
CCc1cnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)nc1-c1cn(CC(N)=O)c2ccccc12
CCc1cnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)nc1-c1cn(CC(=O)NC)c2ccccc12
COc1cc(N(C)C[C@@H]2CCCN2)c(NC(=O)C=C)cc1Nc1ncc(C(=O)OC(C)C)c(n1)-c1cn(C)c2ccccc12 |r|
CNCCN(C)c1cc(OC)c(Nc2ncc(C(=O)OC(C)C)c(n2)-c2cn(C)c3ncccc23)cc1NC(=O)C=C
CCn1cc(-c2nc(Nc3cc(NC(=O)C=C)c(cc3OC)N(C)CCN(C)C)ncc2C(=O)OC(C)C)c2ccccc12
COC(=O)c1cccc2c(cn(C)c12)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(C)c2cc(ccc12)C(=O)OC(C)C
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(C)c2c(cccc12)C(=O)OC(C)C
COC(=O)c1c(-c2ccnc(Nc3cc(NC(=O)C=C)c(cc3OC)N(C)CCN(C)C)n2)c2ccccc2n1C
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1c(C(=O)OC(C)C)n(C)c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1c(C#N)n(C)c2ccccc12
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(C)c2cc(ccc12)C#N
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1c(C(N)=O)n(C)c2ccccc12
CNC(=O)c1c(-c2ccnc(Nc3cc(NC(=O)C=C)c(cc3OC)N(C)CCN(C)C)n2)c2ccccc2n1C
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1c(C(=O)N(C)C)n(C)c2ccccc12
COCCNC(=O)c1c(-c2ccnc(Nc3cc(NC(=O)C=C)c(cc3OC)N(C)CCN(C)C)n2)c2ccccc2n1C
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(C)c2cc(ccc12)-c1cnn(C)c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(c(n1)-c1cn(C)c2ccccc12)P(C)(C)=O
CNC(=O)Nc1cnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)nc1-c1cn(C)c2ccccc12
COc1cc(N2CCC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccccc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccccc2C2(O)CC2)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cnc(F)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)\C=C\CN(C)C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cnc(C)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccc(C)nc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cccnc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccc(F)c(F)c2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccccc2C2(O)COC2)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(Cl)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccc(cc2C(C)(C)O)C(F)(F)F)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccc(Cl)c(F)c2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(Cl)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(Cl)c(F)c2C(C)(C)O)n1
COc1cc(N2CC[C@@H]3CN(C)C[C@H]23)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN2CCCC2)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1
COc1cc(N2CC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)C[C@H]2CCCN2C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CCC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC(CN(C)C)C2)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1
COc1cc(N(C)CCN2CCCCC2)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1
COc1cc(N2CC[C@H]3CN(C)C[C@@H]23)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN2CCCCC2)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@@H]3CN(C)C[C@H]23)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN2CCCC2)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1
COc1cc(N(C)C[C@H]2CCCN2C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CC2CCCN2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc3ccn(C)c3cc2C(C)(C)O)n1
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(cc2C(C)(C)O)C2CC2)n1
COc1cc(N2CCOC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1
COc1cc(N2CC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC(CN(C)C)C2)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1
COc1cc(N2CCOC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@@H]3CN(C)C[C@H]23)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(Cl)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN2CCC[C@@H]2C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CCC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(Cl)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)C[C@@H]2CCCN2C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@@H]3CN(C)C[C@H]23)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(cc2C(C)(C)O)C2CC2)n1 |r|
COc1cc(N2CCC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(cc2C(C)(C)O)C2CC2)n1 |r|
CCC(C)(O)c1cc(F)c(F)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@@H]3CN(C)C[C@H]23)n1 |r|
CCC(C)(O)c1cc(F)c(F)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@H](C2)N(C)C)n1 |r|
CCC(C)(O)c1cc(F)c(F)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
CCC(C)(O)c1cc(F)c(F)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@H]3CN(C)C[C@@H]23)n1 |r|
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(Cl)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(Cl)cc2C(C)(C)O)n1 |r|
CCC(C)(O)c1cc(F)c(F)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@@H]2CN(C)C)n1 |r|
CCC(C)(O)c1cc(F)c(Cl)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@@H]2CN(C)C)n1 |r|
CCC(C)(O)c1cc(F)c(F)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CCC[C@@H]2CN(C)C)n1 |r|
CCC(C)(O)c1cc(F)c(F)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CCC[C@H]2CN(C)C)n1 |r|
CCC(C)(O)c1cc(F)c(Cl)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@H](C2)N(C)C)n1 |r|
COc1cc(N2CC[C@@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(Cl)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(F)c(Cl)cc2C(C)(C)O)n1 |r|
CCC(C)(O)c1cc(F)c(Cl)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CCC[C@@H]2CN(C)C)n1 |r|
CCC(C)(O)c1cc(F)c(Cl)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CCC[C@H]2CN(C)C)n1 |r|
COc1cc(N2CCC[C@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccccc2C(C)(O)C(F)(F)F)n1
CCC(C)(O)c1cc(F)c(Cl)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
CC[C@@](C)(O)c1cc(F)c(Cl)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@H](C2)N(C)C)n1 |r|
CC[C@](C)(O)c1cc(F)c(Cl)cc1Nc1ncnc(Nc2cc(NC(=O)C=C)c(cc2OC)N2CC[C@H](C2)N(C)C)n1 |r|
COc1cc(N2CC[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(Cl)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C2(O)CCC2)n1
CN[C@@H]1CCN(C1)c1cc(OC)c(Nc2ncnc(Nc3cc(Cl)c(F)cc3C(C)(C)O)n2)cc1NC(=O)C=C |r|
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(C3CC3)c(F)cc2C(C)(C)O)n1
COc1cc(N2CC[C@@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1
COc1cc(N2C[C@@H](F)[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
CN[C@@H]1CCN(C1)c1cc(OC)c(Nc2nccc(Nc3cc(Cl)c(F)cc3C(C)(C)O)n2)cc1NC(=O)C=C |r|
COc1cnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)nc1Nc1cc(Cl)c(F)cc1C(C)O
COc1cc(N2CC(F)(F)C[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2C[C@H](N(C)C)C3(CC3)C2)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(c(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1)C(F)(F)F |r|
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(C#N)c(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@@H](CN(C)C)C2)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2C[C@H](F)C[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2C[C@H]3CN(C)[C@H]3C2)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)C[C@H]2C[C@H](C)CN2C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2C[C@@H](C)C[C@@H]2CN(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CC[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(O)C(F)(F)F)n1 |r|
COc1cc(N2C[C@@H](F)[C@H](C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2ccc3[nH]ccc3c2C(C)(C)O)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncnc(Nc2cc3cc[nH]c3cc2C(C)(C)O)n1
COc1cc(N2C[C@@H]3CN(C)C[C@H]23)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2C[C@@H]3CN(C)[C@@H]3C2)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
COc1cc(N2CCC[C@@H]2CN2CCC2)c(NC(=O)C=C)cc1Nc1nccc(Nc2cc(Cl)c(F)cc2C(C)(C)O)n1 |r|
CN(C)C/C=C/C(=O)Nc1cc2c(cc1O[C@H]3CCOC3)ncnc2Nc4ccc(c(c4)Cl)F
COc1cc2ncnc(Nc3ccc(Cl)c(Cl)c3F)c2cc1OC1CCN(CC1)C(=O)C=C
CN(C)C\C=C\C(=O)N1CCCC[C@H](C1)n1c(NC(=O)c2ccnc(C)c2)nc2cccc(Cl)c12 |r|
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)C(CSC(C)=O)CSC(C)=O
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)C1CSSC1
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)CC1CCSS1
OC[C@@H](O)COc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)C[C@H]1CCSS1 |r|
OC[C@@H](O)COc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)CC1CCSS1 |r|
OC[C@H](O)COc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)C[C@@H]1CCSS1 |r|
OC[C@H](O)COc1cc2ncc(C#N)c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)C[C@H]1CCSS1 |r|
Cc1ccc(NC(=O)c2ccc(C)c(c2)C(F)(F)F)cc1C#Cc1nn([C@H]2CC[C@H](O)CC2)c2ncnc(N)c12 |r,wU:26.27,wD:29.31,(-5.46,5.4,;-3.98,5.8,;-3.58,7.29,;-2.09,7.69,;-1,6.6,;.49,7,;1.57,5.91,;1.18,4.42,;3.06,6.31,;3.46,7.79,;4.95,8.19,;6.04,7.1,;7.53,7.5,;5.64,5.62,;4.15,5.22,;6.73,4.53,;8.22,4.93,;6.33,3.04,;7.82,3.44,;-1.4,5.11,;-2.89,4.71,;-3.29,3.22,;-3.68,1.74,;-4.08,.25,;-3.18,-1,;-4.08,-2.24,;-3.68,-3.73,;-2.2,-4.13,;-1.8,-5.62,;-2.89,-6.7,;-2.49,-8.19,;-4.38,-6.31,;-4.77,-4.82,;-5.55,-1.77,;-6.88,-2.54,;-8.22,-1.77,;-8.22,-.23,;-6.88,.54,;-6.88,2.08,;-5.55,-.23,)|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2cnn(C)c2)c2cc[nH]c2n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nc(N2CCOCC2)c2cc[nH]c2n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nc(OC2CN(C2)S(C)(=O)=O)c2ccn(CO)c2n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2cnc3n(C)ccc3c2)c2cc[nH]c2n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2cn(C)c3ccccc23)c2cc[nH]c2n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2cccnc2)c2cc[nH]c2n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2ccccc2)c2cc[nH]c2n1
COc1cc(OCCN(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2cnn(C)c2)c2cc[nH]c2n1
COc1cc(N2CC(C2)N(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2cnn(C)c2)c2cc[nH]c2n1
COc1cc(N2CCN(C)CC2)c(NC(=O)C=C)cc1Nc1nc(-c2cnn(C)c2)c2cc[nH]c2n1
COc1cc(N2CCN(C)CC2)c(NC(=O)C=C)cc1Nc1nc(-c2cnn(C)c2)c2c(Cl)c[nH]c2n1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1nc(-c2cnn(C)c2)c2c(C)c[nH]c2n1
COc1cc(ccc1Nc1nc(-c2cccc(NC(=O)C=C)c2)c2cc[nH]c2n1)N(C)CCN(C)C
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)C1CCN(CC1)S(C)(=O)=O
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCC(CC1)N1CCOCC1
Cc1cccc(Nc2ccnc(Nc3cccc(NC(=O)C=C)c3)n2)c1
Cc1cccc(Nc2nc(Nc3cccc(NC(=O)C=C)c3)ncc2C)c1
Cc1cccc(Nc2nc(Nc3cccc(NC(=O)C=C)c3)ncc2F)c1
CN(C)C\C=C\C(=O)Nc1cccc(Nc2ncc(F)c(Nc3cccc(C)c3)n2)c1
Cc1cnc(Nc2cccc(NC(=O)C=C)c2)nc1Nc1ccccc1
Cc1cnc(Nc2ccccc2)nc1Nc1cccc(NC(=O)C=C)c1
Cc1cccc(Nc2nc(Nc3cc(NC(=O)C=C)ccc3C)ncc2C)c1
Cc1cnc(Nc2cccc(NC(=O)C=C)c2)nc1Nc1cccc(Br)c1
Cc1cnc(Nc2cccc(c2)S(N)(=O)=O)nc1Nc1ccc2CN(CCc2c1)S(=O)(=O)C1CC1
Cc1cnc(Nc2cccc(c2)S(N)(=O)=O)nc1Nc1ccc2CN(CCc2c1)C(=O)CCl
Cc1cnc(Nc2cccc(NC(=O)C=C)c2)nc1Nc1ccc(Oc2ccccc2)cc1
Cc1cnc(Nc2cccc(OCC#C)c2)nc1Nc1cccc(NC(=O)C=C)c1
CN(C)C\C=C\C(=O)Nc1cccc(Nc2nc(Nc3ccccc3)ncc2C)c1
Cc1cnc(Nc2ccccc2)nc1Nc1ccc(NC(=O)C=C)cc1
Cc1ccc(NC(=O)C=C)cc1Nc1nccc(n1)-c1cccnc1
CCC(=O)Nc1cccc(Nc2nc(Nc3ccccc3)ncc2C)c1
COCCOc1ccc(Nc2ncc(F)c(Nc3cccc(NC(=O)C=C)c3)n2)cc1F
CC(C)n5c(Nc1ccccc1)nc4cnc(Nc3ccc(C(=O)NN2CCN(C)CC2)cc3)nc45
CC(C)n1c(Nc2ccc(F)c(Cl)c2)nc2cnc(Nc3ccc(cc3)C(=O)NN3CCN(C)CC3)nc12
CC(=O)Nc5cccc(Nc4nc3cnc(Nc2ccc(C(=O)NN1CCN(C)CC1)cc2F)nc3n4C(C)C)c5
CC(C)n1c(Nc2ccccc2)nc2cnc(Nc3ccc(cc3F)C(=O)NN3CCN(C)CC3)nc12
CC(C)n1c(Nc2ccc(F)c(Cl)c2)nc2cnc(Nc3ccc(cc3F)C(=O)NN3CCN(C)CC3)nc12
COc1cc(ccc1Nc1ncc2nc(Nc3ccccc3)n(C(C)C)c2n1)C(=O)NN1CCN(C)CC1
CC(C)n1c(Nc2ccccc2)nc2cnc(Nc3ccc(cc3)C(=O)NC3CCN(C)CC3)nc12
CC(C)n1c2c(cnc(n2)Nc3ccc(cc3)N4CCN(CC4)C)nc1Nc5ccccc5
CC(C)n1c(Nc2cccc(Br)c2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2cccc(c2)C#C)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2ccc(F)c(Cl)c2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2ccc(Br)cc2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2cccc(c2)C(F)(F)F)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
COc1cccc(Nc2nc3cnc(Nc4ccc(cc4)N4CCN(C)CC4)nc3n2C(C)C)c1
COc1ccc(Nc2nc3cnc(Nc4ccc(cc4)N4CCN(C)CC4)nc3n2C(C)C)cc1
CC(C)n1c(Nc2ccc(OCc3cccc(F)c3)c(Cl)c2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2ccc(NC(=O)Nc3ccc(F)c(Cl)c3)cc2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2ccc(cc2)C(=O)Nc2cccc(F)c2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CN1CCN(CC1)c1ccc(Nc2ncc3nc(Nc4ccccc4)n(C4CC4)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3nc(Nc4ccccc4)n(C)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3nc(Nc4ccccc4)[nH]c3n2)cc1
CN1CCN(CC1)c2ccc(cc2)Nc3ncc4c(n3)n(c(n4)Nc5ccccc5)C6CCCC6
CC(C)n1c(Nc2ccc(cc2)C(F)(F)F)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2cccnc2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(NC2CCCCC2)nc2cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)n1c(Nc2ccccc2)nc2cnc(Nc3cccc(NC(=O)C=C)c3)nc12
COc1cccc(Nc2ncc(Cl)c(Nc3cccc(NC(=O)C=C)c3)n2)c1OC
CN(C)C\C=C\C(=O)Nc1cc2c(Nc3cccc(c3)C#C)ncnc2cc1O[C@H]1CCOC1 |r|
CCN(CC)C\C=C\C(=O)Nc1cc2c(Nc3cccc(c3)C#C)ncnc2cc1O[C@H]1CCOC1 |r|
Nc1c(c(nn1-c1c(Cl)cc(Cl)cc1Cl)-c1ccncc1)-c1ccc(F)cc1 |(-1,-2.52,;-1.47,-1.05,;-2.94,-.58,;-2.94,.96,;-1.47,1.44,;-.56,.19,;.98,.19,;1.74,1.52,;.97,2.85,;3.28,1.52,;4.06,.18,;5.6,.18,;3.29,-1.15,;1.75,-1.15,;.97,-2.48,;-4.18,1.87,;-4.2,3.41,;-5.54,4.16,;-6.87,3.37,;-6.84,1.82,;-5.5,1.08,;-4.18,-1.48,;-5.52,-.72,;-6.85,-1.5,;-6.84,-3.04,;-8.17,-3.82,;-5.49,-3.8,;-4.17,-3.02,)|
COc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCOCC1
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCOCC1
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(=O)CO
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCOCC1
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)C(=O)CO
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCCN(CC1)C(C)=O
COc1cc(ccc1Nc1ncc(Cl)c(Nc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(C)=O
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(C)=O
COc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)C(C)=O
COc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)C(=O)CO
COc1cc(ccc1Nc1ncc(Cl)c(Nc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(=O)CO
FC(F)Oc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCOCC1
FC(F)Oc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCOCC1
COc1cc(ccc1Nc1ncc(Cl)c(Nc2cccc(NC(=O)C=C)c2)n1)N1CCOCC1
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)S(C)(=O)=O
CCOc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(=O)OC(C)(C)C
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCCN(CC1)C(=O)C(F)(F)F
COC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Oc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
CNC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Oc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)S(C)(=O)=O
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(=O)CC(C)(C)C
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(=O)C(F)(F)F
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)S(C)(=O)=O
COc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)S(N)(=O)=O
CNC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
COC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
OCC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC(F)(F)F)c1
OCC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC(F)F)c1
CC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC(F)F)c1
CC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC(F)(F)F)c1
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)C(=O)C(C)(C)C
CCC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1
FC(F)Oc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCOCC1
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCCOCC1
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCCOCC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCCN(CC1)C(=O)OC(C)(C)C
COc1cc(ccc1Nc1ncc(Br)c(Nc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(C)=O
COc1cc(ccc1Nc1ncc(Cl)c(Nc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)S(C)(=O)=O
COc1cc(ccc1Nc1ncc(c(Oc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)C(=O)CC(C)(C)C
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCCN(CC1)C(=O)OC(C)(C)C
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCCN(CC1)C(=O)OC(C)(C)C
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)C(=O)CC(C)(C)C
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(CC1)C(=O)OC(C)(C)C
CC(C)(C)OC(=O)N1CCN(CC1)c1ccc(Nc2ncc(Cl)c(Oc3cccc(NC(=O)C=C)c3)n2)c(OC(F)(F)F)c1
COC(=O)[C@@H]1CN(CCN1C(C)=O)c1ccc(Nc2ncc(c(Nc3cccc(NC(=O)C=C)c3)n2)C(F)(F)F)c(OC)c1 |r|
COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCS(=O)(=O)CC1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ccc2c1
COc1cc(N2CCN(C)CC2)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ncc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ncc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ccc2c1
COc1cc(N(C)CCN(C)N)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(OC)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(c(n1)-c1cnc2n(C)ccc2c1)C(F)(F)F
COc1cc(N2CCN(C)CC2)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ccc2c1
COc1cc(N2CC(C2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ccc2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C(C)=O)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnc2n(C)ncc2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(OC)c(n1)-c1cnc2n(C)ncc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(C)ncc2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(C)ncc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnc2n(C)ncc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(OC)c(n1)-c1cnc2n(C)ncc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)cc(Cl)c2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cccnc1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnn(C)c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnn(C)c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn(C)c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn(C)c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn(C)c1C
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnn(C)c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1c(C)nn(C)c1C |(-1.61,-15.57,;-.28,-14.8,;1.05,-15.57,;1.05,-17.11,;2.39,-17.88,;2.39,-19.42,;3.72,-20.19,;1.05,-20.19,;1.05,-21.73,;2.39,-22.5,;3.72,-21.73,;2.39,-24.04,;3.72,-17.11,;5.05,-17.88,;6.54,-18.28,;7.63,-17.19,;6.94,-19.77,;8.43,-20.17,;3.72,-15.57,;2.39,-14.8,;2.39,-13.26,;3.72,-12.49,;3.72,-10.95,;5.05,-10.18,;6.39,-10.95,;7.72,-10.18,;6.39,-12.49,;5.05,-13.26,;7.72,-13.26,;9.19,-12.79,;9.96,-11.45,;10.09,-14.03,;9.19,-15.28,;9.96,-16.61,;7.72,-14.8,;6.39,-15.57,)|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnn(C)c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cn(C)nc1C
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cn(C)nc1C
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn(c1)C1CCN(CC1)C(=O)OC(C)(C)C
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn(C)c1C
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1ccn(C)c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1ccn(C)c1
COc1cc(N2CCN(C)CC2)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn(C)c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnn(c1)C(F)F
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cn[nH]c1
CCN(C)CCN(C)c1cc(OC)c(Nc2nccc(n2)-c2cnc3n(C)ccc3c2)cc1NC(=O)C=C
CNCCN(C)c1cc(OC)c(Nc2nccc(n2)-c2cnc3n(C)ccc3c2)cc1NC(=O)C=C
CCN(CC)CCN(C)c1cc(OC)c(Nc2nccc(n2)-c2cnc3n(C)ccc3c2)cc1NC(=O)C=C
CCN(C)CCN(C)c1cc(OC)c(Nc2ncc(Cl)c(n2)-c2cnc3n(C)ccc3c2)cc1NC(=O)C=C
CCN(CC)CCN(C)c1cc(OC)c(Nc2ncc(Cl)c(n2)-c2cnc3n(C)ccc3c2)cc1NC(=O)C=C
COc1cc(N(C)CCN2CCCC2)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ccc2c1
COc1cc(N2CC(C2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N(C)CCCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N(C)CCN(C)C(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ccc2c1
CNCCN(C)c1cc(OC)c(Nc2ncc(Cl)c(n2)-c2cnc3n(C)ccc3c2)cc1NC(=O)C=C
COc1cc(OCCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(C)ccc2c1
COc1cc(OCCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnc2n(C)ccc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(C)cc(Cl)c2c1
COc1cc(N2CCC(CC2)N(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnc2n(C)cc(Cl)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cnc2n(C)cc(Cl)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cnc2n(ccc2c1)C(C)C
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(ccc2c1)C(C)C
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cnc2n(ccc2c1)C1CC1
Cc1ccc(NC(=O)C=C)cc1Nc1ncc(C)c(Nc2cccc(Br)c2)n1
C=CC(=O)Nc1cccc(c1)-c1cccc2cnc(Nc3ccc(NC4CCNCC4)cc3)nc12
C/C=C/C(=O)N1CCC[C@H]1c2nc(c3n2ccnc3N)c4ccc(cc4)C(=O)Nc5ccccn5
Nc1ncnc2n(nc(-c3ccc(Oc4ccccc4)cc3)c12)[C@@H]1CCCN(C1)C(=O)C=C
CC#CC(=O)N1CCC[C@H]1c1nc(-c2ccc(OCc3ccccc3)cc2)c2c(N)nccn12 |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN2CCN(Cc3ccc(cc3)-c3cc4c(NCc5ccccc5Cl)ncnc4[nH]3)CC2)C(C)(C)C)cc1 |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN2CCN(Cc3ccc(cc3)-c3cc4c(NCc5ccccc5Cl)ncnc4[nH]3)CC2)C(C)(C)C)cc1 |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCN2CCN(Cc3ccc(cc3)-c3cc4c(NCc5ccccc5Cl)ncnc4[nH]3)CC2)C(C)(C)C)cc1 |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCN2CCN(Cc3ccc(cc3)-c3cc4c(NCc5ccccc5Cl)ncnc4[nH]3)CC2)C(C)(C)C)cc1 |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(Cc3ccc(cc3)-c3cc4c(NCc5ccccc5Cl)ncnc4[nH]3)CC2)C(C)(C)C)cc1 |r|
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(CN2CCN(CCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)cc1
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(CN2CCN(CCOCCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)cc1
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(CN2CCN(CCOCCOCCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)cc1
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(CN2CCN(CCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)cc1
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(OCCOCCOCCOCCNc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(CCOCCNc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(OCCOCCOCCNc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(OCCOCCNc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOc2ccc(cc2)-c2cc3c(NCc4ccccc4Cl)ncnc3[nH]2)C(C)(C)C)cc1 |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(cc2)-c2cc3c(NCc4ccccc4Cl)ncnc3[nH]2)C(C)(C)C)cc1 |r|
Clc1ccccc1CNc1ncnc2[nH]c(cc12)-c1ccc(CN2CCN(CCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)CC2)cc1
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)CCCOCCCOCC(=O)N[C@H](C(=O)N1CC(O)C[C@@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN(C)C\C=C\C(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1OCCCCOCCCCOCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCOCCOc4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCON4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)nc3cn2)n1 |r|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCON4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCOCCOCCON4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCN4CCN(CCOc5ccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c6c5)CC4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)nc3cn2)n1 |r|
COC1(CCN2CCN(CC2)c2ccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3c2)CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(C)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)nc3cn2)n1 |r|
C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CN1CCN(CCCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)CC1)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)nc3cn2)n1 |r|
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCOCCOCCOCCNc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCOCCOCCNc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
C[C@H](NC(=O)[C@H]1C[C@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCOCC#Cc1cccc2CN(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCCN4CCN(CCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(cc5)-c5scnc5C)C(C)(C)C)CC4)nc3cn2)n1 |r|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCN4CCN(CCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(cc5)-c5scnc5C)C(C)(C)C)CC4)nc3cn2)n1 |r|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCN4CCN(CCCCc5ccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c6c5)CC4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCOCCN4CCN(CCOc5ccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c6c5)CC4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCCN4CCN(CCCOc5ccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c6c5)CC4)nc3cn2)n1
C[C@H](NC(=O)[C@H]1C[C@H](O)CN1C(=O)[C@@H](NC(=O)CN1CCN(CCCOCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)CC1)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
C[C@H](NC(=O)[C@H]1C[C@H](O)CN1C(=O)[C@@H](NC(=O)COCCN1CCN(CCCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)CC1)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
C[C@H](NC(=O)[C@H]1C[C@H](O)CN1C(=O)[C@@H](NC(=O)COCCCC#Cc1cccc2CN(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
C[C@H](NC(=O)[C@H]1C[C@H](O)CN1C(=O)[C@@H](NC(=O)COCCCOCCCC#Cc1cccc2CN(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCCCN3CCN(CCOc4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCCCOCCCN3CCN(CC3)c3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCCCN3CCN(CC3)c3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(cc2)-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)C(C)(C)C)cc1 |r|
Clc1ccccc1CNc1ncnc2NC(Cc12)c1ccc(CN2CCN(CCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)CC2)cc1
Clc1ccccc1CNc1ncnc2NC(Cc12)c1ccc(CN2CCN(CCOCCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)CC2)cc1
Clc1ccccc1CNc1ncnc2NC(Cc12)c1ccc(CN2CCN(CCOCCOCCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)CC2)cc1
Clc1ccccc1CNc1ncnc2NC(Cc12)c1ccc(CN2CCN(CCOCCOCCOCCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)CC2)cc1
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCN1CCN(Cc2ccc(cc2)-c2cc3c(NCc4ccccc4Cl)ncnc3[nH]2)CC1)-c1scnc1C |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCN1CCN(Cc2ccc(cc2)-c2cc3c(NCc4ccccc4Cl)ncnc3[nH]2)CC1)-c1scnc1C |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCCN1CCN(Cc2ccc(cc2)-c2cc3c(NCc4ccccc4Cl)ncnc3[nH]2)CC1)-c1scnc1C |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCCOCCN1CCN(Cc2ccc(cc2)-c2cc3c(NCc4ccccc4Cl)ncnc3[nH]2)CC1)-c1scnc1C |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCCOCCOCCN1CCN(Cc2ccc(cc2)-c2cc3c(NCc4ccccc4Cl)ncnc3[nH]2)CC1)-c1scnc1C |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)C(C)(C)C)cc1 |r|
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)C(C)(C)C)cc1 |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCC#Cc1cccc2CN([C@@H](C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)-c1scnc1C |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCCOCC#Cc1cccc2CN([C@@H](C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)-c1scnc1C |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCCOCCOCC#Cc1cccc2CN([C@@H](C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)-c1scnc1C |r|
CC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCCOCCOCCOCC#Cc1cccc2CN([C@@H](C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)-c1scnc1C |r|
Oc1ccc(F)cc1[C@@H](N1Cc2cccc(C#CCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1 |r|
Oc1ccc(F)cc1[C@@H](N1Cc2cccc(C#CCOCCOCCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1 |r|
Oc1ccc(F)cc1[C@@H](N1Cc2cccc(C#CCOCCOCCOCCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1 |r|
Oc1ccc(F)cc1[C@@H](N1Cc2cccc(C#CCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)c2C1=O)C(=O)Nc1nccs1 |r|
Oc1ccc(F)cc1[C@@H](N1Cc2cccc(C#CCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)c2C1=O)C(=O)Nc1nccs1 |r|
Oc1ccc(F)cc1[C@@H](N1Cc2cccc(C#CCOCCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)c2C1=O)C(=O)Nc1nccs1 |r|
Oc1ccc(F)cc1[C@@H](N1Cc2cccc(C#CCOCCOCCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)c2C1=O)C(=O)Nc1nccs1 |r|
C[C@H](NC(=O)[C@H]1C[C@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCC#Cc1cccc2CN([C@@H](C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)-c3ccc(OCCOCCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)cc12 |r|
CC(C)C(N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCCCOc1ccc(cc1)-c1nccc(Nc2cc3n(C(C)C)c(C)nc3cn2)n1)-c1scnc1C |r|
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)-c3ccc(OCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)cc12 |r|
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)-c3ccc(OCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)cc12 |r|
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)-c3ccc(OCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)cc12 |r|
CC(C)C(N1Cc2ccccc2C1=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1OCCOCCOCCOCCOc1ccc(cc1)-c1nccc(Nc2cc3n(C(C)C)c(C)nc3cn2)n1)-c1scnc1C |r|
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)N3CCC4(CCN(CCCOCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(cc5)-c5scnc5C)C(C)(C)C)CC4)CC3)cc12 |r|
Oc1ccc(F)cc1C(N1Cc2cccc(CCCOCCOCCOCCOc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)N3CCC(CC3)OCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@@H](O)C[C@@H]3C(=O)N[C@@H](C)c3ccc(cc3)-c3scnc3C)C(C)(C)C)cc12 |r|
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)N3CCC4(CC3)CN(CCCOCCCOCC(=O)N[C@H](C(=O)N3C[C@@H](O)C[C@@H]3C(=O)N[C@@H](C)c3ccc(cc3)-c3scnc3C)C(C)(C)C)CCO4)cc12 |r|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(nc3cn2)-c2ccc(CN3CCN(CCOc4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)cc2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(c(COCCN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)nc3cn2)C(C)(C)C)n1
COC1CCN(CC1)c1nccc(Nc2cc3[nH]c(COCCN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)nc3cn2)n1
Oc1ccc(F)cc1C(N1Cc2cccc(NCCCCOCCCN3CCN(CC3)c3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCOC3CCN(CC4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c2C1=O)C(=O)Nc1nccs1
CC(C)n1c(C)nc2cnc(Nc3ccnc(n3)N3CCC(CC3)Oc3ccc(CCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)cc12 |r|
COC1(CCN2CCN(CCCOCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(cc3)-c3scnc3C)C(C)(C)C)CC2)CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(C)nc3cn2)n1 |r|
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCN3CCC(CN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(CCCN3CCC(CN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(C#CCOCCOCCOCCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(CCCCCOCCCC3CCN(CC3)c3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(CCCOC3CCN(CC4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c2C1=O)C(=O)Nc1nccs1
Oc1ccc(F)cc1C(N1Cc2cccc(\C=C\COC3CCN(CC4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c2C1=O)C(=O)Nc1nccs1
C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCOCC#Cc1cccc2CN(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C(=O)c12)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
Oc1ccc(F)cc1C(N1Cc2cccc(CCCOCCOCCOCCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)c2C1=O)C(=O)Nc1nccs1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCN4CCN(CC4)c4ccc(OCCCN5CCN(CC5)c5ccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c6c5)cc4)nc3cn2)n1
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCN4CCN(CC4)c4ccc(O[C@H]5C[C@@H](C5)OCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(cc5)-c5scnc5C)C(C)(C)C)cc4)nc3cn2)n1 |r,wU:39.43,46.48,54.58,wD:37.38,51.54,(-10.7,-1.46,;-12.24,-1.46,;-13.01,-.13,;-14.55,-.13,;-15.32,1.2,;-14.55,2.54,;-13.01,2.54,;-12.24,1.2,;-15.32,3.87,;-16.86,3.87,;-17.63,5.2,;-16.86,6.54,;-15.32,6.54,;-14.55,7.87,;-13.01,7.87,;-12.24,6.54,;-10.7,6.54,;-9.67,5.39,;-10.07,3.91,;-8.98,2.82,;-11.56,3.51,;-8.26,6.02,;-6.93,5.25,;-5.6,6.02,;-4.26,5.25,;-2.93,6.02,;-1.59,5.25,;-1.59,3.71,;-.26,2.94,;1.07,3.71,;1.07,5.25,;-.26,6.02,;2.41,2.94,;2.41,1.4,;3.74,.63,;5.07,1.4,;6.41,.63,;7.74,1.4,;9.23,1,;9.63,2.49,;8.14,2.89,;10.96,3.26,;12.3,2.49,;13.63,3.26,;13.63,4.8,;14.96,2.49,;14.96,.95,;13.63,.18,;12.3,.95,;13.63,-1.36,;14.87,-2.27,;14.4,-3.73,;15.17,-5.06,;12.86,-3.73,;12.38,-2.27,;10.9,-1.87,;10.5,-.38,;9.81,-2.96,;8.32,-2.56,;7.23,-3.65,;5.74,-3.25,;4.65,-4.34,;5.05,-5.83,;6.54,-6.22,;7.63,-5.13,;3.96,-6.91,;2.44,-6.67,;1.74,-8.05,;2.83,-9.13,;4.2,-8.44,;5.54,-9.21,;16.3,.18,;17.63,.95,;16.3,-1.36,;17.63,-.59,;5.07,2.94,;3.74,3.71,;-8.42,7.55,;-9.93,7.87,;-10.7,9.21,;-12.24,9.21,;-14.55,5.2,)|
COC1CCN(CC1)c1nccc(Nc2cc3n(C(C)C)c(COCCN4CCN(CC4)c4ccc(OCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(cc5)-c5scnc5C)C(C)(C)C)cc4)nc3cn2)n1 |r|
CC(C)n1c(COCCN2CCN(CC2)c2ccc(O[C@H]3C[C@@H](C3)OCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(cc3)-c3scnc3C)C(C)(C)C)cc2)nc2cnc(Nc3ccnc(n3)-c3cnn(c3)S(=O)(=O)C3CC3)cc12 |r,wU:22.25,29.30,37.40,wD:20.20,34.36,(-8.98,2.82,;-10.07,3.91,;-11.56,3.51,;-9.67,5.39,;-8.26,6.02,;-6.93,5.25,;-5.6,6.02,;-4.26,5.25,;-2.93,6.02,;-1.59,5.25,;-1.59,3.71,;-.26,2.94,;1.07,3.71,;1.07,5.25,;-.26,6.02,;2.41,2.94,;2.41,1.4,;3.74,.63,;5.07,1.4,;6.41,.63,;7.74,1.4,;9.23,1,;9.63,2.49,;8.14,2.89,;10.96,3.26,;12.3,2.49,;13.63,3.26,;13.63,4.8,;14.96,2.49,;14.96,.95,;13.63,.18,;12.3,.95,;13.63,-1.36,;14.87,-2.27,;14.4,-3.73,;15.17,-5.06,;12.86,-3.73,;12.38,-2.27,;10.9,-1.87,;10.5,-.38,;9.81,-2.96,;8.32,-2.56,;7.23,-3.65,;5.74,-3.25,;4.65,-4.34,;5.05,-5.83,;6.54,-6.22,;7.63,-5.13,;3.96,-6.91,;2.44,-6.67,;1.74,-8.05,;2.83,-9.13,;4.2,-8.44,;5.54,-9.21,;16.3,.18,;17.63,.95,;16.3,-1.36,;17.63,-.59,;5.07,2.94,;3.74,3.71,;-8.42,7.55,;-9.93,7.87,;-10.7,9.21,;-12.24,9.21,;-13.01,7.87,;-14.55,7.87,;-15.32,6.54,;-16.86,6.54,;-17.63,5.2,;-16.86,3.87,;-15.32,3.87,;-14.55,5.2,;-14.55,2.54,;-13.02,2.38,;-12.7,.87,;-14.03,.1,;-15.18,1.13,;-14.19,-1.43,;-15.6,-2.06,;-12.95,-2.34,;-14.35,-2.96,;-15.5,-3.99,;-14.03,-4.47,;-12.24,6.54,;-10.7,6.54,)|
CC(C)n1c(COCCN2CCN(CC2)c2ccc(OCCCN3CCN(CC3)c3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)cc2)nc2cnc(Nc3ccnc(n3)-c3cnn(c3)S(=O)(=O)C3CC3)cc12
CC(C)n1c(COCCN2CCN(CC2)c2ccc(OCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(cc3)-c3scnc3C)C(C)(C)C)cc2)nc2cnc(Nc3ccnc(n3)-c3cnn(c3)S(=O)(=O)C3CC3)cc12 |r|
Oc1ccc(F)cc1C(N1Cc2cccc(NCCCCOCCCN3CCC(CC3)N3CCN(CC3)c3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)c2C1=O)C(=O)Nc1nccs1
CC(C)n1nc(N2CC(CNCCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(cc3)-c3scnc3C)C(C)(C)C)C2)c2cnc(Nc3ccnc(n3)-c3cnn(c3)S(=O)(=O)C3CC3)cc12 |r|
C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CN1CCN(CCOCCOCCOCCOCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)CC1)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCOCCN1CCN(CCOCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)CC1)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCN1CCN(CCOCCOCCOCC#Cc2cccc3CN(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C(=O)c23)CC1)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
CC(C)n1nc(N2CCN(CC3CCN(CC3)c3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)CC2)c2cnc(Nc3ccnc(n3)-c3cnn(c3)S(=O)(=O)C3CC3)cc12
CC(C)n1nc(N2CC(CN3CCN(CC4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)C2)c2cnc(Nc3ccnc(n3)-c3cnn(c3)S(=O)(=O)C3CC3)cc12
CC(C)n1nc(N2CC(CN[C@H]3C[C@@H](C3)Oc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)C2)c2cnc(Nc3ccnc(n3)-c3cnn(c3)S(=O)(=O)C3CC3)cc12 |r,wU:11.10,wD:13.15,(-8.98,2.82,;-10.07,3.91,;-11.56,3.51,;-9.67,5.39,;-8.26,6.02,;-8.42,7.55,;-7.28,8.58,;-7.28,10.12,;-5.74,10.12,;-4.64,11.25,;-3.15,10.87,;-2.07,11.97,;-1.59,13.44,;-.06,13.27,;-.56,11.65,;1.22,14.12,;2.56,13.35,;2.72,11.82,;4.12,11.2,;5.37,12.1,;6.88,11.78,;7.43,10.34,;7.65,13.11,;9.18,13.27,;10.08,12.03,;11.61,12.19,;12.24,13.6,;13.77,13.76,;11.34,14.84,;9.8,14.68,;8.9,15.93,;6.62,14.26,;6.86,15.78,;5.21,13.63,;3.8,14.26,;-5.74,8.58,;-9.93,7.87,;-10.7,9.21,;-12.24,9.21,;-13.01,7.87,;-14.55,7.87,;-15.32,6.54,;-16.86,6.54,;-17.63,5.2,;-16.86,3.87,;-15.32,3.87,;-14.55,5.2,;-14.55,2.54,;-13.02,2.38,;-12.7,.87,;-14.03,.1,;-15.18,1.13,;-14.19,-1.43,;-15.6,-2.06,;-12.95,-2.34,;-14.35,-2.96,;-15.5,-3.99,;-14.03,-4.47,;-12.24,6.54,;-10.7,6.54,)|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(OC)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1)C(F)(F)F
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc3CCC(C)(C)n3c2c1
COc1nc2c(F)cc(cc2n1C(C)C)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
COc1nc2c(F)cc(cc2n1C(C)C)-c1ccnc(Nc2cc(NC(=O)C=C)c(OCCN(C)C)cc2OC)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Br)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(cc1Nc1ncc(Br)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1)[N+]([O-])=O
COCCOc1cc(OC)c(Nc2nccc(n2)-c2cc(F)c3nc(C)n(C(C)C)c3c2)cc1NC(=O)C=C
COc1cc(SCCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(OCCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N2CCC(CC2)N2CCOCC2)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COC1CCN(CC1)c1cc(OC)c(Nc2nccc(n2)-c2cc(F)c3nc(C)n(C(C)C)c3c2)cc1NC(=O)C=C
COc1cc(N2CCOCC2)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N2CCC(O)CC2)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(C#N)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C3CC3)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(CF)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NCC=C)cc1Nc1nccc(n1)-c1cnc2nc(C)n(C(C)C)c2c1
COc1nc2ncc(cc2n1C(C)C)-c1ccnc(Nc2cc(NCC=C)c(cc2OC)N(C)CCN(C)C)n1
COc1nc2ccc(cc2n1C(C)C)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2oc(=O)n(C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2cnn(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2cnn(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)c(C(C)C)n2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)cn2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(OC(C)(C)C)c2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2oc(C)nc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)oc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2ocnc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cc(F)c2nc(C)c(C(C)C)n2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2nc(C)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2ncn(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2nc(n(C(C)C)c2c1)C(F)(F)F
COc1cc(N(C)CCN(C)C)c(cc1Nc1nccc(n1)-c1cc(F)c2n(ncc2c1)C1CCCCO1)[N+]([O-])=O
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2n(C)ncc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nn(C)cc2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nn(C)c(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2nn(C)c(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2nccn2n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc2CCCn3c2c(c1)n(C(C)C)c3=O
COc1nc2cc(cc3CCCn1c23)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1ccc2ncsc2c1
CC(C)n1c(C)nc2c(F)cc(cc12)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OC(F)F)N(C)CCN(C)C)n1
CCOc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
CC(C)n1c(C)nc2c(F)cc(cc12)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OCC(F)(F)F)N(C)CCN(C)C)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1
COc1cc(ccc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc(F)c(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1)N1CCN(C)CC1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(F)c(n1)-c1cc(F)c2nc(C)c(C(C)=C)n2c1
COc1cc(ccc1Nc1ncc(F)c(n1)-c1cc(F)c2nc(C)c(C(C)=C)n2c1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc(F)c(n1)-c1cc(F)c2nc(C)cn2c1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc(F)c(n1)-c1cc(F)c2nc(C)c(C(C)C)n2c1)N1CCN(C)CC1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(C(F)F)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(OC(C)C)n(C(C)C)c2c1
CCOc1nc2c(F)cc(cc2n1C(C)C)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(SC)n(C(C)C)c2c1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc(OCC(F)F)n(C(C)C)c2c1
COCc1nc2c(F)cc(cc2n1C(C)C)-c1ccnc(Nc2cc(NC(=O)C=C)c(cc2OC)N(C)CCN(C)C)n1
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cc(F)c2nc3OC(C)(C)Cn3c2c1
COc1cc(N(C)CCN(C)C)c(cc1Nc1nccc(n1)-c1cc(F)c2nc(C)n(C(C)C)c2c1)N(C)C(=O)C=C
COc1cc(N2CCOCC2)c(NC(=O)C=C)cc1Nc1nccc(n1)-n1cc(CN(C)C)c(n1)-c1ccccc1
COCCOc1cc2c(cc1OCCOC)ncnc2Nc3cccc(c3)C#C
COc1cc2c(cc1NC(=O)/C=C/CN3CCCCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
CCCc1nc(cc2n(C)c(C(=O)N3CCN(C)CC3)c(C)c12)-n1ncc2c(C)nc(cc12)-c1cnccc1OC
COCCN1CCN(CC1)c1nc2c(nc(cc2n1C)-n1ncc2c(C)nc(cc12)-c1cnccc1OC)N1C[C@H]2C[C@@H]1CO2 |r|
COc1ccncc1-c1cc2n(ncc2c(C)n1)-c1cc2n(C)c(nc2c(n1)N1CCCCC1)N1CCN(C)CC1
COc1ccncc1-c1cc2n(ncc2c(C)n1)-c1cc2n(C)c(nc2c(n1)N1C[C@H]2C[C@@H]1CO2)N1CCN2CCC[C@@H]2C1 |r|
COc1ccncc1-c1cc2n(ncc2c(C)n1)-c1cc2n(C)c(nc2c(n1)N1C[C@H]2C[C@@H]1CO2)N1CCC(CC1)N1CCN(C)CC1 |r|
COc1ccncc1-c1cc2n(ncc2c(C)n1)-c1cc2n(C)c(nc2c(n1)N1C[C@H]2C[C@@H]1CO2)N1CCN(CC2CC2)CC1 |r|
FC(F)CN1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
COC(=O)N1CCN(CC1)c1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
FC1CNCCC1Nc1ccc(Nc2ncc3cccc(-c4cccc(NC(=O)C=C)c4)c3n2)cc1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3ccccc3)c2c1)-c1ccc(cc1)N1CCNCC1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3ccccc3)c2c1)-c1ccc2[nH]ccc2c1
CN1CCC(CC1)n1cc(cn1)-c1ccc2Nc3ccc(F)cc3N(Cc3ccccc3)C(=O)c2c1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3ccccc3)c2c1)-c1ccc(cc1)-c1cn[nH]c1
Fc1ccc2Nc3ccc(cc3C(=O)N(c3ccccc3)c2c1)-c1ccc(cc1)N1CCNCC1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3cccnc3)c2c1)-c1ccc(cc1)N1CCNCC1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3nccs3)c2c1)-c1ccc(cc1)N1CCNCC1
Fc1ccc2Nc3ccc(cc3C(=O)N(c3ccccc3)c2c1)-c1ccc2[nH]ccc2c1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3cccnc3)c2c1)-c1ccc2[nH]ccc2c1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3nccs3)c2c1)-c1ccc2[nH]ccc2c1
O=C1N(Cc2ccccc2)c2ccccc2Nc2ccc(cc12)-c1ccc(cc1)N1CCNCC1
Fc1cnc2Nc3ccc(cc3C(=O)N(Cc3ccccc3)c2c1)-c1ccc(cc1)N1CCNCC1
O=C1N(Cc2ccccc2)c2cnccc2Nc2ccc(cc12)-c1ccc(cc1)N1CCNCC1
Nc1ccc2Nc3ccc(cc3C(=O)N(Cc3ccccc3)c2c1)-c1ccc2[nH]ccc2c1
CC(=O)Nc1ccc2Nc3ccc(cc3C(=O)N(Cc3ccccc3)c2c1)-c1ccc2[nH]ccc2c1
CCC(=O)Nc1ccc2Nc3ccc(cc3C(=O)N(Cc3ccccc3)c2c1)-c1ccc2[nH]ccc2c1
CN1CCC(CC1)c1ccc(cc1)-c1ccc2Nc3ccc(F)cc3N(Cc3ccccc3)C(=O)c2c1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3cccc4cc[nH]c34)c2c1)-c1ccc(cc1)N1CCNCC1
Fc1ccc2Nc3ccc(cc3C(=O)N(Cc3ccc4cc[nH]c4c3)c2c1)-c1ccc(cc1)N1CCNCC1
CN1CCN(CC1)c1ccc(Oc2ccc3Nc4ccc(F)cc4N(Cc4ccccc4)C(=O)c3c2)cc1
Fc1ccc2Nc3ccc(Oc4ccc(cc4)N4CCNCC4)cc3C(=O)N(Cc3ccccc3)c2c1
CN1CCC(CC1)n1cc(cn1)-c1ccc2Nc3ccc(F)cc3N(Cc3cccc(F)c3)C(=O)c2c1
CN1CCC(CC1)n1cc(cn1)-c1ccc2Nc3ccc(F)cc3N(Cc3cccc(Cl)c3)C(=O)c2c1
CN1CCC(CC1)n1cc(cn1)-c1ccc2Nc3ccc(F)cc3N(Cc3cc(F)cc(F)c3)C(=O)c2c1
CN1CCC(CC1)n1cc(cn1)-c1ccc2Nc3ccc(F)cc3N(Cc3cccc4cc[nH]c34)C(=O)c2c1
Fc1ccc2Nc3ccc(Br)cc3C(=O)N(Cc3ccccc3)c2c1
c1ccc(cc1)CN2c3cc(ccc3Nc4ccccc4C2=O)F
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(C)cc1Nc1ncc(Cl)c(Nc2ccc(C)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(C)cc1Nc1ncc(Br)c(Nc2ccc(C)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N(C)C)c(C)cc1Nc1ncc(Cl)c(Nc2ccc(C)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N(C)C)c(C)cc1Nc1ncc(Br)c(Nc2ccc(C)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(C)cc1Nc1ncc(Br)c(Nc2ccc(F)cc2P(C)(C)=O)n1
CCc1cc(Nc2ncc(Br)c(Nc3ccc(C)cc3P(C)(C)=O)n2)c(OC)cc1N1CCC(CC1)N1CCN(C)CC1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(Cl)cc1Nc1ncc(Br)c(Nc2ccc(C)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(Br)cc1Nc1ncc(Br)c(Nc2ccc(C)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(C)cc1Nc1ncc(Cl)c(Nc2cccc(C)c2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(C)cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccc(C)cc2P(C)(C)=O)n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(N2CCN(C)CC2)c(C)cc1Nc1ncc(Br)c(Nc2ccc(C)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(C)cc1Nc1ncc(Br)c(Nc2ccc(Cl)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(Cl)cc1Nc1ncc(Br)c(Nc2ccc(F)cc2P(C)(C)=O)n1
COc1cc(N2CCC(CC2)N2CCN(C)CC2)c(C)cc1Nc1ncc(Br)c(Nc2ccc(cc2P(C)(C)=O)C(C)C)n1
CCc1cc(Nc2ncc(Br)c(Nc3ccc(cc3P(C)(C)=O)C(C)C)n2)c(OC)cc1N1CCC(CC1)N1CCN(C)CC1
CN1CCN(CC1)C2CCN(CC2)c3ccc(c(c3)OC)Nc4ncc(c(n4)Nc5ccccc5P(=O)(C)C)Cl
C[C@@H]1CCCOc2c(cnn2C)-c2cc(NC(=O)C=C)cc(c2)C(=O)Nc2nc3ccc(Br)cc3n2C1 |r|
C[C@@H]1CCCOc2c(cnn2C)-c2sc(cc2NC(=O)C=C)C(=O)Nc2nc3ccc(Br)cc3n2C1 |r|
Cn1ncc-2c1OCCCOc1ccccc1\C=C\c1n[nH]c3cnc-2cc13 |t:19|
Cn1ncc-2c1OCCCOc1ccccc1\C=C\c1n[nH]c3ccc-2nc13 |t:19|
Cn1ncc-2c1OCCCOc1ccccc1\C=C\c1n[nH]c3ccc-2cc13 |t:19|
Cn1ncc-2c1COCCOc1ccccc1\C=C\c1n[nH]c3cnc-2nc13 |t:19|
CCc1nn(C)c2c1\C=C\c1n[nH]c3cnc(cc13)-c1cc(F)ccc1OCCN(C)C2=O |t:9|
Cn1ncc-2c1COCCOc1ccccc1\C=C\c1n[nH]c3cnc-2cc13 |t:19|
CC1OCCOc2ccc(C)nc2\C=C\c2n[nH]c3cnc(nc23)-c2cnn(C)c12 |t:14|
CN1CCOCCN(c2ccc(F)c(Cl)c2)c2cc3c(\C=C\c4cn(C)nc4C1=O)n[nH]c3cn2 |t:21|
C=CC(=O)NC1=CC(Nc2nccc(N3CC(CN(C)C)C(c4ccccc4)=N3)n2)C(OC)N=C1N1CCOCC1
C=CC(=O)Nc1cc(Nc2ncc(F)c(-n3cc(CN(C)C)c(-c4ccccc4)n3)n2)c(OC)nc1N1CCOCC1
C=CC(=O)Nc1cc(Nc2ncc(C)c(-n3cc(CN(C)C)c(-c4ccccc4)n3)n2)c(OC)nc1N1CCOCC1
C=CC(=O)Nc1cc(Nc2nccc(-n3cc(CN(C)C)c(-c4ccccc4)n3)n2)c(OC(C)C)nc1N1CCOCC1
C=CC(=O)Nc1cc(Nc2nccc(-n3cc(CN(C)C)c(-c4ccccc4)n3)n2)c(OC)nc1N1CCOCC1
O=C(Nc1nccs1)C(c1cccc(F)c1)N1Cc2cnc(Br)cc2C1=O
O=C(Nc1nccs1)C(c1cccc(F)c1)N1Cc2ncc(Br)cc2C1=O
O=C(Nc1ccccn1)C(c1cccc(F)c1)N1Cc2ncc(Br)cc2C1=O
O=C(Nc1nccs1)C(c1cccc(F)c1)N1Cc2ccc(Br)nc2C1=O
O=C(Nc1ccccn1)C(c1cccc(F)c1)N1Cc2ccc(Br)nc2C1=O
CN1CCC(c2ccc(-c3cc4c(cn3)CN(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4=O)cc2)CC1
CN1CCN(c2ccc(-c3cc4c(cn3)CN(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4=O)cc2)CC1
CN1CCN(c2ccc(-c3cnc4c(c3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cn2)CC1
CN1CCC(c2ccc(-c3cnc4c(c3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cc2)CC1
CN1CCN(c2ccc(-c3cnc4c(c3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cc2)CC1
CN1CCC(c2ccc(-c3cnc4c(c3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cc2)C1
CN1CCN(c2ccc(-c3cnc4c(c3)C(=O)N(C(C(=O)Nc3ccccn3)c3cccc(F)c3)C4)cn2)CC1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cc2)CC1
CN1CCN(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cc2)CC1
CN1CCN(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cn2)CC1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cc2)C1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cn2)CC1
CN1CCC(c2ccc(-c3cnc4c(c3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cn2)CC1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)c(F)c2)CC1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4)cc2F)CC1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N(C(C(=O)Nc3ccccn3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3cnc4c(c3)C(=O)N(C(C(=O)Nc3ccccn3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3)cc2F)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5ccccc5)c5nc6ccccc6[nH]5)c(=O)c4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5ccccc5)c5nc6ccccc6[nH]5)c(=O)c4c3F)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3F)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5cccc(F)c5)c5nc6ccccc6[nH]5)c(=O)c4c3F)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3F)cc2F)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5cccc(F)c5)c5nc6ccccc6[nH]5)c(=O)c4n3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4n3)cc2)CC1
CN1CCC(c2ccc(-c3cnc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(C#Cc2ccc3c(c2)C(=O)N(C(c2nc4ccccc4[nH]2)c2cc(F)ccc2O)C3)CC1
Nc1ccc(C#Cc2ccc3c(c2)C(=O)N(C(c2nc4ccccc4[nH]2)c2cc(F)ccc2O)C3)cn1
O=C1c2cc(C#CCN3CCS(=O)(=O)CC3)ccc2CN1C(c1nc2ccccc2[nH]1)c1cc(F)ccc1O
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5cccnc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5cnccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(F)(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2F)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5cncnc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5nccnc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
Oc1ccc(F)cc1C(N1Cc2ccc(cc2C1=O)-c1ccc(cc1)N1CCNCC1)c1nc2ccccc2[nH]1
CN1CCC(c2ccc(-c3ccc4c(c3)CN([C@@H](c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N([C@H](c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3cccc(F)c3)c3nc5cccnc5[nH]3)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3cccc(F)c3)c3nc5ccccc5[nH]3)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)c(F)c2)CC1
Nc1ccc(C#Cc2ccc3c(n2)C(=O)N(C(c2nc4ccccc4[nH]2)c2n[nH]c4c2CCC4)C3)cn1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5cccnc5[nH]3)c3n[nH]c5c3CCC5)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3F)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3n[nH]c5c3CCC5)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4cn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)nc4c3F)cc2)CC1
COc1ccc(F)cc1C(c1nc2ccccc2[nH]1)n1cc2ccc(-c3ccc(C4CCN(C)CC4)cc3)c(F)c2n1
[2H]C(c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)N1Cc2ccc(-c3ccc(C4CCN(C)CC4)cc3)cc2C1=O
[2H][C@@](c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)N1Cc2ccc(-c3ccc(C4CCN(C)CC4)cc3)cc2C1=O
[2H][C@](c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)N1Cc2ccc(-c3ccc(C4CCN(C)CC4)cc3)cc2C1=O
[2H]C1([2H])c2ccc(-c3ccc(C4CCN(C)CC4)cc3)cc2C(=O)N1C([2H])(c1nc2ccccc2[nH]1)c1cc(F)ccc1O
CN(C)CCOc1ccc(-c2ccc3c(c2)C(=O)N(C(c2nc4ccccc4[nH]2)c2cc(F)ccc2O)C3)cc1
CN(C)CCN(C)c1ccc(-c2ccc3c(c2)C(=O)N(C(c2nc4ccccc4[nH]2)c2cc(F)ccc2O)C3)cc1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cccc(F)c3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cccc(Cl)c3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)CN(C(c3nc5ccccc5[nH]3)c3cc(Cl)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3ccn[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5cc(F)ccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5c(Cl)cccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
COc1ccc2[nH]c(C(c3cc(F)ccc3O)N3Cc4ccc(-c5ccc(C6CCN(C)CC6)cc5)cc4C3=O)nc2c1
CN1CC(c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)C1
Cc1ccc2[nH]c(C(c3cc(F)ccc3O)N3Cc4ccc(-c5ccc(C6CCN(C)CC6)cc5)cc4C3=O)nc2c1
COc1cccc2[nH]c(C(c3cc(F)ccc3O)N3Cc4ccc(-c5ccc(C6CCN(C)CC6)cc5)cc4C3=O)nc12
Cc1cccc2[nH]c(C(c3cc(F)ccc3O)N3Cc4ccc(-c5ccc(C6CCN(C)CC6)cc5)cc4C3=O)nc12
CN1CCC(c2ccc(-c3ccc4c(=O)n(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)cc(F)c4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(F)cn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3)cc2)CC1
Cc1c(-c2ccc(C3CCN(C)CC3)cc2)ccc2ncn(C(c3nc4ccccc4[nH]3)c3cc(F)ccc3O)c(=O)c12
CN1CC(Oc2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)C1
Oc1ccc(F)cc1C(c1nc2ccccc2[nH]1)N1Cc2ccc(-c3ccc(-c4cn[nH]c4)cc3)cc2C1
Cn1cc(-c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)cn1
Oc1ccc(F)cc1C(N1Cc2ccc(cc2C1=O)-c1ccc(cc1)N1CCOCC1)c1nc2ccccc2[nH]1
CN1CCC(n2cc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cn2)CC1
Nc1ccc(-c2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)cn1
O=C1c2cc(-c3ccc(C4CCNCC4)cc3)ccc2CN1C(c1nc2ccccc2[nH]1)c1cc(F)ccc1O
CN1CCC(c2ccc(-c3ccc4ccn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3)cc2)CC1
CN1CCC(c2ccc(-c3cc(F)c4c(=O)n(C(c5ccccc5)c5nc6ccccc6[nH]5)ccc4c3)cc2)CC1
CN1CCC(c2ccc(-c3cc(F)c4c(=O)n([C@@H](c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2)CC1
CN1CCC(c2ccc(-c3cc(F)c4c(=O)n([C@H](c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(=O)n([C@@H](c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(=O)n([C@H](c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(=O)n(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2)CC1
CN1CCC(c2ccc(-c3cc(F)c4c(=O)n(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ccn(C(c5ccccc5)c5nc6ccccc6[nH]5)c(=O)c4c3F)cc2)CC1
CN1CCC(c2ccc(-c3cc4ccn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4cc3F)cc2)CC1
CCc1c(-c2ccc(C3CCN(C)CC3)cc2)ccc2ncn(C(c3nc4ccccc4[nH]3)c3cc(F)ccc3O)c(=O)c12
CN1CCC(c2ccc(-c3ccc4ncn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3Cl)cc2)CC1
CN1CCC(c2ccc(-c3ccc4ncn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)c(=O)c4c3C(F)(F)F)cc2)CC1
COc1c(-c2ccc(C3CCN(C)CC3)cc2)ccc2ncn(C(c3nc4ccccc4[nH]3)c3cc(F)ccc3O)c(=O)c12
CN1CCC(c2ccc(-c3ccc4c(c3)C(=S)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC2(c3ccc(-c4ccc5c(c4)C(=O)N(C(c4nc6ccccc6[nH]4)c4cc(F)ccc4O)C5)cc3)CC2C1
CN1CCC(c2ccc(-c3ccc4c(c3F)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2F)CC1
CN1CCC(c2ccc(-c3ccc4c(c3F)C(=O)N(C(c3nc5c(F)cccc5[nH]3)c3cc(F)ccc3O)C4)cc2F)CC1
Cc1c(-c2ccc(C3CCN(C)CC3)cc2)ccc2c1C(=O)N(C(c1nc3ccccc3[nH]1)c1cc(F)ccc1O)C2
CN1CCC(c2ccc(-c3ccc4c(c3)C(=S)N([C@@H](c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(c3)C(=S)N([C@H](c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
Cc1c[nH]c(C(c2cc(F)ccc2O)N2Cc3ccc(-c4ccc(C5CCN(C)CC5)cc4)cc3C2=O)n1
Cc1c[nH]c(C(c2cccc(F)c2)N2Cc3ccc(-c4ccc(C5CCN(C)CC5)cc4)cc3C2=O)n1
Cc1nc(C(c2cc(F)ccc2O)N2Cc3ccc(-c4ccc(C5CCN(C)CC5)cc4)cc3C2=O)[nH]c1C
CN1CCC(Oc2ccc(-c3ccc4c(c3)C(=O)N(C(c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
O=C1c2cc(-c3ccc(OC4CNC4)cc3)ccc2CN1C(c1nc2ccccc2[nH]1)c1cc(F)ccc1O
CN1CCC(c2ccc(-c3ccc4cn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)nc4c3Cl)cc2)CC1
Cc1cnc(C(c2cc(F)ccc2O)N2Cc3ccc(-c4ccc(C5CCN(C)CC5)cc4)c(F)c3C2=O)[nH]1
CC1=CNC([C@H](c2cc(F)ccc2O)N2CC3=CC=C(c4ccc(C5CCN(C)CC5)cc4)C(F)C3C2=O)N1
Cc1c[nH]c([C@H](c2cc(F)ccc2O)N2Cc3ccc(-c4ccc(C5CCN(C)CC5)cc4)c(F)c3C2=O)n1
Cc1c(-c2ccc(C3CCN(C)CC3)cc2)ccc2cn(C(c3nc4ccccc4[nH]3)c3cc(F)ccc3O)nc12
CN1CCC(c2ccc(-c3cc4nn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)cc4cc3O)cc2)CC1
Cc1cc2cn(C(c3nc4ccccc4[nH]3)c3cc(F)ccc3O)nc2cc1-c1ccc(C2CCN(C)CC2)cc1
COc1cc2cn(C(c3nc4ccccc4[nH]3)c3cc(F)ccc3O)nc2cc1-c1ccc(C2CCN(C)CC2)cc1
CN1CCC(c2ccc(-c3ccc4cn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)nc4c3)cc2)CC1
CN1CCC(c2ccc(-c3ccc4cn(C(c5nc6c(F)cccc6[nH]5)c5cc(F)ccc5O)nc4c3F)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(=O)n(C(c5nc6c(F)cccc6[nH]5)c5cc(F)ccc5O)cnc4c3)cc2)CC1
Cc1c[nH]c([C@@H](c2cc(F)ccc2O)N2Cc3ccc(-c4ccc(C5CCN(C)CC5)cc4)cc3C2=O)n1
Cc1c[nH]c([C@H](c2cc(F)ccc2O)N2Cc3ccc(-c4ccc(C5CCN(C)CC5)cc4)cc3C2=O)n1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N([C@@H](c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC(c2ccc(-c3ccc4c(n3)C(=O)N([C@H](c3nc5ccccc5[nH]3)c3cc(F)ccc3O)C4)cc2)CC1
CN1CCC2(c3ccc(-c4ccc5c(=O)n(C(c6nc7ccccc7[nH]6)c6cc(F)ccc6O)ccc5c4)cc3)CC2C1
CN1CCC(c2ccc(-c3ccc4c(=O)n(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2F)CC1
CN1CCC2(c3ccc(-c4cc(F)c5c(=O)n(C(c6nc7ccccc7[nH]6)c6cc(F)ccc6O)ccc5c4)cc3)CC2C1
CN1CCC(c2ccc(-c3cc(F)c4c(=O)n(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)ccc4c3)cc2F)CC1
[2H]C(c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)n1ccc2cc(-c3ccc(C4CCN(C)CC4)cc3)ccc2c1=O
[2H]C(c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)n1ccc2cc(-c3ccc(C4CCN(C)CC4)cc3)cc(F)c2c1=O
[2H][C@](c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)n1ccc2cc(-c3ccc(C4CCN(C)CC4)cc3)ccc2c1=O
[2H][C@@](c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)n1ccc2cc(-c3ccc(C4CCN(C)CC4)cc3)ccc2c1=O
[2H][C@](c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)n1ccc2cc(-c3ccc(C4CCN(C)CC4)cc3)cc(F)c2c1=O
[2H][C@@](c1nc2ccccc2[nH]1)(c1cc(F)ccc1O)n1ccc2cc(-c3ccc(C4CCN(C)CC4)cc3)cc(F)c2c1=O
CN1CCC(c2ccc(-c3cc4nn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)cc4cc3F)cc2)CC1
CN1CCC(c2ccc(-c3cc(F)c4cn(C(c5nc6ccccc6[nH]5)c5cc(F)ccc5O)nc4c3)cc2)CC1