8101 SMILES Strings for Orexin/Hypocretin receptor type 1

Compound Name
SMILES String
CCOC(=O)c1cnc(s1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1ncc(s1)C(C)(C)O |r|
C[C@@H]1CC[C@@H](CN1C(=O)c1ccccc1-n1nccn1)c1ncc(s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnc(s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(cs1)[C@H](O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(cs1)[C@@H](O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(cs1)[C@H](O)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(cs1)[C@@H](O)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1nc(cs1)C(C)(C)O |r|
COC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1nc(cs1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)c1nc(c(C)s1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1csc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)c1csc(n1)C(C)(C)O |r|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2ccccc2-c2cccs2)nc1 |THB:6:7:11.10:13|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1nccc(n1)C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1ccc(cn1)C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1ncccc1C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1cccc(n1)C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccnc(OCC2CC3CCC2N3C(=O)c2cc(C)ccc2-n2nccn2)c1 |THB:7:8:12.11:14|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1cccc(C)n1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(OCC2CC3CCC2N3C(=O)c2cc(C)ccc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1nc(C)cnc1C)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1nc3ccccc3nc1C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cccc3cccnc23)nc1 |THB:6:7:11.10:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cccc3ccccc23)nc1 |THB:6:7:11.10:13|
Cc1ccc2ccccc2c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:19:18:16.15:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2ccccc2-n2cccn2)nc1 |THB:6:7:11.10:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2occc2-c2ccccc2)nc1 |THB:6:7:11.10:13|
CCOc1ccc2ccccc2c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1nc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c(s1)-c1ccccc1F |TLB:12:11:9.8:6|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cc(F)ccc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2c(F)cccc2-c2ncccn2)nc1 |THB:6:7:11.10:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cc(F)ccc2-c2ncccn2)nc1 |THB:6:7:11.10:13|
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
O=C(N1C2CCC1C(COc1cnc3ccccc3n1)C2)c1ccccc1-n1nccn1 |TLB:8:7:5.4:2|
Fc1cccc(c1C(=O)N1C2CCC1C(COc1cnc3ccccc3n1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1cnc3ccccc3n1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Fc1ccc(c(c1)C(=O)N1C2CCC1C(COc1cnc3ccccc3n1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(COc1cnc3ccccc3n1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1nc(C)cc(C)n1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1noc(c1C(=O)N1C2CCC1C(COc1nc(C)cc(C)n1)C2)-c1ccccc1 |TLB:14:13:11.10:8|
CCOc1ccc2ccccc2c1C(=O)N1C2CCC1C(COc1nc(C)cc(C)n1)C2 |TLB:21:20:18.17:15|
CCOc1ccccc1C(=O)N1C2CCC1C(COc1nc(C)cc(C)n1)C2 |TLB:17:16:14.13:11|
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2c(F)cccc2-c2ncccn2)n1 |THB:8:9:13.12:15|
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2cc(F)ccc2-c2ncccn2)n1 |THB:8:9:13.12:15|
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(COc1nc(C)cc(C)n1)C2 |TLB:21:20:18.17:15|
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2ccccc2-c2cccs2)n1 |THB:8:9:13.12:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccc(cn1)C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccc(cn1)C(F)(F)F)C2 |TLB:18:17:15.14:12|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccc(Br)cn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
COc1c(F)cccc1C(=O)N1C2CCC1C(COc1ccc(Br)cn1)C2 |TLB:17:16:14.13:11|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccc(Br)cn1)C2 |TLB:18:17:15.14:12|
Fc1cccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c1-c1ncccn1 |TLB:14:13:11.10:8|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1cccnn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1cccnc1C)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ncccc1C)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccnn1C)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccncc1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1cccnc1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ncccn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1cnccn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccncn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1cccc(OCC2CC3CCC2N3C(=O)c2nc(C)ccc2-n2nccn2)n1 |THB:7:8:12.11:14|
Cc1ccc(-c2ncco2)c(n1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:20:19:17.16:14|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-c1ncccc1C |TLB:15:14:12.11:9|
Cc1noc(n1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1ccn(n1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(N2CCCC2)c(n1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:20:19:17.16:14|
Cc1cc(on1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1cccn1 |TLB:15:14:12.11:9|
Cc1cnc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(c1)-n1nccn1 |TLB:13:12:10.9:7|
Cc1ccnc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c1-n1nccn1 |TLB:14:13:11.10:8|
CN(C)c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
O=C(N1C2CCC1C(COc1ccccn1)C2)c1nc2ccccc2cc1-n1nccn1 |TLB:8:7:5.4:2|
CCOc1ccc2cccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1cnc2ccc(C)c(C(=O)N3C4CCC3C(COc3ccccn3)C4)n12 |TLB:18:17:15.14:12|
Cn1cc(c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2)-c1ccccc1 |TLB:14:13:11.10:8|
Cn1cc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(n1)-c1ccccc1 |TLB:12:11:9.8:6|
Cc1cnc2c(C(=O)N3C4CCC3C(COc3ccccn3)C4)c(C)ccn12 |TLB:14:13:11.10:8|
Cc1ccn2ccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
Cn1ncc(c1C(=O)N1C2CCC1C(COc1ccccn1)C2)-c1ccccc1 |TLB:14:13:11.10:8|
Cc1ccc2nccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
CCOc1ncc2ccccc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cn1ncc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c1-c1ccccc1 |TLB:13:12:10.9:7|
CN1CCN(CC1)c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:22:21:19.18:16|
Cc1ccc(N2CCNCC2)c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(N2CCOCC2)c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
COc1ccc2cccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:20:19:17.16:14|
CCOc1ccc2ccccc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2)-c1ncccc1C |TLB:15:14:12.11:9|
O=C(N1C2CCC1C(COc1ccccn1)C2)c1ncccc1-n1nccn1 |TLB:8:7:5.4:2|
Cc1nc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(s1)-c1ccccc1 |TLB:12:11:9.8:6|
Cc1ccc(-c2ncco2)c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:20:19:17.16:14|
Cc1cc(on1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2)-n1cccn1 |TLB:15:14:12.11:9|
Cc1cnn(c1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(N2CCCC2)c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:20:19:17.16:14|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2)-c1ncccc1C |TLB:15:14:12.11:9|
Cc1cc(on1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(-c2ncco2)c(n1)C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2 |TLB:20:19:17.16:14|
Cc1ccc(N2CCCC2)c(n1)C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2 |TLB:20:19:17.16:14|
Cc1cnn(c1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2)-n1cccn1 |TLB:15:14:12.11:9|
COc1cccc(OC)c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:18:17:15.14:12|
COc1c(F)cccc1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:17:16:14.13:11|
COc1cccc(c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1nccn1 |TLB:16:15:13.12:10|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cc(F)ccc2-c2ccn[nH]2)nc1 |THB:6:7:11.10:13|
Cc1cccc(c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2ncc(Cl)cc2-n2nccn2)nc1 |THB:6:7:11.10:13|
COc1cnc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c(c1)-n1nccn1 |TLB:14:13:11.10:8|
COc1ccc(c(c1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1nccn1 |TLB:16:15:13.12:10|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2c(F)cccc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2ccc(F)cc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cccc(F)c2-n2nccn2)nc1 |THB:6:7:11.10:13|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:18:17:15.14:12|
COc1ccc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c(c1)-n1nccn1 |TLB:14:13:11.10:8|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cc(Cl)ccc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Cc1ccc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c(c1)-n1nccn1 |TLB:13:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c(c1)-c1ncccn1 |TLB:13:12:10.9:7|
Cc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
Fc1ccc(OCC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)nc1 |THB:6:7:11.10:13|
Cc1cccc(C(=O)N2C3CCC2C(COc2ccc(F)cn2)C3)c1-n1nccn1 |TLB:14:13:11.10:8|
OCc1ccc(c(c1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1nccn1 |TLB:16:15:13.12:10|
Cc1noc(n1)-c1ccccc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:20:19:17.16:14|
Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(n1)-n1nccn1 |TLB:13:12:10.9:7|
Fc1cccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c1-n1nccn1 |TLB:14:13:11.10:8|
Cc1ccc(C(=O)N2C3CCC2C(COc2ccccn2)C3)c(n1)-n1ccnn1 |TLB:13:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(n2)C(F)(F)F)C3)c(n1)-n1nccn1 |TLB:13:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(COc2nccc(n2)C(F)(F)F)C3)c(n1)-n1ccnn1 |TLB:13:12:10.9:7|
Cc1noc(n1)-c1ccccc1C(=O)N1C2CCC1C(COc1nccc(n1)C(F)(F)F)C2 |TLB:20:19:17.16:14|
Fc1cccc(C(=O)N2C3CCC2C(COc2nccc(n2)C(F)(F)F)C3)c1-n1nccn1 |TLB:14:13:11.10:8|
Cc1ccc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Cc1ccc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2ccnn2)nc1 |THB:6:7:11.10:13|
Cc1noc(n1)-c1ccccc1C(=O)N1C2CCC1C(COc1ccc(C)cn1)C2 |TLB:20:19:17.16:14|
Cc1ccc(OCC2CC3CCC2N3C(=O)c2cccc(F)c2-n2nccn2)nc1 |THB:6:7:11.10:13|
Cc1cccc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2nccn2)n1 |THB:7:8:12.11:14|
Cc1cccc(OCC2CC3CCC2N3C(=O)c2ccc(C)nc2-n2ccnn2)n1 |THB:7:8:12.11:14|
Cc1noc(n1)-c1ccccc1C(=O)N1C2CCC1C(COc1cccc(C)n1)C2 |TLB:20:19:17.16:14|
Cc1cccc(OCC2CC3CCC2N3C(=O)c2cccc(F)c2-n2nccn2)n1 |THB:7:8:12.11:14|
Cc1ccc(C(=O)N2C3CCC2C(COc2cccc(n2)C(F)(F)F)C3)c(n1)-n1nccn1 |TLB:13:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(COc2cccc(n2)C(F)(F)F)C3)c(n1)-n1ccnn1 |TLB:13:12:10.9:7|
Cc1noc(n1)-c1ccccc1C(=O)N1C2CCC1C(COc1cccc(n1)C(F)(F)F)C2 |TLB:20:19:17.16:14|
Fc1cccc(C(=O)N2C3CCC2C(COc2cccc(n2)C(F)(F)F)C3)c1-n1nccn1 |TLB:14:13:11.10:8|
Cc1ccc(C(=O)N2C3CCC2C(COc2cnc4ccccc4n2)C3)c(n1)-n1ccnn1 |TLB:13:12:10.9:7|
Cc1noc(n1)-c1ccccc1C(=O)N1C2CCC1C(COc1cnc3ccccc3n1)C2 |TLB:20:19:17.16:14|
Fc1cccc(C(=O)N2C3CCC2C(COc2cnc4ccccc4n2)C3)c1-n1nccn1 |TLB:14:13:11.10:8|
Cc1ccc(C(=O)N2C3CCC2C(COc2nc(C)cc(C)n2)C3)c(n1)-n1nccn1 |TLB:13:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(COc2nc(C)cc(C)n2)C3)c(n1)-n1ccnn1 |TLB:13:12:10.9:7|
Cc1noc(n1)-c1ccccc1C(=O)N1C2CCC1C(COc1nc(C)cc(C)n1)C2 |TLB:20:19:17.16:14|
Cc1cc(C)nc(OCC2CC3CCC2N3C(=O)c2cccc(F)c2-n2nccn2)n1 |THB:8:9:13.12:15|
CCOc1nccc(C)c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
Cc1nc2sccn2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:17:16:14.13:11|
CCOc1ncc(Br)cc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
CCOc1nc(C)ccc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
Oc1ccc2cccnc2c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:19:18:16.15:13|
CCOc1ncc(cc1C(=O)N1C2CCC1C(COc1ccccn1)C2)-c1ccccc1 |TLB:17:16:14.13:11|
CCOc1nccc(Br)c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
CCOc1ccnc(Cl)c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:18:17:15.14:12|
CCOc1ccnc(OCC)c1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:20:19:17.16:14|
CCOc1ccccc1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:17:16:14.13:11|
Cc1ccc(C(=O)N2C3CCC2C(COc2cnc4ccccc4n2)C3)c(n1)-n1nccn1 |TLB:13:12:10.9:7|
Fc1ccc(c(c1)C(=O)N1C2CCC1C(CNc1ccccn1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1cc(C)nc(NCC2CC3CCC2N3C(=O)c2cc(F)ccc2-n2nccn2)n1 |THB:8:9:13.12:15|
Fc1ccc(c(c1)C(=O)N1C2CCC1C(CNc1nccc(n1)C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
Fc1ccc(c(c1)C(=O)N1C2CCC1C(CNc1cccc(n1)C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
Fc1ccc(c(c1)C(=O)N1C2CCC1C(CNc1cnc3ccccc3n1)C2)-n1nccn1 |TLB:15:14:12.11:9|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1coc(n1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2 |TLB:21:20:18.17:15|
Cc1coc(n1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
Cc1ccc(c(c1)C(=O)N1C2CCC1C(COc1cc(C)nc(n1)C(F)(F)F)C2)-n1nccn1 |TLB:15:14:12.11:9|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)cn1 |THB:8:9:13.12:15|
Cc1cnc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-n1nccn1 |TLB:14:12:10.9:7|
Cc1cnc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-n1ccnn1 |TLB:14:12:10.9:7|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Cc1cnc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c(c1)-n1nccn1 |TLB:14:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c(n1)-n1nccn1 |TLB:14:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c(n1)-n1ccnn1 |TLB:14:12:10.9:7|
COc1ccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c(c1)-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:18:16:14.13:11|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:19:17:15.14:12|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
FC(F)(F)c1ccc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nc1 |THB:8:9:13.12:15|
Cc1cc(C)nc(NC2CC3CCC2N3C(=O)c2cc(F)ccc2-n2nccn2)n1 |THB:7:8:12.11:14|
Cc1cc(C)nc(NC2CC3CCC2N3C(=O)c2c(F)cccc2-n2nccn2)n1 |THB:7:8:12.11:14|
Cc1cc(C)nc(NC2CC3CCC2N3C(=O)c2ccc(F)cc2-n2nccn2)n1 |THB:7:8:12.11:14|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(C2)Nc1nc(C)cc(C)n1 |TLB:22:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1nc(C)cc(C)n1)-n1nccn1 |TLB:16:14:12.11:9|
Cc1cc(C)nc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)n1 |THB:7:8:12.11:14|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1nc(C)cc(C)n1 |TLB:19:17:15.14:12|
O=C(N1C2CCC1C(C2)Nc1cnc2ccccc2n1)c1ccccc1-n1nccn1 |TLB:9:7:5.4:2|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1cnc2ccccc2n1)-n1nccn1 |TLB:16:14:12.11:9|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1cnc2ccccc2n1 |TLB:18:16:14.13:11|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1cnc2ccccc2n1 |TLB:19:17:15.14:12|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(C2)Nc1cnc2ccccc2n1 |TLB:22:20:18.17:15|
FC(F)(F)c1cccc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)n1 |THB:9:10:14.13:16|
FC(F)(F)c1ccnc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)c1 |THB:9:10:14.13:16|
Clc1ccc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nc1 |THB:5:6:10.9:12|
FC(F)(F)c1ccc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nn1 |THB:8:9:13.12:15|
COc1ccc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nc1 |THB:6:7:11.10:13|
Cc1ccc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nc1 |THB:5:6:10.9:12|
O=C(N1C2CCC1C(C2)Nc1ccccn1)c1ccccc1-n1nccn1 |TLB:9:7:5.4:2|
Clc1ccc2oc(NC3CC4CCC3N4C(=O)c3ccccc3-n3nccn3)nc2c1 |THB:7:8:12.11:14|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(C2)Nc1ccc(Br)cn1 |TLB:22:20:18.17:15|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1ccc(Br)cn1 |TLB:18:16:14.13:11|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1ccc(Br)cn1 |TLB:19:17:15.14:12|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1ccc(Br)cn1)-n1nccn1 |TLB:16:14:12.11:9|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nc1 |THB:8:9:13.12:15|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F |TLB:18:16:14.13:11|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F |TLB:19:17:15.14:12|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1ccc(F)cn1)-n1nccn1 |THB:16:14:12.11:9|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1ccc(F)cn1 |THB:18:16:14.13:11|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
CCOc1ccc2ccccc2c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2cncc3ccccc23)cn1 |THB:8:9:13.12:15|
COc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-n1nccn1 |TLB:15:13:11.10:8|
COc1cccc(c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:17:15:13.12:10|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Cc1nc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(s1)-c1ccc(F)cc1 |TLB:13:11:9.8:6|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
CCOc1ncc2ccccc2c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Cc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(n1)-n1nccn1 |TLB:14:12:10.9:7|
Cc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(n1)-n1ccnn1 |TLB:14:12:10.9:7|
COc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:15:13:11.10:8|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2nc3ccccc3[nH]2)cn1 |THB:8:9:13.12:15|
Cn1c(nc2ccccc12)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:19:17:15.14:12|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
FC(F)Oc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-n1nccn1 |TLB:17:15:13.12:10|
Cc1noc(n1)-c1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
COc1ccc(c(c1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:17:15:13.12:10|
Fc1ccc(c(c1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Fc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-n1nccn1 |TLB:14:12:10.9:7|
Fc1cccc(c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Cc1nc2sccn2c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:18:16:14.13:11|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1nc(C)cc(C)n1 |TLB:18:16:14.13:11|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1cccnn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1cccnn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ccnnc1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1cnccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:14:12:10.9:7|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ccncc1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2nccn3c(Br)cnc23)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2nccn3c(nnc23)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
COC(=O)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1 |THB:8:9:13.12:15|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1I |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1I |TLB:15:13:11.10:8|
Cc1cnc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)cn1 |THB:5:6:10.9:12|
Fc1ccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:14:12:10.9:7|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
CN(C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1)c1cnc(cn1)C(F)(F)F |THB:1:2:6.5:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ncc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:19:17:15.14:12|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ncccc2-n2nccn2)cn1 |THB:8:9:13.12:15|
COc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:23:21:19.18:16|
Fc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
CCOc1ccc2cccnc2c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
COc1cccc(-c2c(C)cnn2C)c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:24:22:20.19:17,(-3.4,-1.05,;-4.89,-.65,;-5.29,.84,;-6.78,1.24,;-7.18,2.72,;-6.09,3.81,;-4.6,3.41,;-3.51,4.5,;-1.97,4.5,;-1.2,3.17,;-1.49,5.97,;-2.74,6.87,;-3.99,5.97,;-5.32,6.74,;-4.2,1.93,;-2.71,1.53,;-1.62,2.62,;-2.31,.04,;-1.54,-1.29,;-3.03,-1.69,;-3.8,-3.02,;-2.31,-2.62,;-.83,-3.02,;-.05,-1.69,;.51,-2.25,;1.84,-3.02,;1.84,-4.56,;3.17,-5.33,;4.51,-4.56,;4.51,-3.02,;3.17,-2.25,;5.84,-5.33,;7.18,-4.56,;5.84,-6.87,;7.18,-6.1,)|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c1-c1ccccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
COC(=O)c1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
COC(=O)c1cc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)ncc1C(F)(F)F
COC(=O)c1cc(O[C@@H]2CC[C@@H](C)N(Cc3ccccc3-n3nccn3)C2)ncc1Br
COC(=O)c1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1Cl
COC(=O)c1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C(=O)OC
COC(=O)c1cc(C)nc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1
COC(=O)c1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1F
COC(=O)c1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(OC)nc2-n2nccn2)c1
COC(=O)c1cc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)ncc1Br |r|
COC(=O)c1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(OC)nc2-c2ncccn2)c1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2OC)c(n1)-c1ncccn1 |r|
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccnc2-n2ncnn2)nccc1C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Cl)ccc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(Cl)cc1-n1nccn1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)C1CC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(c1)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C)cc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cnccc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(C)c1-n1nccn1)Oc1nccc(C#N)c1C |r|
COc1cccc(c1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(C)cccc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CC1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C(F)(F)F)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-c1nccs1)Oc1nccc(C#N)c1C |r|
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1sncc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
CC(C)Oc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-c1cscn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccncc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ncccc1-c1cscn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ncc1-c1cncs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1cscn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncco1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1nccs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1N1CCCC1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1Oc1ccccc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1cscn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1nccs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1cscn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1nccs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)cnc1-c1nccs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1cnn(C)c1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1sccc1-c1nccs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1sccc1-c1cscn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nnc(C)n1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nc(C)sc1-c1ccc(F)cc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1noc(C)n1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1cc(C)cn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1nccs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cn(C)nc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cn(C)nc1-c1nccs1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(C)nsc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-c1ccncc1 |r|
COc1ccc(cn1)-c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nscc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C)cc1C1CC1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(c1)C1CC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1C1CC1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(CO)cc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nscc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1ccccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nc(C)sc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1nc(C)no1)Oc1nccc(C#N)c1C |r|
CCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
CSc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)(F)F)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)C1=C(CCC1)c1ccccn1)Oc1nccc(C#N)c1C |r,t:10|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(OCF)cc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(OC(F)F)cc1-n1nccn1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)C1CCC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cnc(Cl)cc1-n1nccn1)Oc1nccc(C#N)c1C |r|
CCOc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(ccc1-n1nccn1)C#N)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(Cl)nc1-n1nccn1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(OC)n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1sccc1-c1ncccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C)cc1-c1ncccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1nccc(C#N)c1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-c1ccccc1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-c1ccnn1C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-c1cnn(C)c1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-c1ccn(C)n1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-c1cccnc1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-c1ccccn1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(SC)n1 |r|
COc1cc(c(cn1)C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccc(C#N)c1C)-n1nccn1 |r|
CSc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)-n1nccn1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2C)c(n1)N(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(OCF)nc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(Br)nc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C=C)nc1-n1nccn1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc(C#N)c1Cl |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc(C#N)c1C1CC1 |r|
CCc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc(C#N)c1C#N |r|
CSc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(F)c2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(F)ccc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(F)cccc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(C)c2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(C)cc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(C)ccc2-n2nccn2)nccc1C#N |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc(C#N)c2OC)c(n1)-n1nccn1 |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2C2CCC2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-c2ncccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-c2ncccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(F)c2-c2ncccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-c2ncccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(F)ccc2-c2ncccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(F)cccc2-c2ncccn2)nccc1C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Cl)ccc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(C)c1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(Cl)cc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc3c2C(=O)OC3(C)C)c(c1)-n1nccn1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2nccc3c2C(=O)OC3(C)C)c(n1)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)ccnc1-c1noc(C)n1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1noc(C)n1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1noc(C)n1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-c1noc(C)n1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-c1nc(C)no1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1nc(C)no1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1nc(C)no1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1ncccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1ncccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-c1ncccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-c1ncccn1)Oc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1CS(C)(=O)=O)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1nccc2C(=O)OCc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc2COC(=O)c12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Nc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Nc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Nc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Nc1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)N(C)c1nccc2c1C(=O)OC2(C)C |r|
C[C@@H]1OC(=O)c2c1ccnc2N(C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@H]1OC(=O)c2c1ccnc2N(C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-c2nc(C)no2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(OC)nc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(F)c2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(F)ccc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(F)cccc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(F)ccc2-c2nc(C)no2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(F)cccc2-c2nc(C)no2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-c2noc(C)n2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(F)c2-c2noc(C)n2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-c2noc(C)n2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(F)ccc2-c2noc(C)n2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(F)cccc2-c2noc(C)n2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-c2nc(C)no2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(C)c2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(C)cc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(C)ccc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(C)cccc2-n2nccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-c2ncccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(F)c2-c2ncccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-c2ncccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(F)ccc2-c2ncccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(F)cccc2-c2ncccn2)nccc1C#N
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2C2CCC2)nccc1C#N
COc1cc(nc(n1)N(C)C)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
CN(C)c1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
CN(C)c1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
COc1cc(nc(n1)N(C)C)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
COc1cc(nc(n1)N(C)C)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
CN(C)c1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
COc1cc(nc(n1)N(C)C)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1sccc1-n1cccc1
CN(C)c1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccnn1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc2cccnc12
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1sccc1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1occc1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc3ccc(F)cc3s2)c(OC)c1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc3ccccc3s2)c(OC)c1
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1-n1cccn1
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1-c1cccs1
Cc1ccc2ccccc2c1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)c1cccc2OCCOc12
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1cccs1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-n1cccn1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-n1cccc1
Cc1ccc2ccccc2c1C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1C#N
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1-n1cccc1
Fc1ccc(cc1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
Fc1cccc(c1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
Cc1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccco1)c1ccccc1-c1ccccc1
Cc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
O=C(N1CC2CN(CC2C1)c1ccc2ccccc2n1)c1ccccc1-c1cccs1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccco1)c1ccccc1-c1cccs1
CCc1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1cccc2cc[nH]c12
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1cccs1)c1ccccc1-c1cccs1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1cccs1)c1ccccc1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nccn1C
Brc1ccccc1C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
Clc1cccc(c1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
Brc1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
Fc1ccc2nc(sc2c1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(C)ccc2ccccc12
Cc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccc(F)c1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1c(C)ccc2ccccc12
Cc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1c(C)ccc2ccccc12
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccc(F)c1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccc(F)c1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1F
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccc(C)cc1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccc(Cl)c1
CCOc1ccc2ccccc2c1C(=O)N1CC2CN(CC2C1)c1nccc(OC)n1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)c2ccccc12
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1cccc2ccccc12
CCOc1ccccc1C(=O)N1CC2CN(CC2C1)c1nccc(OC)n1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1c(OC)ccc2ccccc12
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1cn[nH]c1)c1ccccc1-c1ccccc1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1cn[nH]c1)c1ccccc1-c1cccs1
Cc1cnc(C)c(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
Cc1cnc(N2CC3CN(CC3C2)C(=O)c2ccccc2-c2ccccc2)c(C)n1
Cc1nc2ccccc2nc1N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
Cc1nc2ccccc2nc1N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1cccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
CCc1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
CCOc1ccc2ccccc2c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1cccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ncoc1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cnoc1-c1ccccc1
CC(C)c1nc(C)cc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1Br
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1-c1nnc[nH]1
O=C(N1CC2CN(CC2C1)c1nc2ccccc2o1)c1ccccc1-c1nnc[nH]1
Cc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
CCOc1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1C(F)(F)F
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)c2ccccc12
CC(C)c1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1cccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c1C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc2ccccc12
FC(F)(F)c1nc2ccccc2nc1N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
Cc1nc2ccccc2nc1N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1cncc(C)n1)-n1nccn1
Cc1cnc(C)c(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cnc1C
Cc1cnc(C)c(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(I)ccc1-n1nccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1cc(C)ccc1-c1ncccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CN(CC2C1)c1cc(C)nc(n1)C(F)(F)F
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
Cc1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ncccn1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
CN(C)c1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
CN(C)c1nc(C)cc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cnc1C)-n1nccn1
CN(C)c1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-n1nccn1
COc1ccc(nc1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
CCOc1ccc2ccccc2c1C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
Cc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(Cl)cc1-n1nccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1)-n1nccn1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-n1nccn1
Cc1nc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(s1)-c1ccccc1F
FC(F)(F)c1cccc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
Cc1cccc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
Cc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1ccnc(c1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
COc1cccc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
O=C(N1CC2CN(CC2C1)c1nc2ccccc2o1)c1ccccc1-c1cccs1
FC(F)(F)c1cccnc1N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cccs1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1nnc[nH]1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1nc(C)sc1-c1ccccc1F
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1cccs1)c1ccccc1-n1nccn1
O=C(N1CC2CN(CC2C1)c1nc2ccccc2o1)c1ccccc1-n1nccn1
CCOc1ccc2ccccc2c1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
CCOc1cccc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CN(CC2C1)c1nccc(n1)C(F)(F)F
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1-n1nccn1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccco1)c1ccccc1-n1nccn1
Fc1ccc(nc1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
FC(F)(F)c1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn[nH]1
Cc1cnc(C)c(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1cncc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1)-n1nccn1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc3ccc(Cl)cc3s2)c(OC)c1
O=C(N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1ccccc1
COc1cccc(OC)c1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
COc1cccc(OC)c1C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nccc(n2)-c2ccccc2)c(OC)c1
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1-c1ccccc1
O=C(N1CC2CN(CC2C1)c1nc2ccccc2s1)c1ccccc1-c1ccccc1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cc(C)c3ccccc3n2)c(OC)c1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc3ccc(OC)cc3s2)c(OC)c1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc3ccc(C)cc3s2)c(OC)c1
Cc1cccc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
Cc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
O=C(N1CC2CN(CC2C1)c1ccc2ccccc2n1)c1ccccc1-c1ccccc1
Fc1ccc2nc(sc2c1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
Cc1cc(nc2ccccc12)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nccc(OC)n2)c(OC)c1
COc1ccccc1C(=O)N1CC2CN(CC2C1)c1nc2ccccc2o1
O=C(N1CC2CN(CC2C1)c1cnc2ccccc2n1)c1ccccc1-c1cccnc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncc[nH]1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc3ccccc3o2)c(OC)c1
O=C(N1CC2CN(CC2C1)c1nc2ccccc2o1)c1ccccc1-c1ccccc1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cccc(C)n2)c(OC)c1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nccc(C)n2)c(OC)c1
COc1ccc2nc(sc2c1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
Cc1ccc2nc(sc2c1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
COc1cccc(OC)c1C(=O)N1CC2CN(CC2C1)c1nc2ccc(Cl)cc2s1
Clc1ccc2nc(sc2c1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ccccc1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cnc3ccccc3n2)c(OC)c1
COc1cccc(OC)c1C(=O)N1CC2CN(CC2C1)c1nc2ccccc2o1
Cc1ccc(cc1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
FC(F)(F)c1ccc(cc1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
Cc1ccc(cc1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
FC(F)(F)c1ccc(cc1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cnc3ccccc3n2)c(C)c1
Clc1cccc(c1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1nccc(n1)-c1ccccc1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1OC
COc1ccccc1C(=O)N1CC2CN(CC2C1)c1nccc(C)n1
COc1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1C#N
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cnnc2ccccc12
Cc1cc(nc(n1)C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1ccnn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1cncn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1ncccc1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ncccc1-c1ccccc1
CCCc1nc(C)cc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1nccc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1cncc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1cnc(C)c(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
Cc1cnc(C)c(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn[nH]1
FC(F)(F)c1cc(nc(n1)N1CCCC1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(C)c1C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1C(F)(F)F
COc1cc(Cl)ccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(Cl)ccc1C
Cc1ccc(C)c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(C)cccc1C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1C
Cc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(C)c1
CCOc1ccc(OCC)c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
CCOc1cccc(OCC)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(C)cccc1Cl
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1I
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccnc1C(F)(F)F
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccnc1Br
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccnc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccnc1-c1ccnn1C1CCCCO1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccnc1-c1ccn[nH]1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccnc1-n1nccn1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccn1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-n1nccn1
COc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)c(C)c(C)n1)-n1nccn1
Fc1ccc2nc(ncc2c1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-n1nccn1
Fc1ccc2nc(ncc2c1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccn1
Fc1cccc(C(=O)N2CC3CN(CC3C2)c2ncc3cc(F)c(F)cc3n2)c1-n1nccn1
COc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1cnc2cc(F)c(F)cc2n1)-n1nccn1
Fc1cccc(c1C(=O)N1CC2CN(CC2C1)c1cnc2cc(F)c(F)cc2n1)-n1nccn1
Fc1ccc2nc(ncc2c1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1Br
Cc1ccc(nc1)-c1cc(F)ccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1cccnc1-c1ccn[nH]1
Cc1nc(cc(=O)[nH]1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1nc(C(=O)N2CC3CN(CC3C2)c2cc(C)nc(C)n2)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CC3CN(CC3C2)c2cc(=O)nc(C)[nH]2)c(s1)-c1ccc(F)cc1
Cc1nc(cc(=O)[nH]1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
COc1cc(OC)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(C)cccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(C)c1-n1nccn1
[O-][N+](=O)c1cnc(nc1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
COC(=O)c1cnc(nc1C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
OC(=O)c1cnc(nc1C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1cnnc1
Cc1cc(nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1)C(O)=O
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)c(F)cc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(C)c1-n1ccnn1
CN(C)C(=O)c1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
CN(C)C(=O)c1cnc(nc1C(F)(F)F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(C)c(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(C)c1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1F
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(c1)-c1ncccn1
COc1cccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c1OC
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1OC(F)(F)F
Cc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(n1)-n1nccn1
COc1cc(C)ccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(C)c1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1F
Cc1cc(nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1)C#N
Fc1cccc(c1C(=O)N1CC2CN(CC2C1)c1nc(cc(n1)C(F)(F)F)C(F)(F)F)-n1nccn1
Cc1cc(O)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1)-c1ccco1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ccn[nH]1
COc1cccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c1-n1nccn1
COc1cccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c1-n1ccnn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-n1ccnn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(c1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(c1)-n1ccnn1
Cc1nc(ncc1F)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Fc1cnc(Cl)nc1N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
Fc1cnc(nc1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1nc(ncc1F)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cnc(nc1C)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
COc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
CCc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
CC(C)c1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
CC(C)c1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
CC(C)c1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(n1)C(C)C)-n1nccn1
Cc1cc(nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1)C(C)(C)C
Cc1cc(nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1)C1CC1
Cc1ncnc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1)N1CCOCC1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
Cc1noc(n1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncnn1C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn(C)n1
Cc1noc(n1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(C)c(C)c(C)n1
Cc1noc(n1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1ncc(F)c(C)n1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn(C)n1
Cc1nc(ncc1F)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn(C)n1
Cc1nc(nc2CCCc12)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1noc(n1)-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1noc(n1)-c1cccc(F)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1nc(ncc1Cl)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1nc(nc(C)c1Cl)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1noc(n1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(C)c(Cl)c(C)n1
Cc1noc(n1)-c1ccccc1C(=O)N1CC2CN(CC2C1)c1nc2CCCc2c(C)n1
Cc1nc(nc(C)c1Cl)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn(C)n1
Cc1nc(ncc1Cl)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn(C)n1
CCc1c(C)nc(nc1C)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1ncn(C)n1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1ncccc1-n1nccn1
Cc1nc(nc(C)c1Cl)N1CC2CN(CC2C1)C(=O)c1ncccc1-n1nccn1
Cc1nc(nc(C)c1F)N1CC2CN(CC2C1)C(=O)c1ncccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc2Cc3ccccc3-c12
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c2OCOc2ccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc2cccc(-n3nccn3)c12
COc1ccc(cc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1)C(C)(C)C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc2ccccc2c1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ncccc1-n1nccn1
COc1cc(Br)c(cc1OC)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc2OCCCOc12
Cc1cccc(n1)-c1cc(F)ccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(n1)-n1ccnn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc2ccccc2c1Br
COc1cc2ccccc2cc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc2ccccc2c1-n1ccnn1
COc1c(ccc2ccccc12)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1cc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(cc1OC)-n1ccnn1
COc1cc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(cc1OC)-n1nccn1
Cc1ccnc(c1)-c1cc(F)ccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
CCCOc1cccnc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-c1ncccc1F
CCCOc1cccnc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
COc1cccc(OC)c1C(=O)N1CC2CN(CC2C1)c1ccc(cn1)C(F)(F)F
COc1cccc(OC)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1ccoc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1ccoc1C(=O)N1CC2CN(CC2C1)c1ccc(cn1)C(F)(F)F
Cc1ccoc1C(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
FC(F)(F)c1ccc(nc1)N1CC2CN(CC2C1)S(=O)(=O)c1ccccc1-c1ccccc1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)S(=O)(=O)c1ccccc1-c1ccccc1
COc1ccccc1S(=O)(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1ccccc1S(=O)(=O)N1CC2CN(CC2C1)c1ccc(cn1)C(F)(F)F
COc1ccccc1S(=O)(=O)N1CC2CN(CC2C1)c1cnc2ccccc2n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-c1ccccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ccccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-c1ncco1
Cc1cccc(n1)-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccc1C |(8.38,.58,;7.29,-.51,;7.69,-2,;6.6,-3.09,;7,-4.58,;5.12,-2.69,;4.72,-1.2,;5.81,-.11,;3.18,-.84,;2.27,.41,;.81,-.07,;-.66,.41,;-1.56,-.84,;-.66,-2.09,;.81,-1.61,;2.27,-2.09,;-3.05,-.04,;-3.05,1.5,;-4.38,-.81,;-4.38,-2.35,;-5.72,-3.12,;-7.05,-2.35,;-7.05,-.81,;-8.38,-.04,;-5.72,-.04,;-5.72,1.5,;-4.38,2.27,;-4.38,3.81,;-5.72,4.58,;-7.05,3.81,;-7.05,2.27,;-8.38,1.5,)|
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccc1Cl |(7.09,-3.97,;6.69,-2.48,;7.78,-1.39,;7.38,.09,;8.47,1.18,;5.89,.49,;4.8,-.6,;5.2,-2.09,;3.31,-.2,;2.41,1.05,;.94,.57,;-.52,1.05,;-1.43,-.2,;-.52,-1.45,;.94,-.97,;2.41,-1.45,;-2.91,.2,;-3.31,1.69,;-4,-.89,;-3.6,-2.38,;-4.69,-3.47,;-6.18,-3.07,;-6.58,-1.58,;-8.07,-1.18,;-5.49,-.49,;-5.89,1,;-4.8,2.09,;-5.2,3.57,;-6.69,3.97,;-7.78,2.88,;-7.38,1.39,;-8.47,.31,)|
Cc1ccnc(c1)-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1ccc(nc1)-c1c(F)ccnc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccc1F |(7.09,-3.97,;6.69,-2.48,;7.78,-1.39,;7.38,.09,;8.47,1.18,;5.89,.49,;4.8,-.6,;5.2,-2.09,;3.31,-.2,;2.41,1.05,;.94,.57,;-.52,1.05,;-1.43,-.2,;-.52,-1.45,;.94,-.97,;2.41,-1.45,;-2.91,.2,;-3.31,1.69,;-4,-.89,;-3.6,-2.38,;-4.69,-3.47,;-6.18,-3.07,;-6.58,-1.58,;-8.07,-1.18,;-5.49,-.49,;-5.89,1,;-4.8,2.09,;-5.2,3.57,;-6.69,3.97,;-7.78,2.88,;-7.38,1.39,;-8.47,.31,)|
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncco1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2ncc(F)c(C)n2)c(c1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2ncc(Cl)c(C)n2)c(c1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)c(F)c(C)n2)c(c1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2ncc(C)c(C)n2)c(c1)-n1nccn1
CCCOc1ncccc1C(=O)N1CC2CN(CC2C1)c1ccc(cn1)C(F)(F)F
CCc1c(C)nc(nc1C)N1CC2CN(CC2C1)C(=O)c1ncccc1-n1nccn1
Cc1noc(n1)-c1cccnc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Fc1cc2ncc(nc2cc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2ncc3cc(F)ccc3n2)c(c1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cnc3cc(F)c(F)cc3n2)c(c1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cc(ncn2)N(C)C)c(c1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cc(nc(C)n2)N(C)C)c(c1)-n1nccn1
Cc1cccc(n1)-c1ccc(F)cc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1ccnc(c1)-c1ccc(F)cc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1ccc(nc1)-c1ccc(F)cc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccc1F
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ccccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncco1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ncccc1C(F)(F)F
CCOc1ccc(C)nc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
CCOc1ncccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-n1nccn1
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
CCCOc1ccc(C)nc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
CCOc1ccc(C)nc1C(=O)N1CC2CN(CC2C1)c1cc(nc(C)n1)N(C)C
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cnc(o1)-c1ccc(C)nc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1ccc(c(c1)C(=O)N1CC2CN(CC2C1)c1cc(nc(C)n1)N(C)C)-n1nccn1
CCCOc1ccc(C)nc1C(=O)N1CC2CN(CC2C1)c1cc(nc(C)n1)N(C)C
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1ncccn1
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ncccn1
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccn1
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1nc(C)ccc1-c1ncccn1
CN(C)c1cc(nc(C)n1)N1CC2CN(CC2C1)C(=O)c1nc(C)ccc1-c1ncc(C)o1
CCCOc1ccc(C)cc1C(=O)N1CC2CN(CC2C1)c1cc(nc(C)n1)N(C)C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1nnc[nH]1
Cc1cc(CO)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1cn(Cc2ccccc2)nn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(CO)n2)c(c1)-n1nccn1
Cc1noc(n1)-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(CO)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1nnc[nH]1
Cc1ccc(c(n1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1)-n1ccnn1
Cc1noc(n1)-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1ncc(F)c(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ncc(Cl)cc1-n1nccn1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1ncc(Cl)cc1-n1nccn1
COc1cnc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(c1)-n1nccn1
COc1cnc(C(=O)N2CC3CN(CC3C2)c2nc(C)c(C)c(C)n2)c(c1)-n1nccn1
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CN(CC2C1)c1nc(C)c(C)c(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(OC(F)F)cc1-n1nccn1
CCOc1ncccc1C(=O)N1CC2CN(CC2C1)c1cnc2cc(F)c(F)cc2n1
CCOc1ncccc1C(=O)N1CC2CN(CC2C1)c1ncc2cc(F)ccc2n1
Fc1cc2ncc(nc2cc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1I
Fc1cccnc1-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1cnc2cc(F)c(F)cc2n1 |(-10.07,1.33,;-9.3,,;-10.07,-1.33,;-9.3,-2.67,;-7.76,-2.67,;-6.99,-1.33,;-7.76,,;-6.99,1.33,;-7.76,2.67,;-9.3,2.67,;-6.99,4,;-5.45,4,;-4.68,2.67,;-5.45,1.33,;-4.68,,;-5.45,-1.33,;-3.14,,;-2.23,1.25,;-.77,.77,;.69,1.25,;1.6,,;.69,-1.25,;-.77,-.77,;-2.23,-1.25,;3.14,,;3.91,1.33,;5.45,1.33,;6.22,,;7.76,,;8.53,-1.33,;10.07,-1.33,;7.76,-2.67,;8.53,-4,;6.22,-2.67,;5.45,-1.33,;3.91,-1.33,)|
Fc1cc2ncc(nc2cc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncco1
Fc1cc2ncc(nc2cc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ccccn1
COc1cccnc1-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1cnc2cc(F)c(F)cc2n1 |(-10.84,1.33,;-9.3,1.33,;-8.53,,;-9.3,-1.33,;-8.53,-2.67,;-6.99,-2.67,;-6.22,-1.33,;-6.99,,;-6.22,1.33,;-6.99,2.67,;-8.53,2.67,;-6.22,4,;-4.68,4,;-3.91,2.67,;-4.68,1.33,;-3.91,,;-4.68,-1.33,;-2.37,,;-1.46,1.25,;,.77,;1.46,1.25,;2.37,,;1.46,-1.25,;,-.77,;-1.46,-1.25,;3.91,,;4.68,1.33,;6.22,1.33,;6.99,,;8.53,,;9.3,-1.33,;10.84,-1.33,;8.53,-2.67,;9.3,-4,;6.99,-2.67,;6.22,-1.33,;4.68,-1.33,)|
Fc1cc2ncc(nc2cc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1cncs1
Fc1cc2ncc(nc2cc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1cscn1
Fc1cn[nH]c1-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1cnc2cc(F)c(F)cc2n1 |(-10.07,1.33,;-9.3,,;-9.78,-1.46,;-8.53,-2.37,;-7.28,-1.46,;-7.76,,;-6.99,1.33,;-7.76,2.67,;-9.3,2.67,;-6.99,4,;-5.45,4,;-4.68,2.67,;-5.45,1.33,;-4.68,,;-5.45,-1.33,;-3.14,,;-2.23,1.25,;-.77,.77,;.69,1.25,;1.6,,;.69,-1.25,;-.77,-.77,;-2.23,-1.25,;3.14,,;3.91,1.33,;5.45,1.33,;6.22,,;7.76,,;8.53,-1.33,;10.07,-1.33,;7.76,-2.67,;8.53,-4,;6.22,-2.67,;5.45,-1.33,;3.91,-1.33,)|
COc1ccc(C(=O)N2CC3CN(CC3C2)c2cnc3cc(F)c(F)cc3n2)c(c1)-c1ncccn1
Cc1cccc(C(=O)N2CC3CN(CC3C2)c2cnc3cc(F)c(F)cc3n2)c1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(O)cc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc2CCOc12
Cc1nc2sccn2c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1cccc(c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1)-n1nccn1
COc1ccc(C(=O)N2CC3CN(CC3C2)c2nc(C)cc(C)n2)c(c1)-c1ncco1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-c1[nH]ncc1F
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1[nH]ncc1F |(7.37,-3.32,;5.89,-3.72,;5.49,-5.2,;4,-5.6,;3.6,-7.09,;2.91,-4.51,;3.31,-3.03,;4.8,-2.63,;2.22,-1.94,;.76,-2.41,;-.15,-1.17,;-1.61,-.69,;-1.61,.85,;-.15,1.32,;.76,.08,;2.22,-.4,;-2.7,1.94,;-4.19,1.54,;-2.3,3.42,;-.82,3.82,;-.42,5.31,;-1.51,6.4,;-3,6,;-4.08,7.09,;-3.39,4.51,;-4.88,4.12,;-5.36,2.65,;-6.9,2.65,;-7.37,4.12,;-6.13,5.02,;-6.13,6.56,)|
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1[nH]ncc1F
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1nccs1
Cc1cnc(s1)-c1cccc(F)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
COc1ncc(s1)-c1cccc(F)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1C1=CC(=O)OC1 |t:29|
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ncccc1F
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1cn(C)cn1
COc1ccnc(n1)-c1cccc(F)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
CSc1nccc(n1)-c1cccc(F)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1cscn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1cncs1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ccnnc1
Cc1ccnc(c1)-c1cccc(F)c1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ccccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-c1ncco1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-c1ncc(F)cc1F
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1cccn1C
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cc(F)ccc1-c1cscn1
Cc1nc(ncc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncco1
COc1c(C)nc(nc1C)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1nc(nc(C)c1O)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1C1(CCC1)C#N)Nc1cc(OCC(F)F)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Nc1cc(OCC(F)F)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1cnnn1)Nc1cc(OCC(F)F)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Nc1cc(OCC(F)F)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccsc1-n1nccn1)Nc1cc(OCC(F)F)ccn1 |r|
CCOc1ncccc1C(=O)N1C[C@@H](C[C@H]1C)Nc1cc(OCC(F)F)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1cccc2CCCc12)Nc1cc(OCC(F)F)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(ccn1)C(F)F |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(F)cn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc2ccccc12 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(ccn1)C(F)(F)F |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(Cl)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(C)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(F)ccn1 |r|
COc1ccnc(N[C@@H]2C[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C#C |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(ccn1)C#N |r|
CC(C)Oc1ccnc(N[C@@H]2C[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
CCOc1ccnc(N[C@@H]2C[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)N(C)c1cc(ccn1)C#N |r|
COc1ccnc(N[C@@H]2C[C@@H](C)N(C2)C(=O)c2ccccc2C2(CC2)C#N)c1 |r|
COc1cccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccsc1-n1nccn1)Nc1cc(ccn1)C(F)F |r|
C[C@@H]1C[C@H](CN1C(=O)c1cscc1-n1nccn1)Nc1cc(ccn1)C(F)F |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Nc1cc(ccn1)C#N |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Nc1cc(ccn1)C#N |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(Br)ccn1 |r|
COC(=O)c1c(OC)ccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
CCOC(=O)c1c(OC)ccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
CCOc1ccnc(N[C@@H]2C[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C(=O)OC |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)N(C)c1cc(Br)ccn1 |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc(C#N)c1C |r|
C[C@@H]1C[C@H](CN1C(=O)c1ccccc1-n1nccn1)N(C)c1nccc(C#N)c1C |r|
COC(=O)c1c(N[C@@H]2C[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
COc1c(N[C@@H]2C[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
COc1cccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1cccnc1-n1cc(C)cn1 |r|
COc1cccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1ccccc1-c1noc(C)n1 |r|
COc1cccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1nccnc1-n1cccn1 |r|
COc1cccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1nccnc1-c1ccccn1 |r|
COc1cccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1ccccc1-c1nc(C)no1 |r|
CCCc1ccccc1C(=O)N1C[C@@H](C[C@H]1C)Nc1ncccc1OC |r|
COc1cccnc1N[C@@H]1C[C@@H](C)N(C1)C(=O)c1ccccc1OC(F)(F)F |r|
CCN(CCn1ncc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCn1ncc(n1)C(C)(O)CC)C(=O)c1ccccc1-n1nccn1
CCN(CCn1ncc(n1)C(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCn1ncc(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1
CCN(CCn1ncc(n1)C(C)(C)O)C(=O)c1ccccc1N1CCCC1
CCN(CCn1ncc(n1)C(C)(C)O)C(=O)c1ccccc1SC(F)(F)F
CCN(CCn1ncc(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)(F)F
CCN(CCn1ncc(n1)C(C)(C)O)C(=O)c1ccccc1OC(C)C
CCOC(=O)c1nn(CCN(CC)C(=O)c2ccccc2-n2nccn2)nc1C
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1cccnc1OC(C)C
CCOc1ncccc1C(=O)N(CC)CCn1nc(C)c(n1)C(C)(C)O
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)(F)F
CCOc1ccccc1C(=O)N(CC)CCn1nc(C)c(n1)C(C)(C)O
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1-n1cccn1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccc(F)cc1-n1nccn1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1cccnc1-c1ccccc1
CCCc1ccccc1C(=O)N(CC)CCn1nc(C)c(n1)C(C)(C)O
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1CC(F)(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1cccnc1CC(F)(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1CC(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1(F)F
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccc(OC)nc1C1CC1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1C1CCC1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1N1CCCC1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1-n1ncnn1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ncccc1-n1nccn1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1ncccc1-c1ccccc1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1nccnc1-c1ccccn1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1nccnc1-n1cccn1
CCN(CCn1nc(C)c(n1)C(C)(C)O)C(=O)c1cccnc1-n1cccn1
CCN(CCn1cc(cn1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCn1ccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-n1nccn1)Nc1nc(C)cc(C)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1c(F)cccc1-c1ncccn1)Nc1nc(C)cc(C)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1c(F)cccc1-n1nccn1)Nc1nc(C)cc(C)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1nc(C)cc(C)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-n1nccn1)Nc1nc(C)cc(C)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)ccc1-c1ncccn1)Nc1nc(C)cc(C)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)ccc1-c1ncccn1)Nc1cc(C)nc(n1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)ccc1-n1nccn1)Nc1cc(C)nc(n1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-c1ncccn1)Nc1cc(C)nc(n1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1c(F)cccc1-n1nccn1)Nc1nccc(n1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1ccnn1)Nc1nccc(n1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@@H]1[C@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
CCOc1ccc(C)nc1C(=O)N1CCC[C@@H](Nc2ccc(cn2)C(F)(F)F)[C@@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
COc1ccc(c(c1)C(=O)N1CCC[C@@H](Nc2ccc(cn2)C(F)(F)F)[C@@H]1C)-n1nccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-c1ncco1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-c1ncccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-c1ncccn1)Nc1ccc(cn1)C(F)(F)F |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2ccc(cn2)C(F)(F)F)[C@@H]1C |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2ccc(cn2)C(F)(F)F)[C@@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ncc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ncc(C)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(nn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(F)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(C)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ncc2ccccc2n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ncc(F)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1nc2ccccc2o1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(Br)cn1 |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2ccc(Br)cn2)[C@@H]1C |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2ccc(Br)cn2)[C@@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1nc2cc(Cl)ccc2o1 |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2nc3cc(Cl)ccc3o2)[C@@H]1C |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2nc3cc(Cl)ccc3o2)[C@@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1cnc2ccccc2n1 |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2cnc3ccccc3n2)[C@@H]1C |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2cnc3ccccc3n2)[C@@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1nccc(n1)-c1ccccc1 |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2nccc(n2)-c2ccccc2)[C@@H]1C |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2nccc(n2)-c2ccccc2)[C@@H]1C |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2ccc(cn2)C(F)(F)F)[C@H]1C |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2ccc(cn2)C(F)(F)F)[C@H]1C |r|
C[C@@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1ccc(Br)cn1 |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2ccc(Br)cn2)[C@H]1C |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2ccc(Br)cn2)[C@H]1C |r|
C[C@@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1nc2cc(Cl)ccc2o1 |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2nc3cc(Cl)ccc3o2)[C@H]1C |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2nc3cc(Cl)ccc3o2)[C@H]1C |r|
C[C@@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1cnc2ccccc2n1 |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2cnc3ccccc3n2)[C@H]1C |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2cnc3ccccc3n2)[C@H]1C |r|
C[C@@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Nc1nccc(n1)-c1ccccc1 |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](Nc2nccc(n2)-c2ccccc2)[C@H]1C |r|
CCOc1ccccc1C(=O)N1CCC[C@@H](Nc2nccc(n2)-c2ccccc2)[C@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1nccn1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1ccnn1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1nc2ccccc2o1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1nccn1)Nc1nc2ccccc2o1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1ccnn1)Nc1nc2ccccc2o1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-c1ncco1)Nc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-c1ncccn1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-c1ncco1)Nc1ccc(Br)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-c1ncccn1)Nc1nc2ccccc2o1 |r|
COc1ccc(C(=O)N2CCC[C@@H](Nc3cnc(cn3)C(F)(F)F)[C@@H]2C)c(c1)-n1nccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-c1ncco1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-c1ncccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-c1ncco1)Nc1cnc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-c1ncco1)Nc1nc2ccccc2o1 |r|
COc1ccc(c(c1)C(=O)N1CCC[C@@H](Nc2ncc(cn2)C(F)(F)F)[C@@H]1C)-n1nccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Nc1ncc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1ccc(Br)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1ccnn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1ncc(cn1)C(F)(F)F |r|
COc1ccc(C(=O)N2CCC[C@@H](Nc3ncc(cn3)C(F)(F)F)[C@@H]2C)c(c1)-n1nccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1ccnn1)Nc1cnc(cn1)C(F)(F)F |r|
COc1ccc(C(=O)N2CCC[C@@H](Nc3ccc(cn3)C(F)(F)F)[C@@H]2C)c(c1)-n1nccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Nc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-n1nccn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-n1nccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-n1nccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncc(F)cn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccnc1-n1nccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccnc1-n1nccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-c1ncccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncc(F)cn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-n1nccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-n1nccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-n1nccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-n1nccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-n1nccn1)Oc1ncc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-n1nccn1)Oc1ncc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-n1nccn1)Oc1ncc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-n1nccn1)Oc1ncc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncc(F)cn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncc(F)cn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-c1ncccn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-c1ncccn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-c1ncc(F)cn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-c1ncccn1)Oc1cnc(cn1)C(F)(F)F |r|
COc1ccc(C(=O)N2CCC[C@@H](Oc3cnc(cn3)C(F)(F)F)[C@@H]2C)c(c1)-n1nccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nccnc1-c1ccccc1)Oc1cnc(cn1)C(F)(F)F |r|
COc1ccc(C(=O)N2CCC[C@@H](Oc3ncc(cn3)C(F)(F)F)[C@@H]2C)c(c1)-n1nccn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-c1ncco1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-n1nccn1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-n1nccn1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nccnc1-c1ccccc1)Oc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-c1ncco1)Oc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)cc1-n1nccn1)Nc1cnc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(O)cc1-n1nccn1)Nc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1cnc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1ncc(Cl)cn1 |r|
COc1ccc(c(c1)C(=O)N1CCC[C@@H](Nc2cnc(cn2)C(F)(F)F)[C@@H]1C)-n1nccn1 |r|
COc1ccc(C(=O)N2CCC[C@@H](Nc3ncc(Cl)cn3)[C@@H]2C)c(c1)-n1nccn1 |r|
COc1ccc(C(=O)N2CCC[C@@H](Nc3cnc(Cl)cn3)[C@@H]2C)c(c1)-n1nccn1 |r|
C[C@H]1C(CCCN1C(=O)c1ncc(C)cc1-n1nccn1)N(C)c1nc2ccccc2o1 |r|
C[C@H]1C(CCCN1C(=O)c1ccc(C)nc1-n1nccn1)N(C)c1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-c1ncccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1nc(C)no1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncccn1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F |r|
COc1ccc(C(=O)N2CCC[C@@H](Nc3ccc(cn3)C(F)(F)F)[C@@H]2C)c(Cl)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-n1nccn1)Nc1nnc(s1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(C)nc1-n1nccn1)Nc1nnc(s1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1nc(C)no1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-n1nccn1)Nc1ncc(cn1)C(F)(F)F |r|
CCOc1ccc(C)nc1C(=O)N1CCC[C@@H](Nc2ncc(cn2)C(F)(F)F)[C@@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-c1ncccn1)Nc1ncc(cn1)C(F)(F)F |r|
COc1ccc(C(=O)N2CCC[C@@H](Nc3ncc(cn3)C(F)(F)F)[C@@H]2C)c(Cl)n1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncccn1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncco1)Nc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-c1ncccn1)Nc1nc2ccccc2o1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncco1)Nc1ncc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncccn1)Nc1nc2ccccc2o1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(F)c1-c1ncccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncco1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncccc1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1c(F)cccc1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-c1ncccn1)Oc1ccc(cn1)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-n1nccn1)Oc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-n1nccn1)Oc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncc(C)cc1-c1ncccn1)Oc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(C)cnc1-c1ncccn1)Oc1ccc(Cl)cn1 |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncccc1-c1ncccn1)Oc1ccc(Cl)cn1 |r|
CCOc1ccc(C)nc1C(=O)N1CCC[C@@H](Oc2ccc(cn2)C(F)(F)F)[C@@H]1C |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cccc(C)c1-c1ncccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1cc(F)ccc1-c1ncccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccc(F)cc1-c1ncccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1nc(C)ccc1-c1ncccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ccccc1-n1nccn1)Oc1ncc(cc1F)C(F)(F)F |r|
C[C@H]1[C@@H](CCCN1C(=O)c1ncccc1-c1ncccn1)Nc1ccc(cn1)C(F)(F)F |r|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:0:1:4.3:17,5:4:18.1:17|
CC1C2CC(Nc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1Br |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccc(C)nc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-c1ncco1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CCOc1ccc(C)nc1C(=O)N1C(C)C2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:18:17:12.13:30,10:12:17.16:30,THB:14:13:17.16:30|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccc(F)cc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccc(F)cc1-c1ncccn1 |TLB:19:18:4.3:17,THB:0:1:4.3:17,5:4:18.1:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc(F)ccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc(F)ccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:0:1:4.3:17,5:4:18.1:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncc(F)cn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncc(F)cn1 |TLB:19:18:4.3:17,THB:0:1:4.3:17,5:4:18.1:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-c1ncc(F)cn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-c1ncc(F)cn1 |TLB:19:18:4.3:17,THB:0:1:4.3:17,5:4:18.1:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:0:1:4.3:17,5:4:18.1:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc(C)cnc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccc(F)cc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc(F)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1c(F)cccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
COc1ccc(C(=O)N2C(C)C3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:14:13:8.9:26,6:8:13.12:26,THB:10:9:13.12:26|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-c1ncccc1F |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(c1)-c1ccc(F)cc1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(nc3)C(F)(F)F)C(C2)N1C(=O)c1ncccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(nc3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(nc3)C(F)(F)F)C(C2)N1C(=O)c1cccc(C)c1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(nc3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(nc3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccc(C)nc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc(C)cnc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccc(F)cc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc(F)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc(cn3)C(F)(F)F)C(C2)N1C(=O)c1c(F)cccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CCOc1ccc(C)nc1C(=O)N1C(C)C2CC(Oc3cnc(cn3)C(F)(F)F)C1C2 |TLB:18:17:12.13:30,10:12:17.16:30,THB:14:13:17.16:30|
COc1ccc(C(=O)N2C(C)C3CC(Oc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:14:13:8.9:26,6:8:13.12:26,THB:10:9:13.12:26|
CC1C2CC(Nc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncccc1-c1ncccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Nc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
Cc1ccc(c(n1)C(=O)N1C(CF)C2CC(Oc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:16:15:9.10:28,7:9:15.14:28,THB:11:10:15.14:28|
FCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1c(F)cccc1-c1ncco1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
Cc1cnc(c(c1)C(=O)N1C(CF)C2CC(Oc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:16:15:9.10:28,7:9:15.14:28,THB:11:10:15.14:28|
FCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C(CF)C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:25:23:20.21:16.15,17:16:23.24:20.21,THB:13:15:23.24:20.21|
FCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1ccccc1-c1ncccn1 |TLB:1:2:7.8:4.5,THB:9:7:4.5:2.20,21:20:7.8:4.5|
FCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1cc(F)ccc1-c1ncccn1 |TLB:1:2:7.8:4.5,THB:9:7:4.5:2.20,21:20:7.8:4.5|
Cc1ccc(c(n1)C(=O)N1C(CF)C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:19:17:14.15:10.9,11:10:17.18:14.15,THB:7:9:17.18:14.15|
FCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1cc(F)ccc1-n1nccn1 |TLB:1:2:7.8:4.5,THB:9:7:4.5:2.20,21:20:7.8:4.5|
FCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1cccc(F)c1-c1ncccn1 |TLB:1:2:7.8:4.5,THB:9:7:4.5:2.20,21:20:7.8:4.5|
FCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1cc(F)ccc1-c1ncc(F)cn1 |TLB:1:2:7.8:4.5,THB:9:7:4.5:2.20,21:20:7.8:4.5|
CC1C2CC(Oc3ccc(cn3)C(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:18:17:4.3:16,THB:5:4:17.1:16,0:1:4.3:16|
CC1C2CC(Oc3ccc(Cl)cn3)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:16:15:4.3:14,THB:5:4:15.1:14,0:1:4.3:14|
CC1C2CC(Oc3ccc(Cl)cn3)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:16:15:4.3:14,THB:5:4:15.1:14,0:1:4.3:14|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1cccc(F)c1-c1ncccn1 |TLB:0:1:6.7:3.4,THB:8:6:3.4:1.19,20:19:6.7:3.4|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:0:1:6.7:3.4,THB:8:6:3.4:1.19,20:19:6.7:3.4|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1ccccc1-n1nccn1 |TLB:0:1:6.7:3.4,THB:8:6:3.4:1.19,20:19:6.7:3.4|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1nc(C)ccc1-c1ncccn1 |TLB:0:1:6.7:3.4,THB:8:6:3.4:1.19,20:19:6.7:3.4|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1ncccc1-n1nccn1 |TLB:0:1:6.7:3.4,THB:8:6:3.4:1.19,20:19:6.7:3.4|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1ncc(C)cc1-n1nccn1 |TLB:0:1:6.7:3.4,THB:8:6:3.4:1.19,20:19:6.7:3.4|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1ncc(C)cc1-c1ncccn1 |TLB:0:1:6.7:3.4,THB:8:6:3.4:1.19,20:19:6.7:3.4|
CC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1cccc(F)c1-c1ncccn1 |TLB:0:1:6.7:3.4,8:6:3.4:1.19,THB:20:19:6.7:3.4|
CC1C2CC(Oc3ccc(C)cn3)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:16:15:4.3:14,THB:5:4:15.1:14,0:1:4.3:14|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1ncc(CCCF)n1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncc(OCCF)cn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1cnc(F)cn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ccc(F)nc1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ccnc(F)c1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1cccc(F)n1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1cccc(n1)[N+]([O-])=O |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1cccc(Br)n1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
Cc1ccc(c(n1)C(=O)N1C(CO)C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:19:17:9.10:15.14,11:10:17.18:15.14,THB:7:9:17.18:15.14|
OCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1c(F)cccc1-n1nccn1 |TLB:1:2:7.8:5.4,THB:9:7:20.2:5.4,21:20:7.8:5.4|
OCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1cc(F)ccc1-c1ncc(F)cn1 |TLB:1:2:7.8:4.5,THB:21:20:7.8:4.5,9:7:4.5:2.20|
COCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:2:3:8.9:5.6,THB:22:21:8.9:5.6,10:8:5.6:3.21|
COCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1nc(C)ccc1-c1ncccn1 |TLB:2:3:8.9:5.6,THB:22:21:8.9:5.6,10:8:5.6:3.21|
COCC1C2CCC(C(C2)Oc2ccc(cn2)C(F)(F)F)N1C(=O)c1ccccc1-c1ncccn1 |TLB:2:3:8.9:5.6,THB:22:21:8.9:5.6,10:8:5.6:3.21|
CC1C2CC(Oc3ccc(cn3)C(F)F)C(C2)N1C(=O)c1nc(C)ccc1-c1ncccn1 |TLB:18:17:4.3:16,THB:5:4:17.1:16,0:1:4.3:16|
CC1C2CC(Oc3cnc4ccccc4n3)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc4ccccc4n3)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc4ccccc4c3)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3cnc4cc(F)ccc4n3)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:20:19:4.3:18,THB:5:4:19.1:18,0:1:4.3:18|
CC1C2CC(Oc3cnc4cc(F)ccc4n3)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:20:19:4.3:18,THB:5:4:19.1:18,0:1:4.3:18|
CC1C2CC(Oc3cnc4cc(F)ccc4n3)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:20:19:4.3:18,THB:5:4:19.1:18,0:1:4.3:18|
CC1C2CC(Oc3cnc4cc(F)c(F)cc4n3)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:21:20:4.3:19,THB:5:4:20.1:19,0:1:4.3:19|
CC1C2CC(Oc3cnc4cc(F)c(F)cc4n3)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:21:20:4.3:19,THB:5:4:20.1:19,0:1:4.3:19|
CC1C2CC(Oc3cnc4cc(F)c(F)cc4n3)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:21:20:4.3:19,THB:5:4:20.1:19,0:1:4.3:19|
CCOC(=O)C1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:23:22:8.7:21,THB:9:8:22.5:21,3:5:8.7:21|
CC1C2CC(Oc3ccc(Cl)cn3)C(C2)N1C(=O)c1ccc(C)nc1-n1nccn1 |TLB:16:15:4.3:14,THB:5:4:15.1:14,0:1:4.3:14|
CC1C2CC(Oc3ccc(Cl)cn3)C(C2)N1C(=O)c1cc(C)cnc1-n1nccn1 |TLB:16:15:4.3:14,THB:5:4:15.1:14,0:1:4.3:14|
CC1C2CC(Oc3ccc(Cl)cn3)C(C2)N1C(=O)c1cccc(F)c1-n1nccn1 |TLB:16:15:4.3:14,THB:5:4:15.1:14,0:1:4.3:14|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccc(OCCF)cc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc2ccccc2nc1OCCO |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc(OCCBr)ccc1-n1nccn1 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cc2ccccc2nc1OCCF |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1c(OCCF)ccc2cccnc12 |TLB:19:18:4.3:17,THB:5:4:18.1:17,0:1:4.3:17|
CC(C)CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:22:21:7.6:20,THB:8:7:21.4:20,3:4:7.6:20|
CC(C)CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-n1nccn1 |TLB:22:21:7.6:20,THB:8:7:21.4:20,3:4:7.6:20|
CC(C)CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncccn1 |TLB:22:21:7.6:20,THB:8:7:21.4:20,3:4:7.6:20|
CC(C)CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:22:21:7.6:20,THB:8:7:21.4:20,3:4:7.6:20|
CC(C)CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-c1ncccn1 |TLB:22:21:7.6:20,THB:8:7:21.4:20,3:4:7.6:20|
CC(C)CC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncc(F)cn1 |TLB:22:21:7.6:20,THB:8:7:21.4:20,3:4:7.6:20|
CCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-n1nccn1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
CCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncccn1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
CCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1nc(C)ccc1-n1nccn1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
CCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ncc(C)cc1-n1nccn1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
CCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1cccc(F)c1-c1ncccn1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
CCC1C2CC(Oc3ccc(cn3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncc(F)cn1 |TLB:20:19:5.4:18,THB:6:5:19.2:18,1:2:5.4:18|
CC1C2CC(Oc3ccc(c(F)n3)C(F)(F)F)C(C2)N1C(=O)c1ccccc1-c1ncccn1 |TLB:20:19:4.3:18,THB:5:4:19.1:18,0:1:4.3:18|
FC(F)(F)c1cnc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3cnc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
CCOc1ncc2ccccc2c1C(=O)N1CC2CC(Oc3cnc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Cc1cnc(C(=O)N2CC3CC(Oc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
CCOc1ncc2ccccc2c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Cc1cnc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
CCOc1ccc2cccnc2c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
COc1ccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
COc1ccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1ccc(c(c1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
COc1cccc(c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:15:14:10.11:27,8:10:14.13:27|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c1-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Cc1cccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c1-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1ccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2cnnc2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Cc1ccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(n1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2ncccc2-n2nccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
COc1c(F)cccc1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:16:15:11.12:28,9:11:15.14:28|
Cc1ccc(OC2CC3CC2N(C3)C(=O)c2cccc(C)c2-c2ncco2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c1-n1ccnn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Cc1ccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(n1)-n1ccnn1 |TLB:12:11:7.8:24,5:7:11.10:24|
CCOc1ccc(C)nc1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:17:16:12.13:29,10:12:16.15:29|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
COc1cccc(-c2ccn[nH]2)c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
COc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:21:20:16.17:33,14:16:20.19:33|
Cc1cnn(C)c1-c1ccccc1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32,(.61,-1.24,;1.38,-2.58,;.9,-4.04,;2.15,-4.95,;3.4,-4.04,;4.73,-4.81,;2.92,-2.58,;4.01,-1.49,;5.5,-1.89,;6.59,-.8,;6.19,.69,;4.7,1.09,;3.61,-0,;2.12,.4,;1.03,-.69,;1.72,1.88,;2.5,3.22,;1.01,3.62,;-.48,3.22,;-1.25,1.88,;-1.25,.34,;-2.58,-.43,;-2.58,-1.97,;-3.92,-2.74,;-5.35,-1.98,;-5.25,-.43,;-3.92,.34,;-6.69,-2.74,;-8.03,-3.49,;-7.44,-1.4,;-5.93,-4.08,;.24,2.28,;.24,4.95,)|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2cccc3cc[nH]c23)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Fc1ccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c1Br |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Oc3ccc(Br)cn3)C1C2 |TLB:20:19:15.16:29,13:15:19.18:29|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(Br)cn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Brc1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ccc(Br)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
FC(F)(F)c1cccnc1OC1CC2CC1N(C2)C(=O)c1ccccc1-n1nccn1 |TLB:18:16:11.12:14,THB:10:11:16.17:14|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ncccc3C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
FC(F)(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1ccc(c(n1)C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Cc1cccc(C(=O)N2CC3CC(Nc4ccc(cn4)C(F)(F)F)C2C3)c1-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
CCOc1ccc2cccnc2c1C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1ccc(c(c1)C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1nc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(s1)-c1ccc(F)cc1 |TLB:11:10:6.7:23,4:6:10.9:23|
Cc1nc2sccn2c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:16:15:11.12:28,9:11:15.14:28|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1ccc(c(n1)C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Cc1ccc(c(n1)C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1cccc(C(=O)N2CC3CC(Nc4ccc(cn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(C(=O)N2CC3CC(Nc4ncc(cn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Oc2cnc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Cc1ccc(c(n1)C(=O)N1CC2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:17:15:12.13:10.9,THB:7:9:15.16:12.13|
Cc1ccc(c(n1)C(=O)N1CC2CCC1C(C2)Oc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:17:15:12.13:10.9,THB:7:9:15.16:12.13|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Cc1ccc(c(n1)C(=O)N1CC2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:17:15:12.13:10.9,THB:7:9:15.16:12.13|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2cccnc2-n2nccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1cnc(c(c1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1cnc(nc1)-c1ccccc1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:21:20:16.17:33,14:16:20.19:33|
Cc1cccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c1-c1ncc(F)cn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2nccnc2-c2ccccc2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Fc1cccc(C(=O)N2CC3CC(Oc4cccc(n4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(C(=O)N2CC3CC(Oc4cc(ccn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(C(=O)N2CC3CC(Oc4ncccc4C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cc(cnc1OC1CC2CC1N(C2)C(=O)c1ccccc1-n1nccn1)C(F)(F)F |TLB:15:13:8.9:11,THB:7:8:13.14:11|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ncc(cc3F)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:27,7:9:13.12:27|
Fc1cc(cnc1OC1CC2CC1N(C2)C(=O)c1ccccc1-c1ncccn1)C(F)(F)F |TLB:15:13:8.9:11,THB:7:8:13.14:11|
Fc1cc(cnc1OC1CC2CC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)C(F)(F)F |TLB:15:13:8.9:11,THB:7:8:13.14:11|
Cc1ccc(OC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
O=C(N1CC2CC(Oc3ccccn3)C1C2)c1ccccc1-n1nccn1 |TLB:7:6:2.3:15,1:2:6.5:15|
Cc1ccc(C(=O)N2CC3CC(Oc4ccccn4)C2C3)c(n1)-n1nccn1 |TLB:12:11:7.8:20,5:7:11.10:20|
Fc1cccc(C(=O)N2CC3CC(Oc4ccccn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:21,6:8:12.11:21|
Cc1ccc(C(=O)N2CC3CC(Oc4ccc(Br)cn4)C2C3)c(n1)-n1nccn1 |TLB:12:11:7.8:21,5:7:11.10:21|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(Br)cn4)C2C3)c1-n1nccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Fc1ccc(C(=O)N2CC3CC(Oc4ccc(Br)cn4)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:21,5:7:11.10:21|
Fc1ccc(c(c1)C(=O)N1CC2CC(Oc3ccc(Br)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
Fc1cccc(c1C(=O)N1CC2CC(Oc3ccc(Br)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
Fc1ccc(C(=O)N2CC3CC(Oc4ccc(Br)cn4)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:21,5:7:11.10:21|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Oc3ccc(Br)cn3)C1C2 |TLB:20:19:15.16:29,13:15:19.18:29|
Clc1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Fc1ccc(c(c1)C(=O)N1CC2CC(Oc3ccc(Cl)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ccc(Cl)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(Cl)cn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Fc1cnc(nc1)-c1ccccc1C(=O)N1CC2CC(Oc3ccc(Cl)cn3)C1C2 |TLB:20:19:15.16:29,13:15:19.18:29|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1CC2CC(Oc3ccc(Cl)cn3)C1C2 |TLB:21:20:16.17:30,14:16:20.19:30|
Fc1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ccc(F)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
Fc1ccc(OC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
FC(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:15:13:8.9:11,THB:7:8:13.14:11|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:25,7:9:13.12:25|
FC(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:15:13:8.9:11,THB:7:8:13.14:11|
Fc1ccc(c(c1)C(=O)N1CC2CC(Oc3cnc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1cccc(C(=O)N2CC3CC(Oc4cnc(cn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1ccc(C(=O)N2CC3CC(Oc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Oc3cnc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Oc3cnc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
FC(F)(F)c1cnc(OC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1cnc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1cnc(OC2CC3CC2N(C3)C(=O)c2nc(C)ccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1cnc(OC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1cnc(OC2CC3CC2N(C3)C(=O)c2ncc(C)cc2-c2ncccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
CCc1cnc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:14:12:7.8:10,THB:6:7:12.13:10|
CCc1cnc(OC2CC3CC2N(C3)C(=O)c2nc(C)ccc2-n2nccn2)nc1 |TLB:14:12:7.8:10,THB:6:7:12.13:10|
CCc1cnc(OC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:14:12:7.8:10,THB:6:7:12.13:10|
CCc1cnc(OC2CC3CC2N(C3)C(=O)c2nc(C)ccc2-c2ncccn2)nc1 |TLB:14:12:7.8:10,THB:6:7:12.13:10|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ccc(nn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1cccc(C(=O)N2CC3CC(Oc4ccc(nn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CC(Oc3ccc(nn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Cc1ccc(C(=O)N2CC3CC(Nc4ccc(cn4)C(F)(F)F)C2C3)c(n1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Fc1cccc(C(=O)N2CC3CC(Nc4ccc(cn4)C(F)(F)F)C2C3)c1-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1ccc(C(=O)N2CC3CC(Nc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Fc1cccc(c1C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
FC(F)(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1cnc(C(=O)N2CC3CC(Nc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Cc1cnc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Cc1noc(n1)-c1cc(F)ccc1C(=O)N1CC2CC(Nc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
CN(C1CC2CC1N(C2)C(=O)c1ccccc1-n1nccn1)c1ccc(cn1)C(F)(F)F |TLB:9:7:2.3:5,THB:1:2:7.8:5|
CN(C1CC2CC1N(C2)C(=O)c1cccc(F)c1-n1nccn1)c1ccc(cn1)C(F)(F)F |TLB:9:7:2.3:5,THB:1:2:7.8:5|
CN(C1CC2CC1N(C2)C(=O)c1cc(F)ccc1-n1nccn1)c1ccc(cn1)C(F)(F)F |TLB:9:7:2.3:5,THB:1:2:7.8:5|
CN(C1CC2CC1N(C2)C(=O)c1nc(C)ccc1-n1nccn1)c1ccc(cn1)C(F)(F)F |TLB:9:7:2.3:5,THB:1:2:7.8:5|
CN(C1CC2CC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)c1ccc(cn1)C(F)(F)F |TLB:9:7:2.3:5,THB:1:2:7.8:5|
CN(C1CC2CC1N(C2)C(=O)c1cc(F)ccc1-c1ncccn1)c1ccc(cn1)C(F)(F)F |TLB:9:7:2.3:5,THB:1:2:7.8:5|
CN(C1CC2CC1N(C2)C(=O)c1c(F)cccc1-c1ncccn1)c1ccc(cn1)C(F)(F)F |TLB:9:7:2.3:5,THB:1:2:7.8:5|
CCN(C1CC2CC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)c1ccc(cn1)C(F)(F)F |TLB:10:8:3.4:6,THB:2:3:8.9:6|
Fc1cccc(C(=O)N2CC3CC(C2C3)N(CC2CC2)c2ccc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:12:8.9:14,6:8:12.11:14|
CC(=O)N(C1CC2CC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)c1ccc(cn1)C(F)(F)F |TLB:3:4:9.10:7,THB:11:9:4.5:7|
COCCN(C1CC2CC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)c1ccc(cn1)C(F)(F)F |TLB:12:10:5.6:8,THB:4:5:10.11:8|
Brc1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Fc1cccc(C(=O)N2CC3CC(Nc4ccc(Br)cn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Nc3ccc(Br)cn3)C1C2 |TLB:20:19:15.16:29,13:15:19.18:29|
Clc1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Fc1cccc(C(=O)N2CC3CC(Nc4ccc(Cl)cn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Fc1ccc(C(=O)N2CC3CC(Nc4ccc(Cl)cn4)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:21,5:7:11.10:21|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Nc3ccc(Cl)cn3)C1C2 |TLB:20:19:15.16:29,13:15:19.18:29|
FC(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:15:13:8.9:11,THB:7:8:13.14:11|
FC(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:15:13:8.9:11,THB:7:8:13.14:11|
COc1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:14:12:7.8:10,THB:6:7:12.13:10|
COc1ccc(NC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:14:12:7.8:10,THB:6:7:12.13:10|
Fc1cc(cnc1NC1CC2CC1N(C2)C(=O)c1ccccc1-n1nccn1)C(F)(F)F |TLB:15:13:8.9:11,THB:7:8:13.14:11|
Cc1ccc(c(n1)C(=O)N1CC2CC(Nc3ncc(cc3F)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:27,7:9:13.12:27|
Fc1cc(cnc1NC1CC2CC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)C(F)(F)F |TLB:15:13:8.9:11,THB:7:8:13.14:11|
FC(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncc(F)cn2)c(F)c1 |TLB:15:13:8.9:11,THB:7:8:13.14:11|
Cc1ccc(c(n1)C(=O)N1CC2CC(Nc3nc4ccccc4o3)C1C2)-n1nccn1 |TLB:14:13:9.10:25,7:9:13.12:25|
Fc1cccc(C(=O)N2CC3CC(Nc4nc5ccccc5o4)C2C3)c1-n1nccn1 |TLB:13:12:8.9:24,6:8:12.11:24|
Fc1cccc(C(=O)N2CC3CC(Nc4nc5ccccc5o4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:24,6:8:12.11:24|
Cc1ccc(NC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)cc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
FC(F)(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2cccc3cc[nH]c23)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
FC(F)(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2cccc3cn[nH]c23)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1cnc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2cccnc2-n2nccn2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2ncccc2-c2ncccn2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1cnc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c1-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1ccc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Fc1ccc(c(c1)C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1cccc(c1C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Cc1cccc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c1-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
COc1ccc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1ccc(C(=O)N2CC3CC(Nc4cnc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Fc1ccc(-c2ncco2)c(c1)C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2 |TLB:19:18:14.15:31,12:14:18.17:31|
Fc1cnc(nc1)-c1ccccc1C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1CC2CC(Nc3cnc(cn3)C(F)(F)F)C1C2 |TLB:21:20:16.17:33,14:16:20.19:33|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2nccnc2-c2ccccc2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ccccc2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2occc2-c2ccccc2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
CN(C1CC2CC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)c1cnc(cn1)C(F)(F)F |TLB:1:2:7.8:5,THB:9:7:2.3:5|
CN(C1CC2CC1N(C2)C(=O)c1cc(F)ccc1-c1ncccn1)c1cnc(cn1)C(F)(F)F |TLB:1:2:7.8:5,THB:9:7:2.3:5|
CN(C1CC2CC1N(C2)C(=O)c1ccccc1-c1ncccn1)c1cnc(cn1)C(F)(F)F |TLB:1:2:7.8:5,THB:9:7:2.3:5|
Fc1cccc(C(=O)N2CC3CC(C2C3)N(CC2CC2)c2cnc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:12:8.9:14,6:8:12.11:14|
Fc1cccc(C(=O)N2CC3CC(Nc4cnc(Cl)cn4)C2C3)c1-n1nccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Fc1ccc(c(c1)C(=O)N1CC2CC(Nc3cnc(Cl)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
Fc1cccc(C(=O)N2CC3CC(Nc4cnc(Cl)cn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Clc1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)cn1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1CC2CC(Nc3cnc(Cl)cn3)C1C2 |TLB:21:20:16.17:30,14:16:20.19:30|
Cc1cnc(NC2CC3CC2N(C3)C(=O)c2cccc(F)c2-n2nccn2)cn1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1cnc(NC2CC3CC2N(C3)C(=O)c2cc(F)ccc2-n2nccn2)cn1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1cnc(NC2CC3CC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)cn1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)cn1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Cc1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)cn1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2cccnc2-n2nccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Fc1cccc(C(=O)N2CC3CC(Nc4ncc(cn4)C(F)(F)F)C2C3)c1-n1nccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1ccc(C(=O)N2CC3CC(Nc4ncc(cn4)C(F)(F)F)C2C3)c(c1)-n1nccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Fc1ccc(c(c1)C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1cccc(c1C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
FC(F)(F)c1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Fc1cnc(nc1)-c1ccccc1C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(-c2ncco2)c1C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2 |TLB:19:18:14.15:31,12:14:18.17:31|
CCOc1ccc(C)nc1C(=O)N1CC2CC(Nc3ncc(cn3)C(F)(F)F)C1C2 |TLB:17:16:12.13:29,10:12:16.15:29|
Fc1cccc(C(=O)N2CC3CC(Nc4ncc(Cl)cn4)C2C3)c1-n1nccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Fc1ccc(c(c1)C(=O)N1CC2CC(Nc3ncc(Cl)cn3)C1C2)-n1nccn1 |TLB:14:13:9.10:23,7:9:13.12:23|
Fc1cccc(C(=O)N2CC3CC(Nc4ncc(Cl)cn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Fc1ccc(C(=O)N2CC3CC(Nc4ncc(Cl)cn4)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:21,5:7:11.10:21|
CN(C1CC2CC1N(C2)C(=O)c1cc(F)ccc1-c1ncccn1)c1ncc(Cl)cn1 |TLB:1:2:7.8:5,THB:9:7:2.3:5|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CC(Nc3ncc(Cl)cn3)C1C2 |TLB:20:19:15.16:29,13:15:19.18:29|
Clc1cnc(NC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
CN(C1CC2CC1N(C2)C(=O)c1ccccc1-c1ncc(F)cn1)c1ncc(Cl)cn1 |TLB:1:2:7.8:5,THB:9:7:2.3:5|
FC(F)(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1ccc(c(n1)C(=O)N1CC2CC(Nc3ccc(nn3)C(F)(F)F)C1C2)-n1nccn1 |TLB:14:13:9.10:26,7:9:13.12:26|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CC(Nc3ccc(nn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(C(=O)N2CC3CC(Nc4ccc(nn4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
FC(F)(F)c1ccc(NC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)cn1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Fc1cccc(C(=O)N2CC3CC(Nc4ccc(nc4)C(F)(F)F)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:25,6:8:12.11:25|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Fc1ccc(C(=O)N2CC3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:15:13:10.11:8.7,THB:5:7:13.14:10.11|
Fc1cnc(nc1)-c1ccccc1C(=O)N1CC2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:23:21:18.19:16.15,THB:13:15:21.22:18.19|
Cc1ccc(c(n1)C(=O)N1CC2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |THB:17:15:12.13:10.9,7:9:15.16:12.13|
FC(F)(F)c1cnc(NC2CC3CCC2N(C3)C(=O)c2ccccc2-n2nccn2)cn1 |TLB:17:15:9.10:12.13,THB:8:9:12.13:16.15|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Cc1cccc(C(=O)N2CC3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Fc1ccc(C(=O)N2CC3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:15:13:10.11:8.7,THB:5:7:13.14:10.11|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:23:21:18.19:16.15,THB:13:15:21.22:18.19|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:23:21:18.19:16.15,THB:13:15:21.22:18.19|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1CC2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:24:22:19.20:17.16,THB:14:16:22.23:19.20|
Cc1cnc(C(=O)N2CC3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:15:13:10.11:8.7,THB:5:7:13.14:10.11|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:23:21:18.19:16.15,THB:13:15:21.22:18.19|
Fc1cc(cnc1OC1CC2CCC1N(C2)C(=O)c1cccc(F)c1-c1ncccn1)C(F)(F)F |TLB:16:14:8.9:11.12,THB:7:8:11.12:15.14|
Cc1ccc(OC2CC3CCC2N(C3)C(=O)c2cccc(F)c2-c2ncccn2)nc1 |TLB:14:12:6.7:9.10,THB:5:6:9.10:13.12|
Brc1ccc(OC2CC3CCC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:14:12:6.7:9.10,THB:5:6:9.10:13.12|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Oc2ccc(Br)cn2)c1-c1ncccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Clc1ccc(OC2CC3CCC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:14:12:6.7:9.10,THB:5:6:9.10:13.12|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Oc2ccc(Cl)cn2)c1-c1ncccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Fc1cnc(nc1)-c1ccccc1C(=O)N1CC2CCC1C(C2)Oc1cnc(cn1)C(F)(F)F |TLB:23:21:18.19:16.15,THB:13:15:21.22:18.19|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1CC2CCC1C(C2)Oc1cnc(cn1)C(F)(F)F |TLB:24:22:19.20:17.16,THB:14:16:22.23:19.20|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CC2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:23:21:18.19:16.15,THB:13:15:21.22:18.19|
Fc1cccc(-c2ncccn2)c1C(=O)N1CC2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:23:21:18.19:16.15,THB:13:15:21.22:18.19|
FC(F)(F)c1cnc(NC2CC3CCC2N(C3)C(=O)c2ccccc2-c2ncccn2)cn1 |TLB:17:15:9.10:12.13,THB:8:9:12.13:16.15|
Fc1cccc(C(=O)N2CC3CCC2C(C3)Oc2ncc(cc2Cl)C(F)(F)F)c1-c1ncccn1 |TLB:16:14:11.12:9.8,THB:6:8:14.15:11.12|
Cc1cnc(C(=O)N2CC3CCC2C(C3)Oc2cnc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:15:13:10.11:8.7,THB:5:7:13.14:10.11|
Cc1cnc(C(=O)N2CC3CCC2C(C3)Oc2ncc(cc2F)C(F)(F)F)c(c1)-c1ncccn1 |TLB:15:13:10.11:8.7,THB:5:7:13.14:10.11|
Fc1cccc(C(=O)N2CC3CC(Oc4ncc(Cl)cn4)C2C3)c1-c1ncccn1 |TLB:13:12:8.9:22,6:8:12.11:22|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CC2CC(Oc3ncc(Cl)cn3)C1C2 |TLB:20:19:15.16:29,13:15:19.18:29|
Cc1ccc(c(n1)C(=O)N1CC2CC(Oc3ccc4cccnc4n3)C1C2)-n1nccn1 |TLB:7:9:13.12:26,14:13:9.10:26|
O=C(N1CC2CC(Oc3ccc4cccnc4n3)C1C2)c1ccccc1-n1nccn1 |TLB:1:2:6.5:19,7:6:2.3:19|
Cc1cnc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:23,5:7:11.10:23|
Cc1cnc(-c2ncccn2)c(c1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Cc1noc(n1)-c1cc(F)ccc1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:20:19:15.16:32,13:15:19.18:32|
Fc1cccc(-c2ncco2)c1C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:19:18:14.15:31,12:14:18.17:31|
Fc1ccc(-c2ncco2)c(c1)C(=O)N1CC2CC(Oc3ccc(cn3)C(F)(F)F)C1C2 |TLB:19:18:14.15:31,12:14:18.17:31|
Cc1cnc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-n1ccnn1 |TLB:12:11:7.8:24,5:7:11.10:24|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2ncccc2-c2ncccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
FC(F)(F)c1ccc(OC2CC3CC2N(C3)C(=O)c2ccccc2-c2ncccn2)nc1 |TLB:16:14:9.10:12,THB:8:9:14.15:12|
Cc1cnc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Clc1cnc(OC2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
COC(=O)c1c(C)ccnc1S[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1cc(cc(C)n1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1ncccc1C(O)=O
COC(=O)c1c(I)ccnc1S[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1ccccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1ccc(cn1)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1nccc(C)c1C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1cc(C)ccn1
COC(=O)c1ccnc(S[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Sc2cc(ccn2)C#N)c(n1)-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-n1nccn1)Sc1cc(ccn1)C#N
COc1cccc(c1C(=O)N1C[C@@H](CC[C@H]1C)Sc1cc(ccn1)C#N)-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(C)c1-n1nccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-n1nccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(Cl)cc1-n1nccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C)cc1-n1nccn1)Sc1cc(ccn1)C#N
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Sc2cc(ccn2)C#N)c(c1)-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Br)ccc1-n1nccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Cl)ccc1-n1nccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ccccc1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1Oc1ccccc1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CC1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1cnn(C)c1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-c1ccccc1)Sc1cc(ccn1)C#N
CC(C)Oc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Sc1cc(ccn1)C#N
CSc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CCCCO1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1N1CCCC1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Sc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1sccc1-c1ncccn1)Sc1cc(ccn1)C#N
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Sc2cc(ccn2)C#N)c(n1)-c1ncccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Sc1cc(ccn1)C#N
COC(=O)c1c(OC)ccnc1S[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1cc(ccn1)C#N
COc1c(N[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Nc1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc(C#N)c1C
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc(C#N)c1C |r|
COc1c(N[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-n2nccn2)nccc1C#N
COc1c(N[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-c2ncccn2)nccc1C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)N(C)c1cc(ccn1)C#N
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)N(C)c1cc(ccn1)C#N |r|
COc1c(ccnc1N(C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccsc1-n1nccn1)C#N |r|
COc1c(ccnc1N(C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccsc1-c1ncccn1)C#N |r|
CCN([C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)N(CC=C)c1cc(ccn1)C#N |r|
CCCN([C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)N(C(C)=O)c1cc(ccn1)C#N
Cc1cccc(C(=O)N2CC3CC(Oc4ccc(cn4)C(F)(F)F)C2C3)c1-c1ncco1 |TLB:13:12:8.9:25,6:8:12.11:25|
Cc1ccc(NC2CC3CC2N(C3)C(=O)c2nc(C)ccc2-n2nccn2)nc1 |TLB:13:11:6.7:9,THB:5:6:11.12:9|
Fc1cnc(nc1)-c1ccccc1C(=O)N1CC2CC(Nc3ncc(cc3F)C(F)(F)F)C1C2 |TLB:20:19:15.16:33,13:15:19.18:33|
Fc1ccc(C(=O)N2CC3CC(Nc4ncc(cn4)C(F)(F)F)C2C3)c(c1)-c1ncccn1 |TLB:12:11:7.8:24,5:7:11.10:24|
Cc1coc(n1)-c1ccc(C)nc1C(=O)N1C2CCC1C(COc1ncc(F)cn1)C2 |TLB:21:20:18.17:15|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2cccc(Cl)c2-c2ncccn2)cn1 |THB:8:9:13.12:15|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(Br)cn2)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(Br)cn2)c1-c1ncccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(Br)cn2)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(Br)cn2)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(Br)cn2)c1-c1ncccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(Br)cn2)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(Br)cn2)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(Br)cn2)c1-c1ncccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(Br)cn2)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c1-c1ccccn1 |TLB:15:13:11.10:8|
Fc1ccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c(c1)-n1nccn1 |TLB:14:12:10.9:7|
Fc1ccc(c(c1)C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Fc1cccc(c1C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Fc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
FC(F)(F)c1ccc(NC2CC3CCC2N3C(=O)c2ccccc2-c2ncccn2)nc1 |THB:8:9:13.12:15|
Fc1cnc(nc1)-c1ccccc1C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:23:21:19.18:16|
FC(F)(F)c1ccc(NC2CC3CCC2N3C(=O)c2cccc(Cl)c2-c2ncccn2)nc1 |THB:8:9:13.12:15|
CN(C1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1)c1ccc(cn1)C(F)(F)F |THB:1:2:6.5:8|
Cc1cnc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(C2)Nc1ccc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Cc1cnc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:14:12:10.9:7|
FC(F)(F)c1ccc(NC2CC3CCC2N3C(=O)c2ncccc2-c2ncccn2)nc1 |THB:8:9:13.12:15|
Fc1cc(cnc1NC1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncccn1)C(F)(F)F |THB:7:8:12.11:14|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2Cl)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2Cl)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cnc(nc1)-c1ccccc1C(=O)N1C2CCC1C(C2)Nc1ncc(cc1Cl)C(F)(F)F |TLB:22:20:18.17:15|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ccccc2-c2ncccn2)c(Cl)c1 |THB:8:9:13.12:15|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ncccc2-c2ncccn2)c(Cl)c1 |THB:8:9:13.12:15|
FC(F)c1ccc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-n2nccn2)nc1 |THB:7:8:12.11:14|
FC(F)c1ccc(NC2CC3CCC2N3C(=O)c2cccc(F)c2-c2ncccn2)nc1 |THB:7:8:12.11:14|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C#N)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C#N)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C#N)c1-c1ncccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C#N)c1-c1ncccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ccc(cn2)C#N)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1cnc(nc1)-c1ccccc1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:23:21:19.18:16|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ncc(F)cn1 |TLB:15:13:11.10:8|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ccccc2-c2ncccn2)cn1 |THB:8:9:13.12:15|
Cc1cnc(c(c1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2cccnc2-n2nccn2)cn1 |THB:8:9:13.12:15|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Cc1cnc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Cc1cnc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:14:12:10.9:7|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ncccc2-c2ncccn2)cn1 |THB:8:9:13.12:15|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ccccc2-c2ccccc2)cn1 |THB:8:9:13.12:15|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c1-c1ccccn1 |TLB:15:13:11.10:8|
Fc1ccc(-c2ncco2)c(c1)C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:21:19:17.16:14|
Fc1cccc(-c2ncco2)c1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:21:19:17.16:14|
Cc1noc(n1)-c1cc(F)ccc1C(=O)N1C2CCC1C(C2)Nc1cnc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
COc1ccc(C(=O)N2C3CCC2C(C3)Nc2cnc(cn2)C(F)(F)F)c(Cl)n1 |TLB:15:13:11.10:8|
Fc1ccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:14:12:10.9:7|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Fc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
FC(F)(F)c1cnc(NC2CC3CCC2N3C(=O)c2ccccc2-c2ncccn2)nc1 |THB:8:9:13.12:15|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2nc(cs2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2nnc(s2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Cc1cnc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2F)C(F)(F)F)c(c1)-n1nccn1 |TLB:14:12:10.9:7|
FC(F)(F)c1ccc(OC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)nc1 |THB:8:9:13.12:15|
Cc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-n1ccnn1 |TLB:15:13:11.10:8|
Fc1cccc(c1C(=O)N1C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
FC(F)(F)c1ccc(OC2CC3CCC2N3C(=O)c2cccnc2-n2nccn2)nc1 |THB:8:9:13.12:15|
Cc1ccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c(n1)-n1nccn1 |TLB:14:12:10.9:7|
Cc1cnc(c(c1)C(=O)N1C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1ccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c(c1)-c1ncccn1 |TLB:14:12:10.9:7|
Fc1cccc(-c2ncccn2)c1C(=O)N1C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
FC(F)(F)c1ccc(OC2CC3CCC2N3C(=O)c2ccccc2-c2ncccn2)nc1 |THB:8:9:13.12:15|
Fc1cnc(nc1)-c1ccccc1C(=O)N1C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:22:20:18.17:15|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1C2CCC1C(C2)Oc1ccc(cn1)C(F)(F)F |TLB:23:21:19.18:16|
Cc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(cn2)C(F)(F)F)c1-c1ncco1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(nc2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(nc2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(c1C(=O)N1C2CCC1C(C2)Oc1ccc(nc1)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ccc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ncc(Br)cn2)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2cnc3ccccc3n2)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2cc(Br)cnc2Cl)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Oc2cnc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2cnc(cn2)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1ccc(C(=O)N2C3CCC2C(C3)Oc2cnc(cn2)C(F)(F)F)c(n1)-n1nccn1 |TLB:14:12:10.9:7|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2cnc(cn2)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cc(cnc1NC1CC2CCC1N2C(=O)c1ccccc1-n1nccn1)C(F)(F)F |THB:7:8:12.11:14|
Fc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2F)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2F)C(F)(F)F)c1-n1nccn1 |TLB:15:13:11.10:8|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1ncc(cc1F)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Cc1ccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2F)C(F)(F)F)c(n1)-n1nccn1 |TLB:14:12:10.9:7|
Cc1cnc(c(c1)C(=O)N1C2CCC1C(C2)Nc1ncc(cc1F)C(F)(F)F)-n1nccn1 |TLB:16:14:12.11:9|
Fc1cc(cnc1NC1CC2CCC1N2C(=O)c1cccc(F)c1-c1ncco1)C(F)(F)F |THB:7:8:12.11:14|
Cc1cnc(-c2ncccn2)c(c1)C(=O)N1C2CCC1C(C2)Nc1ncc(cc1F)C(F)(F)F |TLB:22:20:18.17:15|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1C2CCC1C(C2)Nc1ncc(cc1F)C(F)(F)F |TLB:22:20:18.17:15|
Cc1cnc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2F)C(F)(F)F)c(c1)-c1ncccn1 |TLB:14:12:10.9:7|
Fc1cc(cnc1NC1CC2CCC1N2C(=O)c1ncccc1-c1ncccn1)C(F)(F)F |THB:7:8:12.11:14|
Fc1cc(cnc1NC1CC2CCC1N2C(=O)c1c(F)cccc1-c1ncccn1)C(F)(F)F |THB:7:8:12.11:14|
Fc1cnc(nc1)-c1ccccc1C(=O)N1C2CCC1C(C2)Nc1ncc(cc1F)C(F)(F)F |TLB:22:20:18.17:15|
Fc1cc(cnc1NC1CC2CCC1N2C(=O)c1ccccc1-c1ncccn1)C(F)(F)F |THB:7:8:12.11:14|
Cc1cccc(C(=O)N2C3CCC2C(C3)Nc2ncc(cc2F)C(F)(F)F)c1-c1ncccn1 |TLB:15:13:11.10:8|
Fc1cnc(nc1)-c1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1ncc(cc1F)C(F)(F)F |TLB:23:21:19.18:16|
CC(O)c1cccc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2cccc(c2)C(C)O)c(n1)-n1nccn1
CC(O)c1cccc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-c2ncccn2)c1 |r|
C[C@@H]1CC[C@H](CC1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc(c1)C(C)(O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc(c1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C1(O)CCC1 |r|
CCC(C)(O)c1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)[C@](C)(O)C1CC1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)[C@@](C)(O)C1CC1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc(c1)C(C)(O)C1CC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc(c1)C(C)(O)C1CCCC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc(c1)C(C)(O)C1CCC1 |r|
CCC(C)(O)c1cccc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccc1F)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc(c1F)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2C(O)CCCc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccc2CCC(O)c2c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2[C@H](O)CCc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2[C@@H](O)CCc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccc2CC[C@@H](O)c2c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccc2CC[C@H](O)c2c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2c1CCC[C@@]2(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2c1CCC[C@]2(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2c1CC[C@@]2(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2c1CC[C@]2(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccc2CCC(C)(O)c2c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccc2CC[C@@](C)(O)c2c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccc2CC[C@](C)(O)c2c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc(c1)C(C)(O)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1cccc(c1)C(C)(C)O |r|
Cc1ccc(c(c1)C(=O)N1CCCN(CC1)c1nc2ccc(F)cc2c(=O)[nH]1)-n1nccn1
CC1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1nc2ccc(F)cc2c(=O)[nH]1
Cc1ccc(c(c1)C(=O)N1CCCN(CC1)c1nc2ccc(Cl)cc2c(=O)[nH]1)-n1nccn1
CC1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1nc2ccc(Cl)cc2c(=O)[nH]1
COc1ccc(NC(=O)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c(N)c1 |r|
Cc1nc(C(=O)N2CCC[C@H]2c2nc3cc(Cl)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(Cl)cc(cc3[nH]2)C(F)(F)F)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Cl)c(C)cc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)cc(C)cc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(CO)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(F)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(cccc3[nH]2)C(F)(F)F)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(Br)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Br)cc(C)c3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
COc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
COc1cc2nc([nH]c2cc1OC)C1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(c(F)cc3[nH]2)C(F)(F)F)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(F)c(Br)cc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(Br)cc(F)cc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)c(C)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
CC(C)c1cccc2[nH]c(nc12)C1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c4OCCOc4ccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(cc(cc3[nH]2)C(F)(F)F)C(F)(F)F)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Cl)c(Cl)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@H]2c2nc3c(O)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Br)ccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(ccc3[nH]2)C(F)(F)F)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(C)c(C)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)cccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(ccc3[nH]2)C(C)(C)C)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(Cl)cc(cc3[nH]2)C(F)(F)F)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Cl)c(C)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)cc(C)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(CO)cccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(cccc3[nH]2)C(F)(F)F)c(s1)-c1ccccc1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(Br)cccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Br)cc(C)c3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccccc1
COc1cc2nc([nH]c2cc1OC)C1CCCN1C(=O)c1nc(C)sc1-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(c(F)cc3[nH]2)C(F)(F)F)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(F)c(Br)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(Br)cc(F)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)c(C)ccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@H]2c2nc3cccc(Cl)c3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c4OCCOc4ccc3[nH]2)c(s1)-c1ccccc1
COc1ccc2[nH]c(nc2c1)C1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1nc(C(=O)N2CCC[C@H]2c2nc3c(C)cc(C)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@H]2c2nc3cc(Cl)c(C)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@H]2c2nc3c(C)cc(Br)cc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@H]2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@H]2c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(s1)-c1ccccc1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1c(F)cccc1-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc2ccc(SC)cc2[nH]1)-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1c(C)cccc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc3ccc(SC)cc3[nH]2)c(cc1OC)-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc2ccc(OC)cc2[nH]1)-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1c(C)cccc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(OC)c(OC)cc1-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1c(F)cccc1-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc2cccc(SC)c2[nH]1)-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
COc1ccc(c(C(=O)N2CCC[C@H]2c2nc3cccc(SC)c3[nH]2)c1F)-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1c(C)cccc1-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1cccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1c(F)c(C)ccc1-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1nccn1
CSc1cccc2[nH]c(nc12)[C@@H]1CCCN1C(=O)c1c(F)c(C)ccc1-n1nccn1
CSc1cccc2[nH]c(nc12)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1nccn1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1ccccc1-n1cccn1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1cccn1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1cccn1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1c(F)c(C)ccc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1ccc(Br)cc1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1Cl
COc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CCC[C@H]1c1nc2ccc(OC)cc2[nH]1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(F)c1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1ccc(C)cc1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccc(C)cc1)C1CC1
CCc1ccc(cc1)-c1sc(C)nc1C(=O)N1CCC[C@H]1c1nc2ccc(OC)cc2[nH]1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1ccccc1-c1ccc(C)c(C)c1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(Cl)c(Cl)c1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1cccc(Cl)c1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc2cc(Cl)ccc2[nH]1)-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(Br)c(Cl)c1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(C)c(C)c1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccccc1
COc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(Br)c(Cl)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1ccc(Br)cc1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccccc1)C1CC1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1Cl
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CCC[C@H]1c1nc2ccc(SC)cc2[nH]1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(c1)C(F)(F)F
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(F)c1
COc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1ccc(C)cc1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccc(C)cc1)C1CC1
CCc1ccc(cc1)-c1sc(C)nc1C(=O)N1CCC[C@H]1c1nc2ccc(SC)cc2[nH]1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1nccnc1-c1cc(C)cc(F)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1ccccc1-c1ccc(C)c(C)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(Cl)c(Cl)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(F)cc1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1cccc(Cl)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(Cl)c(Cl)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CC(CN1C=O)c1cnc(nc1)-c1ccc(C)c(C)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(Br)c(Cl)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(C)c(C)c1
COc1cccc(c1)-c1nc(C)ncc1C(=O)N1CCC[C@H]1c1nc2ccc(SC)cc2[nH]1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccccc1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(Br)c(Cl)c1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1cc(Cl)cc(Cl)c1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc2cccc(Cl)c2[nH]1)-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1ccc(Br)cc1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccccc1)C1CC1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1Cl
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CCC[C@H]1c1nc2cccc(SC)c2[nH]1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(c1)C(F)(F)F
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(F)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1ccc(C)cc1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1ccc(F)c(F)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccc(C)cc1)C1CC1
CCc1ccc(cc1)-c1sc(C)nc1C(=O)N1CCC[C@H]1c1nc2cccc(SC)c2[nH]1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)C1CC1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
COc1ccc(cc1)-c1nccnc1C(=O)N1CCC[C@H]1c1nc2cccc(SC)c2[nH]1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nccnc1-c1cccc(c1)C(F)(F)F
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1nccnc1-c1cc(C)cc(F)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1ccccc1-c1ccc(C)c(C)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(C)cc1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(Cl)c(Cl)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(F)cc1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1cccc(Cl)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(Cl)c(Cl)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(C)c(C)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(Br)c(Cl)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(C)c(C)c1
COc1cccc(c1)-c1nc(C)ncc1C(=O)N1CCC[C@H]1c1nc2cccc(SC)c2[nH]1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccccc1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cncnc1-c1cccc(C)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cncnc1-c1cc(Cl)cc(Cl)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1ccc(Br)c(Cl)c1
CSc1cccc2nc([nH]c12)[C@@H]1CCCN1C(=O)c1cnc(C)nc1-c1cc(Cl)cc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Cl)c(Cl)cc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Br)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(ccc3[nH]2)C(F)(F)F)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(C)c(C)cc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3c(C)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(Cl)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(F)c(Cl)cc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCCC2c2nc3cc(ccc3[nH]2)C(C)(C)C)c(s1)-c1cccc(Cl)c1
Cc1ccc(c(c1)C(=O)N1C[C@@H](F)C[C@H]1c1nc2ccc(Cl)c(C)c2[nH]1)-n1nccn1 |r|
Cc1nc(C(=O)N2C[C@H](F)C[C@H]2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1ccc(c(c1)C(=O)N1C[C@H](F)C[C@H]1c1nc2c(C)cccc2[nH]1)-n1nccn1
Cc1nc(C(=O)N2C[C@@H](F)C[C@H]2c2nc3c(C)cccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2C[C@H](F)C[C@H]2c2nc3c(C)cccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CC(F)(F)C[C@H]2c2nc3c(C)cccc3[nH]2)c(s1)-c1ccccc1
Cc1ccc(c(c1)C(=O)N1C[C@H](F)C[C@H]1c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(F)(F)C[C@H]1c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
Cc1nc(C(=O)N2C[C@@H](F)C[C@H]2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CC(F)(F)C[C@H]2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2C[C@H](F)C[C@H]2c2nc3c(C)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
CO[C@H]1C[C@H](N(C1)C(=O)c1cc(C)ccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1 |r|
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(Cl)ccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1c(F)c(OC)ccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(OC)ccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1c(F)c(C)ccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1c(C)cccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1ccc(C)cc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(C)c(C)cc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(F)ccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(Cl)ccc1-n1nccn1)c1nc2ccc(OC)cc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(C)ccc1-n1nccn1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(OC)ccc1-n1nccn1)c1nc2ccc(OC)cc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1ccc(C)cc1-n1nccn1)c1nc2ccc(OC)cc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(C)c(C)cc1-n1nccn1)c1nc2ccc(OC)cc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(F)ccc1-n1nccn1)c1nc2ccc(OC)cc2[nH]1
CO[C@H]1CN(C(=O)c2nc(C)sc2-c2ccccc2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(C)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(C)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)cccc2[nH]1
CO[C@H]1CN(C(=O)c2nc(C)sc2-c2cccc(Cl)c2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2nc(C)sc2-c2cccc(Cl)c2)C(C)(C1)c1nc2c(C)cccc2[nH]1
CO[C@H]1CN(C(=O)c2nc(C)sc2-c2ccccc2)C(C)(C1)c1nc2c(C)cccc2[nH]1
CO[C@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccccc1)c1nc2c(C)cccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(C)ccc2-n2nccn2)[C@@](C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2nc(C)sc2-c2cccc(Cl)c2)[C@@](C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1cccc(C)c1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(sc1-c1ccc(C)c(C)c1)N(C)C)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccc(C)cc1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccc(OC)cc1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1ccccc1-c1ccc(C)c(C)c1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1ccccc1-c1ccccc1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccccc1)c1nc2c(C)cccc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1ccccc1-c1ccc(F)c(C)c1)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(sc1-c1cccc(Cl)c1)N(C)C)c1nc2ccc(Cl)c(C)c2[nH]1
CO[C@H]1CN(C(=O)c2c(F)cccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(F)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(Cl)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2ccccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2c(F)c(OC)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2c(F)c(C)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(C)c(C)cc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2ccc(C)cc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccccc1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(ccc2-n2nccn2)C(F)(F)F)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(OC(F)(F)F)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(OC)c(OC)cc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2cc(C)ccc2-n2cccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2ccccc2-n2cccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2nc(C)ccc2-n2cccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@H]1CN(C(=O)c2nc(C)ccc2-n2nccn2)C(C)(C1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1ccccc1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1)c1nc2c(C)cccc2[nH]1
CO[C@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1)c1nc2c(C)c(Cl)ccc2[nH]1
CO[C@@H]1C[C@H](N(C1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1)c1nc2c(C)c(Cl)ccc2[nH]1
C[C@H]1CCN([C@@H]1c1nc2cccc(C)c2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(F)cc1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1ccccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(F)c(F)cc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
COC(=O)c1cccc2[nH]c(nc12)[C@@H]1[C@@H](C)CCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
COc1cccc2[nH]c(nc12)[C@@H]1[C@@H](C)CCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(CO)cccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(F)cccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(C)ccc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(F)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(F)c(F)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(C)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
CC(C)c1cccc2[nH]c(nc12)[C@@H]1[C@@H](C)CCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1[C@@H](C)CCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(CO)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)cc(C)c2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(C)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc2[nH]c(nc12)[C@@H]1[C@@H](C)CCN1C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(C)cc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(C)ccc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
CC(C)c1cccc2[nH]c(nc12)[C@@H]1[C@@H](C)CCN1C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)cc(C)c2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)cccc2[nH]1)C(=O)c1nc(C)sc1-c1ccccc1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1cc(F)ccc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1c(F)cccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(OC)c(OC)cc2[nH]1)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1c(F)c(C)ccc1-n1nccn1
COc1ccc(c(C(=O)N2CC[C@H](C)[C@H]2c2nc3cc(OC)c(OC)cc3[nH]2)c1F)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1c(C)cccc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1ccccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(C)ccc2[nH]1)C(=O)c1nc(C)sc1-c1ccccc1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1nc(C)sc1-c1ccc(cc1)C(F)(F)F
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1sc(C)nc1-c1ccc(C)cc1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
COc1ccc(cn1)-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(OC)c(OC)cc2[nH]1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1nc(C)sc1-c1ccc(F)cc1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1ncsc1-c1cccc(Cl)c1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1ccccc1-n1cccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1cc(C)ccc1-n1cccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1ccccc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1ccccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2ccccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1ccccc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(C)ccc1-n1cccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1sc(C)nc1-c1ccc(C)cc1
COc1ccc(c(c1)C(=O)N1CC[C@H](C)[C@H]1c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1c(F)c(C)ccc1-n1nccn1
COc1ccc(cn1)-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2c(C)c(Cl)ccc2[nH]1
C[C@H]1CCN([C@@H]1c1nc2c(C)cccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(F)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-n1cccn1
COc1ccc(c(c1)C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(Cl)c(C)cc2[nH]1)-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)c(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1ccccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1ccccc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1sc(C)nc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C#N)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-n1cccn1
COc1ccc(c(c1)C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(C)c(C)cc2[nH]1)-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1ccccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1ccccc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1sc(C)nc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(Cl)c1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(F)cc1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1ccccc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1cc(C)ccc1-n1cccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1sc(C)nc1-c1ccc(C)cc1
COc1ccc(c(c1)C(=O)N1CC[C@H](C)[C@H]1c1nc2c(C)cc(Cl)cc2[nH]1)-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)cc(Cl)cc2[nH]1)C(=O)c1c(F)c(C)ccc1-n1nccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-c1ccccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(Cl)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-c1cccnc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(F)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(F)ccc1-c1ccccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)cccc1-c1cccnc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(ccc1-c1ccccc1)C#N
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1ccc(C)cc1-c1ccccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1ccc(C)cc1-c1cccnc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1ccc(C)cc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)cccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)c(C)ccc1-c1ccccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(ccc1-c1ccccc1)C(F)(F)F
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)c(C)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)c(C)ccc1-c1cccnc1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(F)cc1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2c(Cl)cccc2[nH]1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1cccc(C)c1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(Br)cc1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(C)sc1-c1ccc(F)c(F)c1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1ccsc1-c1ccc(C)c(C)c1
C[C@H]1CCN([C@@H]1c1nc2c(Cl)cccc2[nH]1)C(=O)c1nc(sc1-c1ccc(C)c(C)c1)N(C)C
COc1ccccc1-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2c(Cl)cccc2[nH]1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1ccc(C)cc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(F)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)c(C)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1c(F)cccc1-c1ncccn1
COc1cccc(c1)C#Cc1ccccc1C(=O)N1CC[C@H](C)[C@H]1c1nc2c(C)c(Cl)ccc2[nH]1
COc1cccc(c1)C#Cc1ccccc1C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(Cl)c(C)cc2[nH]1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(C)c1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cc1
COc1ccc(cc1)-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(Br)cc1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)c(F)c1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1ccsc1-c1ccc(C)c(C)c1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccccc1Cl
COc1ccccc1-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F
C[C@H]1CCN([C@@H]1c1nc2cc(ccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(Br)cc1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cc1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)c(F)c1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccccc1Cl
COc1ccccc1-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2c(cccc2[nH]1)C(F)(F)F
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(C)c1
COc1ccc(cc1)-c1sc(C)nc1C(=O)N1CC[C@H](C)[C@H]1c1nc2c(cccc2[nH]1)C(F)(F)F
C[C@H]1CCN([C@@H]1c1nc2c(cccc2[nH]1)C(F)(F)F)C(=O)c1ccsc1-c1ccc(C)c(C)c1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(C)ccc1-c1ccccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(Cl)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(C)ccc1-c1cccnc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(F)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(F)ccc1-c1ccccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(ccc1-c1ccccc1)C#N
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1ccc(C)cc1-c1ccccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1ccc(C)cc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1c(F)cccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(ccc1-c1ccccc1)C(F)(F)F
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1c(F)c(C)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(C)ccc1-c1ccccc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1c(F)c(C)ccc1-c1cccnc1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1ccc(C)cc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(F)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1c(F)c(C)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1c(F)cccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2c(C)c(Cl)ccc2[nH]1)C(=O)c1cc(C)ccc1-c1ncccn1
COc1cc2nc([nH]c2cc1OC)[C@@H]1[C@@H](C)CCN1C(=O)c1cc(C)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2ccc(Cl)c(C)c2[nH]1)C(=O)c1cc(C)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2cc(Cl)cc(C)c2[nH]1)C(=O)c1cc(C)ccc1-c1ncccn1
C[C@H]1CCN([C@@H]1c1nc2cc(C)c(C)cc2[nH]1)C(=O)c1cc(C)ccc1-c1ncccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3cccc(C)c3[nH]2)c(s1)-c1ccccc1 |r|
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1)-n1nccn1
Cc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
COc1cccc(c1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
COc1ccc(cc1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
Cc1cc2nc([nH]c2cc1C)[C@]1(C)CCCN1C(=O)c1ccccc1-c1ccccc1F
Cc1cc2nc([nH]c2cc1C)[C@]1(C)CCCN1C(=O)c1ccccc1-c1ccc(F)cc1
Cc1cc2nc([nH]c2cc1C)[C@]1(C)CCCN1C(=O)c1ccccc1-c1cccc(F)c1
Cc1cccc(c1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
Cc1ccc(cc1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1)-c1ccc(F)cc1C
Cc1ccc(-c2cccc(F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(Cl)ccc2[nH]1)-n1nccn1
COc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
COc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1)-c1ccccc1F
Cc1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1ccc2[nH]c(nc2c1C)[C@]1(C)CCCN1C(=O)c1ccccc1-c1cccc(F)c1
COc1cccc(c1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1cccc(c1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
COc1ccc(cc1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(F)c(Cl)cc2[nH]1)-n1nccn1
Cc1ccc(cc1)-c1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1
Cc1ccc2[nH]c(nc2c1C)[C@]1(C)CCCN1C(=O)c1ccccc1-c1ccccc1F
Cc1ccc2[nH]c(nc2c1C)[C@]1(C)CCCN1C(=O)c1ccccc1-c1ccc(F)cc1
C[C@]1(CCCN1C(=O)c1c(F)cccc1-n1nccn1)c1nc2cc(F)c(Br)cc2[nH]1
Cc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(F)c(Br)cc3[nH]2)c1F)-n1nccn1
COc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(F)c(Br)cc3[nH]2)c(cc1OC)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(F)ccc1-n1nccn1)c1nc2cc(F)c(Br)cc2[nH]1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(F)c(Br)cc3[nH]2)c(cc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(F)c(Br)cc2[nH]1)-n1cccn1
C[C@]1(CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)c1nc2cc(F)c(Br)cc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(C)(C)C)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(F)c(Br)cc3[nH]2)c(c1)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2cc(F)c(Br)cc2[nH]1)-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(F)c(Br)cc3[nH]2)c1F)-n1nccn1
C[C@]1(CCCN1C(=O)c1c(F)cccc1-n1nccn1)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c1F)-n1nccn1
COc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c(cc1OC)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(F)ccc1-n1nccn1)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c(cc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F)-n1cccn1
C[C@]1(CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(Cl)cc(cc2[nH]1)C(F)(F)F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c(c1)-n1nccn1
C[C@]1(CCCN1C(=O)c1ccccc1-n1cccn1)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1ccccc1-n1nccn1)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F)-n1cccn1
C[C@]1(CCCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F)-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c1F)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
COc1ccccc1-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
COc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(Cl)c(C)cc2[nH]1)-n1nccn1
COc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F)-c1ccccc1F
Cc1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(-c2cccc(F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(-c2cccc(c2)C(F)(F)F)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(-c2ccc3OCOc3c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(-c2ccc(cc2)C(F)(F)F)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(-c2ccc(OC(F)(F)F)cc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(-c2cccc(c2)C#N)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)cc(C)cc2[nH]1)-n1nccn1
Cc1ccc(-c2ccc(cc2)C#N)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F)-c1cccc(C)c1C
CCOc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
Cc1ccc(-c2cccc(OC(F)(F)F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1c(F)cccc1-n1nccn1)c1nc2cc(ccc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1cc(F)ccc1-n1nccn1)c1nc2cc(ccc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)c1nc2cc(ccc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1ccccc1-n1nccn1)c1nc2cc(ccc2[nH]1)C(F)(F)F
COc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(ccc3[nH]2)C(F)(F)F)c1F)-n1nccn1
Cc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(ccc3[nH]2)C(F)(F)F)c1F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(cccc2[nH]1)C(F)(F)F)-n1nccn1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(ccc3[nH]2)C(F)(F)F)c(cc1C)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(ccc3[nH]2)C(F)(F)F)c(c1)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F)c1nc2cc(ccc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1)c1nc2cc(ccc2[nH]1)C(F)(F)F
COc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(ccc3[nH]2)C(F)(F)F)c(cc1OC)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-n1cccn1
C[C@]1(CCCN1C(=O)c1ccccc1-n1cccn1)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-n1cccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-n1nccn1
Cc1cccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(ccc3[nH]2)C(F)(F)F)c1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(Br)cccc2[nH]1)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-c1ccc(F)cc1C
Cc1ccc(-c2cccc(F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(-c2ccc(cc2)C(F)(F)F)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(-c2cccc(OC(F)(F)F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
COc1ccccc1-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-c1ccccc1C
Cc1ccc(-c2ccc(OC(F)(F)F)cc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
COc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(Br)cc(C)c2[nH]1)-n1nccn1
Cc1ccc(-c2cccc(c2)C#N)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
COc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(-c2ccc(cc2)C#N)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-c1ccccc1F
Cc1ccc(-c2cccc(c2)C(F)(F)F)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-c1cccc(C)c1C
Cc1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(-c2ccc3OCOc3c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(cc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(OC(F)(F)F)ccc2[nH]1)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)c1nc2c(F)c(F)ccc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(F)c(F)ccc2[nH]1)-n1cccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(c1)-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c1F)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(F)ccc1-n1nccn1)c1nc2c(F)c(F)ccc2[nH]1
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2c(F)c(F)ccc2[nH]1)-n1nccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(s1)-c1ccc(C)cc1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(s1)-c1cccc(C)c1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(s1)-c1ccc(Cl)cc1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(F)c(F)ccc3[nH]2)c(s1)-c1cccc(F)c1
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CCC[C@@]1(C)c1nc2c(F)c(F)ccc2[nH]1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1
Cc1ccc(-c2ccccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1
Cc1ccc(-c2cccnc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(F)cc2[nH]1)C(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(F)c(Br)cc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(Br)cc(F)cc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(Cl)cccc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(F)c(F)ccc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)ccc2[nH]1)-n1nccn1
CC(C)c1cccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccccc1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(SC(F)(F)F)ccc2[nH]1)-n1nccn1
COc1ccc(OC)c2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c3OCCOc3ccc2[nH]1)-n1nccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(c1)-n1nccn1
COc1cc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(cc1OC)-n1nccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(cc1C)-n1nccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1ccccc1-n1cccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1)-n1cccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1)-n1cccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(F)ccc1-n1nccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1ccccc1-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1c(F)cccc1-n1nccn1
Cc1cccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
COc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)cccc2[nH]1)-n1nccn1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)cccc3[nH]2)c(cc1C)-n1nccn1
Cc1cccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1ccccc1-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@]1(C)CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1)-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(C)c(C)cc3[nH]2)c1F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(C)c(C)cc3[nH]2)c(c1)-n1nccn1
COc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(C)c(C)cc3[nH]2)c(cc1OC)-n1nccn1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(C)c(C)cc3[nH]2)c(cc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1)-n1cccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)cccc2[nH]1)-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@]1(C)CCCN1C(=O)c1cc(F)ccc1-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@]1(C)CCCN1C(=O)c1ccccc1-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(F)ccc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1c(F)cccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(OC)c(OC)cc2[nH]1)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1c(F)c(C)ccc1-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC)c(OC)cc3[nH]2)c1F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(Cl)c(Cl)cc2[nH]1)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1ccccc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1nc(C)sc1-c1ccc(cc1)C(F)(F)F
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1sc(C)nc1-c1ccc(C)cc1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
COc1ccc(cn1)-c1sc(C)nc1C(=O)N1CCC[C@@]1(C)c1nc2cc(OC)c(OC)cc2[nH]1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1nc(C)sc1-c1ccc(F)cc1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(Br)ccc2[nH]1)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1ncsc1-c1cccc(Cl)c1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1ccccc1-n1cccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1cccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1nc(C)ccc1-n1cccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1nc(C)ccc1-n1nccn1
COc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC)c(OC)cc3[nH]2)c(cc1OC)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1ccccc1-c1cccc(C)c1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1ccccc1-c1ccc(C)cc1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cnc(C)nc1-c1cccc(C)c1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F)-n1nccn1
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cncnc1-c1ccccc1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1)-c1ccc(F)cc1C
COc1ccccc1-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
COc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
COc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1)-c1ccccc1F
Cc1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
Cc1ccc(-c2cccc(F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1)-c1ccccc1C
Cc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(F)ccc1-c1ccccc1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(F)ccc1-c1ccccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(F)ccc1-c1cccnc1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1c(F)cccc1-c1ccccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1c(F)cccc1-c1ncccn1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1cc(F)ccc1-c1ncccn1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1c(F)cccc1-c1ccccc1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccccc1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccc(F)cc1
Cc1ccccc1-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
COc1ccccc1-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1cccc(c1)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
COc1cccc(c1)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1ccc(cc1)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccccc1F
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1cccc(F)c1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(cc1C)-n1nccn1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(OC(F)(F)F)ccc2[nH]1
COc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(OC(F)(F)F)ccc2[nH]1)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(c1)-n1nccn1
Cc1ccc(-c2ccccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(OC(F)(F)F)ccc2[nH]1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(c1)-c1ccccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(c1)-c1cccnc1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(c1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(s1)-c1ccccc1C
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(s1)-c1cccc(Cl)c1Cl
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(s1)-c1cc(F)cc(F)c1
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CCC[C@@]1(C)c1nc2cc(OC(F)(F)F)ccc2[nH]1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(OC(F)(F)F)ccc3[nH]2)c(s1)-c1ccc(F)cc1
COc1cccc(c1)C#Cc1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)cc(Br)cc2[nH]1
COc1cccc(c1)C#Cc1ccccc1C(=O)N1CCC[C@@]1(C)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1cccc(F)c1F
Cc1cc(ccc1F)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1ccc(-c2nc(C(=O)N3CCC[C@@]3(C)c3nc4c(C)c(Cl)ccc4[nH]3)c(s2)-c2ccc(F)cc2)c(F)c1
Cc1ccc(cc1C)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1cccc(c1)C#N
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccccc1Cl
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1cccc(Cl)c1
Cc1ccc(cc1Cl)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1cc(F)ccc1-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
COc1cc(F)ccc1-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1c(Cl)ccc2[nH]c(nc12)[C@]1(C)CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1cc(F)ccc1F
C[C@]1(CCCN1C(=O)c1cc(Br)ccc1-c1ccccc1)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(cn1)-n1nccn1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c(cn1)-c1ccccc1
C[C@]1(CCCN1C(=O)c1cc(ccc1-c1ccccc1)-c1cccnc1)c1nc2cc(ccc2[nH]1)C(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)c(Br)cc2[nH]1)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(C)c(Br)cc3[nH]2)c(c1C)-n1nccn1
Cc1c(Br)cc2[nH]c(nc2c1C)[C@]1(C)CCCN1C(=O)c1c(F)cccc1-n1nccn1
Cc1c(Br)cc2[nH]c(nc2c1C)[C@]1(C)CCCN1C(=O)c1ccccc1-c1ccccc1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)c(Br)cc2[nH]1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(C)c(Br)cc3[nH]2)c(s1)-c1ccccc1C
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(C)c(Br)cc3[nH]2)c(s1)-c1cccc(Cl)c1Cl
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(C)c(Br)cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(C)c(Br)cc3[nH]2)c(s1)-c1cc(F)cc(F)c1
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(C)c(Br)cc2[nH]1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(C)c(Br)cc3[nH]2)c(s1)-c1ccc(F)cc1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(Br)cc(C)c2[nH]1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cccc(C)c2[nH]1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2[nH]1)C(F)(F)F
COc1cc2nc([nH]c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1ncccn1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(OC(F)(F)F)ccc2[nH]1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(F)c(Br)cc2[nH]1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2ccc(F)c(F)c2[nH]1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2[nH]1
C[C@]1(CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccccc1)c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F
Cc1ccccc1-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(s1)-c1ccc(F)cc1
Cc1cccc(c1)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(s1)-c1ccc(F)cc1
Cc1ccc(cc1)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(s1)-c1ccc(F)cc1
C[C@]1(CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccccc1F)c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1cccc(F)c1)c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccc(F)cc1)c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F
COc1cccc(c1)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(s1)-c1ccc(F)cc1
COc1ccc(cc1)-c1nc(C(=O)N2CCC[C@@]2(C)c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(s1)-c1ccc(F)cc1
C[C@]1(CCCN1C(=O)c1nc(sc1-c1ccc(F)cc1)-c1ccccc1F)c1nc2ccc(cc2[nH]1)C(F)(F)F
C[C@]1(CCCN1C(=O)c1cc(ccc1-n1nccn1)-c1cccc(c1)C#N)c1nc2cc(ccc2[nH]1)C(F)(F)F
COc1cccc(c1)-c1ccc(OC)c(F)c1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1
COc1ccc(cc1)-c1ccc(OC)c(F)c1C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1
COc1ccc(-c2ccccc2F)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2ccc(F)cc2)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2cccc(F)c2)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2cccc(C)c2)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2ccc(C)cc2)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2cccc(c2)C(F)(F)F)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1c(F)c(ccc1-c1ccc2OCOc2c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1
COc1ccc(-c2ccc(cc2)C(F)(F)F)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2ccc(OC(F)(F)F)cc2)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2cccc(c2)C#N)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2ccc(cc2)C#N)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc(-c2cccc(OC(F)(F)F)c2)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)cc(Br)cc3[nH]2)c(cn1)-c1ccccc1
COc1ccc2nc([nH]c2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(sc1-c1ccccc1)C1CC1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1ccc(Br)cc1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1cccc(C)c1
Cc1cccc2nc([nH]c12)[C@@H]1CC(=C)CN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(cn1)-c1sc(C)nc1C(=O)N1CC(=C)C[C@H]1c1nc2cccc(C)c2[nH]1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1cccc(Br)c1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2cccc(C)c2[nH]1)-n1cccn1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1cc(C)cc(C)c1
Cc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(cc1C)-n1nccn1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1ccc(Cl)cc1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cnc(C)nc1-c1cccc(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1ccc(F)c(Br)c1
COc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cccc(C)c2[nH]1)-n1nccn1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1cccc(c1)C(F)(F)F
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cccc(C)c3[nH]2)c(s1)-c1ccc(Cl)c(Cl)c1
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CC(=C)C[C@H]1c1nc2cccc(C)c2[nH]1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2cccc(C)c2[nH]1)-n1nccn1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1ccc(Br)cc1
COc1ccc(cn1)-c1sc(C)nc1C(=O)N1CC(=C)C[C@H]1c1nc2ccc(Cl)c(C)c2[nH]1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1ccc(Cl)cc1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1cccc(c1)C(F)(F)F
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CC(=C)C[C@H]1c1nc2ccc(Cl)c(C)c2[nH]1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1cccc(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1cccc(Br)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1cc(C)cc(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1ccc(F)c(Br)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(s1)-c1ccc(Cl)c(Cl)c1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2ccc(Cl)c(C)c2[nH]1)-n1nccn1
Cc1c(Cl)ccc2nc([nH]c12)[C@@H]1CC(=C)CN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1c(Cl)ccc2nc([nH]c12)[C@@H]1CC(=C)CN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-n1nccn1
Cc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c(cc1C)-n1nccn1
COc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2ccc(Cl)c(C)c2[nH]1)-n1nccn1
Cc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c1F)-n1nccn1
COc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3ccc(Cl)c(C)c3[nH]2)c1F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2ccc(Cl)c(C)c2[nH]1)-n1cccn1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2ccc(Cl)c(C)c2[nH]1)-n1cccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(C)ccc1-n1cccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)ccc1-n1cccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-c1cccc(C)c1
COc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2ccc(OC)cc2[nH]1)-n1nccn1
COc1ccc2nc([nH]c2c1)[C@@H]1CC(=C)CN1C(=O)c1c(F)c(C)ccc1-n1nccn1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(c(Cl)cc3[nH]2)C(F)(F)F)c(s1)-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(C)sc1-c1cccc(C)c1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(sc1-c1ccc(C)c(C)c1)N(C)C
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
COc1ccc(cc1)-c1sc(C)nc1C(=O)N1CC(=C)CC1(C)c1nc2cc(OC)ccc2[nH]1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(C)cc1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1ccccc1-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-c1ccc(C)cc1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1ccccc1-c1ccccc1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1ccccc1-c1ccc(F)c(C)c1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(sc1-c1cccc(Cl)c1)N(C)C
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1nc(C)sc1-c1ccccc1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1ccccc1-n1nccn1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CC(=C)CC1(C)c1nc2cc(OC)ccc2[nH]1)-n1nccn1
COc1ccc2[nH]c(nc2c1)C1(C)CC(=C)CN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cnc(C)nc1-c1ccccc1
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(F)ccc1-n1nccn1
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(Cl)ccc1-n1nccn1
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-n1nccn1
COc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3cc(ccc3[nH]2)C(C)(C)C)c1F)-n1nccn1
Cc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3cc(ccc3[nH]2)C(C)(C)C)c1F)-n1nccn1
Cc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(ccc3[nH]2)C(C)(C)C)c(cc1C)-n1nccn1
Cc1ccc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(ccc3[nH]2)C(C)(C)C)c(c1)-n1nccn1
Cc1cccc(c1C(=O)N1CC(=C)C[C@H]1c1nc2cc(ccc2[nH]1)C(C)(C)C)-n1nccn1
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cncnc1-c1cccc(C)c1
COc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(ccc3[nH]2)C(C)(C)C)c(cc1OC)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(ccc2[nH]1)C(C)(C)C)-n1cccn1
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-n1cccn1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(ccc2[nH]1)C(C)(C)C)-n1cccn1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(ccc2[nH]1)C(C)(C)C)-n1nccn1
Fc1cccc(c1C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1nccn1
Fc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1nccn1
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)[C@@H]1CC(=C)CN1C(=O)c1cc(Cl)ccc1-n1nccn1
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-n1nccn1
COc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c1F)-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(F)ccc1-n1nccn1
Cc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c1F)-n1nccn1
Cc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(cc1C)-n1nccn1
Cc1ccc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(c1)-n1nccn1
Cc1cccc(c1C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1nccn1
FC(F)(F)c1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1nccn1
FC(F)(F)Oc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1nccn1
COc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(cc1OC)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1cccn1
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-n1cccn1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1cccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1c(F)cccc1-n1nccn1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@@H]1CC(=C)CN1C(=O)c1c(F)cccc1-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@@H]1CC(=C)CN1C(=O)c1cc(F)ccc1-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@@H]1CC(=C)CN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-n1nccn1
COc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3cc(C)c(C)cc3[nH]2)c1F)-n1nccn1
Cc1ccc(c(C(=O)N2CC(=C)C[C@H]2c2nc3cc(C)c(C)cc3[nH]2)c1F)-n1nccn1
Cc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(C)c(C)cc3[nH]2)c(cc1C)-n1nccn1
COc1ccc(cc1)-c1sc(C)nc1C(=O)N1CC(=C)C[C@H]1c1nc2cc(OC)ccc2[nH]1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-c1nc(C)no1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccccc1-c1csc(C)n1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(Br)cc1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1Cl
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(F)c(Br)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(sc1-c1ccc(C)c(F)c1)C1CC1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(sc1-c1cccc(C)c1)C1CC1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(sc1-c1ccc(C)c(C)c1)N(C)C
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(sc1-c1cccc(Br)c1)C1CC1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(sc1-c1cccc(F)c1)N1CCCC1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccccc1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1cccc(c1)C(F)(F)F
COc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)C[C@H]1c1nc2cc(OC)ccc2[nH]1)C1CC1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ncsc1-c1cccc(Cl)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1cccc(F)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccccc1Cl
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(sc1-c1ccc(C)cc1)C1CC1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(C)sc1-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1cc(F)cc(F)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccsc1-c1cccc(C)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1ccsc1-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nccnc1-c1ccc(C)cc1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)cccc3[nH]2)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccccc1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3ccccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)cccc3[nH]2)c(s1)-c1cccc(Cl)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1cccc(Cl)c1
COc1ccc2nc([nH]c2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)c(C)ccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
COc1ccc(OC)c2[nH]c(nc12)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
CSc1cccc2[nH]c(nc12)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(Cl)cc1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(Br)cccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(Cl)cccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)cccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(Cl)c(C)cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(C)c(C)cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(ccc3[nH]2)C(C)(C)C)c(s1)-c1ccc(C)c(C)c1
Cc1nc(C(=O)N2CC(=C)C[C@H]2c2nc3c(C)cc(C)cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
CSc1cccc2nc([nH]c12)[C@@H]1CC(=C)CN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nccnc1-c1cccc(C)c1
CSc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(C)c(C)cc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2c(C)cc(C)cc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2c(C)c(C)ccc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2c(Br)cccc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(C)cc2[nH]1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(ccc2[nH]1)C(C)(C)C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)-n1nccn1
COc1ccc(OC)c2[nH]c(nc12)[C@@H]1CC(=C)CN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cccc(Cl)c2[nH]1)-n1nccn1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1cccc(C)c1
COc1ccc2[nH]c(nc2c1)C1CC(=C)CN1C(=O)c1cc(C)sc1-c1ccc(C)c(C)c1
CSc1cccc2nc([nH]c12)C1CC(=C)CN1C(=O)c1cc(C)sc1-c1ccc(C)c(C)c1
CSc1ccc2[nH]c(nc2c1)C1CC(=C)CN1C(=O)c1cc(C)sc1-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3c(C)c(Cl)ccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3cc(C)c(C)cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3c(C)cc(C)cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3c(C)c(C)ccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3c(Br)cccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3c(C)cccc3[nH]2)c(s1)-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3cc(Cl)c(C)cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3cc(ccc3[nH]2)C(C)(C)C)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3cc(Cl)c(cc3[nH]2)C(F)(F)F)c(s1)-c1ccc(C)c(C)c1
COc1ccc(OC)c2[nH]c(nc12)C1CC(=C)CN1C(=O)c1cc(C)sc1-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3cccc(Cl)c3[nH]2)c(s1)-c1ccc(C)c(C)c1
Cc1cc(C(=O)N2CC(=C)CC2c2nc3cc4ccccc4cc3[nH]2)c(s1)-c1ccc(C)c(C)c1
COc1ccc2[nH]c(nc2c1)C1CC(=C)CN1C(=O)c1nc(sc1-c1cccc(C)c1)C1CC1
CSc1cccc2nc([nH]c12)C1CC(=C)CN1C(=O)c1nc(sc1-c1cccc(C)c1)C1CC1
CSc1ccc2[nH]c(nc2c1)C1CC(=C)CN1C(=O)c1nc(sc1-c1cccc(C)c1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2c(C)c(Cl)ccc2[nH]1)C1CC1
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(C)c(C)c1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2cc(C)c(C)cc2[nH]1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2c(C)cc(C)cc2[nH]1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2c(C)c(C)ccc2[nH]1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2c(Br)cccc2[nH]1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2c(C)cccc2[nH]1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2cc(Cl)c(C)cc2[nH]1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2cc(ccc2[nH]1)C(C)(C)C)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2cc(Cl)c(cc2[nH]1)C(F)(F)F)C1CC1
COc1ccc(OC)c2[nH]c(nc12)C1CC(=C)CN1C(=O)c1nc(sc1-c1cccc(C)c1)C1CC1
Cc1cccc(c1)-c1sc(nc1C(=O)N1CC(=C)CC1c1nc2cccc(Cl)c2[nH]1)C1CC1
Cc1ccc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(C)c(C)cc3[nH]2)c(c1)-n1nccn1
Cc1cc2nc([nH]c2cc1C)[C@@H]1CC(=C)CN1C(=O)c1c(C)cccc1-n1nccn1
COc1cc(C(=O)N2CC(=C)C[C@H]2c2nc3cc(C)c(C)cc3[nH]2)c(cc1OC)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(C)c(C)cc2[nH]1)-n1cccn1
Cc1ccc(c(n1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(C)c(C)cc2[nH]1)-n1nccn1
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc(OC)ccc1-n1nccn1)c1nc2ccc(Cl)c(C)c2n1C
Cc1ccc(c(c1)C(=O)N1CC(=C)C[C@H]1c1nc2cc(C)c(C)cc2n1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2n1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(Br)cc(C)c2n1C)-n1nccn1 |r|
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)cccc3n2C)c(s1)-c1cccc(Cl)c1
CCn1c(nc2c(C)cccc12)[C@]1(C)CCCN1C(=O)c1nc(C)sc1-c1cccc(Cl)c1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3n2C)c(s1)-c1ccccc1
CCn1c(nc2c(C)c(Cl)ccc12)[C@]1(C)CCCN1C(=O)c1nc(C)sc1-c1ccccc1
COc1cc2nc(n(C)c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCn1c(nc2cc(OC)c(OC)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nc3cc(C)c(C)cc3n2C)c(c1)-n1nccn1
CCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1cc2nc(n(C)c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCn1c(nc2cc(OC)c(OC)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
Cc1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1C
CCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1ccc(F)cc1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nc3cc(C)c(C)cc3n2C)c(cc1C)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2n1C)-n1nccn1
Cc1c(Cl)ccc2n(C)c(nc12)[C@]1(C)CCCN1C(=O)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(c(Cl)cc2n1C)C(F)(F)F)-n1nccn1
CCn1c(nc2c(C)c(Cl)ccc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1c(Cl)ccc2n(C)c(nc12)[C@]1(C)CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2n1C)-n1nccn1
COc1cc2nc(n(C)c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1C
Cc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CC1CC1
CCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1cccc(C)c1
Cc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CCF
COCCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1cccc(C)c1
Cc1ccc(-c2cccc(F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1C
CCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1cccc(F)c1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(F)c(Br)cc2n1C)-n1nccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3n2C)c(s1)-c1cccc(Cl)c1
Cc1ccc(-c2cccc(F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CC1CC1
Cc1ccc(-c2cccc(F)c2)c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CCF
COCCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1cccc(F)c1
Cc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1C
CCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1ccc(C)cc1
Cc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CC1CC1
Cc1ccc(cc1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CCF
COCCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1ccc(C)cc1
COc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1C
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1C)-c1ccccc1F
CCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1cccc(OC)c1
CCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1ccccc1F
COCCn1c(nc2cc(OC)c(OC)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cc2nc(n(CC3CC3)c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cc2nc(n(CCF)c2cc1OC)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CC1CC1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CC1CC1)-c1ccccc1F
COc1cccc(c1)-c1ccc(C)cc1C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CCF
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc2cc(C)c(C)cc2n1CCF)-c1ccccc1F
COCCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1cccc(OC)c1
COCCn1c(nc2cc(C)c(C)cc12)[C@]1(C)CCCN1C(=O)c1cc(C)ccc1-c1ccccc1F
CCOc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1Br
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(OCc2ccccc2)ccn1
CC(C)Oc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cnccc2-n2nccn2)c1
CC(C)Oc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2ncnn2)c1
CCOc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2ncnn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cccc(F)c2-n2nccn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2C2CC2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2C(F)(F)F)c1
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1cc(OC)ccn1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(OC)nc2-c2ccccc2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2c(F)cccc2-n2nccn2)c1
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2cc(OC(C)C)ccn2)c(n1)-n1nccn1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-n2nccn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(OC)cc2-n2nccn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(OC)nc2C2CC2)c1
CC(C)Oc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccc(F)cc2-n2nccn2)c1
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2cc(OC(C)C)ccn2)c(c1)-n1nccn1
CC(C)Oc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2cc(F)ccc2-n2nccn2)c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(OCC(F)(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1cc(OCC(F)(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ncccc1-n1nccn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-n1nccn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-n1nccn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1nc(C)no1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1noc(C)n1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(OC2CC2)ccn1
CC(C)COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1
CCCOc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1
CC(C)Oc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-c2ncccn2)c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1ncccn1)Oc1cc(OCC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ncccc1-c1ncccn1)Oc1cc(OCC(F)F)ccn1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C
COc1cc(OC)nc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C=O
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C(C)=O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(OC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(OCF)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1cc(OC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)Oc1cc(OC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Oc1cc(OC(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1cc(OC(F)F)ccn1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-c2ncccn2)c1
COc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-n2nccn2)c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1cc(OCC(F)F)ccn1
CC(C)Oc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-n2nccn2)c1
CCOc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-n2nccn2)c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1cc(OCC(F)(F)F)ccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1cc(OCC(F)F)ccn1
CCOc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccsc2-c2ncccn2)c1
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1cc(OCC(F)(F)F)ccn1
CCOC(=O)c1c(C)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
COC(=O)c1c(C)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
COC(=O)c1c(SC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-c1ncccn1
COC(=O)c1c(SC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cc(F)ccc1-c1ncccn1
COC(=O)c1c(SC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(F)cc1-c1ncccn1
COC(=O)c1c(SC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccc(F)c1-c1ncccn1
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1N1CCC1
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1N1CCN(C)CC1
CCc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C(=O)OC
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C(C)C
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C1CC1
COC(=O)c1c(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C1CCC1
CCOC(=O)c1c(CC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3Br)sc2c1 |r|
COc1ccc(Br)nc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1cccnc1C(=O)N(C)[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3-n3nccn3)sc2c1 |r|
COc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2o1 |r|
CC(C)Oc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1ccc(C)nc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3-n3cccn3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3F)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3N3CCCCC3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3N3CCC3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3N3CCCC3)sc2c1 |r|
COC1CN(C1)c1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc2ccccc2n1 |r|
COc1ccc(nc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(F)(F)F |r|
CCOc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3OC(F)(F)F)sc2c1 |r|
FC(F)Oc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Clc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3-n3nccn3)sc2c1 |r|
FC(F)Oc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(Cl)cc2s1 |r|
FC(F)Oc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2o1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ncccc3-n3ccnn3)sc2c1 |r|
FC(F)Oc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(Cl)cc2o1 |r|
CCOc1ccc(C)nc1C(=O)NC1CCCC1Cc1ccc2ccccc2n1
COc1cccc(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2-n2nccn2)c1C(O)=O |r|
CC1(C)OC(=O)c2c1ccnc2O[C@@H]1CC[C@@H](CO)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
OC[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
COC(=O)c1c(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2-n2nccn2)cccc1C#N |r|
Cc1ccnc(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
OC[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(OCC(F)F)ccn1 |r|
Cc1c(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2-n2nccn2)nccc1C#N |r|
COc1ccnc(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1CO)Oc1nccc(C#N)c1OC |r|
COc1c(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2cccnc2OCC(F)(F)F)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2cccnc2OC(C)C)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2OC(F)F)nccc1C#N |r|
COc1c(O[C@@H]2CC[C@@H](CO)N(C2)C(=O)c2ccccc2OC(F)(F)F)nccc1C#N |r|
CC(C)(O)[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
Cc1c(O[C@@H]2CC[C@H](N(C2)C(=O)c2ccccc2-n2nccn2)C(C)(C)O)nccc1C#N |r|
C[C@@H]1CCC(CN1C(=O)c1ccccc1-n1nccn1)c1nc(Br)co1 |r|
COC(=O)C1CC1c1coc(n1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(co1)C1CC1
CCc1ccccc1-c1coc(n1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(co1)-c1cccc(F)n1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(co1)-c1cccc(C)c1
COc1ccc(C(=O)N2C[C@H](CC[C@@H]2C)Oc2cccc(c2)C(C)O)c(n1)-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(C#N)c(N)o1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(C#N)c(Br)o1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(C(=O)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c(Br)o1 |r|
COC(=O)c1nc(oc1Br)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(co1)C(C)(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(co1)-c1ccccc1 |r|
CCOC(=O)C(NC(=O)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1)C(C)=O |r|
Cc1oc(nc1C(C)(C)O)[C@@H]1CCCN(C1)C(=O)c1ccccc1C1(CC1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CCOCC1)C#N)c1nc(c(C)o1)C(C)(C)O
CCOc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccc2ccnn12)c1nc(c(C)o1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CCC(CN1C(=O)c1ccsc1-n1nccn1)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1nc(c(C)o1)C(C)(C)O
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)(F)F)c1nc(c(C)o1)C(C)(C)O
CC(C)Oc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O
COc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O
CC(C)c1sc(Cl)nc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O
COC(=O)c1ccccc1C(=O)N1CC(CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)c1nc(c(C)o1)C(C)(C)O
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O
COCCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cnsc1-n1nccn1)c1nc(c(C)o1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)sc1-n1nccn1)c1nc(C)c(o1)C(C)(C)O |r|
CC[C@](C)(O)c1nc(oc1C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
CC[C@](C)(O)c1nc(oc1C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cscc1-n1nccn1
CC[C@@](C)(O)c1nc(oc1C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cscc1-n1nccn1
CC[C@@](C)(O)c1nc(oc1C)C1CC[C@@H](C)N(C1)C(=O)c1ccsc1-n1nccn1 |r|
CCOC(=O)c1nc(oc1Cl)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
CCOC(=O)C(NC(=O)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1)C(=O)C(F)F |r|
CCOC(=O)C(NC(=O)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1)C(O)(O)C(F)(F)F |r|
CCOC(=O)c1oc(nc1C)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
COC(=O)C(NC(=O)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1)C(=O)c1ccccc1 |r|
COC(=O)c1nc(oc1-c1ccccc1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CCC(CN1C(=O)c1ccccc1-n1nccn1)c1nc(CF)c(o1)-c1ccccc1 |r|
COCc1nc(oc1-c1ccccc1)C1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(c(o1)-c1ccccc1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(C(O)=O)c(o1)-c1ccccc1 |r|
CC(O)c1nc(oc1-c1ccccc1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CCC(CN1C(=O)c1ccccc1-n1nccn1)c1nc(COS(C)(=O)=O)c(o1)-c1ccccc1 |r|
COC(=O)Cc1nc(oc1-c1ccccc1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(CC(C)(C)O)c(o1)-c1ccccc1 |r|
COC(C)(C)Cc1nc(oc1-c1ccccc1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(CCF)c(o1)-c1ccccc1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C(=O)NCC(C)=O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)C(=O)NCC(=O)C(C)(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1ncc(o1)-c1ccccc1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1ncc(o1)C1CCC1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1ncc(o1)C1CC1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)C(=O)NC(C(O)c1ccccc1)c1ccccc1 |r|
CCn1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
CC(C)n1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(CC2CC2)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(c1)C1CCCC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(CC(F)(F)F)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(CC(F)F)c1 |r|
COC(=O)C(C)(C)n1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(c1)C1CCC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(c1)C1CCOC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(CC(C)(C)O)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cnn(c1)C1CC1 |r|
CC(C)n1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccsc1-n1nccn1 |r|
CC(C)n1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccsc1-c1ncccn1 |r|
CC(C)n1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cscc1-n1nccn1 |r|
CC(C)n1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(F)cc1-n1nccn1 |r|
CC(C)n1cc(cn1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1ncnn1 |r|
CCN(CCc1cc(ccn1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1cccnc1OC(C)C
CCOc1ncccc1C(=O)N(CC)CCc1cccc(n1)C(C)(C)O
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)(F)F
CCOc1ccccc1C(=O)N(CC)CCc1cccc(n1)C(C)(C)O
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1cccn1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccc(F)cc1-n1nccn1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1cccnc1-c1ccccc1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1
CCCc1ccccc1C(=O)N(CC)CCc1cccc(n1)C(C)(C)O
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1CC(F)(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccc(OC)nc1C1CC1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1CC(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1cccnc1-n1cccn1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1C1CCC1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ncccc1-c1ccccc1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1N1CCCC1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1ncnn1
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1(F)F
CCN(CCc1cccc(n1)C(C)(C)O)C(=O)c1ccccc1-c1ncccn1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1ccnc(c1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1cncc(Br)c1)C(=O)c1ccccc1-n1nccn1
CCN(CCc1cncc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1ccnc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1ncc(Br)cn1)C(=O)c1ccccc1-n1nccn1
CCN(CCc1nccc(n1)C(=O)OC)C(=O)c1ccccc1-n1nccn1
CCN(CCc1nccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1cnc(Br)cn1)C(=O)c1ccccc1-n1nccn1
CCN(CCc1cc(C)c(Br)cn1)C(=O)c1ccccc1-n1nccn1
CCN(CCc1ccc(C)c(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1cccnc1-n1cccn1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1OC(F)(F)F
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1N1CCCC1
CCCc1ccccc1C(=O)N(CC)CCc1ccc(cn1)C(C)(C)O
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1-n1cccn1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1CC(F)(F)F
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1-n1ncnn1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1cccnc1OCC(F)(F)F
CCOc1ccccc1C(=O)N(CC)CCc1ccc(cn1)C(C)(C)O
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1cccnc1-c1ccccc1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccc(OC)nc1C1CC1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1C1CC1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccc(F)cc1-n1nccn1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1C1CCC1
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1ccccc1C1CC1(F)F
CCN(CCc1ccc(cn1)C(C)(C)O)C(=O)c1cccnc1OCC(F)F
Cc1nc(C(=O)N2CCCCC2CNc2ncc(cn2)C(F)(F)F)c(s1)-c1ccc(F)cc1
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
Cc1nc(C(=O)N2CCCC(C)(C)C2CNc2ncc(cn2)C(F)(F)F)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CC(F)CCC2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CC(F)CCC2CNC(=O)c2cccc3occc23)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CC(F)CCC2CNc2ccc(cn2)C(F)(F)F)c(s1)-c1ccccc1
O[C@@H]1C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
F[C@H]1C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
O=C(NC[C@@H]1CC(=O)CN1C(=O)c1ccccc1-c1ccccc1)c1cccc2cccnc12 |r|
FC1(F)C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNC(=O)c1cccc2cccnc12)C(=O)c1nc(C)sc1-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNC(=O)c1cccc2cccnc12)C(=O)c1sc(C)nc1-c1ccccc1 |r|
COc1c(F)cccc1C(=O)N1CCC[C@@H](C)[C@H]1CNC(=O)c1cccc2cccnc12 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1nc(C)sc1-c1ccccc1 |r|
Cc1nc(C(=O)N2CCC[C@H]([C@H]2CNc2nc3ccccc3o2)C(F)(F)F)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2CCC[C@H]([C@H]2CNc2ccc(cn2)C(F)(F)F)C(F)(F)F)c(s1)-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Br)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CCc1cnc(NC[C@@H]2[C@H](C)CCCN2C(=O)c2nc(C)sc2-c2ccc(F)cc2)nc1 |r|
COc1ccnc(NC[C@@H]2[C@H](C)CCCN2C(=O)c2nc(C)sc2-c2ccc(F)cc2)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccnc(Cl)n1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nccc(Cl)n1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1cc(ccn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncccc1C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1cccc(C)n1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CC1CCCC(CNc2nc3ccccc3o2)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
CC1CCCC(CNc2ccc(cn2)C(F)(F)F)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
CC1CCCC(CNc2ncc(cn2)C(F)(F)F)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
CC1CCCC(CNc2ncc(Cl)cn2)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
CC1CCCC(CNC(=O)c2cccc3cccnc23)N1C(=O)c1sc(C)nc1-c1ccccc1
CC1CCCC(CCOc2ccccc2)N1C(=O)c1sc(C)nc1-c1ccccc1
CC1CCCC(CCOc2ccccc2)N1C(=O)c1ccccc1-c1ccccc1
OC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
Cc1nc(c(s1)C(=O)N1CC(O)CCC1CNC(=O)c1cccc2cccnc12)-c1ccccc1
Cc1nc(c(s1)C(=O)N1CC(F)(F)CCC1CNC(=O)c1cccc2cccnc12)-c1ccccc1
Cc1nc(c(s1)C(=O)N1CC(F)CCC1CNC(=O)c1cccc2cccnc12)-c1ccccc1
FC1(F)CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
F[C@H]1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
F[C@@H]1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
NC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
O=C(NCC1CCC(CN1C(=O)c1ccccc1-c1ccccc1)NCc1ccccc1)c1cccc2cccnc12
CN(C)C1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
OCCNC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
CC(=O)NC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
CNC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1sc(C)nc1-c1ccccc1
CCNC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1sc(C)nc1-c1ccccc1
Cc1nc(c(s1)C(=O)N1CC(CCC1CNC(=O)c1cccc2cccnc12)NCCO)-c1ccccc1
CC(C)NC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
CNC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1
COC1CCC(CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1nc(C)sc1-c1cccc(F)c1
Cc1nc(C(=O)N2CC(O)CCC2CNC(=O)c2cccc3cccnc23)c(s1)-c1cccc(F)c1
Cc1nc(C(=O)N2CC(F)(F)CCC2CNC(=O)c2cccc3cccnc23)c(s1)-c1cccc(F)c1
Cc1nc(C(=O)N2CC(N)CCC2CNC(=O)c2cccc3cccnc23)c(s1)-c1cccc(F)c1
Cc1nc(C(=O)N2CC(CCC2CNC(=O)c2cccc3cccnc23)NCCO)c(s1)-c1cccc(F)c1
Cc1nc(C(=O)N2CC(N)CCC2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CC(F)(F)CCC2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccccc1
Cc1cc2c(cccc2o1)C(=O)NCC1CCC(F)(F)CN1C(=O)c1nc(C)sc1-c1ccc(F)cc1
CC1CCCC(CNC(=O)c2cccc3occc23)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
CC1CCCC(CNC(=O)c2cccc3cccnc23)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
COc1c(F)cccc1C(=O)NCC1CCCC(C)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
CC1CCCC(CNC(=O)c2cccc3oc(C)cc23)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1
C[C@@H]1CCCN([C@@H]1CNC(=O)c1cccc2occc12)C(=O)c1nc(C)sc1-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNC(=O)c1cccc2occc12)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
Cc1nc(c(s1)C(=O)N1C[C@@H]2CCCC[C@@H]2[C@H]1CNC(=O)c1cccc2cccnc12)-c1ccccc1 |r|
Cc1nc(c(s1)C(=O)N1C[C@H]2CCCC[C@@H]2[C@H]1CNC(=O)c1cccc2cccnc12)-c1ccccc1 |r|
O=C(NC[C@@H]1[C@H]2CCCC[C@H]2CN1C(=O)c1ccccc1-c1ccccc1)c1cccc2cccnc12 |r|
O=C(NC[C@@H]1[C@H]2CCCC[C@@H]2CN1C(=O)c1ccccc1-c1ccccc1)c1cccc2cccnc12 |r|
Cc1nc(C(=O)N2C[C@@H]3CCCC[C@@H]3[C@H]2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2C[C@H]3CCCC[C@@H]3[C@H]2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2C[C@@H]3CCCC[C@@H]3[C@H]2CNC(=O)c2cccc3occc23)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2C[C@H]3CCCC[C@@H]3[C@H]2CNC(=O)c2cccc3occc23)c(s1)-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2s1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1cccc2cccnc12)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CC[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CC[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CC[C@@H]1CCCN([C@@H]1CNc1ncc(CC)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1COc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1COc1nc2ccccc2o1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CCc1cnc(OC[C@@H]2[C@H](C)CCCN2C(=O)c2nc(C)sc2-c2ccc(F)cc2)nc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(C)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CC(C)[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1cccc(n1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
COc1cnc(NC[C@@H]2[C@H](C)CCCN2C(=O)c2nc(C)sc2-c2ccc(F)cc2)nc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CO[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CO[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CO[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2s1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
Cc1nc(C(=O)N2C[C@H]3CCC[C@H]3C2CNc2ncc(cn2)C(F)(F)F)c(s1)-c1ccc(F)cc1 |r|
Cc1nc(C(=O)N2C[C@H]3CCC[C@H]3C2CNc2nc3ccccc3o2)c(s1)-c1ccc(F)cc1 |r|
Cc1nc(C(=O)N2C[C@H]3CCC[C@H]3C2COc2ccc(cn2)C(F)(F)F)c(s1)-c1ccc(F)cc1 |r|
Cc1nc(C(=O)N2C[C@H]3CCC[C@H]3C2COc2nc3ccccc3o2)c(s1)-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cccnc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccc(C)nc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccncc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cncnc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccnn1C |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnc(nc1)N1CCN(C)CC1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccc(nc1)N1CCN(C)CC1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnn(CCN2CCOCC2)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ncco1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ccnn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ccnc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1cncn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1ccccc1Oc1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1ccnn1-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nccnc1Cl)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1ccccc1OC(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1cncc(Cl)n1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNC(=O)c1cccc2oc(C)cc12)C(=O)c1nc(C)sc1-c1ccccc1 |r|
C[C@@H]1CCCN([C@@H]1CNC(=O)c1cccc2cccnc12)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
O[C@H]1C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
CO[C@H]1C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
F[C@@H]1C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
CO[C@@H]1C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
Cc1nc(c(s1)C(=O)N1CC[C@H](O)[C@H]1CNC(=O)c1cccc2cccnc12)-c1ccccc1 |r|
CC(=O)O[C@H]1C[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
Cc1nc(c(s1)C(=O)N1CCC(=O)[C@H]1CNC(=O)c1cccc2cccnc12)-c1ccccc1 |r|
Cc1nc(c(s1)C(=O)N1CCC(F)(F)[C@H]1CNC(=O)c1cccc2cccnc12)-c1ccccc1 |r|
Cc1nc(c(s1)C(=O)N1CC[C@@H](O)C[C@H]1CNC(=O)c1cccc2cccnc12)-c1ccccc1 |r|
Cc1nc(c(s1)C(=O)N1CCC(F)(F)C[C@H]1CNC(=O)c1cccc2cccnc12)-c1ccccc1 |r|
C[C@H]1CCCN([C@@H]1CNC(=O)c1cccc2cccnc12)C(=O)c1nc(C)sc1-c1ccccc1 |r|
Cc1nc(C(=O)N2CCC[C@H]([C@H]2CNC(=O)c2cccc3cccnc23)C(F)(F)F)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2CCC[C@H]([C@H]2CNC(=O)c2cccc3occc23)C(F)(F)F)c(s1)-c1ccccc1 |r|
O=C(NCC1C2CCC(CC2)N1C(=O)c1ccccc1-c1ccccc1)c1cccc2cccnc12 |TLB:3:4:9.10:6.7,THB:12:11:9.10:6.7,(1.69,3.81,;1.29,2.32,;-.2,1.92,;-1.29,3.01,;-2.77,2.61,;-4.04,3.34,;-4.04,5.05,;-4.91,3.9,;-4.91,1.9,;-6.48,1.4,;-5.68,2.61,;-3.58,1.3,;-3.18,-.19,;-1.69,-.59,;-4.27,-1.28,;-5.75,-.88,;-6.84,-1.97,;-6.44,-3.45,;-4.96,-3.85,;-3.87,-2.76,;-2.38,-3.16,;-1.98,-4.65,;-.49,-5.05,;.59,-3.96,;.2,-2.47,;-1.29,-2.07,;2.38,1.23,;1.98,-.25,;3.07,-1.34,;4.56,-.94,;4.96,.54,;6.44,.94,;6.84,2.43,;5.75,3.52,;4.27,3.12,;3.87,1.63,)|
Cc1nc(C(=O)N2C3CCC(CC3)C2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccccc1 |TLB:14:13:12.11:9.8,THB:4:6:12.11:9.8,(-7.23,-3.52,;-5.9,-2.75,;-5.42,-1.29,;-3.88,-1.29,;-2.79,-.2,;-1.3,-.6,;-3.19,1.29,;-4.52,1.89,;-4.52,3.89,;-3.65,5.04,;-3.65,3.32,;-5.29,2.6,;-6.09,1.39,;-2.39,2.6,;-.9,3,;.19,1.91,;1.68,2.31,;2.08,3.8,;2.77,1.22,;2.37,-.26,;3.46,-1.35,;4.94,-.96,;5.34,.53,;6.83,.93,;7.23,2.42,;6.14,3.51,;4.65,3.11,;4.25,1.62,;-3.4,-2.75,;-4.65,-3.66,;-1.92,-3.15,;-1.52,-4.64,;-.03,-5.04,;1.06,-3.95,;.66,-2.46,;-.83,-2.06,)|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cn[nH]c1 |r|
COc1ncc(cn1)-c1ccc(C)cc1C(=O)N1CCC[C@@H](C)[C@H]1CNc1ccc(cn1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cncc(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnccc1C |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccc(Cl)cc2o1)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccc(Cl)cc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ncnc1C |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1cnc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccn(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1nccn1C |r|
COc1ccnc(n1)-c1ccc(C)cc1C(=O)N1CCC[C@@H](C)[C@H]1CNc1ccc(cn1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1nn[nH]n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1nccs1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cncs1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-n1cnc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-c1ccnc(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-c1ccc(C)nc1 |r|
C[C@H]1CCCN([C@H]1CNc1nc2ccccc2o1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCCN([C@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)cn1)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-c1ccnn1C |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1cc(C)ccc1-n1cnc(n1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1cc(C)ccc1-c1ccnc(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)cn1)C(=O)c1cc(C)ccc1-n1cnc(n1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1cnc(n1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)cn1)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1cc(C)ccc1-c1ccnn1C |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-n1cnc(n1)C(F)(F)F |r|
C[C@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CC2CCCC2C1CNc1ccc(cn1)C(F)(F)F)-n1nccn1
Cc1ccc(-c2cnn(C)c2)c(c1)C(=O)N1CC2CCCC2C1CNc1ccc(cn1)C(F)(F)F
COc1c(F)cccc1C(=O)N1CCC[C@@H](C)[C@H]1CNc1ccc(cn1)C(F)(F)F |r|
Cc1nc(C(=O)N2CCCC3CN(CC23)c2nc3ccc(Cl)cc3o2)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CCCC3CN(CC23)c2ccc(cn2)C(F)(F)F)c(s1)-c1ccc(F)cc1
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1cccc(C)n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
COc1cccc(NC[C@@H]2[C@H](C)CCCN2C(=O)c2cc(C)ccc2-n2nccn2)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cc1F)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1cccc(C)n1)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncccc1C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncccc1C#N)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cc1F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncccc1C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncccc1C#N)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
COc1cccnc1NC[C@@H]1[C@H](C)CCCN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncccc1C)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncccc1C)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nnc(s1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1cc(C)cn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(F)c1 |r|
CCn1cc(cn1)-c1ccc(C)cc1C(=O)N1CCC[C@@H](C)[C@H]1CNc1ccc(cn1)C(F)(F)F |r|
CC(C)n1cc(cn1)-c1ccc(C)cc1C(=O)N1CCC[C@@H](C)[C@H]1CNc1ccc(cn1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1COc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-n1ccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccc(C)cn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(C)ccc1-n1ccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc2cc(Br)ccc2n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc(cs1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
COc1ccc(NC[C@@H]2[C@H](C)CCCN2C(=O)c2cc(C)ccc2-n2nccn2)nc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(F)ccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C#N)C(=O)c1cc(C)ccc1-n1ccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nnc(s1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1cc(C)ccc1-n1ccc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C#N)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nnc(s1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C1CC1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C1(CC1)C#N)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(F)ccc2o1)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)cn1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C#N)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)nn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cc1F)C#N)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nnc(s1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C#N)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)nn1)C(=O)c1cc(C)ccc1-n1cccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1cc(C)ccc1-n1cccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C#N)C(=O)c1cc(C)ccc1-n1cccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1cccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(C)ccc1-c1ccc(cn1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(C)ccc1-c1ccc(F)cn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nccc(n1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1cccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1cccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1nc(C)ccc1-n1cccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1nc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(F)cc1F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(F)cn1)C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cc1F)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(F)cc1F)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nnc(s1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cc1F)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C#N)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C#N)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nnc(s1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cc1F)C#N)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CN(C)c1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(C)cn1)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cccnn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cccnn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1nc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cc(Cl)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(Cl)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(F)ccc2o1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(F)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CCC(F)(F)C[C@H]1CNc1ccc(Cl)cn1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CCC(F)(F)C[C@H]1CNc1ncc(cn1)C(F)(F)F)-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc2ccc(C)cc2n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc2ccccc2n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2ccccc2o1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1nc2cc(Cl)ccc2o1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc2cc(C)ccc2n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1nc(C)ccc1-c1cccnc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1cccnc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1nc(C)ccc1-c1cccnc1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1nccc2ccccc12 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cc(F)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(F)ccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cccc(F)c1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cccc(F)c1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cccc(F)c1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cccc(F)c1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1c(F)cccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1c(F)cccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1c(F)cccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(F)c(F)cc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)c(F)cc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cc(F)c(F)cc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cc(F)c(F)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cc(F)c(F)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)c(F)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(F)c(F)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1ccc(F)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1ccc(F)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1cccc(F)c1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cccc(F)c1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cccc(F)c1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cccc(F)c1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1c(F)cccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1c(F)cccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1c(F)cccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(Cl)cn1)C(=O)c1c(F)cccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cccc(C)c1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cccc(C)c1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cccc(C)c1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1ccc(C)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1ccc(C)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1ccc(C)cc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cccc(C)c1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cccc(C)c1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1c(C)cccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC(F)(F)CC1CNc1ncc(cn1)C(F)(F)F
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1ccccc1-n1nccn1 |r|
C[C@H]1CCCN([C@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1cnn(C)c1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1ccccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1ccccc1-c1ncccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1c(F)c(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1c(F)c(C)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(ccc1-n1nccn1)C#N |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(ccc1-c1ncccn1)C#N |r|
C[C@@H]1CCCN([C@@H]1CNc1ccc(cn1)C(F)(F)F)C(=O)c1c(F)c(F)ccc1-n1nccn1 |r|
C[C@@H]1CCCN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1c(F)c(F)ccc1-n1nccn1 |r|
COc1ccc(c(C(=O)N2CCC[C@@H](C)[C@H]2CNc2ccc(cn2)C(F)(F)F)c1F)-n1nccn1 |r|
COc1ccc(c(C(=O)N2CCC[C@@H](C)[C@H]2CNc2ncc(cn2)C(F)(F)F)c1F)-n1nccn1 |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2-n2nccn2)nc1C(C)(C)O
CCOc1ncccc1C(=O)N1CCCC[C@@H]1Cc1nc(c(C)o1)C(C)(C)O
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2C2CC2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccc(F)cc2-n2nccn2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2cccnc2OCC(F)(F)F)nc1C(C)(C)O |r|
CC(C)Oc1ncccc1C(=O)N1CCCC[C@@H]1Cc1nc(c(C)o1)C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2N2CCCC2)nc1C(C)(C)O |r|
CCOc1ccccc1C(=O)N1CCCC[C@@H]1Cc1nc(c(C)o1)C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2OC(F)(F)F)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2-n2cccn2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2cccnc2CC(F)(F)F)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2CC(F)F)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2cccnc2-n2cccn2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2cccnc2-c2ccccc2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2OC(F)F)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2cccnc2OCC(F)F)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2OCC(F)(F)F)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2CC(F)(F)F)nc1C(C)(C)O |r|
COc1ccc(C(=O)N2CCCC[C@@H]2Cc2nc(c(C)o2)C(C)(C)O)c(n1)C1CC1 |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ncccc2-n2nccn2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2nccnc2-c2ccccn2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2nccnc2C2CCCC2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2C2CCC2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ncccc2-c2ccccc2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2nccnc2-n2cccn2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2C2CC2(F)F)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2-n2ncnn2)nc1C(C)(C)O |r|
CCCc1ccccc1C(=O)N1CCCC[C@@H]1Cc1nc(c(C)o1)C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2cc(C)ccc2-n2nccn2)nc1C(C)(C)O |r|
Cc1oc(C[C@H]2CCCCN2C(=O)c2ccccc2-c2ncccn2)nc1C(C)(C)O
O=C(N1CC[C@@H]2CCN([C@@H]2C1)c1cc(ccn1)C#N)c1ccccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nccc(n1)C#N)c1ccccc1-n1nccn1
Cc1cc(nc(n1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1)C#N
COc1cc(OC)nc(n1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1ncccn1)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nc2ccccc2o1)c1ccccc1-n1nccn1
OC(=O)c1ccnc(c1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
COC(=O)c1cc(nc(c1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1)C#N
O=C(N1CC[C@H]2CCN([C@H]2C1)c1ccc(nn1)-n1ccnc1)c1ccccc1-n1nccn1
Cc1ccc(C)n1-c1ccc(nn1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
COC(=O)c1ccc(nn1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nncc2scnc12)c1ccccc1-n1nccn1
Clc1cc(C#N)c(cn1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
Cc1cc(ncc1N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1)C#N
CCN1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
CC(C)c1ccnc(N2CC[C@@H]3CCN(C[C@H]23)C(=O)c2ccccc2-n2nccn2)c1C#N
CN(C)c1cc(C)nc(n1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
Clc1c(ccnc1N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1)C#N
Oc1ccnc(c1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
CCc1ccnc(c1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
COCc1ccnc(c1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
Fc1cnc(cc1C#C)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cccc(c1)C#C)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1ncnc2[nH]ccc12)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nccc2ncccc12)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nccc2ccccc12)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1ccnc2ccccc12)c1ccccc1-n1nccn1
COC(=O)c1csc(n1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
COC(=O)c1nc(sc1C)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nccn2nccc12)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nccn2cccc12)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)C1=NC=CC2SCCC12)c1ccccc1-n1nccn1 |c:15,t:13|
O=C(N1CC[C@H]2CCN([C@H]2C1)C1=NC=CC2C=CC=CC12)c1ccccc1-n1nccn1 |c:15,18,20,t:13|
CCOC(=O)c1coc(n1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1ccc2ccccc2n1)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1nccc2C(=O)OCc12)c1ccccc1-n1nccn1
Cc1cnc(cn1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
Cc1ncc(nc1C)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
Cc1nccnc1N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cncc2ccccc12)c1ccccc1-n1nccn1
CC(C)(O)c1csc(n1)-c1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)n1nccn1
CC(C)(O)c1coc(n1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
CC(O)(c1cnc(cn1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1)C(F)(F)F
CC(C)(O)c1cccc(c1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
CC(C)(O)c1ccnc(c1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
CC(C)(O)c1cnc(nc1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
FC(F)COc1ncccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1ccccc1-n1ncnn1
FC(F)(F)Oc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
Cc1nccnc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1cccnc1-n1cccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1nccnc1-n1cccn1
CCOc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
CCCc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
FC(F)(F)Cc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
Fc1ccc(c(c1)C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)-n1nccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1cccnc1-c1ccccc1
CCOc1ncccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
FC(F)(F)COc1ncccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
FC(F)Cc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
FC(F)(F)OCc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
FC(F)COc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
FC(F)(F)Cc1ncccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1ccccc1C1CC1
COc1ccc(C(=O)N2CC[C@H]3CCN([C@H]3C2)c2cc(ccn2)C#N)c(n1)C1CC1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1ccccc1-n1cccn1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1ccccc1C1CCC1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1ccccc1N1CCCC1
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1nccnc1N1CCCC1
Cc1ncccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
CC(C)Oc1ncccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1cccnc1-n1nccn1
FC(F)Oc1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
FC1(F)CC1c1ccccc1C(=O)N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N
O=C(N1CC[C@H]2CCN([C@H]2C1)c1cc(ccn1)C#N)c1ccccc1-c1ccccc1
NC(=O)c1ccc(nc1)N1CC[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1
OC[C@H]1C[C@H]2CCN([C@H]2CN1C(=O)c1ccccc1-c1cc(ccn1)C#N)c1cc(ccn1)C#N
CCOC(=O)[C@H]1C[C@H]2CCN([C@H]2CN1C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N
OC[C@@H]1C[C@H]2CCN([C@H]2CN1C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N
C[C@H]1C[C@H]2CCN([C@H]2CN1C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccc(F)c1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(Cl)cc1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(F)cc1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(F)cc1-c1nc(C)no1
COC(=O)c1c(O)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cc(F)ccc1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1c(F)cccc1-c1noc(C)n1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cc(F)ccc1-c1noc(C)n1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(F)cc1-c1noc(C)n1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccc(F)c1-c1noc(C)n1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1c(F)cccc1-c1nc(C)no1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cc(F)ccc1-c1nc(C)no1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccc(C)c1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(OC)cc1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(OC)nc1-n1nccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccc(F)c1-c1nc(C)no1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccc(F)cc1-c1ncccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccc(F)c1-c1ncccn1
COC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1ncnn1
CCOC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
CCOC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccc(F)c1-n1nccn1
CCOc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1C(=O)OC
CCOC(=O)c1c(OCC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1ncnn1
CCOC(=O)c1c(OC)ccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1ncnn1
CCOc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2ncnn2)c1C(=O)OC
COC(=O)c1c(OC)cccc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
COC(=O)c1c(OC)cccc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccsc1-n1nccn1
COC(=O)c1c(OC)cccc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1ncnn1
COC(=O)c1c(OC)cccc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccsc1-c1ncccn1
COC(=O)c1c(OC)cccc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-c1ncccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1noc(n1)C1CC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1noc(n1)C(C)(C)C |r|
CCc1nc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
CC(C)c1nc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1noc(n1)[C@](C)(O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1noc(n1)[C@H](O)C(F)(F)F |r|
COC(C)(C)c1nc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1noc(n1)[C@@H](O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1noc(n1)[C@@](C)(O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)(F)F)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)c1noc(n1)C(C)(C)O |r|
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)F)c1noc(n1)C(C)(C)O |r|
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1noc(n1)C(C)(C)O |r|
COC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)c1noc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(no1)C(C)(C)C |r|
CC(C)c1noc(n1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(no1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(no1)C1CC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1nsc(n1)C(C)(C)O |r|
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)F)c1nsc(n1)C(C)(C)O |r|
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OCC(F)(F)F)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)(F)F)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1nsc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)c1nsc(n1)C(C)(C)O |r|
COC(C)(C)c1nc(ns1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1nccn1
CCOc1ncccc1C(=O)N1CC2CN(CC2C1)c1nc(c(C)o1)C(C)(C)O
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1cccnc1OCC(F)(F)F
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1OC(F)(F)F
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ncccc1-c1ccccc1
CCCc1ccccc1C(=O)N1CC2CN(CC2C1)c1nc(c(C)o1)C(C)(C)O
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1OCC(F)(F)F
CC(C)Oc1ncccc1C(=O)N1CC2CN(CC2C1)c1nc(c(C)o1)C(C)(C)O
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1cccnc1OCC(F)F
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1cccnc1CC(F)(F)F
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1C1CC1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1C1CCC1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1N1CCCC1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1cccn1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1-n1ncnn1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ncccc1-n1nccn1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1cccnc1-n1cccn1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1cccnc1-c1ccccc1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1nccnc1N1CCCC1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1nccnc1-n1cccn1
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1OC(F)F
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1CC(F)(F)F
Cc1oc(nc1C(C)(C)O)N1CC2CN(CC2C1)C(=O)c1ccccc1C1CC1(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ccccc1)n1ncc(n1)C(C)(C)O |r|
CCCc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O |r|
CCCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O |r|
CC(C)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CC1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OC(F)F)n1ncc(n1)C(C)(C)O |r|
COC(=O)c1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CC(F)(F)F)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-n1cc(C)cn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1SC(F)(F)F)n1ncc(n1)C(C)(C)O |r|
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)n1ncc(n1)C(C)(C)O
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OCC(F)(F)F)n1ncc(n1)C(C)(C)O
CC(C)Oc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OCC(F)F)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)(F)F)n1ncc(n1)C(C)(C)O
COC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)F)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1[C@@H]1CC1(F)F)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1[C@H]1CC1(F)F)n1ncc(n1)C(C)(C)O
COC(=O)c1cnn(n1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1ncc(n1)[C@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1ncc(n1)[C@@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1ncc(n1)-c1ccccc1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1ncc(Br)n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1noc(C)n1)n1ncc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1sccc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1nc(C)no1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1nc(C)no1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-c1noc(C)n1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1noc(C)n1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1nc(C)no1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-c1ccccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-n1cccn1)n1ncc(n1)C(C)(C)O |r|
COCCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)n2ncc(n2)C(C)(C)O)c(n1)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(C)c1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1noc(C)n1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-c1nc(C)no1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1N1CCCC1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(Oc2ccccc2)c1)n1ncc(n1)C(C)(C)O |r|
COc1cccc(c1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(C)cccc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)n2ncc(n2)C(C)(C)O)c(c1)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C)nc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
COCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc2ccnn12)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ncccc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-n1nccn1)n1ncc(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1C1CC1)n1ncc(n1)C(C)(C)O |r|
CC(O)c1cnn(n1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1cccnc1OCC(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1nc(C)c(n1)C(C)(C)O
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)n1nc(C)c(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)n1nc(C)c(n1)C(C)(C)O |r|
CCOc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)F)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)(F)F)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)n1nc(C)c(n1)C(C)(C)O |r|
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CC1)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1cccn1)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-c1ccccc1)n1nc(C)c(n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1nnc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1cc(cn1)C(C)(C)O
CCCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1cc(cn1)C(C)(C)O
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CC1)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OCC(F)F)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OCC(F)(F)F)n1cc(cn1)C(C)(C)O |r|
CC(C)Oc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1cc(cn1)C(C)(C)O |r|
CC(C)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)(F)F)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)F)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1[C@@H]1CC1(F)F)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1[C@H]1CC1(F)F)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CCC1)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1SC(F)(F)F)n1cc(cn1)C(C)(C)O |r|
CCOc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-n1cccn1)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-c1ccccc1)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1cccn1)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-n1cccn1)n1cc(cn1)C(C)(C)O |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)n2cc(cn2)C(C)(C)O)c(n1)C1CC1 |r|
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CC(F)F)n1cc(cn1)C(C)(C)O |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)n2cc(cn2)C(C)(C)O)c(n1)C1CCC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-n1nccn1)n1cc(cn1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1cc(cn1)[C@@H](O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1cc(cn1)[C@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1cc(cn1)C(C)(O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1cc(cn1)[C@@](C)(O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1cc(cn1)[C@](C)(O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1cc(c(C)n1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)n1ncc(c1C)C(C)(C)O |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1ncc(cn1)C(F)(F)F |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ncc(cn1)C(F)(F)F)-n1nccn1 |r|
CCc1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2cc(C)ccc2-n2nccn2)nc1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(Cl)cn1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F |r|
Cc1ccc(c(c1)C(=O)N[C@@H]1CCC[C@@H]1Nc1cnc(Cl)cn1)-n1nccn1 |r|
Fc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F)-n1nccn1 |r|
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2cccn2)nc1 |r|
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)nc1 |r|
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-c2ncccn2)nc1 |r|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1ncc(cn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)cn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)nc1 |r|
FC(F)(F)c1cnc(O[C@@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)cn1 |r|
FC(F)(F)c1ccnc(O[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)c1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Oc1cc(ccn1)C(F)(F)F |r|
FC(F)(F)c1ccnc(CC2CCCC2NC(=O)c2ccccc2-n2nccn2)c1
FC(F)(F)c1ccc(CC2CCCC2NC(=O)c2ccccc2-n2nccn2)nc1
Cc1ccc(c(c1)C(=O)NC1CCCC1Cc1ccc(cn1)C(F)(F)F)-n1nccn1
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1cccc(n1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2Br)cn1 |r|
CCOc1ccc(C)cc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
CCOc1ccc(C)nc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2cccn2)cn1 |r|
Fc1cccc(c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |r|
Fc1cccc(F)c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2ccnn2)cn1 |r|
Fc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |r|
COc1ccc(C)cc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-c2ncccn2)cn1 |r|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2c(Cl)cccc2-n2nccn2)cn1 |r|
Fc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1ccnn1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1ccnn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-n2cccn2)cn1 |r|
Cc1nnc(o1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
FC(F)(F)c1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |r|
Fc1cccc(c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1cccn1 |r|
Fc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1cccn1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1cccn1 |r|
COc1cccc(Br)c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
COc1cccc(c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1cccn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2N2CCCCC2)cn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2cc(Cl)ccc2-n2nccn2)cn1 |r|
Fc1cccc(C(=O)N[C@H]2CCC[C@@H]2Nc2cnc(cn2)C(F)(F)F)c1-n1nccn1 |r|
FC(F)(F)c1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1ccnn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2cc(Cl)ccc2-n2ccnn2)cn1 |r|
Fc1ccc(c(C(=O)N[C@H]2CCC[C@@H]2Nc2cnc(cn2)C(F)(F)F)c1F)-n1nccn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2cc(ccc2-n2nccn2)C2CC2)cn1 |r|
FC(F)(F)Oc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2cc(Cl)ccc2-n2cccn2)cn1 |r|
CCOc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
Fc1cc(F)c(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2C(F)(F)F)cn1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2C2CC2)cn1 |r|
Fc1ccc(F)c(c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F)-n1nccn1 |r|
FC(F)c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
Fc1cccc(C2CC2)c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(nc1)C(F)(F)F)-n1nccn1 |r|
COc1cccc(OC)c1C(=O)N(C1CCC1)[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F |r|
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2Cl)nc1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2Cl)nc1 |r|
COc1cccc(F)c1C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F |r|
Fc1cccc(F)c1C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F |r|
CN([C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)c1cnc(cn1)C(F)(F)F |r|
CN([C@H]1CCC[C@@H]1NC(=O)c1cc(F)ccc1-n1nccn1)c1cnc(cn1)C(F)(F)F |r|
CN([C@H]1CCC[C@@H]1NC(=O)c1c(F)cccc1-n1nccn1)c1cnc(cn1)C(F)(F)F |r|
Cc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-n1nccn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1ncccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
Cc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)C(F)(F)F |r|
Cc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-c1ncccn1)C(F)(F)F |r|
Cc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1cc(F)ccc1-c1ncccn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
CC1(CCCC1NC(=O)c1ccccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F
C[C@]1(CCC[C@H]1NC(=O)c1ccccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1cc(F)ccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1ncccc1-n1cccn1)Nc1cnc(cn1)C(F)(F)F |r|
CCOc1cccnc1C(=O)N[C@H]1CCC[C@]1(C)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1c(Cl)cccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1c(F)cccc1F)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1ncccc1C1CC1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1ncccc1OC(F)(F)F)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1ccccc1-c1ncccn1)Nc1cnc(cn1)C(F)(F)F |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1cc(Cl)ccc1-n1nccn1)Nc1cnc(cn1)C(F)(F)F |r|
CC1(CCCC1NC(=O)c1ccccc1-n1nccn1)Nc1ncc(cn1)C(F)(F)F
CC1(CCCC1NC(=O)c1ccccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F
CC1(CCCC1NC(=O)c1ccccc1-n1nccn1)Nc1ccc(OC(F)(F)F)cn1
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2cc(Cl)ccc2-n2nccn2)nc1 |r|
Fc1cccc(C(=O)N[C@H]2CCC[C@@H]2Nc2ccc(cn2)C(F)(F)F)c1-n1nccn1 |r|
Fc1cc(F)c(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F)-n1nccn1 |r|
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-n2nccn2)nc1 |r|
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-n2cccn2)nc1 |r|
Fc1cccc(c1C(=O)N[C@H]1CCC[C@@H]1Nc1ccc(cn1)C(F)(F)F)-n1nccn1 |r|
CC1(CCCC1NC(=O)c1ncccc1-n1nccn1)Nc1ncc(cc1F)C(F)(F)F
NC(=O)c1cccc([C@@H]2CCC[C@@H]2Nc2ncc(cc2F)C(F)(F)F)c1-n1nccn1
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)c(Cl)c1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)c(Br)c1 |r|
Cc1cc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)c(n1)C1CC1 |r|
CC(C)c1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)C(F)(F)F |r|
CCc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)C(F)(F)F |r|
O=C(N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C1CC1)c1ccccc1-n1nccn1 |r|
CC(C)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)cn1 |r|
CCc1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)cn1 |r|
FC(F)(F)Oc1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)nc1 |r|
FC(F)(F)Oc1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2cc(Cl)ccc2-n2nccn2)nc1 |r|
Brc1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)nc1 |r|
COc1cc(Br)cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1 |r|
FC(F)(F)c1ccnc(N[C@H]2CCC[C@@H]2NC(=O)c2ccccc2-n2nccn2)c1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-n2nccn2)c(Cl)c1 |r|
Fc1cc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-n1nccn1)C(F)(F)F |r|
Cc1cc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-n1nccn1)C(F)(F)F |r|
CCc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-n1nccn1)C(F)(F)F |r|
FC(F)(F)c1cnc(NC2CC(F)(F)CC2NC(=O)c2ccccc2-n2nccn2)cn1
FC(F)(F)c1cnc(NC2CC(F)(F)CC2NC(=O)c2ccccc2-n2nccn2)nc1
FC(F)(F)c1ccc(NC2CC(F)(F)CC2NC(=O)c2ccccc2-n2nccn2)nc1
FC(F)(F)Oc1ccc(N[C@H]2CC(F)(F)C[C@@H]2NC(=O)c2ccccc2-n2nccn2)nc1 |r|
Fc1cc(cnc1N[C@H]1CC(F)(F)C[C@@H]1NC(=O)c1ccccc1-n1nccn1)C(F)(F)F |r|
CCOc1cnc(nc1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
COc1cccc(F)c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F |r|
Cc1cc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-c1ncccn1)C(F)(F)F |r|
Fc1cc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-c1ncccn1)C(F)(F)F |r|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ncc(cc1F)C(F)(F)F |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1ncc(cc1F)C(F)(F)F |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1ncc(nc1C)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-n2nccn2)c(n1)C1CC1 |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-c2ncccn2)c(n1)C1CC1 |r|
C[C@@]1(CCC[C@@H]1NC(=O)c1ncccc1-c1ncccn1)Nc1cnc(cn1)C(F)(F)F |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@H]1CCC[C@]1(C)Nc1cnc(cn1)C(F)(F)F |r|
CC1(CCCC1NC(=O)c1ncccc1-c1ncccn1)Nc1ncc(cc1F)C(F)(F)F
Fc1cc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-c1ncccn1)C(F)(F)F |r|
FC(F)(F)c1cnc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-c2ncccn2)c(Cl)c1 |r|
CCc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-c1nc(C)no1)C(F)(F)F |r|
CCc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-c1ncccn1)C(F)(F)F |r|
CCc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-c1ncccn1)C(F)(F)F |r|
CC1(CCCC1NC(=O)c1ncccc1-c1ncccn1)Nc1ncc(cn1)C(F)(F)F
CC1(CCCC1NC(=O)c1ncccc1-n1nccn1)Nc1ncc(cn1)C(F)(F)F
CC1(CCCC1NC(=O)c1ncccc1-n1nccn1)Nc1ccc(cn1)C(F)(F)F
CC1(CCCC1NC(=O)c1ncccc1-c1ncccn1)Nc1ccc(cn1)C(F)(F)F
FC(F)Oc1ccc(N[C@H]2CC(F)(F)C[C@@H]2NC(=O)c2ccccc2-n2nccn2)nc1 |r|
CCc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1cc(F)ccc1-c1ncccn1)C(F)(F)F |r|
Cc1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ncccc1-c1ncccn1)C(F)(F)F |r|
Cc1nnc(o1)-c1ccccc1C(=O)N[C@H]1CCC[C@]1(C)Nc1cnc(cn1)C(F)(F)F |r|
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1-n1nccn1
CCN(CCNc1nc(C)cc(C)n1)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1cccc(c1)C1CC1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1cccnc1OC(C)C
CCOc1ncccc1C(=O)N(CC)CCN(C)c1nc(C)cc(C)n1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1OC(F)(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1OC(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1cccnc1-c1ccccc1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1cccnc1OCC(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1cccnc1OCC(F)(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccc(F)cc1-n1nccn1
CCOc1ccccc1C(=O)N(CC)CCN(C)c1nc(C)cc(C)n1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1-n1cccn1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1nccnc1-n1nccn1
CCCc1ccccc1C(=O)N(CC)CCN(C)c1nc(C)cc(C)n1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1OCC(F)(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1CC(F)(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccc(OC)nc1C1CC1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1OCC(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1cccnc1CC(F)(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ncccc1-n1nccn1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1CC(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1cccnc1-n1cccn1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1nccnc1N1CCCC1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1C1CCC1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ncccc1-c1ccccc1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1nccnc1-n1cccn1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1C1CC1(F)F
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1N1CCCC1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1-n1ncnn1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1ccccc1-c1ncccn1
CCN(CCN(C)c1nc(C)cc(C)n1)C(=O)c1nccnc1-c1ccccn1
CCN(CCN(CC)c1nc(C)cc(C)n1)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C(C)C)c1nc(C)cc(C)n1)C(=O)c1ccccc1-n1nccn1
CCN(CCN(CC(F)F)c1nc(C)cc(C)n1)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1nccc(C#N)c1C)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1nccc(C#N)c1Cl)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1nc(OC)cc(OC)n1)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1nccc(n1)C#N)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1nc(Cl)cc(n1)N(C)C)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1cccc(n1)C#N)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1ncc(Cl)c(n1)C(F)(F)F)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1OC(F)(F)F
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-c1nnn[nH]1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1cccnc1OCc1ccccc1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1cccnc1Oc1ccccc1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1cccnc1C(F)(F)F
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1ccnc1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1C1(CCOCC1)C#N
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-c1cnccn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1cccn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1OCCF
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1OCC(F)(F)F
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1c(F)cccc1-n1nccn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1COC
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1c(F)cccc1-n1ccnn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1cccc2[nH]c(=O)oc12
CCOc1nc2cccc(C(=O)N(CC)CCN(C)c3cc(ccn3)C#N)c2[nH]1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1cc(C)ccc1-n1nccn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1cc(C)nn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1N1CCCC1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1cccc2oc(=O)[nH]c12
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-c1ncc[nH]1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1cnnn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1C1(CC1)C#N
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-c1nc(C)no1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1ccnn1
CCOc1cccc(C(=O)N(CC)CCN(C)c2cc(ccn2)C#N)c1OC
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1cc(F)ccc1-n1nccn1
CCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccc(OCC(F)(F)F)nc1
CN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1nccn1
CCCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1nccn1
CCCCN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1nccn1
CN(CCN(Cc1ccccc1)C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N
CN(CCN(CC1CC1)C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N
CC(C)CN(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1nccn1
CC(C)N(CCN(C)c1cc(ccn1)C#N)C(=O)c1ccccc1-n1nccn1
CN(CCN(CC(F)(F)F)C(=O)c1ccccc1-n1nccn1)c1cc(ccn1)C#N
CCN(CC(NC)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1cccnc1OC(C)C
CCOc1ncccc1C(=O)N(CC)CCN(C)c1nccc(n1)C(C)(C)O
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)F
CCCc1ccccc1C(=O)N(CC)CCN(C)c1nccc(n1)C(C)(C)O
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1CC(F)(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1cccnc1CC(F)(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1CC(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)(F)F
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccc(OC)nc1C1CC1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1ncnn1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1cccnc1-c1ccccc1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ncccc1-c1ccccc1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1nccnc1-n1cccn1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1cccnc1-n1cccn1
CCN(CCN(C)c1nccc(n1)C(C)(C)O)C(=O)c1ncccc1-n1nccn1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)F
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ncccc1-n1nccn1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1cccn1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1nccnc1-n1cccn1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)(F)F
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OC(F)F
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)(F)F
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1cccnc1OCC(F)F
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1OCC(F)(F)F
CCOc1ccccc1C(=O)N(CC)CCN(C)c1cccc(n1)C(C)(C)O
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1cccnc1CC(F)(F)F
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1C1CC1(F)F
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1cccnc1OC(C)C
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ncccc1-c1ccccc1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1ccccc1-n1ncnn1
CCN(CCN(C)c1cccc(n1)C(C)(C)O)C(=O)c1cccnc1-n1cccn1
CCOc1ncccc1C(=O)N(CC)CCN(C)c1cccc(n1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(on1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1cc(on1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Cl)ccc1-n1nccn1)c1cc(on1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-n1nccn1)c1cc(on1)C(C)(C)O
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(on1)C(C)(C)O |r|
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(on1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)c1cc(on1)C(C)(C)O
CCC(O)(CC)c1cc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(on1)C(C)(O)C1CC1
CC[C@@](C)(O)c1cc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
CC[C@](C)(O)c1cc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(on1)C1(O)CCC1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(on1)C(C)(O)C(F)(F)F
C[C@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(on1)C(C)(O)C(F)(F)F
CC(C)C(C)(O)c1cc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
CC(C)C(C)(O)c1cc(no1)[C@H]1CC[C@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(on1)[C@](C)(O)C(F)F |r|
COC(C)(C)c1cc(no1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
CCOC(=O)c1cc(on1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
COCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(no1)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1cc(no1)C(C)(C)O
CCOc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-n1nccn1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-n1cccn1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ccccc1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Cl)ccc1-n1nccn1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-c1ccccn1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1cc(no1)C(C)(C)O
COC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(no1)C(C)(C)O
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-c1ccccc1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ncccc1-c1ccccc1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OCC(F)F)c1cc(no1)C(C)(C)O
CC(C)(O)c1cc(on1)[C@@H]1CCCN(C1)C(=O)c1ccccc1OCC(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1cnccn1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1CC1(F)F)c1cc(no1)C(C)(C)O
CC[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(no1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(no1)[C@@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(no1)[C@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1cc(no1)[C@@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1cc(no1)[C@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1cc(no1)[C@@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1cc(no1)[C@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1cc(no1)[C@@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1cc(no1)[C@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1cc(no1)[C@@H](O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1cc(no1)[C@@H](O)C(F)(F)F
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1cc(no1)[C@H](O)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1cc(no1)[C@H](O)C(F)(F)F
CON(C)C(=O)c1cc(on1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(no1)C(C)(O)C1CC1
CCC(C)(O)c1cc(on1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(no1)C1CCCO1 |r|
COC(C)(C)c1cc(on1)[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)c1cc(sn1)C(C)(C)O
CC(C)(O)c1cc(ns1)[C@@H]1CCCN(C1)C(=O)c1cscc1-n1nccn1
COC(=O)c1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)c1cc(sn1)C(C)(C)O
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)c1cc(sn1)C(C)(C)O
COCCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)c1cc(sn1)C(C)(C)O
O=S(=O)(NC1CC1)c1ccc(cc1)S(=O)(=O)N1CCCc2ccccc12
Cc1c(oc2ccccc12)C(=O)Nc1ccc(cc1)N1CCOCC1
O=C(Nc1cccc(NC(=O)N2CCN(CC2)c2ccccc2)c1)N1CCN(CC1)c1ccccc1
[#8]-c1ccccc1-c1csc(n1)-[#6](\C#N)=[#6]-1/[#6]-[#6]-[#6]-[#6]-1
COc1ccc(cc1)-c1cc2nc(cc(N3CCC4(CC3)OCCO4)n2n1)-c1ccccc1
CCN1C(C)=C(C)S\C1=C1/SC(=S)N(CC)C1=O |t:4|
O=C(N1CCCC(C1)c1nc(no1)-c1ccc(cc1)S(=O)(=O)NCc1ccccc1)c1ccco1
CN1C(=O)C2(N=c3ccccc3=N2)c2ccccc12 |c:12,t:5|
Oc1ccccc1-c1nc(NCC2CCCO2)c2ccccc2n1
COc1ccc(cc1)-c1nn2c(nnc2s1)-c1ccccc1
CNc1oc(nc1C#N)-c1cccc2ccccc12
Nc1nc(cc(-c2cccs2)c1C#N)-c1ccccn1
COC(=O)c1ccccc1NC(=O)c1sc(=S)n(C)c1N
O=C(OC1CCOC1=O)c1ccc(s1)-c1nc2ccccc2s1
Cc1ccnc2ccc(cc12)-c1nc2ccccc2o1
N#C\[#6](=[#6]-1/[#16]-[#6]=[#6]-[#16]-1)-c1nc(cs1)-c1ccccc1 |c:5|
COC(=O)c1ccccc1NC(=O)CSc1nc(O)cc(=O)n1C1CCCC1
Cc1noc(C)c1COC(=O)c1ccc2C(=O)c3ccccc3S(=O)(=O)c2c1
N#CC(C1=NCCC1)c1nc(cs1)-c1ccccc1 |t:3|
Nn1c(nc2sc3CCCCc3c2c1=O)-c1cccs1
CCn1c(C)nc2cc(ccc12)-c1nc2-c3ccccc3Cn2n1
Cc1cnc(NC(=O)c2ccc(o2)-c2nc3ccccc3s2)s1
CCn1c(C)cs\c1=N/C(=O)c1ccccc1O
O=c1sc(Nc2ccccc2)nc2ccsc12
CSc1nc2ccc3nc(NC(=O)c4cccs4)sc3c2s1
COc1cccc(c1)-c1cc(no1)C(=O)Nc1ccccc1SC
C=CCNc1nc(nc(n1)-n1ccnc1)N(c1ccccc1)c1ccccc1
COc1ccc(cc1O)-c1nc2ccccc2s1
CSc1cccc(NC(=O)C2CCCN(C2)S(=O)(=O)c2ccc(F)cc2)c1
Cc1ccc(NC(=O)c2ccc3ccccc3n2)nc1
CCn1c(SCC(=O)Nc2ccc3n(CC)c4ccccc4c3c2)nnc1-c1cnccn1
CCN(CC)c1ccc(NC(=O)c2cc3ccccc3o2)c(C)c1
CCOC(=O)c1c(C)nc2c3ccccc3ccn12
c1ccc2oc(nc2c1)-c1ccc2ccccc2n1
Cn1c2ccc(Cl)cc2c2nc3ccccc3nc12
O=C(C1CCCN1S(=O)(=O)c1cccc2cccnc12)N1CCn2c1nc1ccccc21
Cc1ccc2nc(Nc3ccccc3)c(CN=O)c(=O)n2c1
CCn1c2ccccc2c2nc3ccccc3nc12
C1CN(CCN1c1ccccc1)c1ncnc2c3ccccc3oc12
OC(CN1c2ccccc2Sc2ccccc12)Cn1nnc2ccccc12
Cc1nn(C)c(C)c1N=Cc1c(O)ccc2ccccc12 |w:8.8|
Nc1c(oc2ccccc12)C(=O)c1ccc(Br)s1
Cc1csc(n1)-c1coc2cc(O)cc(C)c2c1=O
CCN(CC)c1ccc2cc(-c3nc4ccccc4n3C)c(=O)oc2c1
COc1ccccc1C(=O)Nc1nc(cs1)-c1ccc(cc1)S(=O)(=O)N1CCOCC1
Cc1nc2ccc(cc2[nH]1)-c1nc2ccccc2o1
Cc1nn2c(N)c(-c3ccccc3)c(C)nc2c1-c1ccccc1
Cc1cc(NC(=O)CCC(=O)N(Cc2cccs2)C(C(=O)NC2CCCC2)c2ccccc2)no1
CCOC(=O)c1ccc2[nH]c(C)c(C)c2c1
O=C(OCC#CCSc1nc2ccccc2o1)c1cc2ccccc2o1
Cc1cccc(c1)-c1cc2nc(cc(N3CCC4(CC3)OCCO4)n2n1)-c1ccccc1
Cc1ccc(cc1)-c1cc2nc(cc(N3CCC4(CC3)OCCO4)n2n1)-c1ccccc1
Cc1c(\C=C\C(=O)c2cccs2)cnn1C
Cc1c(c(=O)n(-c2ccccc2)n1C)C1(C(=O)Nc2c1cc(Br)cc2C)c1c(C)n(C)n(-c2ccccc2)c1=O
Clc1ccc(cc1)C1=CC(=O)N(Nc2ccccc2)C1=O |t:8|
CSc1cccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc(Br)s2)c1
COc1ccc(CN=Nc2snc(SC)c2C#N)cc1OC |w:8.8|
CSc1nc2ccc3nc(NC(=O)c4ccccc4)sc3c2s1
COC(=O)C(C(C)=O)=C1C=C(NS(=O)(=O)c2ccc(C)cc2)c2ccccc2C1=O |w:8.30,t:9|
Clc1cccc(-c2ccc(C=NNC(=O)C3C(CNC3=O)c3ccccc3)o2)c1Cl
COc1ccc(C=c2sc3nc(nn3c2=O)-c2ccccc2OC)c(OC)c1
CCn1c(SCC(=O)c2ccc3ccccc3c2)nnc1-c1cccs1
CN(C(c1ccccc1)c1ccccc1)C(=O)CSc1nc(cn1N)-c1ccccc1
Cc1cc(SCC(=O)c2ccc3OCOc3c2)nc2ccccc12
Cc1noc(C)c1COc1ccc(cc1)C(=O)OCC(=O)N1CC(=O)Nc2ccccc12
CCSc1nnc(NC(=O)c2ccc3ccccc3n2)s1
Cc1cnc(NC(=O)c2cc3c(C)nn(-c4ccccc4)c3s2)s1
Cc1nc2cc(NC(=O)COc3ccccc3C#N)ccc2n1-c1ccccc1
Cc1cccc(NC(=O)NNC(=O)c2cc(nc3ccccc23)-c2ccccc2Cl)c1
Cc1ccc(cc1)C(=O)OCn1ncc(Cl)c(Cl)c1=O
Clc1ccccc1C(=O)Nc1ccc2sc3ccccc3c(=O)c2c1
NC(=S)NN=Cc1ccccc1OCc1cccc(Cl)c1 |w:4.3|
Cc1ccc(\C=C2/Sc3ccccc3C2=O)s1
CCSC1=NC(O)(C(C(C1C#N)c1ccccc1Cl)C(=O)c1cccs1)C(F)(F)F |t:3|
Cc1cc(oc1C(=O)N(CC(=O)NC1CCCC1)c1ccccc1C)C(C)(C)C
Cc1cc(C)nc([N-]\C(N)=[NH+]\c2ccc(F)c(c2)[N+]([O-])=O)n1
CCn1c2ccccc2c2cc(NC(=O)c3cccc(OC)c3)ccc12
COc1ccc-2c(c1)NC(=O)c3c2c4ccccc4s3
Cc1[nH]c2ccccc2c1C(=O)CSc1nc2ccccc2[nH]1
Cc1cccc(C=NNC(=O)c2cc3CCc4ccccc4-c3s2)c1
CC(=O)NC(NC(=S)Nc1ccc(cc1)N=Nc1ccccc1)C(Cl)(Cl)Cl |w:15.15|
Cc1nn(c(C)c1C=NNC(=O)c1cc(n[nH]1)-c1ccccc1)-c1ccccc1 |w:8.9|
C\C(\C=C1\SC(=NC1=O)N1CCOCC1)=C\c1ccccc1 |c:5|
[O-][N+](=O)c1cccc(c1)-c1nc(-c2cccs2)c([nH]1)-c1cccs1
Brc1cccc(C=C(NC(=O)c2ccccc2)c2n[nH]c(=S)[nH]2)c1 |w:6.5|
COc1ccc(C=Cc2nnc([nH]2)-c2ccccc2O)cc1OC |w:7.7|
Cc1ccc(cc1Cl)-c1nnc(SCc2ccc(cc2)C(=O)Nc2nccs2)n1CC=C
CCn1c2ccccc2c2cc(NC(=O)c3cccc(OC)c3OC)ccc12
[O-][N+](=O)c1ccc(cc1)-c1c[nH]c(SC(c2ccccc2)c2ccccc2)n1
COc1ccc(C=Cc2nc(N)nc(n2)-c2ccccc2O)cc1OC |w:6.5|
CC(NS(=O)(=O)c1ccc(OCC(=O)Nc2cccc(c2)[N+]([O-])=O)cc1)c1ccccc1
CN(\[NH+]=C\[c-]1cc(ccc1=O)[N+]([O-])=O)c1ccccc1
[#6]-[#8]-c1ccc(cc1-[#8]-[#6])-[#6](=O)-[#8]\[#7]=[#6]-1/c2ccccc2-c2ccccc-12
OC1(N=C(SCC=C)C(C#N)C(C1C(=O)c1cccs1)c1ccccc1Cl)C(F)(F)F |t:2|
Cc1ccc(cc1)C(=O)N\C(=C\c1ccc(o1)-c1cccc(c1)[N+]([O-])=O)C(=O)NC(C)(C)C
Cc1nn(c(C)c1C=NNC(=O)c1cc(n[nH]1)-c1cccs1)-c1ccccc1 |w:8.9|
COCCCNC(=O)CCC(=O)NNc1nc2ccccc2c2nc(nn12)-c1ccccc1
CCCCNC(=O)CCC(=O)NNc1nc2ccccc2c2nc(nn12)-c1ccccc1
CN(C)c1c(F)c(F)c2c(C)c3ccccc3nc2c1F
CCn1c2ccccc2c2cc(NC(=O)c3cc(OC)cc(OC)c3)ccc12
Clc1[nH]c2ccccc2c1C=NNC(=O)c1sc2ccccc2c1Cl |w:11.13|
Cc1nc2c(ccc3nc(NC(=O)Cc4cccc5ccccc45)sc23)s1
O=C(Nc1nnc(o1)-c1ccccc1)c1cc(nc2ccccc12)-c1cccs1
Cc1cc(Cl)ccc1OCCCC(=O)NCCN1C(=O)S\C(=C/c2cccnc2)C1=O
COc1ccccc1-c1nnc(SCc2csc(n2)-c2ccc(Cl)cc2)n1CC=C
COc1ccc2c(Cl)c(sc2c1)C(=O)NN=Cc1c(C)[nH]c2ccccc12 |w:15.16|
Cc1cc(nc2ccccc12)-c1ccc(cc1)N1CCOCC1
COc1ccccc1NS(=O)(=O)c1cccc(NC(=O)c2ccc3ccccc3n2)c1
CCN(CC)c1ccc(NC(=O)Cn2c(nc3ccccc23)C(C)NC(=O)c2ccccc2)cc1
COc1ccc(CNC(=O)COC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2cccs2)cc1
CNC(=O)NC(=O)C(C)OC(=O)c1c2CC\C(=C/c3cccs3)c2nc2ccccc12
Cc1c(oc2c1ccc1ccccc21)C(=O)OCC(=O)NCCN1C(=O)CSC1=O
Oc1cccc(c1)C(=O)OCc1cc(=O)n2c(n1)sc1ccccc21
O=C(Nc1cccc(c1)S(=O)(=O)NCc1ccco1)c1cc(nc2ccccc12)-c1ccccc1
Fc1ccc(cc1)-c1cc(C(=O)Nc2cccc(c2)S(=O)(=O)NCc2ccco2)c2ccccc2n1
Clc1cc(Cl)c(cc1C(=O)NCCN1C(=O)S\C(=C/c2ccccc2)C1=O)S(=O)(=O)N1CCOCC1
Cc1ccsc1C=NNC1=c2ccccc2=NC1=O |w:7.8,c:10,17|
Oc1cc(C=Cc2c(F)cccc2Cl)nc2ccccc12 |w:4.3|
Clc1ccccc1NS(=O)(=O)c1cccc(c1)C(=O)NNC1=c2ccccc2=NC1=O |c:23,30|
Clc1ccc(C=NNC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)c2cccs2)cc1
Clc1cccc2c(Br)ccc(SCC(=O)Nc3ccc(cc3)S(=O)(=O)Nc3nccs3)c12
CN(C)c1ccc(cc1)-c1nnc(o1)-c1cccs1
OCC1(Cc2cccc(Cl)c2)CCCN(Cc2ccc3cc(F)ccc3n2)C1
O=C(NC(=S)Nc1nc(cs1)-c1ccccc1)c1ccco1
Brc1ccc(C=NNC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)c2cccs2)cc1
S=c1[nH]nc(-c2cc([nH]n2)-c2ccccc2)n1N=Cc1c2ccccc2cc2ccccc12 |w:17.19|
O=c1c2ccccc2nc2c3ccccc3c(NCc3ccccn3)nn12
CCc1c(C)sc(NC(=S)Nc2nc(C)cc(C)n2)c1C(=O)OC
Oc1ccc(NC(=S)NNC2=c3ccccc3=NC2=O)cc1 |c:10,17|
COc1cccc(CN=Nc2cc(C)nc(n2)-c2ccccc2O)c1O |w:9.9|
O=C(NC(=S)Nc1cccc2cccnc12)c1cccs1
COc1cc(OC)c(cc1OC)-c1nc2ccccc2s1
NS(=O)(=O)c1ccc(CNC(=O)c2cc(nc3ccc(Cl)cc23)-c2ccccn2)cc1
Cc1ccc(o1)-c1cc([nH]n1)C(=O)NN=CC(Br)=Cc1ccccc1 |w:14.15,18.20|
COc1ccccc1C(=O)Nc1nc2cc3OCCOc3cc2s1
O=C(CSc1ccc(nn1)-c1cccs1)c1cccs1
CCOC(=O)N1CCN(CC1)C(=O)CSc1ccc(nn1)-c1ccccc1
O=C(CSc1ccc(nn1)-c1ccccc1)c1cccs1
COc1ccc(OCc2n(CC(=O)OC3CC(C)CCC3C(C)C)c3ccccc3[n+]2C)cc1
CN(C)\C=C1\Oc2c(ccc3ccccc23)C1=O
Cc1nc2c(cnn2c2CCCc12)-c1ccc(Cl)cc1
Cc1ccc(C)n1-c1ccsc1-c1cc2nc(C)cc(=O)n2[nH]1 |(13.85,-2.9,;12.31,-2.9,;11.41,-4.14,;9.94,-3.67,;9.94,-2.13,;8.7,-1.22,;11.41,-1.65,;11.88,-.18,;13.35,.29,;13.35,1.83,;11.88,2.31,;10.98,1.06,;9.44,1.06,;8.54,-.18,;7.08,.29,;5.75,-.48,;4.41,.29,;3.08,-.48,;4.41,1.83,;5.75,2.6,;5.75,4.14,;7.08,1.83,;8.54,2.3,)|
N#Cc1cccn1-c1nccc(n1)-c1cccs1
Nc1c(sc2nc3CCCCc3cc12)-c1nc(N)nc(n1)N1CCOCC1
C=CCNC(=O)CCC(=O)NNc1nc2ccccc2c2nc(nn12)-c1ccccc1
OC(=O)c1ccc(cc1)-n1c(O)cc(SC(NCc2ccc3OCOc3c2)=Nc2ccc(F)cc2)c1O |w:27.30|
Cc1cc(O)cc2c1sc1ccccc1c2=O
CCOC(=O)c1ccc2[nH]c3ccccc3c2c1
CCN(CC)P(=O)(Nc1cccc(c1)C(F)(F)F)c1ccc(cc1NC(=O)c1ccco1)N(C)C
OC1CN(Cc2cc(=O)n3ccsc3n2)c2c(C1)ccc1ccccc21
CCN(C(=O)CSc1ncnc2sc(CC)cc12)c1c(N)n(Cc2ccccc2)c(=O)[nH]c1=O
Cc1cc(C)nc(NC(N)=Nc2ccc(SC(F)F)cc2)n1 |w:10.10|
CN(C1CCCCC1)C(=O)COC(=O)c1cccc(c1)S(=O)(=O)Nc1c(C)n(C)n(-c2ccccc2)c1=O
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(=O)N2CCN(CC2)c2ccccn2)cc1
Cc1nn(c(C)c1P(=S)(c1nccn1C=C)c1nccn1C=C)-c1ccccc1
COc1cc2c(cc1NC(=O)CSc1nnc(-c3cnccn3)n1CC=C)oc1ccccc21
Cc1ccc(NC2=NC(=O)C(S2)=Cc2cccn2C)cc1C |w:12.13,t:6|
COc1ccc(OC)c(C=NNC(=O)c2cc3c(OC)cc(OC)cc3[nH]2)c1
CCN(CC)c1ccc(C=NNC(=O)c2ccco2)c(O)c1 |w:10.10|
Cc1ccc(cc1)-c1csc2nnc(SCC(=O)Nc3nsc(n3)-c3ccccc3)n12
S=c1[nH]nc(-c2cc([nH]n2)-c2ccccc2)n1N=Cc1cccs1 |w:17.19|
CN(C)S(=O)(=O)c1ccc(cc1)-c1csc(N=NCc2ccco2)n1 |w:16.16|
CC(C)n1c(=O)[nH][nH]c1=S
Cc1ccc(C)n1-c1nn(c2cccc(F)c12)S(=O)(=O)c1cccc2cccnc12 |(6.6,-5.67,;8.06,-5.19,;9.31,-6.09,;10.56,-5.18,;10.07,-3.72,;10.98,-2.47,;8.53,-3.72,;7.62,-2.48,;8.09,-1.02,;6.85,-.12,;5.62,-1.02,;4.11,-.71,;3.08,-1.85,;3.56,-3.32,;5.07,-3.63,;5.54,-5.1,;6.09,-2.49,;6.85,1.42,;5.31,1.42,;8.39,1.42,;6.85,2.96,;5.52,3.73,;5.52,5.27,;6.85,6.04,;8.19,5.27,;9.57,6.09,;10.96,5.3,;10.96,3.69,;9.57,2.9,;8.19,3.73,)|
Cn1c(N)c(sc1=S)C(=O)NN=Cc1ccccc1
Cc1noc(C)c1S(=O)(=O)Nc1ccc(O)c2c1oc(cc2=O)-c1ccccc1Cl
COc1ccc(cc1OC)S(=O)(=O)Nc1c(O)ccc2ccccc12
Oc1ccc2ccccc2c1NS(=O)(=O)c1cccc2ccccc12
CCOc1ccccc1C(=O)NCCCCNC(=O)c1ccccc1OCC
CCOc1ccccc1C(=O)NCCNC(=O)c1ccccc1OCC
COc1cccc(OP(=O)(Nc2ccccc2)Oc2cccc(OC)c2)c1
C(N1CCN(CC1)C1CCCSc2ccccc12)c1ccccc1
Cc1cccc(OCCSc2nc3ccccc3n2CCC(O)=O)c1
Cc1cc(C)n2nc(cc2n1)-c1cccc(Br)c1
OC(=O)CCn1c(SCCOc2ccccc2)nc2ccccc12
N#CCSc1nc(nc2ccccc12)-c1ccccc1
Cc1ccc(O)c(NC(=O)c2cc(on2)-c2ccccc2Cl)c1
[O-][N+](=O)c1c(-c2ccccc2)c2cc(Cl)ccc2[nH]c1=O
CCOc1cc(cc(Br)c1OS(=O)(=O)c1ccccc1)C(=S)N1CCOCC1
COc1ccc(NC(=O)C(=O)Nc2cccc3cccnc23)cc1OC
Cn1c2ccc(F)cc2c2nc3ccccc3nc12
Clc1ccc(CN2CC[C@H]3C=CC[C@H]([C@H]3C2=O)C(=O)Nc2ccccc2)cc1Cl |c:10|
COc1ccc(CN2CC[C@H]3C=CC[C@H]([C@H]3C2=O)C(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1OC |c:11|
Cc1cccc2c3nc4ccccc4nc3n(C)c12
COC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CCCc1c[nH]c2ccccc12
O=c1c2ccccc2oc2cc(ccc12)-c1ccc2[nH]ccc2c1
CNc1nc(Nc2ccc(C)c(Cl)c2)c2cnn(C)c2n1
Cn1cc(\C=C(/C#N)C(=O)Nc2ccccc2O)c2ccccc12
Cc1nn(-c2ccccc2)c2nc(N)c(C#N)c(C3CC(=O)C(=O)C=C3)c12 |c:25|
COc1cc(Cn2cc(O)n(-c3ccccc3Cl)c2=S)cc(OC)c1OC |(5.14,3.81,;6.48,4.58,;7.81,3.81,;7.81,2.27,;9.14,1.5,;9.14,-.04,;7.81,-.81,;6.4,-.19,;5.37,-1.33,;3.84,-1.17,;6.14,-2.67,;5.52,-4.07,;6.42,-5.32,;5.8,-6.73,;4.26,-6.89,;3.36,-5.64,;3.99,-4.23,;3.08,-2.99,;7.65,-2.35,;8.79,-3.38,;10.48,2.27,;10.48,3.81,;11.81,4.58,;13.15,3.81,;9.14,4.58,;9.14,6.12,;10.48,6.89,)|
CC(NC(=O)COc1cccc(NC(C)=O)c1)c1ccc2ccccc2c1
Cc1ccc(cc1)S(=O)(=O)N1CCCN(CC1)C(=O)c1cc2ccccc2[nH]1
Cc1ccc(C)c(NP(=O)(Oc2ccccc2)Oc2ccccc2)c1
CN(C)c1ccc(NC(=S)c2ccc3ccccc3n2)cc1
Fc1cccc(Nc2nc3ccccc3n3cnnc23)c1
Cc1cc(C(=O)NCc2cccc(Cl)c2)c2ccccc2n1
COC(=O)C1=C(C)N(Cc2ccccc2)C(NCc2ccccc2)=N[C@H]1c1cccc(F)c1 |c:4,25|
Cc1noc(C)c1S(=O)(=O)N(CC(=O)NCCc1ccc(Cl)cc1)c1ccc(C)cc1
CSc1cccc(NC(=O)C2CCCN(C2)S(=O)(=O)c2cccs2)c1
Cc1ccc(\C=C2\Sc3ccccc3N(CC(=O)NCC3CCCO3)C2=O)cc1
COc1cccc(\C=C2\Oc3ccccc3N(CC(=O)NCC3CCCO3)C2=O)c1
Brc1cccc(\C=C2\Oc3ccccc3N(CC(=O)NCC3CCCO3)C2=O)c1
Cc1cc(C)cc(NC(=O)C2CCCN2S(=O)(=O)c2cccc3cccnc23)c1
OC(=O)c1ccccc1NS(=O)(=O)c1cccc(c1)-n1sc2ccccc2c1=O
CCOc1ccc(cc1)S(=O)(=O)N1CCCC(C1)C(=O)Nc1cc(C)cc(C)c1
COc1cccc2oc3cc(ccc3c(=O)c12)-c1ccc2[nH]ccc2c1
COc1ccc(cc1)N(CC(=O)NCCc1cccc(C)c1)S(=O)(=O)c1c(C)noc1C
CN(Cc1ccccc1)C(=O)c1nc[nH]c1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC(C)(C)C
COc1cc2ccccc2cc1C(=O)Nc1ccc(cc1)N1CCOCC1
CCOc1ccccc1C(=O)Nc1ccc2nc3CCCCCn3c(=O)c2c1
Fc1cccc(NC2CCCN(C2)C(=O)c2cccc(c2)N2CCNC2=O)c1
CCOC(=O)C1C(C)NC(=O)N=C1COC(=O)C=Cc1cccc(OC)c1 |w:17.17,c:11|
CCc1cc(sc1C)C(=O)OCC(=O)N1CCC(=N1)c1ccccc1 |c:18|
Cc1ccc(NC2CCCN(C2)C(=O)c2cn(C)c3ccccc23)cc1C
COc1cccc(C=NNC(=O)c2nnn(c2CN(C)c2ccccc2)-c2nonc2N)c1
CN(Cc1c(nnn1-c1nonc1N)C(=O)NN=Cc1cccc(O)c1)c1ccccc1
COc1cccc2oc3ccc(cc3c(=O)c12)C#Cc1ccccn1
Cn1c2ccccc2c(=O)c2cc(ccc12)C#Cc1ccccn1
Cc1ccc(NC2CCCN(C2)C(=O)c2cccc(c2)-c2ncc[nH]2)cc1C
COc1ccc(OC)c(c1)S(=O)(=O)NCC(N1CCc2ccccc12)c1ccco1
CSc1cccc(c1)N1CC(CC1=O)C(=O)NCCN1C(=O)S\C(=C/c2cccnc2)C1=O
CN(c1ccc(C)cc1)S(=O)(=O)c1cccc(c1)C(=O)NCC(N1CCOCC1)c1cccs1
CSc1ccc(CN(C)C(=O)c2cc(ccc2C)S(=O)(=O)NCc2ccccc2)cc1
COc1ccc(cc1)[C@@H]1CC=C([C@@H](N1S(=O)(=O)c1ccccc1C)c1cccc(Cl)c1)C(O)=O |c:11|
CCOc1ccccc1N1CCN(CC1)C(=O)c1ccc(cc1)S(=O)(=O)Nc1ccccc1
CC(NC(C)c1ccccc1Cl)C(=O)Nc1cccc(c1)S(=O)(=O)N1CCCCC1
CCN(C(=O)CON=Cc1ccc(OC)cc1OC)c1c(N)n(Cc2ccccc2)c(=O)[nH]c1=O |w:7.6|
Cc1ccccc1NC(=O)C1CCCN1S(=O)(=O)c1ccccc1C(F)(F)F
CCOC(=O)C1C(C)NC(=O)N=C1COC(=O)c1ccc2ccccc2c1O |c:11|
Cc1nc2ccc(NC(=O)c3oc4ccc(F)cc4c3C)cc2s1
CCSc1ccc(cc1OC)[C@@H]1[C@@H]2[C@@H](C(=O)N(CC)C2=O)[C@@]2(CCCCN12)C(=O)OC
CC(C)(O)c1cc2ccc(cc2c(=O)o1)C#Cc1ccsc1
O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)c1cccc2[nH]ccc12
COc1cc(OC)cc(c1)C#Cc1ccc2n(CC=C)c3ccccc3c(=O)c2c1
Cn1c2ccccc2c(=O)c2cc(ccc12)C#Cc1cccc(N)c1
C=CCn1c2ccccc2c(=O)c2cc(ccc12)C#Cc1ccccn1
COc1ccc2sc(c(C#CCO)c2c1)-c1ccc(cc1)N(C)C
COC(=O)C1=C(C[C@@H]2CC[C@H]1N2C(=O)NCCOc1ccccc1Cl)c1ccccc1OCc1ccccc1 |t:4,TLB:2:4:11:8.9|
COc1ccccc1NC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)cc1
CC(OC(=O)c1oc2ccccc2c1C)C(=O)N(C)Cc1ccccc1
OCCN(Cc1ccccc1)C(=O)C[C@H]1C\C=C/C[C@H](Cc2ccc(F)cc2)C(=O)OC[C@@H](NC1=O)c1ccccc1 |c:17|
CC(C)(C)OC(=O)C[C@@H]1C\C=C/C[C@H](CC(=O)N[C@@H](CO)Cc2ccccc2)C(=O)N[C@@H](COC1=O)C(C)(C)C |c:10|
COc1cccc(c1)-c1sc2ccc(OC)cc2c1-c1ccc(OCCN(C)C)cc1
C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc2c(NC(=O)Nc3ccc(F)cc3)cccc2C1=O
Cc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Cl)cc2)c1
Cc1ccc(cc1)[C@@H]1CC=C([C@@H](N1S(=O)(=O)c1ccccc1C)c1cccc(Cl)c1)C(O)=O |c:10|
CC[C@@]12[C@H](C[C@H](CC(=O)NC\C=C(/C)CCC=C(C)C)C(=O)N1CCc1c2[nH]c2cc(ccc12)-c1ccco1)C(=O)N1CCN(CC1)C(=O)c1ccco1 |wU:5.5,wD:2.1,3.43,(11.18,3.81,;12.32,2.78,;13.68,3.5,;14.15,1.97,;15.72,1.62,;16.79,2.81,;18.3,2.5,;19.33,3.65,;18.84,5.11,;20.83,3.33,;21.86,4.48,;23.37,4.17,;24.39,5.31,;23.91,6.78,;25.9,5,;26.93,6.15,;28.43,5.83,;29.46,6.98,;30.97,6.67,;28.98,8.44,;16.29,4.33,;17.3,5.49,;14.71,4.64,;14.24,6.11,;12.73,6.43,;11.7,5.28,;12.17,3.82,;10.93,2.92,;9.7,3.82,;8.14,3.47,;7.06,4.64,;7.56,6.16,;9.12,6.48,;10.17,5.28,;5.56,4.31,;4.41,5.34,;3.08,4.56,;3.41,3.06,;4.94,2.9,;13.11,.83,;11.61,1.17,;13.57,-.64,;12.52,-1.77,;12.98,-3.24,;14.49,-3.58,;15.53,-2.45,;15.07,-.97,;14.94,-5.05,;16.45,-5.39,;13.9,-6.18,;12.37,-6,;11.73,-7.4,;12.86,-8.44,;14.2,-7.69,)|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1noc(C)n1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(C)cccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(C)c1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(Cl)cc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C)cc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nscc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cn(C)nc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(C)nsc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1sccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Br)ccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(Cl)ccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2cc(ccn2)C#N)c(n1)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(ccc1-n1nccn1)C(N)=O)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(cc1-n1nccn1)C#N)Oc1cc(ccn1)C#N |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2cc(ccn2)C#N)c(n1)C1CC1 |r|
CCOc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2cc(ccn2)C#N)c(c1)-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(OCF)cc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(OC(F)F)cc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(OCCO)cc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(C)nc1-n1nccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(nc1-n1nccn1)C(F)(F)F)Oc1cc(ccn1)C#N |r|
COc1ccc(C(=O)N2C[C@@H](CC[C@H]2C)Oc2cc(ccn2)C#N)c(Cl)n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1sccc1-c1ncccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccc(F)c1-c1ncccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-c1ncccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(F)ccc1-c1ncccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1c(F)cccc1-c1ncccn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)Oc1ncccc1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)Oc1cccc(C)n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc2ccccc12 |r|
O=C1N(Cc2cc3ccccc3[nH]2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc3ccccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc3[nH]ccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc3OCCOc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc(c2)-c2cccnc2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2ccccc2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2ccc3OCOc3c2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc3OCOc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc3ccccc23)CCCC11CCN(CC1)c1nc2ccccc2[nH]1
Cc1cc2c(CN3CCCC4(CCN(CC4)c4cnc5ccccc5n4)C3=O)cccc2[nH]1
FC(F)(F)c1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
Cc1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
Cc1cc(C)cc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
Cc1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1C
Cc1ccc(C)c(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
O=C1N(Cc2cccc3cccnc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc(c2)-c2ccccc2)CCCC11CCN(CC1)c1cnc2ccccc2n1
FC(F)(F)c1ccccc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
Cn1ccc2c(CN3CCCC4(CCN(CC4)c4cnc5ccccc5n4)C3=O)cccc12
Clc1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
Clc1cccc(CN2CCCC3(CCN(CC3)c3nccc(n3)-c3ccccc3)C2=O)c1
COc1ccc(cc1)-c1nnc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)o1
Cc1noc(c1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)-c1ccccc1
Cc1cc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c2ccccc2n1
Cc1onc(c1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)-c1ccccc1
O=C1N(Cc2noc3ccccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1CCCC2(CCN(CC2)c2cnc3ccccc3n2)N1Cc1cccc2[nH]ccc12
Cc1noc(n1)-c1ccccc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1nc2ccccc2o1
Cc1ccc(C)c(CN2C(=O)CCCC22CCN(CC2)c2cnc3ccccc3n2)c1
O=C1CCCC2(CCN(CC2)c2nc3ccccc3o2)N1Cc1cccc2[nH]ccc12
O=C1CCCC2(CCN(CC2)c2cnc3ccccc3n2)N1Cc1c[nH]c2ccccc12
Cn1ccc2c(CN3C(=O)CCCC33CCN(CC3)c3cnc4ccccc4n3)cccc12
O=C1N(Cc2cccc(c2)-n2ccnn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc(c2)-n2nccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1cnc2ccccc2c1
O=C1N(Cc2ccccc2-n2nccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1nc2ccccc2s1
O=C1N(Cc2cccc(c2)-c2ccccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc3cnccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2ccnc(c2)N2CCOCC2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2c[nH]c3ncccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc(c2)-c2ccncc2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc(c2)-n2cccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc(c2)-c2ncccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2ccnc(c2)-n2cccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cccc(c2)-c2cnccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cn2nnc3ccccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1nc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c(s1)-c1cccc(C)c1
O=C1N(Cc2cnc3ccccn23)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1nc2ccccn2c1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
Brc1cc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)ccn1
Cc1nc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c(s1)-c1cccc(F)c1
CC(N1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)c1c[nH]c2ccccc12
O=C1N(Cc2cccc3nonc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
N=CC(CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)c1ccccn1
COCc1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
O=C1N(Cc2cccc(n2)-n2cccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
Clc1cc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c2OCOCc2c1
COc1ccnc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1OC
O=C1N(Cc2cccc(c2)C#N)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2nccc3ccccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
Fc1ccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)cc1C#N
O=C1N(Cc2ncoc2-c2ccccc2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cc(=O)[nH]c3ccccc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1nc(no1)-c1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
Fc1ccc(cc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)C#N
O=C1N(Cc2ccc(cc2)-c2ncccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
COc1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1F
O=C1N(Cc2cccc(n2)N2CCCC2)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1noc(n1)-c1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
CNc1c(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)cccc1C=N
Cn1ncc2c(CN3CCCC4(CCN(CC4)c4cnc5ccccc5n4)C3=O)cccc12
CC(=N)OC(=N)c1ccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)cc1
O=C1N(Cc2cncn2-c2ccccc2)CCCC11CCN(CC1)c1cnc2ccccc2n1
COc1cccc(c1)-n1cncc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
COc1ccccc1-n1ccnc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
O=C1N(Cc2cccc3nsnc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1oc(nc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)-c1cscn1
Cc1oc(nc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)-c1ccoc1
Cc1ncc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c2COC(C)(C)Oc12
O=C1N(Cc2cncn2Cc2ccccc2)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1nc(oc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)-c1ccccc1
Fc1cc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c2OCOCc2c1
O=C1N(Cc2ccccc2C#N)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1ccc(N)c(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
O=C1N(Cc2cccc3NCCc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2cc(ccn2)-n2cccn2)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1ccc(cc1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O)-n1nccn1
Nc1ccccc1C(=N)CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
Cn1cc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c2ccccc12
O=C1N(Cc2cccc3NCCOc23)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cc1[nH]c2ccccc2c1CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
c1ccc(cc1)CN2C(=O)CCCC23CCN(CC3)c4cnc5ccccc5n4
O=C1CCCC2(CCN(CC2)c2cnc3ccccc3n2)N1Cc1noc2ccccc12
Clc1ccc2oc(nc2c1)N1CCC2(CCCC(=O)N2Cc2cccc3[nH]ccc23)CC1
O=C1CCCC2(CCN(CC2)c2nnc(o2)-c2ccccc2)N1Cc1cccc2[nH]ccc12
O=C1CCCC2(CCN(CC2)c2nc3ccccc3[nH]2)N1Cc1cccc2[nH]ccc12
Clc1ccc2nc(oc2c1)N1CCC2(CCCC(=O)N2Cc2cccc3[nH]ccc23)CC1
Cc1ccc2oc(nc2c1)N1CCC2(CCCC(=O)N2Cc2cccc3[nH]ccc23)CC1
O=C1CCCC2(CCN(CC2)c2cnc3ccccc3n2)N1Cc1c[nH]c2ncccc12
CNc1ccccc1C(=N)CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
Cn1cc(CN2C(=O)CCCC22CCN(CC2)c2cnc3ccccc3n2)c2cccnc12
CN1CCOc2c(CN3CCCC4(CCN(CC4)c4cnc5ccccc5n4)C3=O)cccc12
CN1CCc2c1cccc2CN1CCCC2(CCN(CC2)c2cnc3ccccc3n2)C1=O
Cc1cnc(o1)-c1cccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)c1
O=C1N(Cc2ccccc2-c2ncco2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2ccccc2-c2ccco2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1nc2ccccc2[nH]1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1nccc(n1)-c1ccccc1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1ncnc2[nH]ccc12
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1nccc2occc12
Cc1nnc(N2CCC3(CCCN(Cc4c[nH]c5ccccc45)C3=O)CC2)c2ccccc12
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1ccc2ccccc2n1
O=C1CC2(CCCN(Cc3c[nH]c4ccccc34)C2)CCN1c1nccc2ccccc12
Cc1cc(nc2ccccc12)N1CCC2(CCCN(Cc3c[nH]c4ccccc34)C2=O)CC1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1cc(ncn1)-c1ccccc1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1nccc(n1)-c1ccncc1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1cc2nccnc2cn1
N=C(\C=C/c1ncc[nH]1)N1CCC2(CCCN(Cc3c[nH]c4ccccc34)C2=O)CC1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1ncc2ccccc2n1
Cc1nc2ccccc2nc1N1CCC2(CCCN(Cc3c[nH]c4ccccc34)C2=O)CC1
O=C1N(Cc2c[nH]c3ccccc23)CCCC11CCN(CC1)c1nnc(s1)-c1ccccc1
Cc1cc(nc(n1)N1CCC2(CCNC(Cc3c[nH]c4ccccc34)C2=O)CC1)-n1cccn1
O=C1C(Cc2c[nH]c3ccccc23)NCCC11CCN(CC1)c1nccc(n1)-n1cccn1
O=C1N(Cc2ccc3ccccc3c2)CCCC11CCN(CC1)c1cnc2ccccc2n1
O=C1N(Cc2ccccc2)CCCC11CCN(CC1)c1nc2ccccc2[nH]1
Cn1c(nc2ccccc12)N1CCC2(CCCN(Cc3cccc4ccccc34)C2=O)CC1
FC(F)(F)c1ccc(CN2CCCC3(CCN(CC3)c3cnc4ccccc4n3)C2=O)cc1
O=C1N(Cc2ccc3OCCOc3c2)CCCC11CCN(CC1)c1cnc2ccccc2n1
Cn1c(nc2ccccc12)N1CCC2(CCCN(Cc3ccccc3)C2=O)CC1
O=C1N(Cc2cccc3OCCOc23)CCCC11CCN(CC1)c1nccc2occc12
Cc1ccc(c(c1)C(=O)N1CCCC(COc2ccc(F)nc2)C1)-n1nccn1
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1cnccn1 |r|
C[C@@H]1CC[C@@H](COc2cccc(C)n2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(ccc1-n1nccn1)C(O)=O |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(CO)ccc1-n1nccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(ccc1-c1ncccn1)C(O)=O |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(CO)ccc1-c1ncccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1nccs1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(F)ccc1-n1nccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1ccccc1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(F)ccc1-c1ncccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1cn[nH]c1 |r|
CCOc1ccccc1C(=O)N1C[C@H](COc2ccc(F)cn2)CC[C@H]1C |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cccc2cc[nH]c12 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1ccccc1-c1ncccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1c(F)cccc1-c1ncccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1ccccc1-n1cccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)cn2)CN1C(=O)c1ncccc1-c1ccccc1 |r|
C[C@@H]1CC[C@@H](COc2ccc(Br)nc2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CC[C@@H](COc2ccnc(Cl)c2)CN1C(=O)c1ccccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CCCCC(COc2ccc(F)c(C)c2)C1)-n1nccn1
CC1CCCC(COc2ccc(F)c(C)c2)CN1C(=O)c1cc(C)ccc1-n1nccn1
CC1CCCC(COc2ccc(F)c(C)c2)CN1C(=O)c1ccccc1-n1nccn1
CC1CCCC(COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-n1nccn1
CC1CCCC(COc2ccc(F)cn2)CN1C(=O)c1ccccc1-n1nccn1
CC1CCCC(COc2ccc(F)c(C)c2)CN1C(=O)c1cc(C)ccc1-c1nccs1
CC1CCCC(COc2ccc(F)c(C)c2)CN1C(=O)c1cc(C)ccc1-c1ncccn1
CC1CCCC(COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1ncco1
CC1CCCC(COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1nccs1
CC1CCCC(COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-c1ncccn1
CC1COCC(COc2ccc(F)c(C)c2)CN1C(=O)c1cc(C)ccc1-n1nccn1
CC1COCC(COc2ccc(F)c(C)c2)CN1C(=O)c1ccccc1-n1nccn1
COc1ccnc(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
Cc1cnc(C)c(n1)N1CC2CN(CC2C1)C(=O)c1ccccc1-c1nnc[nH]1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccnc1-c1cc[nH]n1
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1cccnc1-c1cc[nH]n1
Cc1nc([nH]c(=O)n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1nc(C(=O)N2CC3CN(CC3C2)c2cc(=O)[nH]c(C)n2)c(s1)-c1ccc(F)cc1
Cc1cc(=O)[nH]c(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1cc[nH]n1
CN1CNC(=N1)c1ccccc1C(=O)N1CC2CN(CC2C1)c1ncc(Cl)c(C)n1 |c:4|
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1cnccc1-n1ccnn1
Cc1ccc(nc1)-c1c(F)cccc1C(=O)N1CC2CN(CC2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1ccccc1-c1cccs1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1ccccc1-c1ccco1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1ccccc1-c1ccccc1
O=C(N1CCC2CN(C2C1)c1cnc2ccccc2n1)c1ccccc1-c1cccs1
O=C(N1CCC2CN(C2C1)c1cnc2ccccc2n1)c1ccccc1-c1ccco1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1ccccc1-n1cccc1
O=C(N1CCC2CN(C2C1)c1cnc2ccccc2n1)c1ccccc1-c1ccccc1
O=C(N1CCC2CN(C2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1ccccc1
Cc1ccc(cc1)-c1ccccc1C(=O)N1CCC2CN(C2C1)c1cnc2ccccc2n1
O=C(N1CCC2CN(C2C1)c1nc2ccccc2o1)c1ccccc1-c1ccccc1
COc1cccc(CO)c1C(=O)N1CCC2CN(C2C1)c1cnc2ccccc2n1
Brc1ccccc1C(=O)N1CCC2CN(C2C1)c1cnc2ccccc2n1
O=C(N1CCC2CN(C2C1)c1cnc2ccccc2n1)c1ccccc1-c1cccnc1
COc1cccc(CO)c1C(=O)N1CCC2CN(C2C1)c1nccc(n1)-c1ccccc1
COc1cccc(CO)c1C(=O)N1CCC2CN(C2C1)c1nc2ccccc2o1
Cc1ccc(C)c(c1)S(=O)(=O)N1CCC2CN(C2C1)c1nccc(n1)-c1ccccc1
Cc1ccc(C(=O)N2CCC3CN(C3C2)c2cnc3ccccc3n2)c(C)c1
Cc1ccc(C)c(c1)S(=O)(=O)N1CCC2CN(C2C1)c1cnc2ccccc2n1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1c(F)cccc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1cc(F)ccc1-c1ncccn1
CCOc1ccc2ccccc2c1C(=O)N1CCC2CN(C2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC2CN(C2C1)c1nc(C)cc(C)n1)-n1nccn1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC2CN(C2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1ccccc1-c1ncccn1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1c(F)cccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1ccc(F)cc1-n1nccn1
Cc1cc(nc(C)n1)N1CC2CCN(CC12)C(=O)c1c(F)cccc1-n1nccn1
Fc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC2CN(C2C1)c1cnc2ccccc2n1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CCN(CC12)C(=O)c1ccc(F)cc1-n1nccn1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CCN(CC12)C(=O)c1ccccc1-n1nccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CCN(CC12)C(=O)c1ccc(F)cc1-n1nccn1
O=C(N1CCC2CN(C2C1)c1cnc2ccccc2n1)c1ccccc1-n1nccn1
CN(C)c1nc(C)cc(n1)N1CC2CCN(CC12)C(=O)c1cc(F)ccc1-n1nccn1
Cc1cc(C)nc(n1)N1CC2CCN(CC12)C(=O)c1cc(F)ccc1-n1nccn1
Cc1cc(nc(n1)C(F)(F)F)N1CC2CCN(CC12)C(=O)c1cc(F)ccc1-n1nccn1
CN(C)c1nc(C)cc(n1)N1CC2CCN(CC12)C(=O)c1ccccc1-n1nccn1
CN(C)c1nc(C)cc(n1)N1CC2CCN(CC12)C(=O)c1c(F)cccc1-n1nccn1
CN(C)c1nc(C)cc(n1)N1CC2CCN(CC12)C(=O)c1ccc(F)cc1-n1nccn1
CN(C)c1nc(cc(n1)C(F)(F)F)N1CC2CCN(CC12)C(=O)c1cc(F)ccc1-n1nccn1
O=C(N1CC2CN(C2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1ccccc1
O=C(N1CC2CN(C2C1)c1cnc2ccccc2n1)c1ccccc1-c1ccccc1
O=C(N1CC2CN(C2C1)c1cnc2ccccc2n1)c1ccccc1-c1cccs1
O=C(N1CC2CN(C2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1cccs1
Cc1nc(C(=O)N2CC3CN(C3C2)c2cnc3ccccc3n2)c(s1)-c1ccccc1F
Cc1nc(C(=O)N2CC3CN(C3C2)c2nccc(n2)-c2ccccc2)c(s1)-c1ccccc1F
COc1ccccc1C(=O)N1CC2CN(C2C1)c1nccc(n1)-c1ccccc1
COc1ccccc1C(=O)N1CC2CN(C2C1)c1cnc2ccccc2n1
O=C(N1C[C@@H]2CN([C@@H]2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1cccs1 |r|
O=C(N1C[C@H]2CN([C@H]2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-c1cccs1 |r|
Cc1cc(C)nc(n1)N1CC2CN(CC12)C(=O)c1ccccc1-c1cccs1
Cc1cc(C)nc(n1)N1CC2CN(CC12)C(=O)c1ccccc1Br
Cc1ccnc(n1)N1CC2CN(CC12)C(=O)c1ccccc1Br
Cc1ccnc(n1)N1CC2CN(CC12)C(=O)c1ccccc1-c1cccs1
Cc1ccnc(n1)N1CC2CN(CC12)C(=O)c1ccccc1-c1ccccc1
COc1ccnc(n1)N1CC2CN(CC12)C(=O)c1ccccc1-c1cccs1
COc1ccnc(n1)N1CC2CN(CC12)C(=O)c1ccccc1-c1ccccc1
CCOc1ccc2ccccc2c1C(=O)N1CC2CN(C2C1)c1nc(OC)cc(OC)n1
CCOc1ccc2ccccc2c1C(=O)N1CC2CN(C2C1)c1nc(C)cc(C)n1
Cc1cc(C)nc(n1)N1CC2CN(CC12)C(=O)c1ccccc1-n1nccn1
O=C(N1CC2CN(C2C1)c1nccc(n1)-c1ccccc1)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CN(C2C1)c1nc(C)cc(C)n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CN(C2C1)c1nccc(n1)-c1ccccc1)-n1nccn1
Fc1ccc(c(c1)C(=O)C1CC[C@H]2CN([C@H]2C1)c1cnnc(Cl)c1)-n1nccn1 |r|
Cc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc(C)cc(C)n2)c(n1)-n1ccnn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccnc1C(F)(F)F |r|
Cc1nc(nc(C)c1C)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1 |r|
Cc1cc(nc(n1)C(F)(F)F)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1c(F)cccc1-c1ncccn1 |r|
Cc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nccc(n2)C(F)(F)F)c(n1)-n1ccnn1 |r|
Fc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1nccc(n1)C(F)(F)F)-n1nccn1 |r|
Fc1cccc(c1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nccc(n1)C(F)(F)F)-n1nccn1 |r|
Cc1cnc(C)c(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1 |r|
Cc1cnc(C)c(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1cnc(C)c(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1c(F)cccc1-n1nccn1 |r|
Cc1cnc(C)c(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-n1nccn1 |r|
Cc1cnc(cn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1 |r|
Cc1cnc(cn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1c(F)cccc1-n1nccn1 |r|
Cc1cnc(cn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccc(F)cc1-n1nccn1 |r|
Cc1cnc(cn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-n1nccn1 |r|
Cc1cnc(cn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1nccnc1N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1 |r|
Cc1nccnc1N1C[C@@H]2CCN(C[C@H]12)C(=O)c1c(F)cccc1-n1nccn1 |r|
Cc1nccnc1N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1nccnc1N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccc(F)cc1-n1nccn1 |r|
Cc1nccnc1N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-n1nccn1 |r|
Cc1cncc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-n1nccn1 |r|
Cc1cncc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1cncc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1 |r|
Cc1cncc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1c(F)cccc1-n1nccn1 |r|
Cc1cncc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccc(F)cc1-n1nccn1 |r|
Fc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cnc3ccccc3n2)c(c1)-n1nccn1 |r|
Fc1cccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cnc3ccccc3n2)c1-n1nccn1 |r|
Fc1cccc(c1C(=O)N1CC[C@H]2CN([C@H]2C1)c1cnc2ccccc2n1)-n1nccn1 |r|
Fc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cnc2ccccc2n1)-n1nccn1 |r|
Clc1ccc2oc(nc2c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1 |r|
Fc1cccc(c1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc2cc(Cl)ccc2o1)-n1nccn1 |r|
Fc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc2cc(Cl)ccc2o1)-n1nccn1 |r|
Fc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc3cc(Cl)ccc3o2)c(c1)-n1nccn1 |r|
Fc1cccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc3cc(Cl)ccc3o2)c1-n1nccn1 |r|
Cc1cccc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1c(F)cccc1-n1nccn1 |r|
Cc1cccc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-n1nccn1 |r|
Cc1cccc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1ccnc(c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1cc(C)nc(c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Fc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cccc(n1)C(F)(F)F)-n1nccn1 |r|
Fc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cc(ccn1)C(F)(F)F)-n1nccn1 |r|
Cc1ccc(nc1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccnc2ncccc12 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(C)c1-n1cccn1 |r|
COc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1)-n1nccn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(C)c1-n1nccn1 |r|
COc1cnc(C)nc1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1nccnc1-c1ccccc1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(C)c1-n1ccnn1 |r|
COc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cc(C)ccn1)-n1nccn1 |r|
COc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cc(ccn1)C(F)(F)F)-n1nccn1 |r|
CN(C)c1ccnc(c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(C)c1-n1nccn1 |r|
COc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cc(ccn2)N(C)C)c(c1)-n1nccn1 |r|
CN(C)c1ccnc(c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-c1ncccn1 |r|
CN(C)c1ccnc(c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-n1nccn1 |r|
Fc1cccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cc(ccn2)C(F)(F)F)c1-n1nccn1 |r|
COc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cc(ccn2)C(F)(F)F)c(c1)-n1nccn1 |r|
Cc1cccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cc(ccn2)C(F)(F)F)c1-n1nccn1 |r|
Cc1cc(C)nc(c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-n1nccn1 |r|
COc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cc(C)cc(C)n2)c(c1)-n1nccn1 |r|
COc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cc(ccn1)N(C)C)-n1nccn1 |r|
COc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cc(C)cc(C)n1)-n1nccn1 |r|
Fc1cccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cc(ccn2)C(F)(F)F)c1-c1ncccn1 |r|
Cc1cc(C)nc(c1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-c1ncccn1 |r|
COc1ccc(Br)c(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc(C)cc(C)n2)c1F |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-n1cccn1 |r|
COc1ccc(-c2ncccn2)c(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc(C)cc(C)n2)c1F |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(C)c(C)nc1-n1nccn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(C)c(C)nc1-n1ccnn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccc(nc1-n1ccnn1)C(F)(F)F |r|
Cc1cnc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1)-n1nccn1 |r|
Cc1cnc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1)-n1ccnn1 |r|
COc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc(C)cc(C)n2)c(n1)-n1nccn1 |r|
COc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc(C)cc(C)n2)c(n1)-n1ccnn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1Br |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-c1cncnc1 |r|
CN(C)c1ccc(cn1)-c1ccc(F)cc1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc2Cc3ccccc3-c12 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc2C(=O)c3ccccc3-c12 |r|
Cc1noc(n1)-c1ccccc1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-c1cc[nH]n1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ccccc1-c1nnc[nH]1 |r|
Cc1nc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2nc(C)cc(C)n2)c(s1)-c1ccc(C)cc1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1c[nH]nc1-c1ccccc1 |r|
Cc1onc(c1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1)-c1ccccc1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cnoc1-c1ccccc1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ncoc1-c1ccccc1F |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ncoc1-c1cccc(Cl)c1 |r|
Cc1cc(no1)-c1onc(C)c1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1 |r|
Cc1nnsc1-c1onc(C)c1C(=O)N1CC[C@H]2CN([C@H]2C1)c1nc(C)cc(C)n1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ncccc1Br |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ncccc1-n1ccnn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1ncccc1-n1nccn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-c1cc[nH]n1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cccc(F)c1-c1ncccn1 |r|
Cc1cc(nc(N)n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
CNc1nc(C)cc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-c1ccn(C)n1 |r|
CN(C)c1cc(ncn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
CNc1cc(ncn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1nc(N)cc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Nc1cc(nc(N)n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1cc(ncn1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Fc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1cc(NC2CC2)ncn1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CC[C@H]2CN([C@H]2C1)c1ccnc(n1)-c1ccccc1)C(F)(F)F |r|
FC(F)C(F)(F)Oc1ccccc1C(=O)N1CC[C@H]2CN([C@H]2C1)c1ccnc(n1)-c1ccccc1 |r|
Cc1onc(c1C(=O)N1CC[C@H]2CN([C@H]2C1)c1ccnc(n1)-c1ccccc1)-c1ccccc1 |r|
Cc1ccc(C(=O)N2CC[C@H]3CN([C@H]3C2)c2cc(C)nc(n2)C(F)(F)F)c(n1)-n1ccnn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccnc2c(F)cccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)Nc1nccc2ccccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2ocnc12 |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1F)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(c2c(n[nH]c2n1)-c1ccccc1)C(F)(F)F)c1ccccc1 |r|
Cn1nc(-c2ccccc2)c2c(cc(OCC(=O)N[C@H]3CCc4ccccc34)nc12)C(F)(F)F |r|
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F |r|
C[C@H](CNC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1c(C)n[nH]c1C |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ccccc1)c1ccccc1 |r|
CC(CCc1ccccc1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ccccc1
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1ccccc1 |r|
CC(NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1ccccc1
COc1cccc(c1)-c1nn(C)c2nc(OCC(=O)N[C@@H](C)c3ccccc3)cc(c12)C(F)(F)F |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1cccc(F)c1)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccc(F)cc1)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1cccc(C)c1)C(F)(F)F)c1ccccc1 |r|
Cc1ccc(CNC(=O)COc2cc(c3c(nn(C)c3n2)-c2ccccc2)C(F)(F)F)cc1
CC(NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1c(C)n[nH]c1C
CCn1nccc1C(C)NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F
COc1ccc(CNC(=O)COc2cc(c3c(nn(C)c3n2)-c2ccccc2)C(F)(F)F)cc1
COc1ccc(cc1)C(C)NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F
COc1cccc(c1)C(C)NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccc(C)cc1)C(F)(F)F)c1ccccc1 |r|
COc1ccccc1-c1nn(C)c2nc(OCC(=O)N[C@@H](C)c3ccccc3)cc(c12)C(F)(F)F |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1cccc(Cl)c1)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1cccc(Br)c1)C(F)(F)F)c1ccccc1 |r|
Cn1nc(-c2cccc(F)c2)c2c(cc(OCC(=O)N[C@H]3CCc4ccccc34)nc12)C(F)(F)F |r|
COc1ccc(cn1)C(C)NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F
CC(NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1c(C)nn(C)c1C
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1 |r|
CC(Oc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)C(=O)N[C@@H](C)c1ccccc1 |r|
CC(NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1ccc(C)nc1
C[C@H](NC(=O)COc1cc(c2c(cn(C)c2n1)-c1ccccc1)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ncccc1F)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ncco1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1cnn(C)c1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ncccn1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1cnccn1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ccc(C)cn1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1nc(C)cs1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1nccs1)c1ccc(C)cc1 |r|
COc1ccnc(n1)-c1nn(C)c2nc(OCC(=O)N[C@@H](C)c3ccc(C)cc3)cc(C)c12 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1cncs1)c1ccc(C)cc1 |r|
COc1nc(cs1)-c1nn(C)c2nc(OCC(=O)N[C@@H](C)c3ccc(C)cc3)cc(C)c12 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ncc(C)s1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1cccc(C)n1)c1ccc(C)cc1 |r|
Cc1ccc2[C@H](CCc2n1)NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)C1CC1 |r|
COc1ccc2C(CCc2c1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1
COc1ccc2[C@H](CCc2c1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1 |r|
Cc1ccc(cc1)C(C)(C)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)C1CC1 |r|
C[C@H](NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)C1CC1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)C1CC1)C(F)(F)F)c1ccc(C)cc1 |r|
COc1ccc(cn1)C(C)NC(=O)COc1cc(c2c(nn(C)c2n1)C1CC1)C(F)(F)F
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(c2c(nn(C)c2n1)C1CC1)C(F)(F)F |r|
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)-c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)-c1ccccc1)c1ccc(C)cc1 |r|
COc1ccc(cn1)C(C)NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)-c1ccccc1
COc1ccccc1-c1nn(C)c2nc(OCC(=O)N[C@@H](C)c3ccc(C)cc3)ccc12 |r|
C[C@H](NC(=O)COc1ccc2c(nn(C)c2n1)C(C)(C)C)c1ccc(C)cc1 |r|
CC(C)c1nn(C)c2nc(OCC(=O)N[C@@H](C)c3ccc(C)cc3)cc(C)c12 |r|
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1cc(C)oc1C |r|
CC(NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1cc(C)oc1C)c1c(C)nn(C)c1C
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1ccoc1C |r|
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(C)c2c(nn(C)c2n1)-c1cc(OC)cc(OC)c1 |r|
COc1ccnc(c1)-c1nn(C)c2nc(OCC(=O)N[C@@H](C)c3ccc(C)cc3)cc(C)c12 |r|
Cc1cc(c(C)o1)-c1nn(C)c2nc(OCC(=O)N[C@H]3CCc4nc(C)ccc34)cc(C(F)F)c12 |r|
COc1ccc(cc1)[C@H](C)NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)-c1cc(C)oc1C |r|
Cc1ccc2C(CCc2c1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1
COc1ccc2[C@H](CCc2c1)NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)C1CC1 |r|
COc1ccc2[C@H](CCc2c1)NC(=O)COc1cc(c2c(nn(C)c2n1)C1CC1)C(F)(F)F |r|
Cc1ccc2[C@H](CCc2c1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1 |r|
CC(NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1)c1cnc2[nH]ccc2c1
CC(NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1)c1ccc2n(C)ccc2c1
Cc1ccc2C(CCc2n1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1
Cc1ccc2[C@H](CCc2n1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1 |r|
CCOc1ccc2[C@H](CCc2c1)NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1 |r|
COc1ccc2[C@H](CCc2c1)NC(=O)C(C)Oc1cc(C)c2c(nn(C)c2n1)C1CC1 |r|
Cc1cc(c(C)o1)-c1nn(C)c2nc(OCC(=O)N[C@H]3CCc4nc(C)ccc34)cc(c12)C(F)(F)F |r|
COc1cc2CCC(NC(=O)COc3cc(C)c4c(nn(C)c4n3)C3CC3)c2cc1OC
C[C@H](NC(=O)COc1cc(C)c2c(nn(C)c2n1)C1CC1)c1ccc(C)cc1 |r|
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Br)s2)c1
FC(F)(F)Oc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Br)s2)c1
COc1cccc(c1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(SC)c1
CCCc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(SC)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc3N(C)CCOc3c2)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(SC)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cccc(Cl)c2)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(cc2)C(F)(F)F)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Cl)cc2)c1
COc1ccc(cc1OC)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(SC)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cccc(Br)c2)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(C)c(Cl)c2)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Br)cc2)c1
CSc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Cl)c(Cl)c2)c1
Brc1ccc(s1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccccc1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(c1)C(F)(F)F
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(Cl)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(Br)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(C)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(OC)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(c1)N(C)C
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccc(C)c(C)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc2ccccc12
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cccc(c1)C#N
Cc1cc(cc(c1)NC(=O)[C@@H]2CCCN2S(=O)(=O)c3ccc(cc3)OC)C
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(OC)cc(OC)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(C)ccc1Cl
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(OC)ccc1Cl
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccc(F)c(Cl)c1
CCOc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(OC)cc2)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccc2CCCc2c1
CCc1cccc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(OC)cc2)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)ccc1OC
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccc(F)c(F)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccc(F)c(C)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(C)ccc1F
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccc(Cl)c(C)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1ccc(Cl)c(Cl)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Br)cc2)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cccc3ccccc23)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc3ccccc3c2)c1
COc1ccc(cc1OC)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(C)cc(C)c1
COc1cc(C)ccc1S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(C)cc(C)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Cl)cc2)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(C=C)cc2)c1
COc1ccc(C)cc1S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(C)cc(C)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(cc2)S(C)(=O)=O)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc(ccc2Cl)C(F)(F)F)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(cc2Cl)C(F)(F)F)c1
Cc1ccc(c(Br)c1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(C)cc(C)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Cl)c(c2)C(F)(F)F)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Cl)c(Cl)c2)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc(C)c(Cl)cc2C)c1
Cc1ccc(c(C)c1)S(=O)(=O)N1CCC[C@H]1C(=O)Nc1cc(C)cc(C)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Br)cc2C)c1
Cc1cc(C)cc(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(Br)cc2Cl)c1
COc1ccc(cc1)S(=O)(=O)N1CCC[C@@H]1C(=O)Nc1cc(C)cc(C)c1
C[C@@H]1CS[C@@H](COc2ccccn2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CS[C@@H](COc2ccc(F)cn2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CS[C@@H](COc2ccc(C)cn2)CN1C(=O)c1ccccc1-n1nccn1
C[C@@H]1CS[C@@H](COc2ccc(Cl)cn2)CN1C(=O)c1ccccc1-n1nccn1
C[C@@H]1CS[C@@H](COc2ccc(cn2)C#N)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CS[C@@H](COc2ccc(cn2)C(F)(F)F)CN1C(=O)c1ccccc1-n1nccn1
C[C@@H]1CS[C@@H](COc2ncccc2Cl)CN1C(=O)c1ccccc1-n1nccn1
C[C@@H]1CS[C@@H](COc2ncccc2C#N)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CS[C@@H](COc2cc(C)ccn2)CN1C(=O)c1ccccc1-n1nccn1
C[C@@H]1CS[C@@H](COc2ncccn2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CS[C@@H](COc2ncc(Cl)c(C)n2)CN1C(=O)c1ccccc1-n1nccn1
C[C@@H]1CS[C@@H](COc2ncc(C)c(Cl)n2)CN1C(=O)c1ccccc1-n1nccn1
COc1cnc(OC[C@H]2CN([C@H](C)CS2)C(=O)c2ccccc2-n2nccn2)nc1Cl
C[C@@H]1CS[C@@H](COc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-n1nccn1
C[C@@H]1CS(=O)[C@@H](COc2ccc(F)cn2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CS(=O)(=O)[C@@H](COc2ccc(F)cn2)CN1C(=O)c1ccccc1-n1nccn1 |r|
C[C@@H]1CS[C@@H](CSc2ccccn2)CN1C(=O)c1ccccc1-n1nccn1 |r|
COc1ccc(c(n1)C(=O)N1C2CCC1C(COc1ccc(F)cn1)C2)-n1nccn1 |TLB:16:15:13.12:10|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F |THB:18:16:14.13:11|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F |THB:19:17:15.14:12|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1ncc(cn1)C(F)(F)F)-n1nccn1 |THB:16:14:12.11:9|
CCOc1ccc(C)nc1C(=O)N1C2CCC1C(C2)Nc1cnc2ccccc2n1 |THB:19:17:15.14:12|
Cc1ccc(c(n1)C(=O)N1C2CCC1C(C2)Nc1cnc2ccccc2n1)-n1nccn1 |THB:16:14:12.11:9|
COc1c(F)cccc1C(=O)N1C2CCC1C(C2)Nc1cnc2ccccc2n1 |THB:18:16:14.13:11|
FC(F)(F)c1ccnc(NC2CC3CCC2N3C(=O)c2ccccc2-n2nccn2)c1 |TLB:9:10:14.13:16|
Fc1cccc(C(=O)N2C3CCC2C(C3)Oc2ncc(cn2)C(F)(F)F)c1-c1ncccn1 |THB:15:13:11.10:8|
O=C(N1CCOC[C@H]1Cc1cccc(c1)-c1ncon1)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ncon1)-n1nccn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ccccn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1cccnc1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ncccn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1cnccn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1cccnn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1nccs1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ncco1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1cccs1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)c1ccccc1-n1nccn1
O=C(N1CCOC[C@@H]1Cc1cccc(c1)-n1nccn1)c1ccccc1-n1nccn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-n1cccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1ccnn1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-n1cccn1)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ncccn1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-c1ncccn1)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1cccn1)-n1nccn1
Fc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1cccn1)-n1nccn1
Cc1ccc(c(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2cccn2)c1F)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2cccn2)c(c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1cncn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ccccn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1cccnc1)-n1nccn1
Fc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ccncc1)-n1nccn1
Cc1ccc(c(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c1F)-n1nccn1
Clc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)c1cc(ccc1-n1nccn1)C#N
COc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1
COc1ccc(c(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c1F)-n1nccn1
COc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(cc1OC)-n1nccn1
Cc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(cc1C)-n1nccn1
Fc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(c1)-n1nccn1
COc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(cc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1cccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1nccc(C)n1)-n1nccn1
Cc1ccnc(n1)-c1cccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)c1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1cnccn1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-c1ncco1)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1nccs1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-c1nccs1)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1cccs1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-c1cccs1)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1cccnn1)-n1nccn1
O=C(N1CCOC[C@H]1Cc1cccc(c1)-c1cccnn1)c1ccccc1-n1nccn1
Cc1ccc(c(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncccn2)c1F)-n1nccn1
COc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ncccn1)-n1nccn1
Clc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ncccn1)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1cccn1)-n1nccn1
Fc1cccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c1-n1nccn1
O=C(N1CCC[C@H]1Cc1cccc(c1)-n1nccn1)c1ccccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1 |r|
O=C(N1CCCC[C@H]1Cc1cccc(c1)-n1nccn1)c1ccccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CCCC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1 |r|
Oc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ncccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cc(ccc1F)-n1nccn1)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccccc1-n1nccn1)-n1nccn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2cc(C)ccc2-n2nccn2)cc1-c1ncon1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ncon1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccc(C)cc2-n2nccn2)cc1-c1ncon1
COc1ccc(C[C@@H]2COCCN2C(=O)c2ccc(F)cc2-n2nccn2)cc1-c1ncon1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c(c1)-n1nccn1
COc1ccc(C[C@@H]2COCCN2C(=O)c2c(C)cccc2-n2nccn2)cc1-c1ncon1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1ccc(C)c(c1)-n1nccn1)-n1nccn1
Cc1cccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c1-n1nccn1
Cc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2ccc(C)c(c2)-n2nccn2)c(c1)-n1nccn1
C[C@@H]1COC[C@@H](Cc2cccc(c2)-n2nccn2)N1C(=O)c1ccccc1-n1nccn1
C[C@@H]1COC[C@@H](Cc2cccc(c2)-n2nccn2)N1C(=O)c1ccc(C)cc1-n1nccn1
C[C@@H]1COC[C@@H](Cc2cccc(c2)-n2nccn2)N1C(=O)c1cccc(C)c1-n1nccn1
C[C@H]1COC[C@@H](Cc2cccc(c2)-n2nccn2)N1C(=O)c1ccc(C)cc1-n1nccn1
C[C@H]1COC[C@@H](Cc2cccc(c2)-n2nccn2)N1C(=O)c1cccc(C)c1-n1nccn1
C[C@H]1COC[C@@H](Cc2cccc(c2)-n2nccn2)N1C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1COC[C@@H](Cc2cccc(c2)-n2nccn2)N1C(=O)c1cc(C)c(C)cc1-n1nccn1
Cc1cc(C)c(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1
FC(F)(F)c1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(c1)-n1nccn1
Clc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(c1)-n1nccn1
COc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(cc1F)-n1nccn1
Cc1cc(C(=O)N2CCOC[C@H]2Cc2ccc(C)c(c2)-c2ncon2)c(cc1C)-n1nccn1
Fc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncon2)c(cc1F)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncon2)c(c1)-n1nccn1
Fc1cccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncon2)c1-n1nccn1
Cc1cccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncon2)c1-n1nccn1
Clc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ncon1)-n1nccn1
Cc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncon2)c(cc1C)-n1nccn1
Clc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncon2)c(c1)-n1nccn1
FC(F)(F)c1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-c2ncon2)c(c1)-n1nccn1
Fc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ncon1)-n1nccn1
Cc1cc(C)c(c(c1)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-c1ncon1)-n1nccn1
Clc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ncon1
Fc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(cc1F)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(c1C)-n1nccn1
COc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(c1)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c(c1C)-n1nccn1
COc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c(c1)-n1nccn1
C[C@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1cccc(C)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1cc(C)c(C)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1ccc(C)c(C)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@@]1(C)Cc1cccc(c1)-n1nccn1)-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CCOC[C@H]1Cc1cccc(c1)-n1nccn1)-n1nccn1
COc1cc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c(cc1Cl)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(Cl)cc(c2)-n2nccn2)c(c1)-n1nccn1
Cc1cccc(C(=O)N2CCOC[C@H]2Cc2cc(Cl)cc(c2)-n2nccn2)c1-n1nccn1
Clc1cccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-c2ncccn2)CO1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-c2ncccn2)CO1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-c2ncccn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-c2ncccn2)CO1)C(=O)c1cccc(C)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-c2ncccn2)CO1)C(=O)c1ccc(C)c(C)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-c2ncccn2)CO1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-c2ncccn2)CO1)C(=O)c1ccc(Cl)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2nccn2)CO1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2nccn2)CO1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2nccn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2nccn2)CO1)C(=O)c1cccc(C)c1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cc(ccc1C)-n1nccn1)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2Cl)-n2nccn2)c(c1)-n1nccn1
Cc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccccc1-n1nccn1)-n1nccn1
Cc1cccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2Cl)-n2nccn2)c1-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2C)-n2nccn2)c(c1)-n1nccn1
Cc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cccc(C)c1-n1nccn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cc(ccc1Cl)-n1nccn1)-n1nccn1
Clc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccccc1-n1nccn1)-n1nccn1
Cc1cccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c1-n1nccn1
Cc1cc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c(cc1C)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccc(Cl)cc1-n1nccn1)-n1nccn1
COc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cc(ccc1F)-n1nccn1)-n1nccn1
Cc1ccc(c(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c1F)-n1nccn1
COc1ccc(c(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c1F)-n1nccn1
COc1cc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c(cc1C)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cccc(Cl)c1-n1nccn1)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1c(F)cccc1-n1nccn1)-n1nccn1
Fc1cc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c(cc1F)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccc(cc1-n1nccn1)C(F)(F)F)-n1nccn1
COc1cc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-n2nccn2)c(cc1Cl)-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2ccnn2)CO1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2ccnn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
CC[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1cc(C)ccc1-n1nccn1
CC[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1ccccc1-n1nccn1
CC[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
Fc1cc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc(c1)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(F)cc(c2)-n2nccn2)c(c1)-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1cccc(C)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1ccc(C)c(C)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1ccc(Cl)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2ncccn2)CO1)C(=O)c1cccc(Cl)c1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cc(ccc1F)-c1ncccn1)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2ncccn2)c(c1)-n1nccn1
Cc1cccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2ncccn2)c1-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2ncccn2)c(c1C)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)-c1ncccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccc(Cl)cc1-n1nccn1)-c1ncccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cccc(Cl)c1-n1nccn1)-c1ncccn1
C[C@@H]1OCCN([C@@H]1Cc1cccc(c1)-n1nccn1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@@H]1OCCN([C@@H]1Cc1cccc(c1)-n1nccn1)C(=O)c1ccc(C)cc1-n1nccn1
C[C@@H]1OCCN([C@@H]1Cc1cccc(c1)-n1nccn1)C(=O)c1cccc(C)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-c2cccnn2)CO1)C(=O)c1ccc(C)cc1-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2cccnn2)c(c1)-n1nccn1
C[C@H]1OCCN([C@@H]1Cc1cccc(c1)-n1nccn1)C(=O)c1cc(C)ccc1-n1nccn1
C[C@H]1OCCN([C@@H]1Cc1cccc(c1)-n1nccn1)C(=O)c1ccc(C)cc1-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2Cl)-n2nccn2)c(c1C)-n1nccn1
Clc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2Cl)-n2nccn2)c(c1)-n1nccn1
Clc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cccc(Cl)c1-n1nccn1)-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1cccc(Cl)c1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2nccn2)CO1)C(=O)c1cccc(Cl)c1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cc(ccc1F)-c1ncon1)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2ncon2)c(c1)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)-c1ncon1
Cc1cccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2ncon2)c1-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccc(Cl)cc1-n1nccn1)-c1ncon1
Cc1cc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2ncon2)c(cc1C)-n1nccn1
Fc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cccc(Cl)c1-n1nccn1)-c1ncon1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2F)-c2ncon2)c(c1C)-n1nccn1
FC(F)(F)c1cccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2)-n2nccn2)c1-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cccc(c2F)-n2nccn2)c(c1)-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cccc(c2)-n2nccn2)CO1)C(=O)c1ccc(Cl)cc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2nccn2)CO1)C(=O)c1cc(Cl)ccc1-n1nccn1
C[C@@H]1CN([C@H](Cc2cc(ccc2F)-n2nccn2)CO1)C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC[C@H]1Cc1cc(ccc1C)-n1cccn1)-n1nccn1
Cc1ccc(C(=O)N2CCOC[C@H]2Cc2cc(ccc2C)-n2cccn2)c(c1)-n1nccn1
Cc1ccc(cc1C[C@@H]1COCCN1C(=O)c1cccc(C)c1-n1nccn1)-n1cccn1
Cc1ccc(cc1C[C@@H]1COCCN1C(=O)c1ccc(Cl)cc1-n1nccn1)-n1nccn1
Cc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ncccn1
Cc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1nccs1
Clc1ccc(C[C@@H]2COCCN2C(=O)c2ccccc2-n2nccn2)cc1-c1ncccn1
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(Cl)cn1)-n1nccn1 |r|
Fc1cc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)C(F)(F)F |r|
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cnc2ccccc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2sc(C)nc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2ncccc2c1
COc1cccc(OC)c1[C@H]1CCCC(=O)N1Cc1ccc2ccccc2n1
COc1cccc(OC)c1[C@@H]1CCCC(=O)N1Cc1ccc2ccccc2n1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2ccccc2n1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cnc(OC(F)F)c(Cl)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(n1)-c1ccc(F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1cccnc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cncc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccncc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(n1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccnc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)N1CCCCC1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1nccs1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc2ccccc12
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)N1CCOCC1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(s1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-n1cccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2nccnc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cnc(s1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc(ccn1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-n1cncn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)N1CCCC1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc(on1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cnn(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-n1ccnc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(n1)N1CCCCC1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ncccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1nc2ccccc2s1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2n(C)c3ccccc3c2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1noc(C)n1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccnc(c1)N1CCCC1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1csc(n1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccnc(Br)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1F)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(n1)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(n1)-c1nccs1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc(ccc1F)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(F)c(c1)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1cncs1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ncc(C)s1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-n1nccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1cscn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-n1ccnn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2nc(C)sc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc(ccc1Cl)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc(Cl)cc(c1)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccnc(c1)-c1ccccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(n1)-n1cccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccnc(c1)-n1cccn1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1nccs1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccn1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1csc(n1)-c1ccccc1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1ccc2nc(C)sc2c1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1ccc(F)c(c1)-c1ccccn1
COc1ccnc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1nccs1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccn1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1csc(n1)-c1ccccc1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1cccc(n1)-n1cccn1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-n1nccn1
COc1cncc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cnc(OC(F)F)c(C)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cnc(OC(F)F)c(c1)C1CC1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1csc(C)n1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc(Oc2ccccc2)cc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(Oc2ccccc2)c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc2ccccc2c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc2ccccc12
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc(cc1)-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccccc1-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc2ccccc2n1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cnc2ccccc2c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccnc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(n1)-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1ncccn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1ccccn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1nccs1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc2n(C)c3ccccc3c2c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1cccnc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)N1CCCCC1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cnc(OC(F)F)c(Cl)c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cncc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)N1CCCC1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cnn(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc2sc(C)nc2c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1ccncc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-n1cccn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1csc(n1)-c1ccccc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1cncs1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1ncc(C)s1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-n1nccn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1cscn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccnc(c1)-n1cccn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(n1)-n1cccn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc2nc(C)sc2c1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1F)-c1ccccn1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc(F)c(c1)-c1ccccn1
COc1cc(OC)c(C2CCC(=O)N2Cc2ccc(OC(F)(F)F)cc2)c(OC)c1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cnc2ccccc2c1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc2ccccc2n1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc2ccccc2c1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cnc(OC(F)F)c(Cl)c1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc(cc1)-c1ccccc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)-c1cccnc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc2ccccc12
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(Oc2ccccc2)c1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc(Oc2ccccc2)cc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)-c1ccccn1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccnc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(n1)-c1ccccc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ccccc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)N1CCCC1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)-c1nccs1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)-n1cccn1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1cccc(OC)c1C1CCC(=O)N1Cc1nc2ccccc2s1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)N1CCCCC1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(n1)N1CCCCC1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2ccccc2c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1nccs1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)N1CCCCC1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-n1cccn1
COc1cccc(OC)c1C1CCC(=O)N1Cc1cccc(c1)-c1noc(C)n1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(n1)-c1ccccc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-c1ccccc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ccccn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1cccnc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ncccn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1noc(C)n1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cnn(c1)-c1ccccc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1csc(n1)-c1ccccc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1F)-c1ccccn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1cncs1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ncc(C)s1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-n1nccn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1cscn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2nc(C)sc2c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cc(Cl)cc(c1)-c1ccccn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(F)c(c1)-c1ccccn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-n1cccn1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(n1)-n1cccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(Cl)cc1
COc1ccc(CN2C(CCCC2=O)c2c(OC)cccc2OC)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)c(F)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)c(Cl)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(SC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(cc1)C(F)(F)F
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(Oc2ccccc2)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2OCOc2c1
COc1cc(Cl)cc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(cc1)-n1cccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(cc1)-n1cccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2nonc2c1
COc1ccc2cc(CN3C(CCCC3=O)c3c(OC)cccc3OC)ccc2c1
COc1cc(OC)c(C2CCCC(=O)N2Cc2ccc(OC(F)(F)F)cc2)c(OC)c1
COc1cccc(OC)c1C1CC(C)CC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CC(C)(C)CC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(OC(F)(F)F)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OCCF)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)F)nc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(OC(F)F)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(Oc2ccccc2)c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc2ccccc2o1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc2ccccc2s1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2OC(F)(F)Oc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(OC(F)F)n1
COc1cccc(OC)c1C1CCCC(=O)N1C(C)c1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1C(C)c1cnc(OC(F)F)c(Cl)c1
CCC(N1C(CCCC1=O)c1c(OC)cccc1OC)c1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)F)cn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc(OC(F)F)ccn1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccccc1-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccccc1Oc1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(Oc2ccccc2)nc1
COc1cccc(OC)c1C1CCCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
CCOc1ccccc1C1CCC(=O)N1Cc1ccc(F)cc1
CCOc1ccccc1C1CCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc(F)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OC(F)F)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)F)nc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OC(F)(F)F)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OC(F)F)n1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccnc(OC(F)F)c1
CCC(N1C(CC(C)C1=O)c1c(OC)cccc1OC)c1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cc(OC(F)F)ccn1
CCOc1ccc(CN2C(CCCC2=O)c2c(OC)cccc2OC)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(C)C)cc1
CCCOc1ccc(CN2C(CCCC2=O)c2c(OC)cccc2OC)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OCC2CC2)cc1
COc1cccc(OCCCO)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OCC2CC2)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COCCOc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
CCOc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OCCO)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OCC(O)CO)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCC(C)(C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCC(C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CC(C)(C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccnc(c1)-c1nccs1
COc1cccc(F)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(Cl)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(C)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1)C(F)(F)F
Fc1cccc(F)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cc(F)c(C2CCCC(=O)N2Cc2ccc(OC(F)(F)F)cc2)c(F)c1
Cc1ccc(F)c(C2CCCC(=O)N2Cc2ccc(OC(F)(F)F)cc2)c1F
Fc1cccc(c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1)C(F)(F)F
FC(F)(F)Oc1ccc(CN2C(CCCC2=O)c2c(Cl)cccc2Cl)cc1
Fc1cccc(Cl)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC(C)C)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
CCOc1cccc(OCC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cc(F)cc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cc(C)cc(OC)c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cc(F)cc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1ccc2c(C)noc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1ccccc1C1CCCC(=O)N1Cc1ccc2ccccc2c1
COc1ccccc1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2ccccc2c1
FC(F)(F)c1ccccc1C1CCCC(=O)N1Cc1ccc2ccccc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2NCCCc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2n(C)ccc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cn2ccccc2n1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2n(C)nnc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(cc1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(cc1)N1CCCC1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(OCC(F)(F)F)cc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1cc2ccccc2n1C
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc(cc1)S(C)(=O)=O
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2oc(C)nc2c1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccc2sccc2c1
CCOc1ccccc1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
FC(F)(F)Oc1ccc(CN2C(CCCC2=O)c2ccccc2OC(F)(F)F)cc1
COc1cccc(OC)c1[C@@H]1C[C@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CO[C@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |o1:2,4|
COc1cccc(OC)c1[C@@H]1C[C@@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1cccc(OC)c1C1CC(F)(F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1cccc(OC)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1cccc(OC)c1[C@@H]1C[C@H](C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1cccc(OC)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1cccc(OC)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CO[C@@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |o1:2,4|
CC[C@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |o1:2,4|
COc1cccc(OC)c1[C@@H]1C[C@@H](C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1cccc(F)c1[C@@H]1C[C@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(OC)c1C1COCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CNCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1CN(C)CC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1ncnc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1ncnc(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1ncnc(OC)c1C1CCCC(=O)N1Cc1csc(n1)-c1ccccc1
Cc1nc(cs1)-c1cccc(CN2C(CCCC2=O)c2cccc3OCCOc23)c1
O=C1CCCC(N1Cc1cccc(c1)-c1ccccc1)c1cccc2OCCOc12
COc1cncc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cncc(OC)c1C1CCCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1cncc(OC)c1C1CCCCC(=O)N1Cc1ccc2n(C)c3ccccc3c2c1
COc1cncc(OC)c1C1CCCCC(=O)N1Cc1csc(n1)-c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1csc(Oc2ccccc2)n1
COc1ccc2nc(C)oc2c1C1CCCC(=O)N1Cc1ccc2ccccc2n1
COc1ccc2ncoc2c1C1CCCC(=O)N1Cc1ccc2ccccc2n1
COc1ccc(Cl)c(OC)c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc(Oc2nccs2)cc1
Cc1nc(cs1)-c1cccc(CN2C(CCCC2=O)c2ccccc2-c2ccccc2)c1
O=C1CCCC(N1Cc1cccc(c1)-c1ccccc1)c1ccccc1-c1ccccc1
O=C1CCC(N1Cc1cccc(c1)-c1ccccc1)c1ccccc1-c1ccccc1
Cc1nc(cs1)-c1cccc(CN2C(CCC2=O)c2ccccc2-c2ccccc2)c1
FC(F)(F)Oc1ccc(CN2C(CCC2=O)c2ccccc2-c2ccccc2)cc1
O=C1CCC(N1Cc1csc(n1)-c1ccccc1)c1ccccc1-c1ccccc1
CC1CC(N(Cc2cccc(c2)-c2ccccc2)C1=O)c1ccccc1-c1ccccc1
CC1CC(N(Cc2cccc(c2)-c2csc(C)n2)C1=O)c1ccccc1-c1ccccc1
CC1CC(N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1ccccc1-c1ccccc1
COc1cccc(OC)c1C1CCC(=O)N1Cc1ccc(Oc2nc(C)cs2)cc1
COc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(Cl)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
O[C@@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1cccc2OCCOc12 |o1:1,3|
COc1cc(F)ccc1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1ccccc1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:8,10|
COc1ccccc1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:8,10|
CCOc1ccccc1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
CCOc1ccccc1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(Cl)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cc(F)ccc1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
CCOc1ccccc1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(Cl)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
FC(F)(F)Oc1ccc(CN2[C@@H](C[C@H](Cl)C2=O)c2cccc3OCCOc23)cc1 |o1:11,13|
COc1cc(F)ccc1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(C)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
CCOc1c(F)cccc1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1ccc(F)c(OC)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1ccc2ccccc2c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:12,14|
COc1c(F)ccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1ccc(Cl)c(OC)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1ccc2ccccc2c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:12,14|
COc1ccc2ccccc2c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:12,14|
COc1c(F)ccc(F)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1ccc(Cl)c(OC)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1ccc(Cl)c(OC)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1c(F)ccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1c(F)ccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
FC(F)(F)Oc1ccc(CN2[C@@H](C[C@@H](Cl)C2=O)c2cccc3OCCOc23)cc1 |o1:11,13|
COc1cc(F)ccc1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(F)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(C)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
COc1cccc(C)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:9,11|
CCOc1c(F)cccc1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1ccc(F)c(OC)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
CCOc1c(F)cccc1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1ccc(F)c(OC)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
CCOc1c(F)cccc1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1ccc(F)c(OC)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
CCOc1cccc(F)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cc(F)ccc1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
COc1cccc(OC)c1C1CC(F)(F)C(=O)N1Cc1cccc(c1)-c1ccccc1
CCOc1cccc(OC)c1C1CC(F)(F)C(=O)N1Cc1cccc(c1)-c1ccccc1
CCOc1ccc(F)c(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
CCOc1ccc(F)c(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
CCOc1ccc(F)c(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
CCOc1cc(F)ccc1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cc(F)ccc1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1ccc(F)c(F)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cnc2ccccc2c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2ccccc2n1
COc1ccnc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ncc(C)s1
COc1ccnc(OC)c1C1CC(C)C(=O)N1Cc1csc(n1)-c1ccc(C)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-c1ncc(C)s1
COc1ccnc(OC)c1C1CC(C)C(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1cccc(OC)c1C1CC(F)(F)C(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1ccnc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ccccc1
COc1ccnc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1nc(Cl)cs1
COc1ccnc(OC)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1cccc(OC)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:10,12|
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1cnc2ccccc2c1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc2ccccc2n1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-c1ncc(C)s1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-n1cccn1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc2oc3ccccc3c2c1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1csc(n1)-c1ccc(C)cc1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ncc(C)s1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1nc(Cl)cs1
COc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-c1nc(C)cs1
COc1cccc(OC)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:10,12|
COc1cccc(OC)c1[C@@H]1C[C@@H](F)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:10,12|
COc1cccc(OC)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:10,12|
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1cccc(OC(F)(F)F)c1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)(F)F)c(F)c1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)F)cc1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1cccc(OC(F)F)c1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)F)c(Cl)c1
CCOc1cccc(CN2C(CC(C)C2=O)c2c(F)cccc2OCC)c1
CCCOc1ccc(CN2C(CC(C)C2=O)c2c(F)cccc2OCC)cc1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1cnc2ccccc2c1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc2ccccc2n1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-c1ncc(C)s1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-n1cccn1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc2oc3ccccc3c2c1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1csc(n1)-c1ccc(C)cc1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1ncc(C)s1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1cccc(c1)-c1nc(Cl)cs1
CCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccnc(c1)-c1nc(C)cs1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2n(C)c3ccccc3c2c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cc2ccccc2n1C
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cc2ccccc2[nH]1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cc2cc(F)ccc2n1C
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2n(C)ccc2c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2[nH]ccc2c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2sc(C)nc2c1
CC(C)Oc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1cccc(F)c1[C@@H]1C[C@@H](F)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:9,11|
COc1cccc(F)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:9,11|
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(C)C)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(SC(F)(F)F)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)(F)C(F)F)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)(F)F)c(F)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)F)c(Cl)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)F)cc1
COc1ccc(OC(F)(F)F)cc1CN1C(CC(C)C1=O)c1c(OC)cccc1OC
COc1ccc(CN2C(CC(C)C2=O)c2c(OC)cccc2OC)cc1OC(F)(F)F
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccccc1OC(F)(F)F
COc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:9,11|
CC(C)Oc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:9,11|
CC(C)Oc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1cccc(F)c1C1CC(F)(F)C(=O)N1Cc1ccc2oc3ccccc3c2c1
CC(C)Oc1cccc(F)c1C1CC(F)(F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |o1:9,11|
CC(C)Oc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
CC1CC(N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cccc1OCCF
CCCOc1cccc(F)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1
CC1CC(N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cccc1OCCO
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OCC(F)(F)F)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OCC(F)(F)F)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OCC(F)F)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OCC(F)F)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OCCF)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OCCF)cc1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OC(C)C)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1cccc(OC(F)(F)C(F)F)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc(OC(F)F)c(OC)c1
COc1cccc(OC)c1C1CC(C)C(=O)N1Cc1ccc2sc3ccccc3c2c1
CCOc1cccc(Cl)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)c(F)c1 |o1:10,12|
CCOc1cccc(F)c1C1CC(O)C(=O)N1Cc1ccc(OC(F)(F)F)c(Cl)c1
COc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1cccc(OC(F)(F)F)c1 |o1:9,11|
CCOc1cc(F)cc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
O[C@@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cccc1OCCF |o1:1,3|
CCOc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccccc1OC(F)(F)F |o1:10,12|
CCOc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)c(F)c1 |o1:10,12|
CCOc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)c(F)c1 |o1:10,12|
CCOc1cccc(Cl)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cccc(Cl)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:10,12|
CCOc1cc(F)cc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
CCOc1cc(F)cc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |o1:11,13|
COc1ccc2nc(C)oc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1ccc2nc(C)oc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
CCc1nc2ccc(OC)c(C3CCCC(=O)N3Cc3cccc(c3)-c3csc(C)n3)c2o1
COc1ccc2OCCOc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1ccc2OCCOc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1ncc(C)s1
COc1ccc2ccccc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1ncccn1
COc1ccc2ccccc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1ncc(C)s1
COc1ccc2ccccc2c1C1CCCC(=O)N1Cc1cccc(Oc2ccccc2)c1
COc1ccc2OCOc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
COc1ccc2OCOc2c1C1CCCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
O=C1CCCCC(N1Cc1cccc(c1)-c1nccs1)c1ccccc1-c1ccncc1
O=C1CCCCC(N1Cc1cccc(c1)-c1nccs1)c1ccccc1-c1cncs1
O=C1CCCCC(N1Cc1cccc(c1)-c1nccs1)c1ccccc1-c1cscn1
O=C1CCCCC(N1Cc1cccc(c1)-c1nccs1)c1ccccc1-c1cccnc1
O=C1CCCCC(N1Cc1cccc(c1)-c1nccs1)c1ccccc1-c1ccccc1
COc1ccc2ncoc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1csc(C)n1
O=C1CCCC(N1Cc1cccc(c1)-c1ccccc1)c1ccnn1-c1ccccc1
COc1ccc2OCOc2c1C1CCCC(=O)N1Cc1cccc(c1)-c1ccccc1
COc1ccc2OCOc2c1C1CCCC(=O)N1Cc1cccc(Oc2ccccc2)c1
COc1ccc2OCOc2c1C1CCCC(=O)N1Cc1csc(n1)-c1ccccc1
COc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1cccc(OC(F)(F)F)c1 |o1:9,11|
CCOc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)c(Cl)c1 |o1:10,12|
CCOc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)c(Cl)c1 |o1:10,12|
COc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1cccc(OC(F)(F)F)c1 |o1:9,11|
Cc1ccc(c(c1)C(=O)N1CCOC1Cn1ccc(n1)-c1ccc(F)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC1Cn1cc(cn1)-c1ccc(F)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cn1ccc(n1)-c1ccc(F)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cn1cc(cn1)-c1ccc(F)cn1)-n1nccn1
C[C@H]1CN([C@H](Cn2cc(cn2)-c2ccc(F)cn2)O1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CN([C@H](Cn2cc(cn2)-c2ccc(F)cn2)O1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CO[C@@H](Cn2ccc(n2)-c2ccc(F)cn2)N1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CO[C@@H](Cn2cc(cn2)-c2ccc(F)cn2)N1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@H]1CO[C@@H](Cn2ccc(n2)-c2ccc(F)cn2)N1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@H]1CO[C@@H](Cn2cc(cn2)-c2ccc(F)cn2)N1C(=O)c1cc(C)ccc1-n1nccn1 |r|
Fc1ccc(nc1)-c1ccn(CC2OCCN2C(=O)c2ccccc2-n2nccn2)n1 |w:12.12|
Fc1ccc(nc1)-c1ccn(CC2OCCN2C(=O)c2cc(F)ccc2-n2nccn2)n1 |w:12.12|
Cc1ccc(c(c1)C(=O)N1CCOC1Cn1ccc(n1)-c1ccc(F)cn1)-c1ncccn1 |w:13.15|
Fc1ccc(nc1)-c1ccn(CC2OCCN2C(=O)c2ccccc2-c2ncccn2)n1 |w:12.12|
Fc1ccc(nc1)-c1ccn(CC2OCCN2C(=O)c2cc(F)ccc2-c2ncccn2)n1 |w:12.12|
Cc1ccc(c(c1)C(=O)N1CCOC1Cn1ccc(n1)-c1ccc(F)cc1)-n1nccn1 |w:13.15|
Fc1ccc(cc1)-c1ccn(CC2OCCN2C(=O)c2ccccc2-n2nccn2)n1 |w:12.12|
Fc1ccc(cc1)-c1ccn(CC2OCCN2C(=O)c2cc(F)ccc2-n2nccn2)n1 |w:12.12|
Cc1ccc(c(c1)C(=O)N1CCOC1Cn1ccc(n1)-c1ccc(F)cc1)-c1ncccn1 |w:13.15|
Fc1ccc(cc1)-c1ccn(CC2OCCN2C(=O)c2cc(F)ccc2-c2ncccn2)n1 |w:12.12|
Cc1ccc(c(n1)C(=O)N1CCOC1Cn1cc(cn1)-c1ccc(F)cc1)-n1nccn1 |w:13.15|
Cc1ccc(c(c1)C(=O)N1CCOC1Cn1cc(cn1)-c1ccc(F)cc1)-c1ncccn1 |w:13.15|
Fc1ccc(cc1)-c1cnn(CC2OCCN2C(=O)c2cc(F)ccc2-c2ncccn2)c1 |w:12.12|
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCCOC1Cc1noc(n1)-c1ccc(F)cn1 |w:20.23|
Cc1ccc(c(n1)C(=O)N1CCOC1Cn1ccc(n1)-c1ccc(F)cc1)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCCOC1Cn1ccc(n1)-c1ccc(F)cc1)-n1nccn1
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CCCOC1Cn1ccc(n1)-c1ccc(F)cc1
Fc1ccc(nc1)-c1ccn(CC2OCCCN2C(=O)c2cc(F)ccc2-n2nccn2)n1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cn1ccc(n1)-c1ccc(F)cn1)-c1ncccn1
Cc1ccc(c(n1)C(=O)N1CCCOC1Cn1cc(cn1)-c1ccc(F)cc1)-n1nccn1
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1CCCOC1Cn1cc(cn1)-c1ccc(F)cc1
Fc1ccc(nc1)-c1ccn(CC2OCCCN2C(=O)c2cc(F)ccc2-c2ncccn2)n1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cn1cc(cn1)-c1ccc(F)cc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cc1noc(n1)-c1ccc(F)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cc1noc(n1)-c1ccc(F)cc1)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCCOC1Cc1noc(n1)-c1ccc(F)cc1)-n1nccn1
C[C@H]1CCO[C@@H](Cn2cc(cn2)-c2ccc(F)cn2)N1C(=O)c1cc(C)ccc1-n1nccn1 |r|
CC1COC(Cn2cc(cn2)-c2ccc(F)cn2)N(C1)C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cn1ccc(n1)-c1ccc(F)cc1)-c1ncccn1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cc1cnn(c1)-c1ccc(F)cn1)-c1ncccn1 |w:14.16|
Cc1ccc(c(c1)C(=O)N1CCCOC1Cn1cc(cn1)-c1ccc(F)cc1)-c1ncccn1
Fc1ccc(nc1)-n1cc(CC2OCCCN2C(=O)c2cc(F)ccc2-c2ncccn2)cn1
Cc1ccc(c(c1)C(=O)N1CCOC1Cc1ccn(n1)-c1ccc(F)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCOC1Cc1cnn(c1)-c1ccc(F)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCOC1Cc1cnn(c1)-c1ccc(F)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(F)c1C)-n1nccn1
Cc1ccc(cc1)-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc(c1)-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
CCCOc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1c(C)cccc1F)-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1cc(C)ccc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1cc(F)cc(F)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1ccc(F)c(F)c1)-n1nccn1
Cc1cccc(c1)-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1Cl)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(F)c2OC)c(cc1C)-n1nccn1
Cc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@H]1CCN1C(=O)c1ccc(C)cc1-n1nccn1
Cc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(cc1C)-n1nccn1
Cc1ccc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(c1)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1F)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1F)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(cc1F)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(F)c2OC)c(cc1F)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1 |r|
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(cc1C)-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(OC)c(F)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1cccnc1OC1CCC1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1)-n1nccn1
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(s1)-c1ccccc1F
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(s1)-c1cccc(C)c1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(s1)-c1ccccc1
CN(C)c1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(s1)-c1ccccc1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ncsc1-c1ccccc1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ncsc1-c1cccc(Cl)c1
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(s1)-c1ccc(C)cc1
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(s1)-c1ccccc1C
Cc1cccc(c1C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
FC(F)(F)Oc1ccc(c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
Cc1cccc(c1)-c1ocnc1C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccccc1-n1nccn1
Cc1cccc(c1)-c1scnc1C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(o1)-c1cccc(C)c1
Cc1onc(c1C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-c1ccccc1Cl
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccccc1-c1ccccc1
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1ccccc1F
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1cccc(C)c1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1ccccc1
CN(C)c1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1ccccc1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ncsc1-c1ccccc1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ncsc1-c1cccc(Cl)c1
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1ccc(C)cc1
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1ccccc1C
Cc1cccc(c1C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
Cc1cccc(c1)-c1ocnc1C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccccc1-n1nccn1
Cc1cccc(c1)-c1scnc1C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
Cc1nc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(o1)-c1cccc(C)c1
Cc1onc(c1C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-c1ccccc1Cl
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccccc1-c1ccccc1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1Cl)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1Cl)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccc(Cl)cc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1ccc(C(=O)N2CC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(c1)-n1nccn1
Cc1ccc(C(=O)N2CC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(Cl)ccc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1noc(n1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(cc1F)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(F)c2OC)c(cc1C)-n1nccn1
Cc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(F)c2C)c(cc1C)-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1noc(n1)-c1cccc(F)c1C)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(cc1Cl)-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CC[C@H]1c1noc(n1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(F)c2C)c(cc1Cl)-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
Cc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1noc(n1)-c1cccc(Cl)c1C)-n1nccn1
Cc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1Cl)-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CC[C@H]1c1noc(n1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(c1)-n1nccn1
Cc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1ccc(cc1-n1nccn1)C(F)(F)F
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(Cl)c2OC)c(cc1C)-n1nccn1 |r|
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(Cl)c2OC)c(cc1Cl)-n1nccn1
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CC[C@H]1c1noc(n1)-c1cccc(Cl)c1C
Cc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1cc(F)ccc1-c1ncccn1
COc1cc(C(=O)N2CC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1C)-c1ncccn1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CC[C@H]1c1noc(n1)-c1cccc(Cl)c1C
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nnc([nH]1)-c1ccccc1)-n1nccn1
Cc1ccc(C(=O)N2CC[C@H]2c2nnc([nH]2)-c2ccccc2)c(c1)-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCN1C(=O)c1ccc(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nnc([nH]1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1c(Cl)cccc1-c1nnc([nH]1)[C@@H]1CCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(C(=O)N2CC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
Cc1cc(C(=O)N2CC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1cc(C(=O)N2CC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(cc1Cl)-n1nccn1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCN1C(=O)c1ccc(Cl)cc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCN1C(=O)c1ccc(cc1-n1nccn1)C(F)(F)F
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1[C@H]2CC[C@@H]1[C@@H](COc1ccccn1)C2 |r,TLB:21:20:18.17:15|
Cc1ccc(-c2ncccn2)c(n1)C(=O)N1[C@@H]2CC[C@H]1[C@H](COc1ccccn1)C2 |r,TLB:21:20:18.17:15|
Cc1ccc(c(n1)C(=O)N1[C@@H]2CC[C@H]1[C@H](COc1ccccn1)C2)-n1nccn1 |r,TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1[C@H]2CC[C@@H]1[C@@H](COc1ccccn1)C2)-n1nccn1 |r,TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1[C@H]2CC[C@@H]1[C@H](COc1ccccn1)C2)-n1nccn1 |r,TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1[C@@H]2CC[C@H]1[C@H](COc1ccc(F)cn1)C2)-n1nccn1 |r,TLB:15:14:12.11:9|
Cc1ccc(c(n1)C(=O)N1[C@H]2CC[C@@H]1[C@@H](COc1ccc(F)cn1)C2)-n1nccn1 |r,TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1[C@@H]2CC[C@H]1[C@H](COc1ccc(F)cn1)C2)-n1nccn1 |r,TLB:15:14:12.11:9|
Cc1ccc(c(c1)C(=O)N1[C@H]2CC[C@@H]1[C@@H](COc1ccc(F)cn1)C2)-n1nccn1 |r,TLB:15:14:12.11:9|
Cn1cc(c(n1)C(=O)N1[C@@H]2CC[C@H]1[C@H](COc1ccccn1)C2)-c1ccccc1 |r,TLB:14:13:11.10:8|
Cn1cc(C(=O)N2[C@@H]3CC[C@H]2[C@H](COc2ccccn2)C3)c(n1)-c1ccccc1 |r,TLB:12:11:9.8:6|
Cc1ccc(C2CCNCC2)c(n1)C(=O)N1C2CCC1C(COc1ccccn1)C2 |TLB:21:20:18.17:15|
CCOc1ncc2ccccc2c1C(=O)N1[C@@H]2CC[C@H]1[C@H](COc1ccccn1)C2 |r,TLB:21:20:18.17:15|
FC(F)(F)c1cnc(N[C@@H]2C[C@H]3CC[C@@H]2N3C(=O)c2ccccc2-n2nccn2)cn1 |r,THB:8:9:13.12:15|
FC(F)(F)c1cnc(N[C@H]2C[C@@H]3CC[C@H]2N3C(=O)c2ccccc2-n2nccn2)cn1 |r,THB:8:9:13.12:15|
Fc1cccc(C(=O)N2[C@@H]3CC[C@H]2[C@@H](C3)Nc2ccc(cn2)C(F)(F)F)c1-c1ncccn1 |r,TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2[C@@H]3CC[C@H]2[C@@H](C3)Oc2ncc(cn2)C(F)(F)F)c1-c1ncccn1 |r,TLB:15:13:11.10:8|
Fc1cccc(C(=O)N2[C@H]3CCC2[C@H](C3)Oc2ncc(cn2)C(F)(F)F)c1-c1ncccn1 |r,THB:15:13:11.10:8|
Fc1ccc(OC[C@@H]2C[C@H]3CC[C@@H]2N3C(=O)c2ccccc2-c2cccs2)nc1 |r,THB:6:7:11.10:13|
Fc1ccc(OC[C@H]2C[C@@H]3CC[C@H]2N3C(=O)c2ccccc2-c2cccs2)nc1 |r,THB:6:7:11.10:13|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@H]1Nc1cnc2ccccc2n1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc2ccccc2n1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccccc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@H]1Nc1nc2ccccc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2cc(Cl)ccc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@H]1Nc1nc2ccccc2o1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1N(C)c1nc2ccc(F)cc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccccc2o1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(Cl)cc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@@H]1CCC[C@H]1Nc1nc2ccccc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@@H]1CCC[C@H]1Nc1nc2ccccc2o1 |r|
COc1cccc(OC)c1C(=O)N[C@@H]1CCC[C@@H]1Nc1nc2ccc(Cl)cc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@@H]1CCC[C@H]1Nc1nc2ccc(Cl)cc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@H]1Nc1nc2ccc(Cl)cc2s1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)-n1nccn1 |r|
CCOc1cccc(OCC)c1C(=O)N[C@@H]1CCC[C@@H]1Nc1nc2ccccc2o1 |r|
CCOc1cccc(OCC)c1C(=O)N[C@H]1CCC[C@H]1Nc1nc2ccccc2o1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccccc2s1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ccc2ccccc2n1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N[C@@H]1CCC[C@@H]1Nc1cnc2ccccc2n1)-n1nccn1 |r|
COc1cccc(OC)c1C(=O)NC1CN(CC1Nc1nc2ccc(Cl)cc2s1)C(=O)OCc1ccccc1
CCOC(=O)N1CC(NC(=O)c2c(OC)cccc2OC)C(C1)Nc1nc2ccc(Cl)cc2s1
COc1cccc(OC)c1C(=O)NC1COCC1Nc1nc2ccc(Cl)cc2s1
COc1cccc(OC)c1C(=O)N[C@@H]1C[C@@H](O)C[C@@H]1Nc1nc2ccc(Cl)cc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@@H]1CC(F)C[C@@H]1Nc1nc2ccc(Cl)cc2s1 |r|
Cc1ccc(c(c1)C(=O)NC1CCCC1Cc1ccc2ccccc2n1)-n1nccn1
CCOc1ccc(C)cc1C(=O)NC1CCCC1Cc1ccc2ccccc2n1
COc1cccc(OC)c1C(=O)NC1CCCC1Cc1ccc2ccccc2n1
CCOc1cccc(OCC)c1C(=O)NC1CCCC1Cc1ccc2ccccc2n1
COc1cccc(OC)c1C(=O)NC1CCCC1Cc1nc2ccc(Cl)cc2s1
Cc1ccc(c(c1)C(=O)NC1CCCC1Cc1nc2ccc(Cl)cc2s1)-n1nccn1
COc1cccc(OC)c1C(=O)N(C)[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3cccn3)sc2c1 |r|
Fc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)-n1nccn1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3Cl)sc2c1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)-n1ccnn1 |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-c3ncccn3)sc2c1 |r|
COc1ccc(OC)c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc(-c2ncccn2)c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3ccnc3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3cncn3)sc2c1 |r|
Fc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)-n1ccnn1 |r|
COc1cccc(F)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3c(F)cccc3F)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3F)sc2c1 |r|
CCOc1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Cc1ccccc1C(=O)N[C@@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@H]3NC(=O)c3c(Cl)cccc3Cl)sc2c1 |r|
COc1ccc(F)cc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1c(F)cccc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
FC(F)Oc1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
COc1cccc(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Cc1cccc(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3C3CC3)[nH]c2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)[nH]c2c1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Nc1ncc2ccccc2n1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N[C@H]1CCC[C@@H]1Cc1ccc2ccccc2n1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N[C@@H]1CCC[C@H]1Cc1ccc2ccccc2n1)-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)NC1CCCC1Cc1cnc2ccccc2n1)-n1nccn1
COc1cccc(OC)c1C(=O)NC1COCC1Nc1nc2ccc(F)cc2s1
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2o1 |r|
COc1ccc(C)cc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Cc1cccc(C)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3c(F)cccc3-n3nccn3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3c(F)cccc3Cl)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3c(Cl)cccc3-n3nccn3)sc2c1 |r|
Cc1nnc(o1)-c1ccccc1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3ccnn3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3cc(Cl)ccc3-n3cccn3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)sc2c1 |r|
CN([C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(=O)c1c(F)cccc1F |r|
COc1ccccc1C(=O)N(C)[C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1 |r|
CN([C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(=O)c1ccccc1Cl |r|
CN([C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(=O)c1ccccc1-n1cccn1 |r|
CN([C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(=O)c1ccccc1-n1nccn1 |r|
CN([C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
CN([C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(=O)c1ccccc1-c1ncccn1 |r|
CN([C@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2s1)C(=O)c1ccccc1-c1nc(C)no1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2cc(F)ccc2s1 |r|
COc1cccc(OC)c1C(=O)N[C@H]1CCC[C@@H]1Nc1nc2cc(F)ccc2o1 |r|
O=C(N[C@H]1CCC[C@@H]1Nc1nc2ccccc2o1)c1ccccc1-n1nccn1 |r|
Fc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)oc2c1 |r|
Fc1ccc2oc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)nc2c1 |r|
Clc1ccc2sc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)nc2c1 |r|
O=C(N[C@H]1CCC[C@@H]1Nc1nc2ccccc2s1)c1ccccc1-n1nccn1 |r|
Clc1ccc2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)sc2c1 |r|
Fc1ccc2sc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)nc2c1 |r|
Fc1cc(F)c2nc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)sc2c1 |r|
Fc1cccc2sc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)nc12 |r|
O=C(N[C@H]1CCC[C@@H]1Nc1nc2cccnc2s1)c1ccccc1-n1nccn1 |r|
Clc1cncc2sc(N[C@H]3CCC[C@@H]3NC(=O)c3ccccc3-n3nccn3)nc12 |r|
O=C(N[C@@H]1CCC[C@@H]1Nc1nc2ccncc2s1)c1ccccc1-n1nccn1 |r|
Cc1noc(n1)-c1ccccc1C(=O)N[C@@H]1CCC[C@@H]1Nc1nc2ccc(F)cc2o1 |r|
Fc1ccc2nc(NC3COCC3NC(=O)c3ccccc3-n3nccn3)sc2c1
Cc1ccc(c(c1)C(=O)NC1COCC1Cc1nc2ccccc2s1)-n1nccn1
Fc1ccc2nc(N[C@@H]3CC(F)(F)C[C@@H]3NC(=O)c3ccccc3-n3nccn3)sc2c1 |r|
Fc1ccc2nc(N[C@H]3CC(F)(F)C[C@H]3NC(=O)c3ccccc3-n3nccn3)sc2c1 |r|
FC1(F)C[C@H](NC(=O)c2ccccc2-n2nccn2)[C@@H](C1)Nc1nc2ccc(Cl)cc2s1 |r|
FC1(F)C[C@@H](NC(=O)c2ccccc2-n2nccn2)[C@H](C1)Nc1nc2ccc(Cl)cc2s1 |r|
CC1(CCCC1NC(=O)c1ccccc1-n1nccn1)Nc1nc2ccc(F)cc2s1
CC1(CCCC1NC(=O)c1ccccc1-n1nccn1)Nc1nc2ccc(Cl)cc2s1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1)-n1nccn1
Cc1cccc(c1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc(c1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccnc1)-n1nccn1
Cc1ccc(cc1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1C1CC1)-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cc(F)cc(F)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(F)c1F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cc(C)cc(C)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cc(C)cc(C)n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(C)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(F)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1c[nH]c2ccccc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccc2OC(F)(F)Oc2c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccc(F)c(F)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1Cl)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccc2OCOc2c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1c(C)cccc1Cl)-n1nccn1
CCc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(F)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(C)c1Cl)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccnc1Cl)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1C(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1nccnc1Cl)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1O)-n1nccn1
COc1cc(ccn1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)F)-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc(-c2noc(n2)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c1F
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1c(C)ccnc1Cl)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1c(C)cncc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc2OCCOc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc2[nH]ccc12)-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc2[nH]cc(-c3noc(n3)[C@@H]3CCCN3C(=O)c3cc(C)ccc3-n3nccn3)c2c1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(OC(F)F)c1)-n1nccn1
COCc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc2cc[nH]c12)-n1nccn1
COc1cc(OC)cc(c1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccnc1OC1CCC1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccnc1OC1CCCC1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1c[nH]c2ncccc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cn(C)c2ncccc12)-n1nccn1
CCc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(c1C)C(F)(F)F)-n1nccn1
CCOc1cnccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cn(C)c2ccccc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cnccc1C)-n1nccn1
COc1cccc(-c2noc(n2)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c1OC
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cnn(C)c1)-n1nccn1
CCc1cnc(cc1C)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cc(C)c(C)cn1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccc(C)c(C)n1)-n1nccn1
COc1cc(O)ccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cc(C)nc(C)c1)-n1nccn1
COc1cc(cc(C)n1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CC(C)Cc1cc(C)cc(n1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccnc(C)c1)-n1nccn1
COc1ccc(F)c(-c2noc(n2)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c1F
COc1cccc(-c2noc(n2)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c1Cl
CC(C)Oc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc(F)c1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccnc(Cl)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc2n(C)ccc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccnc2[nH]ccc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1c(C)cccc1F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc2ccn(C)c12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccnc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1c[nH]c2cccc(C)c12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccc(C)c(C)c1)-n1nccn1
Cc1ccc(-c2noc(n2)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c(C)c1
COc1ccc(cc1OC)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ncccc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cc(C)ccc1C)-n1nccn1
CC(=O)n1cc(-c2noc(n2)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c2ccccc12
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccnc1OC(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1CCO)-n1nccn1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1cccn1
Cc1ccc(-c2ccccn2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1nc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(o1)-c1cccc(C)c1
Cc1cccc(c1)-c1ocnc1C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ncsc1-c1cccc(Cl)c1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(c1)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
Cc1cccc(c1C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
COc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1[nH]cnc1-c1ccccc1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1C)-n1cccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1cccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccnc1-c1ccccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1cccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)c(F)cc1-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(F)cc1-n1cccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(F)cc1-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-n1cccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1C)-n1cccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-c1ccn[nH]1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-c1ccn[nH]1
COc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(c1)-n1nccn1
Cc1cc(C)c(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-c1ncco1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(cc1-n1nccn1)C(F)(F)F
Cc1nc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1cccc(F)c1
Cc1nc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1ccccc1F
Cc1nc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1ccc(F)cc1
Cc1nc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(s1)-c1cccc(C)c1
Cc1ncc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(n1)-c1cccc(Cl)c1
COc1cccc(c1)-c1nccnc1C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(c1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1F)-n1nccn1
Cc1ccc(-c2ncco2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1cc(F)cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1OC)-n1nccn1
Cc1noc(n1)-c1ccccc1C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-c1ccccc1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1cccn1
Cc1ccc(-c2ccccn2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
Cc1nc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(o1)-c1cccc(C)c1
Cc1cccc(c1)-c1ocnc1C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ncsc1-c1cccc(Cl)c1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c1F)-n1nccn1
Cc1ccc(c(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c1F)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F
Cc1cccc(c1C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
FC(F)(F)Oc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1[nH]cnc1-c1ccccc1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
Fc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1cccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccnc1-c1ccccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1cccn1
Fc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1F)-n1nccn1
Fc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(c1)-n1cccn1
Fc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
Fc1cccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c1-n1cccn1
Fc1cccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c1-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1cccn1
Fc1ccc(-c2ccn[nH]2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
Fc1cccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c1-c1ccn[nH]1
COc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
Cc1cc(C)c(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-c1ncco1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(cc1-n1nccn1)C(F)(F)F
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1F)-n1nccn1
Cc1ccc(-c2ncco2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F
Cc1cc(F)cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1OC)-n1nccn1
FC(F)(F)c1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
FC(F)(F)c1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2C(F)(F)F)c(c1)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2C(F)(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2C(F)(F)F)c(cc1C)-n1nccn1
Fc1cccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2C(F)(F)F)c1-c1ccn[nH]1
Cc1ccc(-c2ccccn2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1C(F)(F)F
FC(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
FC(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)F)c(c1)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)F)c(cc1C)-n1nccn1
FC(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-c1ccn[nH]1
Cc1ccc(-c2ccccn2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)F
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)cc(C)c1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(C)c1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(F)c1OC)-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2OC)c(cc1C)-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-c1ccn[nH]1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-c1ccccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(cc1-n1nccn1)C(F)(F)F
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2OC)c(cc1F)-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)cc(C)c1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2OC)c(cc1OC)-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)cc(C)c1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-c1ccn[nH]1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-c1ccccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(C)c1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)ccc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(cc1-n1nccn1)C(F)(F)F
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(F)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-c1ncco1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)cc(C)c1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(OC)cc1-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC)c(cc1C)-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC)-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-c1ccn[nH]1
COc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1nccn1
Clc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1Cl)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2Cl)c(c1)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2Cl)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2Cl)c(cc1C)-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1Cl)-n1nccn1
Fc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1Cl)-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1Cl)-n1nccn1
Clc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
Cc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
Cc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(c1)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(cc1C)-n1nccn1
COc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(F)c1C)-n1nccn1
Cc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
Cc1cccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2C)c1-n1nccn1
Cc1ccc(c(n1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(F)c1C)-n1nccn1
Cc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-c1ccn[nH]1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(F)c1-c1ccn[nH]1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1nc(C)ccc1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)ccc1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(C)c1-n1nccn1
CCOc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(F)ccc1-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(c(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c1F)-n1nccn1
Cc1ccc(c(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c1F)-n1nccn1
Cc1noc(n1)-c1ccccc1C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-c1ccccc1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1C)-c1ncccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(OC(F)(F)F)c1)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(c1C)-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(C)c(C)c1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(C)c(C)c1-n1nccn1
Cc1ccc(-c2ncccn2)c(c1)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
Cc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(ccc1-n1nccn1)C#N
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(Cl)c2C)c(cc1Cl)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1Cl)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2OC)c(cc1Cl)-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2ccccc2OC(F)(F)F)c(cc1C)-c1ncccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2OC)c(cc1C)-c1ncccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-c1ncccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(OC)c(F)cc1-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nc(no2)-c2cccc(F)c2C)c(cc1Cl)-n1nccn1
Cc1c(Cl)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(Cl)c1-n1nccn1
COc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(Cl)c1-n1nccn1
FC(F)(F)Oc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccc(Cl)c1-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
CCOc1c(F)cccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
CCOc1ncccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
Cc1cccc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cccc2CCOc12)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
CCOc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(F)c2C)c(cc1C)-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1n[nH]c2ccccc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cnc2sccn12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cccc(n1)C(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cc(ccn1)C(F)(F)F)-n1nccn1
COc1cc(Cl)cc(n1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cc(Cl)cc(C)n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cccc(Cl)c1C)-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1F)-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(F)cc1-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)ccc1-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(F)cc1-n1nccn1
Cc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
COc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cccc(F)c1C)-n1nccn1
COc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(F)c2C)c(c1)-n1nccn1
COc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(F)c2C)c(cc1C)-n1nccn1
COc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(F)c2OC)c(cc1C)-n1nccn1
Cc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(Cl)c2OC)c(cc1Cl)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(Cl)c2OC)c(cc1C)-n1nccn1
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cc(C)ccc2OC)c(cc1Cl)-n1nccn1
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cc(C)cc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
COc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(OC)c2C)c(cc1Cl)-n1nccn1
COc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2cc(C)c(C)cc2-n2nccn2)c1C
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(OC)c2C)c(cc1C)-n1nccn1
COc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2cc(C)ccc2-n2nccn2)c1C
COc1c(Cl)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2cc(Cl)ccc2-n2nccn2)c1C
COc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2ccc(Cl)cc2-n2nccn2)c1C
COc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cccc(Cl)c1-n1nccn1
COc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2ccc(C)cc2-n2nccn2)c1C
Cc1cc(c(cc1Cl)C(=O)N1CCC[C@H]1c1noc(n1)-c1ccccc1OC(F)(F)F)-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(Cl)c2C)c(cc1Cl)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(F)c2OC)c(cc1Cl)-n1nccn1
CCOc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CCC[C@H]1c1noc(n1)-c1cccc(Cl)c1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(F)c2C)c(cc1F)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(F)c2OC)c(cc1F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2ccccc2OC(F)(F)F)c(cc1Cl)-n1nccn1
FC(F)(F)Oc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1c(F)cccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
CCOc1ncccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
COc1ccc(C)cc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
COc1cc(C)cc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1ccc(C)cc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cc(C)cc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
COc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cc(C)ccc2OC)c(cc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cccc(C)c1C)-n1nccn1
CCc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1noc(n1)-c1cc(C)ccc1C)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(C)c2C)c(c1)-n1nccn1
CCc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
Cc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
Cc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2cc(Cl)ccc2-n2nccn2)c1C
CCc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2ccc(Cl)cc2-n2nccn2)c1C
CCc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1cccc(-c2nc(no2)[C@@H]2CCCN2C(=O)c2cc(C)c(C)cc2-n2nccn2)c1C
CCc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
Cc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(C)c2C)c(cc1C)-n1nccn1
CCc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cc(C)ccc2C)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cccc(C)c2C)c(cc1Cl)-n1nccn1
CCc1ccccc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2noc(n2)-c2cc(C)ccc2C)c(cc1Cl)-n1nccn1
COc1cc(C)cc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc(C)cc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cc(C)cc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1ccc(C)cc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1cc(C)cc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1ccc(C)cc1-c1nc(no1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
COc1cc(C)cc(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
COc1ccc(C)c(c1)-c1nc(no1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(no1)-c1ccccc1)-n1nccn1
Cc1nc(C(=O)N2CCC[C@H]2c2cc(no2)-c2ccccc2)c(s1)-c1cccc(Cl)c1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(no1)-c1cccc(C)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(no1)-c1cc(C)cc(C)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(no1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1ncccc1-c1cc(on1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CC(C)Oc1ncccc1-c1cc(on1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1cc(on1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1c(F)cccc1-c1cc(on1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(on1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(on1)-c1cccc(Cl)c1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2cc(on2)-c2ccccc2)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2cc(on2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(on1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2cc(on2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2cc(on2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2cc(on2)-c2ccccc2OC(F)(F)F)c(cc1Cl)-n1nccn1
Cc1cccc(c1)-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(o1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(o1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(o1)-c1ccccc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(o1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1nc(C(=O)N2CCC[C@H]2c2nnc(o2)-c2ccccc2OC(F)(F)F)c(s1)-c1cccc(F)c1
Cc1nc(C(=O)N2CCC[C@H]2c2nnc(o2)-c2ccccc2OC(F)(F)F)c(s1)-c1ccccc1F
COc1cc(C(=O)N2CCC[C@H]2c2nnc(o2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc(o2)-c2cccc(Cl)c2C)c(cc1Cl)-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nnc(o2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
COc1c(F)cccc1-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1c(F)cccc1-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(o1)-c1cc(C)cc(C)c1)-n1nccn1
CCc1ccccc1-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(o1)-c1cccc(F)c1C)-n1nccn1
CCOc1ccccc1-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(o1)-c1cccc(Cl)c1)-n1nccn1
COc1cccc(c1)-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc(cc1)-c1nnc(o1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc(s1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(co1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc(co1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncc(o1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncc(o1)-c1ccccc1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1ccccc1)-n1nccn1
COc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
COc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC)c(cc1Cl)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC)c(cc1C)-n1nccn1
COc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
COc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
COc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2cccc(F)c2OC)c(cc1Cl)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2cccc(F)c2OC)c(cc1C)-n1nccn1
COc1c(F)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
COc1c(F)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
COc1c(F)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
COc1c(F)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(OC)c(Cl)cc1-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(OC)c(C)cc1-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ncsc1-c1ccccc1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ncoc1-c1ccccc1
Cc1cccc(c1)-c1scnc1C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F
Cc1cccc(c1)-c1ocnc1C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(Cl)c(C)cc1-n1nccn1
COc1c(Cl)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1c(Cl)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2cccc(Cl)c2OC)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2cccc(Cl)c2OC)c(cc1Cl)-n1nccn1
COc1c(Cl)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)c(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1cccc(F)c1C)-n1nccn1
CCOc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCOc1ncccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1c(F)cccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccccc1-n1nccn1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1nc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(o1)-c1cccc(C)c1
Cc1nc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(s1)-c1ccccc1
Cc1nc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(s1)-c1cccc(C)c1
FC(F)(F)Oc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1ccccc1-c1ccccc1
COc1cc(C(=O)N2CCC[C@H]2c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(cc1Cl)-n1nccn1
Cc1cccc(c1C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nnc([nH]1)-c1cc(C)cc(C)c1)-n1nccn1
CCc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1cccc(c1)-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccc(cc1)-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
CCCOc1ccccc1-c1nnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
COc1ccccc1-c1cnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2ncc([nH]2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
CCOc1ccccc1-c1cnc([nH]1)[C@@H]1CCCN1C(=O)c1ccc(C)cc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cnc([nH]1)-c1ccccc1)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2cnc([nH]2)-c2ccccc2)c(c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cnc([nH]1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2cnc([nH]2)-c2cccc(Cl)c2C)c(c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncc([nH]1)-c1cccc(Cl)c1)-n1nccn1
COc1cccc(c1)-c1cnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncc([nH]1)-c1cccc(Cl)c1C)-n1nccn1
CCOc1ccccc1-c1cnc([nH]1)[C@@H]1CCCN1C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncc([nH]1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncc([nH]1)-c1ccccc1C(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(n[nH]1)-c1ccccc1)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2cc(n[nH]2)-c2cccc(Cl)c2C)c(c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(n[nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@H]2c2cc(n[nH]2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cc(n[nH]1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1ncn(n1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1cn(nn1)-c1ccccc1)-n1nccn1
C[C@]1(CCCN1C(=O)c1ccccc1-n1nccn1)c1nc(no1)-c1ccccc1
C[C@]1(CCCN1C(=O)c1ncsc1-c1cccc(Cl)c1)c1nc(no1)-c1ccccc1
Cc1cccc(c1)-c1ocnc1C(=O)N1CCC[C@@]1(C)c1nc(no1)-c1ccccc1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc(no1)-c1ccccc1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nc(no1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nnc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(c1)-n1nccn1
C[C@]1(CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1)c1nnc([nH]1)-c1ccccc1OC(F)(F)F
Cc1cc(c(cc1Cl)C(=O)N1CCC[C@@]1(C)c1nnc([nH]1)-c1ccccc1OC(F)(F)F)-n1nccn1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(cc1C)-n1nccn1
C[C@]1(CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1)c1nnc([nH]1)-c1ccccc1OC(F)(F)F
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nnc([nH]2)-c2ccccc2OC(F)(F)F)c(c1)-c1ccccc1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nnc([nH]1)-c1ccccc1OC(F)(F)F
Cc1ccc(c(c1)C(=O)N1CCC[C@@]1(C)c1nnc([nH]1)-c1cccc(Cl)c1C)-n1nccn1
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nnc([nH]2)-c2cccc(Cl)c2C)c(c1)-n1nccn1
Cc1cc(c(cc1Cl)C(=O)N1CCC[C@@]1(C)c1nnc([nH]1)-c1cccc(Cl)c1C)-n1nccn1
Cc1cc(C(=O)N2CCC[C@@]2(C)c2nnc([nH]2)-c2cccc(Cl)c2C)c(cc1C)-n1nccn1
Cc1c(Cl)cccc1-c1nnc([nH]1)[C@]1(C)CCCN1C(=O)c1cc(Cl)ccc1-n1nccn1
Cc1c(Cl)cccc1-c1nnc([nH]1)[C@]1(C)CCCN1C(=O)c1ccc(Cl)cc1-n1nccn1
Cc1ccc(-c2ccccc2)c(c1)C(=O)N1CCC[C@@]1(C)c1nnc([nH]1)-c1cccc(Cl)c1C
Cc1ccc(C(=O)N2CCC[C@@]2(C)c2nnc([nH]2)-c2cccc(Cl)c2C)c(c1)-c1ccccc1
O=C(N1CCC[C@H]1c1nc(no1)-c1ccccc1)c1cccs1
Clc1cccc(c1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccs1
Cc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1cccs1
O=C(N1CCC[C@H]1c1nc(no1)-c1ccccc1)c1ccoc1
Clc1cccc(c1)-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccoc1
Cc1ccccc1-c1noc(n1)[C@@H]1CCCN1C(=O)c1ccoc1
Cc1onc(c1C(=O)N1CCC[C@H]1c1nc(no1)-c1cccc(Cl)c1C)-c1ccccc1Cl
Cc1onc(c1C(=O)N1CCC[C@H]1c1noc(n1)-c1cccc(Cl)c1C)-c1ccccc1Cl
Cc1onc(c1C(=O)N1CCC[C@H]1c1nnc(o1)-c1cccc(Cl)c1C)-c1ccccc1Cl
Cc1onc(c1C(=O)N1CCC[C@H]1c1nc(no1)-c1ccccc1OC(F)(F)F)-c1ccccc1Cl
CN([C@@H]1CC[C@]2([C@H]3Cc4ccc(c5c4[C@]2([C@H]1O5)CCN3CC6CC6)O)O)C(=O)/C=C/c7ccoc7
COc1ccc2C[C@H]3N(CC[C@@]45[C@@H](Oc1c24)[C@@H](CC[C@@]35O)N(C)Cc1ccccc1)C(=O)OC(C)(C)C |r|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1C)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(C)c1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(C)cc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1C(F)(F)F)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1[N+]([O-])=O)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1C#N)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(F)c1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(Cl)c1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1Br)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(Br)c1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1c(C)cc(C)cc1C)ccc3OC |r,THB:29:9:5.4.6:13|
COc1ccc2C[C@H]3N(CC[C@@]45[C@@H](Oc1c24)[C@@H](CC[C@@]35O)N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc2cccnc12 |r,TLB:18:19:6.5.15:8.10.9,20:19:6.5.15:8.10.9|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)CCCC)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)C1CC1)ccc3OC |r,THB:29:9:5.4.6:13|
COc1ccc2C[C@H]3N(CC[C@@]45[C@@H](Oc1c24)[C@@H](CC[C@@]35O)N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(cc1)N(C)C |r,TLB:18:19:6.5.15:8.10.9,20:19:6.5.15:8.10.9|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)C(=O)C1CC1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)C(=O)c1ccc(C)cc1)ccc3OC |r,THB:29:9:5.4.6:13|
COc1ccc2C[C@H]3N(CC[C@@]45[C@@H](Oc1c24)[C@@H](CC[C@@]35O)N(C)Cc1ccccc1)S(=O)(=O)c1ccccc1 |r|
COc1ccc2C[C@H]3N(CC[C@@]45[C@@H](Oc1c24)[C@@H](CC[C@@]35O)N(C)C(=O)Nc1ccccc1)S(=O)(=O)c1ccccc1 |r,TLB:18:19:6.5.15:8.10.9,20:19:6.5.15:8.10.9|
COc1ccc2C[C@H]3N(CC[C@@]45[C@@H](Oc1c24)[C@@H](CC[C@@]35O)N(C)C(=O)NCc1ccccc1)S(=O)(=O)c1ccccc1 |r,TLB:18:19:6.5.15:8.10.9,20:19:6.5.15:8.10.9|
COc1ccc2C[C@H]3N(CC[C@@]45[C@@H](Oc1c24)C1(CC[C@@]35O)OCCO1)S(=O)(=O)c1ccccc1[N+]([O-])=O |r|
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-c1ccccc1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1cccc(C)c1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1cccc(F)c1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccc(F)cc1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1C1CC1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1cccnc1-n1cccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1cc(F)ccc1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccc(OC)cc1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-n1ncnn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1cccnc1OCC(F)F
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1C1(CC1)C#N
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-c1nc(C)no1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1sccc1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccsc1-n1nccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1cccnc1OCC(F)(F)F
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1CC(F)(F)F
CCOc1ccccc1C(=O)N(CC)CCc1nc(c(C)o1)C(C)(C)O
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1C(=O)OC
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-n1cccn1
CCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1C1(CC1)C(F)F
CCN(CCc1nc(C(=O)N(C)OC)c(C)o1)C(=O)c1ccccc1-n1nccn1
Cc1oc(CCN(CC=C)C(=O)c2ccccc2-n2nccn2)nc1C(O)=O
CCCN(CCc1nc(C(=O)OCC)c(C)o1)C(=O)c1ccccc1-n1nccn1
CCOC(=O)c1nc(CCN(CC2CC2)C(=O)c2ccccc2-n2nccn2)oc1C
COC(=O)C(NC(=O)CCN(CC(F)F)C(=O)c1ccccc1-n1nccn1)C(C)=O
Cc1oc(CCN(CCCO)C(=O)c2ccccc2-n2nccn2)nc1C(C)(C)O
Cc1oc(CCN(CCO)C(=O)c2ccccc2-n2nccn2)nc1C(C)(C)O
COCCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
CN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
COC(=O)C(NC(=O)CCN(C1CC1)C(=O)c1ccccc1-n1nccn1)C(C)=O
Cc1oc(CCN(C2CCC2)C(=O)c2ccccc2-n2nccn2)nc1C(C)(C)O
COCCCN(CCc1nc(c(C)o1)C(C)(C)O)C(=O)c1ccccc1-n1nccn1
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CC(F)(F)F)Oc1nccn2ccnc12 |r|
CCCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccn2cc(C)nc12
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)Oc1nccn2cc(C)nc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-c1ccccc1)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-n1cccn1)Oc1nccn2cc(C)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccn2cc(C)nc12 |r|
CC(C)c1cn2ccnc(O[C@@H]3CC[C@@H](C)N(C3)C(=O)c3ccccc3-n3nccn3)c2n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2cc(nc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccn2cc(nc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccn2cc(nc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2cc(nc12)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2cc(CO)nc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(Cl)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Oc1nccn2c(Cl)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccn2c(Cl)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccn2c(Cl)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Nc1nccn2c(Cl)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(F)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(Br)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(C)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(cnc12)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(C=C)cnc12 |r|
CCc1cnc2c(O[C@@H]3CC[C@@H](C)N(C3)C(=O)c3ccccc3-n3nccn3)nccn12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)Oc1nccn2c(CF)cnc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#C)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1nccn2c(cnc12)C(F)F |r|
COCc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-n1cccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-c1ccccn1)Oc1nccn2c(cnc12)C(F)F |r|
COC(=O)c1nccnc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ncccc1-c1ccccc1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1NCC(F)(F)F)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-n1cccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1cnccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-c1ncccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1nccn2c(cnc12)C(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CS(C)(=O)=O)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ncccc1-c1ccccc1)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)(F)F)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1OCC(F)F)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cccnc1-n1cccn1)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1nccn2c(cnc12)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(cnc12)C(O)C(F)F |r|
CC(O)c1cnc2c(O[C@@H]3CC[C@@H](C)N(C3)C(=O)c3ccccc3-n3nccn3)nccn12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2nccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1nccn2nccc12
C[C@@H]1CC[C@H](CN1C(=O)c1cscc1-n1nccn1)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1C1(CC1)C#N)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccc(F)cc1-n1nccn1)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-c1ncccn1)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-c1ccccn1)Oc1nccn2ccnc12 |r|
COC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nccnc1-n1nccn1)Oc1nccn2ccnc12 |r|
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccn2ccnc12 |r|
CC(C)Oc1ncccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccn2ccnc12 |r|
CC(C)Oc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1nccn2ccnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ncccn1)Oc1nccn2nccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccn2nccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Sc1nccn2nccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2ncc(Br)c12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2ncc(C)c12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccn2nccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccnc2ocnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1ccnc2ocnc12 |r|
COC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1ccnc2ocnc12
CCOc1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1ccnc2ocnc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc2n(C)ncc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc2n(C)ncc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc2nn(C)cc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc2n(C)cnc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc2ncn(C)c12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc2ncn(C)c12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Nc1nccc2n(C)cnc12
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2cncc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccn2c(C)ncc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1nccc2nc(C)nn12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccn2c1nn(C)c2=O |r|
CCc1cnc(N[C@H]2CCC[C@H]2NC(=O)c2cc(C)ccc2-n2nccn2)nc1 |r|
Cc1ccc(c(c1)C(=O)N[C@@H]1CCC[C@@H]1Nc1ccc(Cl)cn1)-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)nn1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(ccc1-n1nccn1)C(F)(F)F |r|
COc1ccc(c(n1)C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1ccc(cn1)C(F)(F)F)-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(Cl)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(Cl)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1COc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(C)cn1 |r|
C[C@@H]1CC(F)(F)CN(C1COc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(C)c1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cc1 |r|
COc1ccc(cc1)-c1cn(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1ccc(cn1)C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(C)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1COc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cc(C)ccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cn1 |r|
COc1ccc(nc1)-c1cn(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1ncc(cn1)C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1sc(C)nc1-c1ccccc1 |r|
COc1cccc(c1)-c1cn(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1ncc(cn1)C(F)(F)F |r|
COc1ccc(nc1)-c1cn(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1cnc(cn1)C(F)(F)F |r|
COc1cccc(n1)-c1cn(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1cnc(cn1)C(F)(F)F |r|
COc1cccc(c1)-c1cn(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1cnc(cn1)C(F)(F)F |r|
COc1ccc(cc1)-c1cn(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1cnc(cn1)C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(C)c1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccc(C)n1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(C)c1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cc(C)ccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccc(C)c1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(C)cn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(C)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(C)cn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ncccc1C |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cc(C)ccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(C)cn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccc1C |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccc(C)c1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(C)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccc1C |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccc(C)n1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccc1F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccc1F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccc(F)c1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-c1nnn(C)n1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-c1nnn(C)n1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)oc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccn1 |r|
COc1cccc(c1)-c1sc(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1cnc(cn1)C(F)(F)F |r|
COc1ccc(cc1)-c1sc(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1cnc(cn1)C(F)(F)F |r|
COc1cccc(n1)-c1sc(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1cnc(cn1)C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cc(F)ccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(C)n1 |r|
COc1ccc(nc1)-c1sc(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)C1CNc1ncc(cn1)C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cn(C)nc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cnn(C)c1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cn(C)nc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cnn(C)c1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1cn(C)nc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)oc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncccn1)C(=O)c1nc(C)oc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)oc1-c1cccnc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)oc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccnc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cc(C)sc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccnc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
CCc1cnc(NCC2[C@H](C)CC(F)(F)CN2C(=O)c2nn(C)cc2-c2ccccc2)nc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)nc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)oc1-c1ccc(F)cc1 |r|
CCc1cnc(NCC2[C@H](C)CC(F)(F)CN2C(=O)c2nn(C)cc2-c2ccc(F)cn2)nc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)nc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)nc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1nn(C)cc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(C)nc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)sc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-c1nc(C)no1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cc(ccc1-n1nccn1)C#N |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(ccc1-n1nccn1)C#N |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1nn(C)cc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(F)cc1 |r|
COc1nc(NCC2[C@H](C)CC(F)(F)CN2C(=O)c2nn(C)cc2-c2ccccn2)ncc1C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cc(Cl)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccn1 |r|
COc1nc(NCC2[C@@H](C)CC(F)(F)CN2C(=O)c2nn(C)cc2-c2ccccn2)ncc1C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1nc(C)ccc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cc(ccc1-c1ccc(F)cc1)C#N |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1ncnn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1nc(C)sc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cc(C)ccc1-c1nnn(C)n1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-c1nnn(C)n1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1ncc(C)n1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-n1nccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1cccc(F)c1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccccc1F |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(Cl)cn1)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ccc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-c1nnn(C)n1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(Cl)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(C)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1nccc(C)n1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(cn1)C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cc(Cl)ccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cc1F)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cccc(n1)C(F)(F)F |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccc(Cl)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cnccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1cncnc1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ccc(C)cn1 |r|
CCn1cc(c(n1)C(=O)N1CC(F)(F)C[C@@H](C)[C@H]1CNc1ncc(cn1)C(F)(F)F)-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)c(C)c1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1C#CC1CC1 |r|
CC#Cc1ccc(C)nc1C(=O)N1CC(F)(F)C[C@@H](C)[C@H]1CNc1ncc(cn1)C(F)(F)F |r|
CC(C)n1cc(c(n1)C(=O)N1CC(F)(F)C[C@@H](C)[C@H]1CNc1ncc(cn1)C(F)(F)F)-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(CC(F)(F)F)cc1-c1ncccn1 |r|
CCc1cnc(NC[C@@H]2[C@H](C)CC(F)(F)CN2C(=O)c2nc(C)sc2-c2ccc(F)cc2)nc1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1nnn(C)n1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccncn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cc1F)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ncc(cc1F)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ncc(cc1F)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1COc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)nc1-c1ccc(Cl)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-c1nnn(C)n1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(Cl)cn1)C(=O)c1cn(C)nc1-c1ccccc1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CN(C)c1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncc(F)cn1 |r|
C[C@@H]1CC(F)(F)CN([C@@H]1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nn(C)c(C)c1-c1ncc(F)cn1 |r|
Cc1ccc(c(c1)C(=O)N1CCC[C@H]1c1nc2c(cccc2[nH]1)[N+]([O-])=O)-n1nccn1
CSc1ccc2nc([nH]c2c1)[C@@H]1CCCN1C(=O)c1cncnc1-c1ccc(Br)c(C)c1
Cc1ccc(c(c1)C(=O)N1C[C@@H](F)C[C@H]1c1nc2c(C)c(Cl)ccc2[nH]1)-n1nccn1
CO[C@H]1C[C@H](N(C1)C(=O)c1cc(C)ccc1-n1nccn1)c1nc2c(C)c(Cl)ccc2[nH]1
C[C@H]1CCN([C@@H]1c1nc2c(C)cccc2[nH]1)C(=O)c1cc(C)ccc1-n1nccn1
Cc1nc(C(=O)N2CCC[C@@]2(C)c2nc3c(C)cccc3[nH]2)c(s1)-c1ccccc1
Cc1cc(ccc1-c1nc(cs1)C(=O)N1CCC[C@@]1(C)c1nc2c(C)c(Cl)ccc2[nH]1)-c1ccc(F)cc1
COc1ccc(-c2ccc3OCOc3c2)c(C(=O)N2CCC[C@@]2(C)c2nc3c(C)c(Cl)ccc3[nH]2)c1F
COc1ccc2[nH]c(nc2c1)[C@@H]1CC(=C)CN1C(=O)c1nc(C)sc1-c1ccc(F)cc1
COCCn1c(nc2cc(C)c(C)cc12)C1CCCN1C(=O)c1cc(C)ccc1-c1cccc(OC)c1
Fc1cccc(C(=O)N2CC3CN(CC3C2)c2cnc3cc(F)c(F)cc3n2)c1-n1nccn1
Cc1nc(nc(=O)[nH]1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Fc1cc2cnc(nc2cc1F)N1CC2CN(CC2C1)C(=O)c1cccc(F)c1-c1ncccn1
CO[C@@H]1CN(CC[C@@H]1[C@H]1C[C@@H]2CC[C@H](C1)N2[C@H](C1CC1)C(N)=O)c1ncc(F)cn1 |r,TLB:16:15:9.8.14:12.11|
CO[C@@H]1CN(CC[C@@H]1[C@H]1C[C@@H]2CC[C@H](C1)N2[C@H](C(C)C)C(N)=O)c1ncc(F)cn1 |r|
CCO[C@@H]1CN(CC[C@@H]1[C@H]1C[C@@H]2CC[C@H](C1)N2[C@H](C1CC1)C(N)=O)c1ncc(Cl)cn1 |r|
C[C@H]1C[C@H](CCN1c1ncc(F)cn1)[C@H]1C[C@@H]2CC[C@H](C1)N2[C@H](C1CC1)C(N)=O |r,TLB:22:21:15.14.20:18.17|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(F)cc2)c(s1)-c1ccccc1 |THB:4:6:8:10,(-7.3,-.22,;-5.81,-.61,;-4.78,.53,;-3.37,-.1,;-2.04,.67,;-.7,-.1,;-2.04,2.21,;-3.37,2.98,;-3.37,4.52,;-2.04,5.29,;-2.04,3.75,;-.7,4.52,;-.7,2.98,;.63,2.21,;1.96,2.98,;3.3,2.21,;4.63,2.98,;5.96,2.21,;5.96,.67,;7.3,-.1,;4.63,-.1,;3.3,.67,;-3.53,-1.63,;-5.04,-1.95,;-2.44,-2.72,;-.96,-2.32,;.13,-3.41,;-.27,-4.89,;-1.75,-5.29,;-2.84,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2cc3ccccc3cn2)c(s1)-c1ccccc1 |(-7.96,-.22,;-6.48,-.61,;-5.45,.53,;-4.04,-.1,;-2.71,.67,;-1.37,-.1,;-2.71,2.21,;-4.04,2.98,;-4.04,4.52,;-2.71,5.29,;-2.71,3.75,;-1.37,4.52,;-1.37,2.98,;-.04,2.21,;1.3,2.98,;2.63,2.21,;3.96,2.98,;5.3,2.21,;6.63,2.98,;7.96,2.21,;7.96,.67,;6.63,-.1,;5.3,.67,;3.96,-.1,;2.63,.67,;-4.2,-1.63,;-5.71,-1.95,;-3.11,-2.72,;-1.62,-2.32,;-.53,-3.41,;-.93,-4.89,;-2.42,-5.29,;-3.51,-4.2,)|
Cc1ccc(c(n1)C(=O)N1C2CC(C2)CC1COc1ccc(F)cc1)-n1nccn1 |(-7.34,.24,;-6,-.53,;-6,-2.07,;-4.67,-2.84,;-3.33,-2.07,;-3.33,-.53,;-4.67,.24,;-2,.24,;-.67,-.53,;-2,1.78,;-3.33,2.55,;-3.33,4.09,;-2,4.86,;-2,3.32,;-.67,4.09,;-.67,2.55,;.67,1.78,;2,2.55,;3.33,1.78,;4.67,2.55,;6,1.78,;6,.24,;7.34,-.53,;4.67,-.53,;3.33,.24,;-2,-2.84,;-2,-4.38,;-.54,-4.86,;.37,-3.61,;-.54,-2.37,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(F)cc2)c(s1)-c1ccccc1F |THB:4:6:8:10,(-7.3,-.22,;-5.81,-.61,;-4.78,.53,;-3.37,-.1,;-2.04,.67,;-.7,-.1,;-2.04,2.21,;-3.37,2.98,;-3.37,4.52,;-2.04,5.29,;-2.04,3.75,;-.7,4.52,;-.7,2.98,;.63,2.21,;1.96,2.98,;3.3,2.21,;3.3,.67,;4.63,-.1,;5.96,.67,;7.3,-.1,;5.96,2.21,;4.63,2.98,;-3.53,-1.63,;-5.04,-1.95,;-2.44,-2.72,;-.96,-2.32,;.13,-3.41,;-.27,-4.89,;-1.75,-5.29,;-2.84,-4.2,;-4.33,-4.6,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2cccc(F)c2)c(s1)-c1ccccc1 |THB:4:6:8:10,(-7.3,-.22,;-5.81,-.61,;-4.78,.53,;-3.37,-.1,;-2.04,.67,;-.7,-.1,;-2.04,2.21,;-3.37,2.98,;-3.37,4.52,;-2.04,5.29,;-2.04,3.75,;-.7,4.52,;-.7,2.98,;.63,2.21,;1.96,2.98,;3.3,2.21,;3.3,.67,;4.63,-.1,;5.96,.67,;5.96,2.21,;7.3,2.98,;4.63,2.98,;-3.53,-1.63,;-5.04,-1.95,;-2.44,-2.72,;-.96,-2.32,;.13,-3.41,;-.27,-4.89,;-1.75,-5.29,;-2.84,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccccc2F)c(s1)-c1ccccc1 |(-6.63,-.22,;-5.14,-.61,;-4.11,.53,;-2.71,-.1,;-1.37,.67,;-.04,-.1,;-1.37,2.21,;-2.71,2.98,;-2.71,4.52,;-1.37,5.29,;-1.37,3.75,;-.04,4.52,;-.04,2.98,;1.3,2.21,;2.63,2.98,;3.96,2.21,;3.96,.67,;5.3,-.1,;6.63,.67,;6.63,2.21,;5.3,2.98,;5.3,4.52,;-2.87,-1.63,;-4.37,-1.95,;-1.78,-2.72,;-.29,-2.32,;.8,-3.41,;.4,-4.89,;-1.09,-5.29,;-2.18,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(Br)cc2)c(s1)-c1ccccc1 |(-7.32,-.61,;-5.78,-.61,;-4.75,.53,;-3.35,-.1,;-2.01,.67,;-.68,-.1,;-2.01,2.21,;-3.35,2.98,;-3.35,4.52,;-2.01,5.29,;-2.01,3.75,;-.68,4.52,;-.68,2.98,;.66,2.21,;1.99,2.98,;3.32,2.21,;4.66,2.98,;5.99,2.21,;5.99,.67,;7.32,-.1,;4.66,-.1,;3.32,.67,;-3.51,-1.63,;-5.01,-1.95,;-2.42,-2.72,;-.93,-2.32,;.16,-3.41,;-.24,-4.89,;-1.73,-5.29,;-2.82,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(F)c(F)c2)c(s1)-c1ccccc1 |(-7.32,-.61,;-5.78,-.61,;-4.75,.53,;-3.35,-.1,;-2.01,.67,;-.68,-.1,;-2.01,2.21,;-3.35,2.98,;-3.35,4.52,;-2.01,5.29,;-2.01,3.75,;-.68,4.52,;-.68,2.98,;.66,2.21,;1.99,2.98,;3.32,2.21,;3.32,.67,;4.66,-.1,;5.99,.67,;7.32,-.1,;5.99,2.21,;7.32,2.98,;4.66,2.98,;-3.51,-1.63,;-5.01,-1.95,;-2.42,-2.72,;-.93,-2.32,;.16,-3.41,;-.24,-4.89,;-1.73,-5.29,;-2.82,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(C)cc2)c(s1)-c1ccccc1 |(-7.32,-.61,;-5.78,-.61,;-4.75,.53,;-3.35,-.1,;-2.01,.67,;-.68,-.1,;-2.01,2.21,;-3.35,2.98,;-3.35,4.52,;-2.01,5.29,;-2.01,3.75,;-.68,4.52,;-.68,2.98,;.66,2.21,;1.99,2.98,;3.32,2.21,;4.66,2.98,;5.99,2.21,;5.99,.67,;7.32,-.1,;4.66,-.1,;3.32,.67,;-3.51,-1.63,;-5.01,-1.95,;-2.42,-2.72,;-.93,-2.32,;.16,-3.41,;-.24,-4.89,;-1.73,-5.29,;-2.82,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(Cl)cc2)c(s1)-c1ccccc1 |(-7.32,-.61,;-5.78,-.61,;-4.75,.53,;-3.35,-.1,;-2.01,.67,;-.68,-.1,;-2.01,2.21,;-3.35,2.98,;-3.35,4.52,;-2.01,5.29,;-2.01,3.75,;-.68,4.52,;-.68,2.98,;.66,2.21,;1.99,2.98,;3.32,2.21,;4.66,2.98,;5.99,2.21,;5.99,.67,;7.32,-.1,;4.66,-.1,;3.32,.67,;-3.51,-1.63,;-5.01,-1.95,;-2.42,-2.72,;-.93,-2.32,;.16,-3.41,;-.24,-4.89,;-1.73,-5.29,;-2.82,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(F)cc2)c(s1)-c1ccc(F)cc1 |(-7.32,-.27,;-5.78,-.27,;-4.75,.88,;-3.35,.25,;-2.01,1.02,;-.68,.25,;-2.01,2.56,;-3.35,3.33,;-3.35,4.87,;-2.01,5.64,;-2.01,4.1,;-.68,4.87,;-.68,3.33,;.66,2.56,;1.99,3.33,;3.32,2.56,;4.66,3.33,;5.99,2.56,;5.99,1.02,;7.32,.25,;4.66,.25,;3.32,1.02,;-3.51,-1.28,;-5.01,-1.6,;-2.42,-2.37,;-.93,-1.97,;.16,-3.06,;-.24,-4.55,;.85,-5.64,;-1.73,-4.95,;-2.82,-3.86,)|
Fc1ccc(OCC2CC3CC(C3)N2C(=O)c2nc(Cl)sc2-c2ccccc2)cc1 |(7.32,-.1,;5.99,.67,;5.99,2.21,;4.66,2.98,;3.32,2.21,;1.99,2.98,;.66,2.21,;-.68,2.98,;-.68,4.52,;-2.01,5.29,;-3.35,4.52,;-3.35,2.98,;-2.01,3.75,;-2.01,2.21,;-2.01,.67,;-.68,-.1,;-3.35,-.1,;-4.75,.53,;-5.78,-.61,;-7.32,-.61,;-5.01,-1.95,;-3.51,-1.63,;-2.42,-2.72,;-.93,-2.32,;.16,-3.41,;-.24,-4.89,;-1.73,-5.29,;-2.82,-4.2,;3.32,.67,;4.66,-.1,)|
COc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(F)cc2)c(s1)-c1ccccc1 |(-7.85,.83,;-7.32,-.61,;-5.78,-.61,;-4.75,.53,;-3.35,-.1,;-2.01,.67,;-.68,-.1,;-2.01,2.21,;-3.35,2.98,;-3.35,4.52,;-2.01,5.29,;-2.01,3.75,;-.68,4.52,;-.68,2.98,;.66,2.21,;1.99,2.98,;3.32,2.21,;4.66,2.98,;5.99,2.21,;5.99,.67,;7.32,-.1,;4.66,-.1,;3.32,.67,;-3.51,-1.63,;-5.01,-1.95,;-2.42,-2.72,;-.93,-2.32,;.16,-3.41,;-.24,-4.89,;-1.73,-5.29,;-2.82,-4.2,)|
Fc1ccc(OCC2CC3CC(C3)N2C(=O)c2nc(sc2-c2ccccc2)C2CC2)cc1 |(8.04,-.1,;6.71,.67,;6.71,2.21,;5.37,2.98,;4.04,2.21,;2.71,2.98,;1.37,2.21,;.04,2.98,;.04,4.52,;-1.29,5.29,;-2.63,4.52,;-2.63,2.98,;-1.29,3.75,;-1.29,2.21,;-1.29,.67,;.04,-.1,;-2.63,-.1,;-4.04,.53,;-5.07,-.61,;-4.3,-1.95,;-2.79,-1.63,;-1.7,-2.72,;-.21,-2.32,;.88,-3.41,;.48,-4.89,;-1.01,-5.29,;-2.1,-4.2,;-6.55,-.22,;-7.64,.87,;-8.04,-.61,;4.04,.67,;5.37,-.1,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2nc3ccc(F)cc3s2)c(s1)-c1ccccc1 |(-8.47,-.61,;-6.93,-.61,;-5.9,.53,;-4.49,-.1,;-3.16,.67,;-1.82,-.1,;-3.16,2.21,;-4.49,2.98,;-4.49,4.52,;-3.16,5.29,;-3.16,3.75,;-1.82,4.52,;-1.82,2.98,;-.49,2.21,;.85,2.98,;2.18,2.21,;2.34,.68,;3.85,.36,;4.62,-.97,;6.16,-.97,;6.93,.36,;8.47,.36,;6.16,1.7,;4.62,1.7,;3.59,2.84,;-4.65,-1.63,;-6.16,-1.95,;-3.56,-2.72,;-3.96,-4.2,;-2.87,-5.29,;-1.38,-4.89,;-.98,-3.41,;-2.07,-2.32,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc(cn2)C(F)(F)F)c(s1)-c1ccccc1 |(-7.99,-.61,;-6.45,-.61,;-5.42,.53,;-4.01,-.1,;-2.68,.67,;-1.35,-.1,;-2.68,2.21,;-4.01,2.98,;-4.01,4.52,;-2.68,5.29,;-2.68,3.75,;-1.35,4.52,;-1.35,2.98,;-.01,2.21,;1.32,2.98,;2.66,2.21,;3.99,2.98,;5.32,2.21,;5.37,.65,;3.99,-.1,;2.66,.67,;6.7,-.12,;8.04,-.89,;5.93,-1.46,;7.47,1.21,;-4.17,-1.63,;-5.68,-1.95,;-3.08,-2.72,;-3.48,-4.2,;-2.39,-5.29,;-.91,-4.89,;-.51,-3.41,;-1.6,-2.32,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ccc3ccccc3n2)c(s1)-c1ccccc1 |(-7.99,-.61,;-6.45,-.61,;-5.42,.53,;-4.01,-.1,;-2.68,.67,;-1.35,-.1,;-2.68,2.21,;-4.01,2.98,;-4.01,4.52,;-2.68,5.29,;-2.68,3.75,;-1.35,4.52,;-1.35,2.98,;-.01,2.21,;1.32,2.98,;2.66,2.21,;2.66,.67,;3.99,-.1,;5.32,.67,;6.66,-.1,;7.99,.67,;7.99,2.21,;6.66,2.98,;5.32,2.21,;3.99,2.98,;-4.17,-1.63,;-5.68,-1.95,;-3.08,-2.72,;-3.48,-4.2,;-2.39,-5.29,;-.91,-4.89,;-.51,-3.41,;-1.6,-2.32,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2ncc3ccn(C)c3n2)c(s1)-c1ccccc1 |(-7.84,-.61,;-6.3,-.61,;-5.27,.53,;-3.86,-.1,;-2.53,.67,;-1.2,-.1,;-2.53,2.21,;-3.86,2.98,;-3.86,4.52,;-2.53,5.29,;-2.53,3.75,;-1.2,4.52,;-1.2,2.98,;.14,2.21,;1.47,2.98,;2.8,2.21,;2.8,.67,;4.14,-.1,;5.47,.67,;6.94,.2,;7.84,1.44,;6.94,2.69,;7.33,4.18,;5.47,2.21,;4.14,2.98,;-4.03,-1.63,;-5.53,-1.95,;-2.94,-2.72,;-3.33,-4.2,;-2.25,-5.29,;-.76,-4.89,;-.36,-3.41,;-1.45,-2.32,)|
Cc1nc(C(=O)N2C3CC(C3)CC2COc2cnc3ccccc3n2)c(s1)-c1ccccc1 |(-7.99,-.61,;-6.45,-.61,;-5.42,.53,;-4.01,-.1,;-2.68,.67,;-1.35,-.1,;-2.68,2.21,;-4.01,2.98,;-4.01,4.52,;-2.68,5.29,;-2.68,3.75,;-1.35,4.52,;-1.35,2.98,;-.01,2.21,;1.32,2.98,;2.66,2.21,;2.66,.67,;3.99,-.1,;5.32,.67,;6.66,-.1,;7.99,.67,;7.99,2.21,;6.66,2.98,;5.32,2.21,;3.99,2.98,;-4.17,-1.63,;-5.68,-1.95,;-3.08,-2.72,;-3.48,-4.2,;-2.39,-5.29,;-.91,-4.89,;-.51,-3.41,;-1.6,-2.32,)|
Cc1nc(C(=O)N2C3CC(C3)CC2CNc2cc3ccccc3cn2)c(s1)-c1ccccc1 |(-7.96,-.22,;-6.48,-.61,;-5.45,.53,;-4.04,-.1,;-2.71,.67,;-1.37,-.1,;-2.71,2.21,;-4.04,2.98,;-4.04,4.52,;-2.71,5.29,;-2.71,3.75,;-1.37,4.52,;-1.37,2.98,;-.04,2.21,;1.3,2.98,;2.63,2.21,;3.96,2.98,;5.3,2.21,;6.63,2.98,;7.96,2.21,;7.96,.67,;6.63,-.1,;5.3,.67,;3.96,-.1,;2.63,.67,;-4.2,-1.63,;-5.71,-1.95,;-3.11,-2.72,;-1.62,-2.32,;-.53,-3.41,;-.93,-4.89,;-2.42,-5.29,;-3.51,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2CNc2ccc3ccccc3n2)c(s1)-c1ccccc1 |(-7.96,-.22,;-6.48,-.61,;-5.45,.53,;-4.04,-.1,;-2.71,.67,;-1.37,-.1,;-2.71,2.21,;-4.04,2.98,;-4.04,4.52,;-2.71,5.29,;-2.71,3.75,;-1.37,4.52,;-1.37,2.98,;-.04,2.21,;1.3,2.98,;2.63,2.21,;2.63,.67,;3.96,-.1,;5.3,.67,;6.63,-.1,;7.96,.67,;7.96,2.21,;6.63,2.98,;5.3,2.21,;3.96,2.98,;-4.2,-1.63,;-5.71,-1.95,;-3.11,-2.72,;-1.62,-2.32,;-.53,-3.41,;-.93,-4.89,;-2.42,-5.29,;-3.51,-4.2,)|
Cc1nc(C(=O)N2C3CC(C3)CC2CNc2nc3ccc(F)cc3s2)c(s1)-c1ccccc1 |(-8.47,-.61,;-6.93,-.61,;-5.9,.53,;-4.49,-.1,;-3.16,.67,;-1.82,-.1,;-3.16,2.21,;-4.49,2.98,;-4.49,4.52,;-3.16,5.29,;-3.16,3.75,;-1.82,4.52,;-1.82,2.98,;-.49,2.21,;.85,2.98,;2.18,2.21,;2.34,.68,;3.85,.36,;4.62,-.97,;6.16,-.97,;6.93,.36,;8.47,.36,;6.16,1.7,;4.62,1.7,;3.59,2.84,;-4.65,-1.63,;-6.16,-1.95,;-3.56,-2.72,;-3.96,-4.2,;-2.87,-5.29,;-1.38,-4.89,;-.98,-3.41,;-2.07,-2.32,)|
Cc1nc(C(=O)N2C3CC(C3)[C@@H](F)[C@@H]2COc2ccc(F)cn2)c(s1)-c1ccccc1 |r,wU:11.12,wD:13.15,(-7.32,6.59,;-5.79,6.43,;-4.76,7.58,;-3.35,6.95,;-2.02,7.72,;-.68,6.95,;-2.02,9.26,;-3.35,10.03,;-3.35,11.57,;-2.02,12.34,;-2.02,10.8,;-.68,11.57,;.65,12.34,;-.68,10.03,;.65,9.26,;1.98,10.03,;3.32,9.26,;3.32,7.72,;4.65,6.95,;5.99,7.72,;7.32,6.95,;5.99,9.26,;4.65,10.03,;-3.51,5.42,;-5.02,5.1,;-2.37,4.39,;-2.69,2.88,;-1.54,1.85,;-.08,2.33,;.24,3.83,;-.9,4.87,)|
C[C@@H]1C2CC(C2)N([C@H]1COc1cc2ccccc2cn1)C(=O)c1nc(C)sc1-c1ccccc1 |r,wU:1.0,wD:7.9,(-.04,5.29,;-1.37,4.52,;-2.71,5.29,;-4.04,4.52,;-4.04,2.98,;-2.71,3.75,;-2.71,2.21,;-1.37,2.98,;-.04,2.21,;1.3,2.98,;2.63,2.21,;3.96,2.98,;5.3,2.21,;6.63,2.98,;7.96,2.21,;7.96,.67,;6.63,-.1,;5.3,.67,;3.96,-.1,;2.63,.67,;-2.71,.67,;-1.37,-.1,;-4.04,-.1,;-5.45,.53,;-6.48,-.61,;-7.96,-.22,;-5.71,-1.95,;-4.2,-1.63,;-3.11,-2.72,;-1.62,-2.32,;-.53,-3.41,;-.93,-4.89,;-2.42,-5.29,;-3.51,-4.2,)|
C[C@H]1C2CC(C2)N([C@H]1COc1cc2ccccc2cn1)C(=O)c1nc(C)sc1-c1ccccc1 |r,wD:7.9,1.0,(-.04,5.29,;-1.37,4.52,;-2.71,5.29,;-4.04,4.52,;-4.04,2.98,;-2.71,3.75,;-2.71,2.21,;-1.37,2.98,;-.04,2.21,;1.3,2.98,;2.63,2.21,;3.96,2.98,;5.3,2.21,;6.63,2.98,;7.96,2.21,;7.96,.67,;6.63,-.1,;5.3,.67,;3.96,-.1,;2.63,.67,;-2.71,.67,;-1.37,-.1,;-4.04,-.1,;-5.45,.53,;-6.48,-.61,;-7.96,-.22,;-5.71,-1.95,;-4.2,-1.63,;-3.11,-2.72,;-1.62,-2.32,;-.53,-3.41,;-.93,-4.89,;-2.42,-5.29,;-3.51,-4.2,)|
C[C@H]1C2CC(C2)N([C@H]1COc1ccc(F)cc1)C(=O)c1nc(C)ccc1-c1ncccn1 |r,wD:7.9,1.0,(.67,5,;-.67,4.23,;-2,5,;-3.33,4.23,;-3.33,2.69,;-2,3.47,;-2,1.93,;-.67,2.69,;.67,1.93,;2,2.69,;3.33,1.93,;4.67,2.69,;6,1.93,;6,.39,;7.34,-.38,;4.67,-.38,;3.33,.38,;-2,.38,;-.67,-.38,;-3.33,-.38,;-4.67,.38,;-6,-.38,;-7.34,.38,;-6,-1.93,;-4.67,-2.69,;-3.33,-1.93,;-2,-2.69,;-.67,-1.92,;.67,-2.69,;.67,-4.23,;-.67,-5,;-2,-4.23,)|
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C[C@@H]1C2CC(C2)N(C1COc1ccc(F)cc1)C(=O)c1nc(C)sc1-c1ncccn1 |r,wU:1.0,TLB:0:1:3:5,THB:17:6:3:5,(.63,5.29,;-.7,4.52,;-2.04,5.29,;-3.37,4.52,;-3.37,2.98,;-2.04,3.75,;-2.04,2.21,;-.7,2.98,;.63,2.21,;1.96,2.98,;3.3,2.21,;4.63,2.98,;5.96,2.21,;5.96,.67,;7.3,-.1,;4.63,-.1,;3.3,.67,;-2.04,.67,;-.7,-.1,;-3.37,-.1,;-4.78,.53,;-5.81,-.61,;-7.3,-.22,;-5.04,-1.95,;-3.53,-1.63,;-2.44,-2.72,;-.96,-2.32,;.13,-3.41,;-.27,-4.89,;-1.75,-5.29,;-2.84,-4.2,)|
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C[C@H]1C2CC(C2)N(C1CNc1ncc2ccccc2n1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wD:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;6.67,-.61,;8,.16,;8,1.7,;6.67,2.47,;5.33,1.7,;4,2.47,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@H]1C2CC(C2)N(C1CNc1nc2ccccc2s1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wD:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;3.12,.16,;4.63,-.16,;5.4,-1.49,;6.94,-1.49,;7.71,-.16,;6.94,1.18,;5.4,1.18,;4.37,2.32,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cc2ccccc2cn1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;4,2.47,;5.33,1.7,;6.67,2.47,;8,1.7,;8,.16,;6.67,-.61,;5.33,.16,;4,-.61,;2.67,.16,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccc(F)cc2s1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(-.48,4.78,;-1.81,4.01,;-3.14,4.78,;-4.48,4.01,;-4.48,2.47,;-3.14,3.24,;-3.14,1.7,;-1.81,2.47,;-.48,1.7,;.86,2.47,;2.19,1.7,;2.35,.16,;3.86,-.16,;4.63,-1.49,;6.17,-1.49,;6.94,-.16,;8.48,-.16,;6.17,1.18,;4.63,1.18,;3.6,2.32,;-3.14,.16,;-1.81,-.61,;-4.48,-.61,;-5.81,.16,;-7.14,-.61,;-8.48,.16,;-7.14,-2.15,;-5.81,-2.92,;-4.48,-2.15,;-3.14,-2.92,;-2.98,-4.46,;-1.48,-4.78,;-.71,-3.44,;-1.74,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ncc2ccccc2n1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;6.67,-.61,;8,.16,;8,1.7,;6.67,2.47,;5.33,1.7,;4,2.47,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(Cl)cn1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.67,4.78,;-.67,4.01,;-2,4.78,;-3.33,4.01,;-3.33,2.47,;-2,3.24,;-2,1.7,;-.67,2.47,;.67,1.7,;2,2.47,;3.33,1.7,;3.33,.16,;4.67,-.61,;6,.16,;7.34,-.61,;6,1.7,;4.67,2.47,;-2,.16,;-.67,-.61,;-3.33,-.61,;-4.67,.16,;-6,-.61,;-7.34,.16,;-6,-2.15,;-4.67,-2.92,;-3.33,-2.15,;-2,-2.92,;-1.84,-4.46,;-.33,-4.78,;.44,-3.44,;-.59,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2cc(F)ccc2s1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;3.12,.16,;4.63,-.16,;5.4,-1.49,;6.94,-1.49,;7.71,-2.82,;7.71,-.16,;6.94,1.18,;5.4,1.18,;4.37,2.32,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2ccccc2n1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;6.67,-.61,;8,.16,;8,1.7,;6.67,2.47,;5.33,1.7,;4,2.47,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc2ccccc2n1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;6.67,-.61,;8,.16,;8,1.7,;6.67,2.47,;5.33,1.7,;4,2.47,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccc(F)cc2s1)C(=O)c1nc(C)sc1-c1ncccn1 |r,wU:1.0,(.26,5.29,;-1.08,4.52,;-2.41,5.29,;-3.75,4.52,;-3.75,2.98,;-2.41,3.75,;-2.41,2.21,;-1.08,2.98,;.26,2.21,;1.59,2.98,;2.92,2.21,;4.33,2.84,;5.36,1.7,;6.9,1.7,;7.67,.36,;6.9,-.97,;7.67,-2.31,;5.36,-.97,;4.59,.36,;3.08,.68,;-2.41,.67,;-1.08,-.1,;-3.75,-.1,;-5.15,.53,;-6.18,-.61,;-7.67,-.22,;-5.41,-1.95,;-3.91,-1.63,;-2.82,-2.72,;-3.22,-4.2,;-2.13,-5.29,;-.64,-4.89,;-.24,-3.41,;-1.33,-2.32,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccc(F)cc2s1)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;7.71,-2.82,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccc(F)cc2s1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;7.71,-2.82,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
CCOc1ccc(C)nc1C(=O)N1C2CC(C2)[C@@H](C)C1CNc1nc2ccc(F)cc2s1 |r,wU:17.19,(-1.04,-5,;-2.37,-4.23,;-2.37,-2.69,;-3.71,-1.93,;-5.04,-2.69,;-6.37,-1.93,;-6.37,-.38,;-7.71,.38,;-5.04,.38,;-3.71,-.38,;-2.37,.38,;-1.04,-.38,;-2.37,1.93,;-3.71,2.69,;-3.71,4.23,;-2.37,5,;-2.37,3.47,;-1.04,4.23,;.29,5,;-1.04,2.69,;.29,1.93,;1.63,2.69,;2.96,1.93,;4.37,2.55,;5.4,1.41,;6.94,1.41,;7.71,.07,;6.94,-1.26,;7.71,-2.59,;5.4,-1.26,;4.63,.07,;3.12,.39,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccc(F)cc2s1)C(=O)c1cc(ccc1-n1nccn1)C#N |r,wU:1.0,(.96,4.78,;-.37,4.01,;-1.71,4.78,;-3.04,4.01,;-3.04,2.47,;-1.71,3.24,;-1.71,1.7,;-.37,2.47,;.96,1.7,;2.29,2.47,;3.63,1.7,;5.03,2.32,;6.07,1.18,;7.61,1.18,;8.38,-.16,;7.61,-1.49,;8.38,-2.82,;6.07,-1.49,;5.3,-.16,;3.79,.16,;-1.71,.16,;-.37,-.61,;-3.04,-.61,;-4.37,.16,;-5.71,-.61,;-5.71,-2.15,;-4.37,-2.92,;-3.04,-2.15,;-1.71,-2.92,;-1.55,-4.46,;-.04,-4.78,;.73,-3.44,;-.3,-2.3,;-7.04,.16,;-8.38,.93,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccccc2s1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2cccnc2s1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2ccccc2n1)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(.67,4.78,;-.67,4.01,;-2,4.78,;-3.33,4.01,;-3.33,2.47,;-2,3.24,;-2,1.7,;-.67,2.47,;.67,1.7,;2,2.47,;3.33,1.7,;4.67,2.47,;6,1.7,;6,.16,;7.34,-.61,;7.34,-2.15,;6,-2.92,;4.67,-2.15,;4.67,-.61,;3.33,.16,;-2,.16,;-.67,-.61,;-3.33,-.61,;-4.67,.16,;-6,-.61,;-7.34,.16,;-6,-2.15,;-4.67,-2.92,;-3.33,-2.15,;-2,-2.92,;-1.84,-4.46,;-.33,-4.78,;.44,-3.44,;-.59,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(F)c(C)n1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.67,4.78,;-.67,4.01,;-2,4.78,;-3.33,4.01,;-3.33,2.47,;-2,3.24,;-2,1.7,;-.67,2.47,;.67,1.7,;2,2.47,;3.33,1.7,;3.33,.16,;4.67,-.61,;6,.16,;7.34,-.61,;6,1.7,;7.34,2.47,;4.67,2.47,;-2,.16,;-.67,-.61,;-3.33,-.61,;-4.67,.16,;-6,-.61,;-7.34,.16,;-6,-2.15,;-4.67,-2.92,;-3.33,-2.15,;-2,-2.92,;-1.84,-4.46,;-.33,-4.78,;.44,-3.44,;-.59,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cccc(n1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;5.38,1.72,;4,2.47,;6.72,2.49,;8.05,3.26,;7.49,1.16,;5.95,3.83,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2cc(F)ccc2n1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(-.67,4.78,;-2,4.01,;-3.33,4.78,;-4.67,4.01,;-4.67,2.47,;-3.33,3.24,;-3.33,1.7,;-2,2.47,;-.67,1.7,;.67,2.47,;2,1.7,;2,.16,;3.33,-.61,;4.67,.16,;6,-.61,;7.34,.16,;8.67,-.61,;7.34,1.7,;6,2.47,;4.67,1.7,;3.33,2.47,;-3.33,.16,;-2,-.61,;-4.67,-.61,;-6,.16,;-7.34,-.61,;-8.67,.16,;-7.34,-2.15,;-6,-2.92,;-4.67,-2.15,;-3.33,-2.92,;-3.17,-4.46,;-1.67,-4.78,;-.9,-3.44,;-1.93,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2cc(F)c(F)cc2n1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(-.67,4.78,;-2,4.01,;-3.33,4.78,;-4.67,4.01,;-4.67,2.47,;-3.33,3.24,;-3.33,1.7,;-2,2.47,;-.67,1.7,;.67,2.47,;2,1.7,;2,.16,;3.33,-.61,;4.67,.16,;6,-.61,;7.34,.16,;8.67,-.61,;7.34,1.7,;8.67,2.47,;6,2.47,;4.67,1.7,;3.33,2.47,;-3.33,.16,;-2,-.61,;-4.67,-.61,;-6,.16,;-7.34,-.61,;-8.67,.16,;-7.34,-2.15,;-6,-2.92,;-4.67,-2.15,;-3.33,-2.92,;-3.17,-4.46,;-1.67,-4.78,;-.9,-3.44,;-1.93,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(F)cc1)C(=O)c1cc(C)ccc1-c1nccs1 |r,wU:1.0,(.67,4.78,;-.67,4.01,;-2,4.78,;-3.33,4.01,;-3.33,2.47,;-2,3.24,;-2,1.7,;-.67,2.47,;.67,1.7,;2,2.47,;3.33,1.7,;4.67,2.47,;6,1.7,;6,.16,;7.34,-.61,;4.67,-.61,;3.33,.16,;-2,.16,;-.67,-.61,;-3.33,-.61,;-4.67,.16,;-6,-.61,;-7.34,.16,;-6,-2.15,;-4.67,-2.92,;-3.33,-2.15,;-2,-2.92,;-.59,-2.3,;.44,-3.44,;-.33,-4.78,;-1.84,-4.46,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;5.33,1.7,;4,2.47,;6.67,-.61,;8,.16,;6.67,-2.15,;8,-1.38,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2ncccc2n1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;6.67,-.61,;8,.16,;8,1.7,;6.67,2.47,;5.33,1.7,;4,2.47,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2cc(F)ccc2n1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(-.67,4.78,;-2,4.01,;-3.33,4.78,;-4.67,4.01,;-4.67,2.47,;-3.33,3.24,;-3.33,1.7,;-2,2.47,;-.67,1.7,;.67,2.47,;2,1.7,;2,.16,;3.33,-.61,;4.67,.16,;6,-.61,;7.34,.16,;8.67,-.61,;7.34,1.7,;6,2.47,;4.67,1.7,;3.33,2.47,;-3.33,.16,;-2,-.61,;-4.67,-.61,;-6,.16,;-7.34,-.61,;-8.67,.16,;-7.34,-2.15,;-6,-2.92,;-4.67,-2.15,;-3.33,-2.92,;-3.17,-4.46,;-1.67,-4.78,;-.9,-3.44,;-1.93,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ccccc1 |r,wU:1.0,(-.01,5.26,;-1.34,4.49,;-2.68,5.26,;-4.01,4.49,;-4.01,2.95,;-2.68,3.72,;-2.68,2.18,;-1.34,2.95,;-.01,2.18,;1.32,2.95,;2.66,2.18,;2.66,.64,;3.99,-.13,;5.32,.64,;5.32,2.18,;3.99,2.95,;6.66,-.13,;7.99,.64,;6.66,-1.67,;7.99,-.9,;-2.68,.64,;-1.34,-.13,;-4.01,-.13,;-5.26,.78,;-6.5,-.13,;-7.99,.27,;-6.03,-1.59,;-4.49,-1.59,;-3.4,-2.68,;-1.91,-2.28,;-.82,-3.37,;-1.22,-4.86,;-2.71,-5.26,;-3.8,-4.17,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r,wU:1.0,(-.01,5.26,;-1.34,4.49,;-2.68,5.26,;-4.01,4.49,;-4.01,2.95,;-2.68,3.72,;-2.68,2.18,;-1.34,2.95,;-.01,2.18,;1.32,2.95,;2.66,2.18,;2.66,.64,;3.99,-.13,;5.32,.64,;5.32,2.18,;3.99,2.95,;6.66,-.13,;7.99,.64,;6.66,-1.67,;7.99,-.9,;-2.68,.64,;-1.34,-.13,;-4.01,-.13,;-5.26,.78,;-6.5,-.13,;-7.99,.27,;-6.03,-1.59,;-4.49,-1.59,;-3.4,-2.68,;-1.91,-2.28,;-.82,-3.37,;-1.22,-4.86,;-2.71,-5.26,;-3.8,-4.17,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(C)cn1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.67,4.78,;-.67,4.01,;-2,4.78,;-3.33,4.01,;-3.33,2.47,;-2,3.24,;-2,1.7,;-.67,2.47,;.67,1.7,;2,2.47,;3.33,1.7,;3.33,.16,;4.67,-.61,;6,.16,;7.34,-.61,;6,1.7,;4.67,2.47,;-2,.16,;-.67,-.61,;-3.33,-.61,;-4.67,.16,;-6,-.61,;-7.34,.16,;-6,-2.15,;-4.67,-2.92,;-3.33,-2.15,;-2,-2.92,;-1.84,-4.46,;-.33,-4.78,;.44,-3.44,;-.59,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cncc(n1)C(F)(F)F)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;5.33,1.7,;4,2.47,;6.67,2.47,;8,1.7,;6.67,4.01,;8,3.24,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccc(F)cc2o1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;7.71,-2.82,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2cc(F)ccc2n1)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(-.67,4.78,;-2,4.01,;-3.33,4.78,;-4.67,4.01,;-4.67,2.47,;-3.33,3.24,;-3.33,1.7,;-2,2.47,;-.67,1.7,;.67,2.47,;2,1.7,;2,.16,;3.33,-.61,;4.67,.16,;6,-.61,;7.34,.16,;8.67,-.61,;7.34,1.7,;6,2.47,;4.67,1.7,;3.33,2.47,;-3.33,.16,;-2,-.61,;-4.67,-.61,;-6,.16,;-7.34,-.61,;-8.67,.16,;-7.34,-2.15,;-6,-2.92,;-4.67,-2.15,;-3.33,-2.92,;-3.17,-4.46,;-1.67,-4.78,;-.9,-3.44,;-1.93,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2ccccc2o1)C(=O)c1nc(C)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2cccnc2s1)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2cccnc2s1)C(=O)c1cc(ccc1-n1nccn1)C#N |r,wU:1.0,(.96,4.78,;-.37,4.01,;-1.71,4.78,;-3.04,4.01,;-3.04,2.47,;-1.71,3.24,;-1.71,1.7,;-.37,2.47,;.96,1.7,;2.29,2.47,;3.63,1.7,;5.03,2.32,;6.07,1.18,;7.61,1.18,;8.38,-.16,;7.61,-1.49,;6.07,-1.49,;5.3,-.16,;3.79,.16,;-1.71,.16,;-.37,-.61,;-3.04,-.61,;-4.37,.16,;-5.71,-.61,;-5.71,-2.15,;-4.37,-2.92,;-3.04,-2.15,;-1.71,-2.92,;-1.55,-4.46,;-.04,-4.78,;.73,-3.44,;-.3,-2.3,;-7.04,.16,;-8.38,.93,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2cccnc2s1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1cc(ccc1-n1nccn1)C#N |r,wU:1.0,(.67,4.78,;-.67,4.01,;-2,4.78,;-3.33,4.01,;-3.33,2.47,;-2,3.24,;-2,1.7,;-.67,2.47,;.67,1.7,;2,2.47,;3.33,1.7,;3.33,.16,;4.67,-.61,;6.05,.13,;6,1.7,;4.67,2.47,;7.38,-.64,;8.72,-1.41,;6.61,-1.98,;8.15,.69,;-2,.16,;-.67,-.61,;-3.33,-.61,;-4.67,.16,;-6,-.61,;-6,-2.15,;-4.67,-2.92,;-3.33,-2.15,;-2,-2.92,;-1.84,-4.46,;-.33,-4.78,;.44,-3.44,;-.59,-2.3,;-7.34,.16,;-8.67,.93,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc2cc(F)ccc2n1)C(=O)c1cc(ccc1-n1nccn1)C#N |r,wU:1.0,(,4.58,;-1.33,3.81,;-2.67,4.58,;-4,3.81,;-4,2.27,;-2.67,3.04,;-2.67,1.5,;-1.33,2.27,;,1.5,;1.33,2.27,;2.67,1.5,;2.67,-.04,;4,-.81,;5.33,-.04,;6.67,-.81,;8,-.04,;9.34,-.81,;8,1.5,;6.67,2.27,;5.33,1.5,;4,2.27,;-2.67,-.04,;-1.33,-.81,;-4,-.81,;-5.33,-.04,;-6.67,-.81,;-6.67,-2.35,;-5.33,-3.12,;-4,-2.35,;-2.67,-3.12,;-2.19,-4.58,;-.65,-4.58,;-.18,-3.12,;-1.42,-2.21,;-8,-.04,;-9.34,.73,)|
C[C@@H]1C2CC(C2)N(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;4,2.47,;5.33,1.7,;5.33,.16,;4,-.61,;2.67,.16,;6.67,-.61,;8,.16,;6.67,-2.15,;8,-1.38,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1nc2cccnc2o1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(.29,4.78,;-1.04,4.01,;-2.37,4.78,;-3.71,4.01,;-3.71,2.47,;-2.37,3.24,;-2.37,1.7,;-1.04,2.47,;.29,1.7,;1.63,2.47,;2.96,1.7,;4.37,2.32,;5.4,1.18,;6.94,1.18,;7.71,-.16,;6.94,-1.49,;5.4,-1.49,;4.63,-.16,;3.12,.16,;-2.37,.16,;-1.04,-.61,;-3.71,-.61,;-5.04,.16,;-6.37,-.61,;-7.71,.16,;-6.37,-2.15,;-5.04,-2.92,;-3.71,-2.15,;-2.37,-2.92,;-2.21,-4.46,;-.71,-4.78,;.06,-3.44,;-.97,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nn(C)cc1-c1ncccn1 |r,wU:1.0,(-.01,5.26,;-1.34,4.49,;-2.68,5.26,;-4.01,4.49,;-4.01,2.95,;-2.68,3.72,;-2.68,2.18,;-1.34,2.95,;-.01,2.18,;1.32,2.95,;2.66,2.18,;2.66,.64,;3.99,-.13,;5.32,.64,;5.32,2.18,;3.99,2.95,;6.66,-.13,;7.99,.64,;6.66,-1.67,;7.99,-.9,;-2.68,.64,;-1.34,-.13,;-4.01,-.13,;-5.26,.78,;-6.5,-.13,;-7.99,.27,;-6.03,-1.59,;-4.49,-1.59,;-3.4,-2.68,;-1.91,-2.28,;-.82,-3.37,;-1.22,-4.86,;-2.71,-5.26,;-3.8,-4.17,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1ccc(Cl)cc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.33,.16,;5.33,1.7,;4,2.47,;6.67,-.61,;8,.16,;6.67,-2.15,;8,-1.38,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-6.67,-2.15,;-8,-2.92,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ccc(nn1)C(F)(F)F)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r,wU:1.0,(,5,;-1.33,4.23,;-2.67,5,;-4,4.23,;-4,2.69,;-2.67,3.46,;-2.67,1.92,;-1.33,2.69,;,1.92,;1.33,2.69,;2.67,1.93,;2.67,.38,;4,-.38,;5.38,.36,;5.33,1.93,;4,2.7,;6.72,-.41,;8.05,-1.18,;5.95,-1.75,;7.49,.92,;-2.67,.38,;-1.33,-.39,;-4,-.39,;-5.33,.38,;-6.67,-.39,;-8,.38,;-6.67,-1.93,;-5.33,-2.7,;-4,-1.93,;-2.67,-2.7,;-1.33,-1.92,;,-2.69,;,-4.23,;-1.33,-5,;-2.67,-4.24,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1nc(C)ccc1-c1ncccn1 |r,wU:1.0,(,5.01,;-1.33,4.24,;-2.67,5.01,;-4,4.24,;-4,2.7,;-2.67,3.47,;-2.67,1.93,;-1.33,2.7,;,1.93,;1.33,2.7,;2.67,1.93,;2.67,.39,;4,-.38,;5.38,.36,;5.33,1.93,;4,2.69,;6.72,-.41,;8.05,-1.18,;5.95,-1.75,;7.49,.92,;-2.67,.39,;-1.33,-.38,;-4,-.38,;-5.33,.39,;-6.67,-.38,;-8,.39,;-6.67,-1.92,;-5.33,-2.69,;-4,-1.92,;-2.67,-2.69,;-1.33,-1.93,;,-2.7,;,-4.24,;-1.33,-5.01,;-2.67,-4.23,)|
C[C@@H]1C2CC(C2)N(C1CNc1ncc(cn1)C(F)(F)F)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-8,.16,;-6.67,-2.15,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1ccc(F)cc1-n1nccn1 |r,wU:1.0,(,4.78,;-1.33,4.01,;-2.67,4.78,;-4,4.01,;-4,2.47,;-2.67,3.24,;-2.67,1.7,;-1.33,2.47,;,1.7,;1.33,2.47,;2.67,1.7,;2.67,.16,;4,-.61,;5.38,.13,;5.33,1.7,;4,2.47,;6.72,-.64,;8.05,-1.41,;5.95,-1.98,;7.49,.69,;-2.67,.16,;-1.33,-.61,;-4,-.61,;-5.33,.16,;-6.67,-.61,;-6.67,-2.15,;-8,-2.92,;-5.33,-2.92,;-4,-2.15,;-2.67,-2.92,;-2.51,-4.46,;-1,-4.78,;-.23,-3.44,;-1.26,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1c(F)cccc1-n1nccn1 |r,wU:1.0,(-.77,4.78,;-2.1,4.01,;-3.44,4.78,;-4.77,4.01,;-4.77,2.47,;-3.44,3.24,;-3.44,1.7,;-2.1,2.47,;-.77,1.7,;.56,2.47,;1.9,1.7,;1.9,.16,;3.23,-.61,;4.61,.13,;4.56,1.7,;3.23,2.47,;5.95,-.64,;7.28,-1.41,;5.18,-1.98,;6.72,.69,;-3.44,.16,;-2.1,-.61,;-4.77,-.61,;-6.1,.16,;-6.1,1.7,;-7.44,-.61,;-7.44,-2.15,;-6.1,-2.92,;-4.77,-2.15,;-3.44,-2.92,;-3.28,-4.46,;-1.77,-4.78,;-1,-3.44,;-2.03,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r,wU:1.0,(-.1,4.78,;-1.44,4.01,;-2.77,4.78,;-4.1,4.01,;-4.1,2.47,;-2.77,3.24,;-2.77,1.7,;-1.44,2.47,;-.1,1.7,;1.23,2.47,;2.56,1.7,;2.56,.16,;3.9,-.61,;5.28,.13,;5.23,1.7,;3.9,2.47,;6.61,-.64,;7.95,-1.41,;5.84,-1.98,;7.38,.69,;-2.77,.16,;-1.44,-.61,;-4.1,-.61,;-5.44,.16,;-6.77,-.61,;-8.11,.16,;-6.77,-2.15,;-5.44,-2.92,;-4.1,-2.15,;-2.77,-2.92,;-2.61,-4.46,;-1.1,-4.78,;-.33,-3.44,;-1.36,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C1CC1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(-.1,4.78,;-1.44,4.01,;-2.77,4.78,;-4.1,4.01,;-4.1,2.47,;-2.77,3.24,;-2.77,1.7,;-1.44,2.47,;-.1,1.7,;1.23,2.47,;2.56,1.7,;2.56,.16,;3.9,-.61,;5.23,.16,;5.23,1.7,;3.9,2.47,;6.57,-.61,;7.34,-1.95,;8.11,-.61,;-2.77,.16,;-1.44,-.61,;-4.1,-.61,;-5.44,.16,;-6.77,-.61,;-8.11,.16,;-6.77,-2.15,;-5.44,-2.92,;-4.1,-2.15,;-2.77,-2.92,;-2.61,-4.46,;-1.1,-4.78,;-.33,-3.44,;-1.36,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1cnc(cn1)C1CC1)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(-.1,4.78,;-1.44,4.01,;-2.77,4.78,;-4.1,4.01,;-4.1,2.47,;-2.77,3.24,;-2.77,1.7,;-1.44,2.47,;-.1,1.7,;1.23,2.47,;2.56,1.7,;2.56,.16,;3.9,-.61,;5.23,.16,;5.23,1.7,;3.9,2.47,;6.57,-.61,;7.34,-1.95,;8.11,-.61,;-2.77,.16,;-1.44,-.61,;-4.1,-.61,;-5.44,.16,;-6.77,-.61,;-8.11,.16,;-6.77,-2.15,;-5.44,-2.92,;-4.1,-2.15,;-2.77,-2.92,;-2.61,-4.46,;-1.1,-4.78,;-.33,-3.44,;-1.36,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ncc(cn1)C1CC1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r,wU:1.0,(-.1,4.78,;-1.44,4.01,;-2.77,4.78,;-4.1,4.01,;-4.1,2.47,;-2.77,3.24,;-2.77,1.7,;-1.44,2.47,;-.1,1.7,;1.23,2.47,;2.56,1.7,;3.9,2.47,;5.23,1.7,;5.23,.16,;3.9,-.61,;2.56,.16,;6.57,-.61,;7.34,-1.95,;8.11,-.61,;-2.77,.16,;-1.44,-.61,;-4.1,-.61,;-5.44,.16,;-6.77,-.61,;-8.11,.16,;-6.77,-2.15,;-5.44,-2.92,;-4.1,-2.15,;-2.77,-2.92,;-2.61,-4.46,;-1.1,-4.78,;-.33,-3.44,;-1.36,-2.3,)|
C[C@@H]1C2CC(C2)N(C1CNc1ncc(cn1)C1CC1)C(=O)c1cc(F)ccc1-n1nccn1 |r,wU:1.0,(-.1,4.78,;-1.44,4.01,;-2.77,4.78,;-4.1,4.01,;-4.1,2.47,;-2.77,3.24,;-2.77,1.7,;-1.44,2.47,;-.1,1.7,;1.23,2.47,;2.56,1.7,;3.9,2.47,;5.23,1.7,;5.23,.16,;3.9,-.61,;2.56,.16,;6.57,-.61,;7.34,-1.95,;8.11,-.61,;-2.77,.16,;-1.44,-.61,;-4.1,-.61,;-5.44,.16,;-6.77,-.61,;-8.11,.16,;-6.77,-2.15,;-5.44,-2.92,;-4.1,-2.15,;-2.77,-2.92,;-2.61,-4.46,;-1.1,-4.78,;-.33,-3.44,;-1.36,-2.3,)|
Cc1nc(nc(C)c1C)N1CC2CN(CC2C1)C(=O)c1ccc(F)cc1-n1nccn1
CC(=O)Nc1cc(F)c(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)c1
CC(=O)Nc1ccc(-c2ncccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)c1F
CC(=O)Nc1ccc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
Nc1ccc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
CC(=O)Nc1ccc(-n2nccn2)c(C(=O)N(C)[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
CC(=O)Nc1ccc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(Cl)cc2)n1
CC(=O)Nc1ccc(-n2nccn2)c(C(=O)N(C(C)C)[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
[2H]C([2H])(Oc1ccc(F)cc1)[C@H]1CCC[C@@H]1NC(=O)c1nc(NC(C)=O)ccc1-n1nccn1
CC(=O)Nc1ccc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)c(F)c2)n1
COC(=O)Nc1ccc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
O=C(N[C@H]1CCC[C@@H]1COc1ccc(F)cc1)c1nc(NC(=O)C(F)F)ccc1-n1nccn1
Nc1ccc(-c2ncccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
O=C(N[C@H]1CCC[C@@H]1COc1ccc(F)cc1)c1nc(NC(=O)C2CC2)ccc1-n1nccn1
CC(=O)Nc1ccc(-c2ncccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
CC(=O)Nc1ccc(-c2ncccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(Cl)cc2)n1
COCC(=O)Nc1ccc(-c2ncccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
CC(=O)Nc1ccc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2F)n1
CC(=O)Nc1ccc(-c2ncccn2)c(C(=O)N(C)[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
O=C(N[C@H]1CCC[C@@H]1COc1ccc(F)cc1)c1nc(NCC(F)F)ccc1-n1nccn1
O=C(N[C@H]1CCC[C@@H]1COc1ccc(F)cc1)c1nc(NCCO)ccc1-n1nccn1
CC(=O)Nc1ccc(-c2ncc(F)cn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
Nc1ccc(-c2ncc(F)cn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)n1
CC(=O)Nc1cc(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)c(-n2nccn2)cn1
CC(=O)Nc1cc(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)c(-c2ncccn2)cn1
CC(=O)Nc1cnc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cc2)c1
CC(=O)Nc1ccc(-n2nccn2)c(C(=O)N[C@H]2CCC[C@@H]2COc2ccc(F)cn2)n1
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1c(F)cccc1-n1nccn1 |r|
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)C4C(c5ccccc5)=CN5C=CC=CC45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccn5)cn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ncccc5F)cn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccc(C)s5)cn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5cccs5)nn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccn5)nn5ccccc45)C[C@H]3C2)n1
Cc1nc(N2C[C@H]3CN(C(=O)c4c(-c5ncccc5F)cn5ccccc45)C[C@H]3C2)nc2ccoc12
Cc1nc(N2C[C@H]3CN(C(=O)c4c(-c5ncccc5F)cn5ccccc45)C[C@H]3C2)nn2cccc12
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5nccs5)cn5ccccc45)C[C@H]3C2)n1
O=C(c1c(-c2ncccc2F)cn2ccccc12)N1C[C@@H]2CN(c3cnc4ccccc4n3)C[C@@H]2C1
Cc6cc(C)nc(N5C[C@@H]4CN(C(=O)c2c(c1ncccc1C(F)(F)F)cn3ccccc23)C[C@@H]4C5)n6
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccc5)nn5cccnc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccc5)nn5ccncc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccc5)nn5ncccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccc5F)cn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccsc5)cn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ncccc5F)cn5cc(F)ccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccn5)cn5cc(F)ccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ncco5)cn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ncccn5)cn5ccccc45)C[C@H]3C2)n1
Cc1nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccn5)cn5ccccc45)C[C@H]3C2)nc(C)c1F
Cc1nc(N2C[C@H]3CN(C(=O)c4c(-c5ncccc5F)cn5ccccc45)C[C@H]3C2)nc2c1CCC2
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5cccs5)cn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccccn5)nn5cc(F)ccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5ccncc5)nn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5cccnc5)nn5ccccc45)C[C@H]3C2)n1
Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4c(-c5cccs5)nn5cc(F)ccc45)C[C@H]3C2)n1
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cc1)C(=O)c1ccccc1-n1nccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cc1)C(=O)c1cc(F)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cc1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cc1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cc1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1cc(nn1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1ccc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H](Cn1cc(cn1)-c1ccc(F)cn1)N(C)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H](Cn1ccc(n1)-c1ccc(F)cn1)N(C)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H](Cn1ccc(n1)-c1ccc(F)cn1)NC(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN(CCn1cc(cn1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1
CN(CCn1cc(cn1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1
CN(CCn1ccc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)NCCn1cc(cn1)-c1ccc(F)cn1)-n1nccn1
CC(C)[C@@H](Cn1ccc(n1)-c1ccc(F)cn1)N(C)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN([C@H](C)Cn1ccc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cc1)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cc1)C(=O)c1nc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cc1)C(=O)c1ccccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cc1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cn1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cc1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cc1)C(=O)c1nc(C)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cc1)C(=O)c1cc(F)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cn1nnc(n1)-c1ccc(F)cc1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cc1)C(=O)c1nc(C)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cn1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
CCN([C@@H](C)Cc1noc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-c1ncccn1 |r|
CCN([C@@H](C)Cn1cc(cn1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H](Cn1cc(cn1)-c1ccc(F)cn1)NC(=O)c1cc(C)ccc1-n1nccn1 |r|
CCN(CCn1ccc(n1)-c1ccc(F)cn1)C(=O)c1cc(C)ccc1-n1nccn1
Cc1ccc(c(c1)C(=O)NCCn1ccc(n1)-c1ccc(F)cn1)-n1nccn1
CC[C@@H](Cn1ccc(n1)-c1ccc(F)cn1)N(C)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12Oc3cccc4C[C@@]5([H])N(CC[C@@]1(c34)[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1 |r,THB:32:11:7.15.8:16|
[H][C@]12Cc3ccc(OC)cc3[C@@]3(CCN1S(=O)(=O)c1ccccc1)C[C@H](CC[C@@]23O)N(C)C(=O)\C=C\c1ccoc1 |r,THB:15:14:3.10.2:28|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@]12Cc3ccc(OC)cc3[C@@]3(CCN1S(=O)(=O)c1ccccc1)C[C@@H](CC[C@@]23O)N(C)C(=O)\C=C\c1ccoc1 |r,THB:15:14:3.10.2:28|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5([H])CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1)ccc3OC |r,THB:29:9:13:6.4.5|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14C5=CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1)ccc3OC |r,t:16,THB:28:9:13:6.4.5|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14C5=CC[C@@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1)ccc3OC |r,t:16,THB:28:9:13:6.4.5|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5([H])CC[C@@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1)ccc3OC |r,THB:29:9:13:6.4.5|
CCOc1ccc(cc1)-c1cc(C(=O)c2ccccc2)c2ccc(ccc12)C(O)=O
COC(=O)c1cccc2c(C=O)cc(I)c2c1
COC(=O)c1cc(CN2CCOCC2)c2ccc(Cl)ccc12
CC1(C)OC[C@H](NC(=O)Nc2ccc(Br)cc2Cl)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2-c2cccc(Cl)c2)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](NC(=O)Nc2ccccc2-c2ccccc2)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](NC(=O)Nc2ccc(Br)cc2)[C@@H](O1)c1ccccc1 |r|
Cc1ccc(Cl)c(NC(=O)N[C@H]2COC(C)(C)O[C@H]2c2ccccc2)c1 |r|
CC1(C)OC[C@H](NC(=O)Nc2c(Cl)cccc2Cl)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccc(Cl)cc2Cl)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](\N=C(/S)Nc2ccc(Cl)cc2Cl)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](NC(=O)Nc2ccccc2F)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2-c2cccs2)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](\N=C(/S)Nc2ccccc2Br)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](NC(=O)Nc2ccccc2I)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2-c2ccccc2Cl)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](NC(=O)Nc2ccccc2C(F)(F)F)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2Br)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2cc(Cl)ccc2Cl)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2cccc(Br)c2)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2Cl)[C@@H](O1)c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)c2ccc(Cl)cc2Cl)[C@@H](O1)c1ccccc1
CC(C)c1ccccc1NC(=O)N[C@H]1COC(C)(C)O[C@H]1c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2-c2ccsc2)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](NC(=O)Cc2ccccc2Br)[C@@H](O1)c1ccccc1
Cc1ccc(NC(=O)N[C@H]2COC(C)(C)O[C@H]2c2ccccc2)c(C)c1 |r|
CC1(C)OC[C@H](NC(=O)Nc2ccccc2-c2cccnc2)[C@@H](O1)c1ccccc1
Cc1ccc(\N=C(/NC#N)N[C@H]2COC(C)(C)O[C@H]2c2ccccc2)c(Br)c1
Cc1cc(Br)ccc1NC(=O)N[C@H]1COC(C)(C)O[C@H]1c1ccccc1 |r|
COc1ccccc1NC(=O)N[C@H]1COC(C)(C)O[C@H]1c1ccccc1 |r|
CC1(C)OC[C@H](NC(=O)Oc2ccccc2Cl)[C@@H](O1)c1ccccc1
CC1(C)OC[C@H](NC(=O)Nc2ccc(Br)cc2Br)[C@@H](O1)c1ccccc1 |r|
CCN(Cc1cccnc1)C(=O)CN(c2ccc(nc2)OC)S(=O)(=O)c3ccccc3C
CS(=O)(=O)c1cc(cnc1)N2C(=O)N(c3c(cccn3)S2(=O)=O)Cc4c(cc(cc4F)F)F
Cc1nc2ccc(cc2o1)NC(=O)Nc3ccnc4c3nccc4
Cc1cc(c2cc(cc(c2n1)F)F)NC(=O)Nc3ccc(cc3)N(C)C
c1ccc(cc1)S(=O)(=O)N2CCCC23CCN(CC3)c4nc5ccccc5o4
C[C@H]1CC[C@H](N(C1)C(=O)c2cccc(c2OC)F)CNc3ccc(cn3)Br
COc1cc(cnc1OC)N2C(=O)N(c3c(cccn3)S2(=O)=O)Cc4c(cc(cc4F)F)F
Cc1c(cnc(n1)C)OC[C@]2(C[C@H]2C(=O)Nc3ccc(cn3)F)c4cccc(c4)F
Cc1ccc(c(c1)C(=O)N2CCN(CC[C@H]2C)c3nc4cc(ccc4o3)Cl)n5nccn5
[H][C@]12C[C@H](CC[C@@]1(O)[C@@H](Cc1ccc(OC)cc21)N(CC1CC1)S(=O)(=O)c1ccccc1)N(C)C(=O)\C=C\c1ccoc1 |r|
[H][C@]12C[C@@H](CC[C@@]1(O)[C@@H](Cc1ccc(OC)cc21)N(CC1CC1)S(=O)(=O)c1ccccc1)N(C)C(=O)\C=C\c1ccoc1 |r|
[H][C@]12Oc3c4c(C[C@@H](N(CC5CC5)S(=O)(=O)c5ccccc5)[C@]([H])(CC[C@H]1N(C)C(=O)\C=C\c1ccoc1)[C@]24[H])ccc3OC |r|
[H][C@]12Oc3c4c(C[C@@H](N(CC5CC5)S(=O)(=O)c5ccccc5)[C@](O)(CC[C@H]1N(C)C(=O)\C=C\c1ccoc1)[C@]24[H])ccc3OC |r|
[H][C@@]12CC[C@@H](C[C@]1([H])c1cc(OC)ccc1C[C@H]2N(CC1CC1)S(=O)(=O)c1ccccc1)N(C)C(=O)\C=C\c1ccoc1 |r|
[H][C@]12Oc3c4c(C[C@@H](N(CC5CC5)S(=O)(=O)c5ccccc5)[C@]([H])(CC[C@@H]1N(C)C(=O)\C=C\c1ccoc1)[C@]24[H])ccc3OC |r|
[H][C@]12Oc3c4c(C[C@@H](N(CC5CC5)S(=O)(=O)c5ccccc5)[C@](O)(CC[C@@H]1N(C)C(=O)\C=C\c1ccoc1)[C@]24[H])ccc3OC |r|
[H][C@@]12CC[C@H](C[C@]1([H])c1cc(OC)ccc1C[C@H]2N(CC1CC1)S(=O)(=O)c1ccccc1)N(C)C(=O)\C=C\c1ccoc1 |r|
CN([C@@H]1CC[C@@]2(O)[C@H]3CC4=C(CCCC4)[C@@]2(CCN3S(=O)(=O)c2ccccc2)C1)C(=O)\C=C\c1ccoc1 |r,t:9,THB:19:18:9.10.8:5|
COc1ccc2C[C@H]3N(CC[C@@]4(C[C@H](CC=C34)N(C)C(=O)\C=C\c3ccoc3)c2c1)S(=O)(=O)c1ccccc1 |r,t:15,THB:30:8:5.28.6:16|
COc1ccc2C[C@H]3N(CC[C@@]4(C[C@@H](CC=C34)N(C)C(=O)\C=C\c3ccoc3)c2c1)S(=O)(=O)c1ccccc1 |r,t:15,THB:30:8:5.28.6:16|
CN([C@H]1CC[C@@]2(O)[C@H]3Cc4ccccc4[C@@]2(CCN3S(=O)(=O)c2ccccc2)C1)C(=O)\C=C\c1ccoc1 |r,THB:19:18:9.14.8:5|
CN([C@@H]1CC[C@@]2(O)[C@H]3Cc4ccccc4[C@@]2(CCN3S(=O)(=O)c2ccccc2)C1)C(=O)\C=C\c1ccoc1 |r,THB:19:18:9.14.8:5|
[H][C@@]12CC[C@H](C[C@@]11CCN([C@@H]2Cc2ccc(OC)cc12)S(=O)(=O)c1ccccc1)N(C)C(=O)\C=C\c1ccoc1 |r,THB:20:9:12.19.11:1|
[H][C@@]12CC[C@@H](C[C@@]11CCN([C@@H]2Cc2ccc(OC)cc12)S(=O)(=O)c1ccccc1)N(C)C(=O)\C=C\c1ccoc1 |r,THB:20:9:12.19.11:1|
CN([C@H]1CC[C@@]2(O)[C@H]3CC4=C(CCCC4)[C@@]2(CCN3S(=O)(=O)c2ccccc2)C1)C(=O)\C=C\c1ccoc1 |r,t:9,THB:19:18:9.10.8:5|
FC1(F)CCN(CC1Oc1ccc2ccccc2n1)C(=O)c1nccc2[nH]cnc12
COc1ccc(CCNC(=O)Cn2c(nc3ccccc23)-c2nonc2N)cc1OC
COc1ccc(cc1)N(CC(=O)NC(C)c1ccccc1)S(=O)(=O)c1ccc(OC)c(OC)c1
COC(=O)CN(C(c1ccccc1)c1cc(Br)ccc1NC(=O)c1ccccc1Cl)C(C)=O
Cc1ccc(cc1)C(O)(C(=O)NNc1cc(Cl)ccc1Cl)c1ccc(C)cc1
COc1ccccc1OCCNC[C@@H](O)COc1cccc2[nH]c3ccccc3c12 |r|
Cc1cccc2c3nnc(N\N=C/c4c5ccccc5cc5ccccc45)nc3[nH]c12
O=C(CSc1nnc(-c2cccs2)n1Cc1ccco1)Nc1ccc2OCCOc2c1
CCOC(=O)c1c(NC(=O)C(C)Sc2nnc(CNC(=O)c3cc(OC)cc(OC)c3)n2-c2ccccc2OC)sc2CCCc12 |(63.07,-14.05,;64.53,-14.53,;64.86,-16.03,;66.32,-16.51,;67.47,-15.47,;66.65,-18.01,;65.61,-19.17,;64.08,-19.01,;63.18,-20.25,;63.81,-21.66,;61.65,-20.1,;61.02,-18.69,;60.74,-21.34,;59.21,-21.18,;58.44,-19.85,;56.93,-20.17,;56.78,-21.71,;55.45,-22.48,;54.11,-21.72,;52.78,-22.49,;52.78,-24.03,;51.44,-21.72,;51.44,-20.17,;50.1,-19.41,;50.1,-17.87,;51.43,-17.09,;48.77,-20.18,;48.77,-21.72,;47.44,-22.49,;47.44,-24.03,;50.11,-22.49,;58.18,-22.33,;58.51,-23.84,;59.97,-24.3,;60.3,-25.8,;59.15,-26.84,;57.69,-26.37,;57.36,-24.87,;55.9,-24.39,;54.75,-25.42,;66.39,-20.49,;67.9,-20.17,;69.31,-20.79,;70.34,-19.64,;69.56,-18.31,;68.05,-18.64,)|
C\C(\C=C\c1ccccc1)=N\Nc1nc(Nc2ccccc2)nc(n1)-n1nc(C)cc1C
COc1ccccc1N1C(=O)c2ccccc2NC11C(=O)N(CC=C)c2ccccc12
[H][C@@]12Oc3c4C1[C@@](O)(CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)[C@@H](Cc4ccc3OC)N(CC1CC1)C(=O)OC(C)(C)C |r|
[H][C@@]12Oc3c4C1[C@@](O)(CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)[C@@H](Cc4ccc3OC)N(CC1CC1)C(C)=O |r|
[H][C@@]12Oc3c4C1[C@@](O)(CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)[C@@H](Cc4ccc3OC)N(CC1CC1)C(=O)C1CC1 |r|
[H][C@@]12Oc3c4C1[C@@](O)(CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)[C@@H](Cc4ccc3OC)N(CC1CC1)C(=O)c1ccccc1 |r|
[H][C@@]12Oc3c4C1[C@]1(CC[C@H]2N(C)C(=O)\C=C\c2ccoc2)OC(=O)N(CC2CC2)[C@]1([H])Cc4ccc3OC |r|
[H][C@@]12Oc3c4C1[C@]1(CC[C@H]2N(C)C(=O)\C=C\c2ccoc2)OS(=O)(=O)N(CC2CC2)[C@]1([H])Cc4ccc3OC |r|
[H][C@@]12Oc3c4C1[C@@]([H])(CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)[C@@H](Cc4ccc3OC)N(CC1CC1)C(=O)OC(C)(C)C |r|
[H][C@@]12Oc3c4C1[C@@]([H])(CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)[C@@H](Cc4ccc3OC)NCC1CC1 |r|
[H][C@@]12Oc3c4C1[C@@]([H])(CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)[C@@H](Cc4ccc3OC)N(C)CC1CC1 |r|
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CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N4CCC[C@H]4C(=O)N5CCC[C@H]5C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CSCC[C@H](N)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)CCSC)[C@@H](C)O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
Nc1nc2ccc(NC(=O)Nc3ccnc4cccnc34)cc2o1
Cc1nc(C(=O)N2CCC[C@H]2Cc2nnc(o2)-c2ccccc2)c(s1)-c1ccccc1F |r|
CN(Cc1[nH]cc[n+]1C)C(=O)C[C@H]1CN(Cc2ccccc2)CCO1 |r|
Fc1ccccc1COc1ccc2ccccc2c1C=C1C(=O)NC(=O)NC1=O
Cc1nn(c(N2CCCC2)c1\C=N\n1cnc2n(ncc2c1=O)-c1ccccc1)-c1ccccc1
O=C1N(c2ccccc2\C1=C/c1ccc(cc1)N1CCOCC1)c1ccccc1
COc1ccc2cc(CN(C)C(=O)COC(=O)c3c(F)cccc3F)ccc2c1
Cc1nc(COc2ccc(cc2)C(=O)N2CCC[C@@H]2c2ccc3OCCOc3c2)cs1 |r|
COc1cc(=O)n2CCN(CCc2c1C(=O)N(C)[C@H](C)c1ccco1)C(=O)C1(CC1)c1ccccc1 |r|
Fc1cccc(\C=C\C(=O)N2CCOc3c(C2)cc(cc3OC[C@H]2CCCCO2)-c2cccnc2)c1 |r|
COc1cc(=O)n2CCN(CCc2c1C(=O)N(C)Cc1nonc1C)C(=O)C1(CC1)c1ccccc1
Fc1cccc2sc(C(=O)N3CCN(Cc4ccco4)CC3)c(Cl)c12
Cc1[nH]c2ccccc2c1[C@H]1N(CCC(=O)N2CCN(CC2)c2ccccn2)C(=O)c2ccccc12 |r|
Cc1c(oc2c(C)c(C)ccc12)C(=O)N1CCN(Cc2ccccn2)CC1
Cc1[nH]c2ccc(cc2c1C)C(=O)N1CCN(Cc2ccc3OCOc3c2)CC1
Cc1ccc(CSCc2ccc(o2)-c2nc(no2)-c2ccccn2)cc1
O=C(N1CCC[C@@H]1c1ccc2OCCOc2c1)c1ccc(OCc2cn3ccccc3n2)cc1 |r|
CN(Cc1c(F)cccc1Cl)C(=O)Cc1csc(n1)-c1ccc(C)o1
Cc1ccc(nn1)N1CCCN(CC1)C(=O)c1cn(C)c2ccccc12
C[C@@H](Oc1ccc2c(c1)oc(=O)c1ccccc21)C(=O)c1ccccc1 |r|
O=S(=O)(N1CCN(Cc2nc(cs2)-c2ccco2)CC1)c1ccc2OCCOc2c1
Clc1ccc(cc1C(=O)N1CCn2c1nc1ccccc21)S(=O)(=O)N1CCOCC1
Cn1c(c(C(=O)COC(=O)c2ccc3c(c2)nc2CCCn2c3=O)c2ccccc12)-c1ccccc1
Cc1nc(no1)-c1ccc(Cl)c(c1)S(=O)(=O)N1CCC[C@H](C1)C(=O)N1CCc2ccccc12 |r|
COc1ccc([C@H]2CCCN2C(=O)c2ccc(OCc3cn4ccccc4n3)cc2)c(OC)c1 |r|
Cc1nc2cc(F)cc(C(=O)NCCOc3ccc4ccccc4c3)c2nc1C
CN(CCc1cccc2ccccc12)C(=O)c1c[nH]c(=O)c(Cl)c1
CN1C(=O)c2ccc(cc2C1=O)C(=O)OCCCn1c2ccccc2[nH]c1=O
OC1=NC(=O)N(C(=O)\C1=C\c1ccccc1OCc1ccccc1F)c1ccc2OCOc2c1 |t:1|
C[C@@H]1CN(C(=O)CN1C(=O)c1cccc2ccccc12)c1cccc(Cl)c1 |r|
Fc1ccc(CN(C2CC2)C(=O)c2cccc(c2)N2CCCC2=O)cc1
C[C@H](Oc1cccc(c1)N1C(=O)C2C3CC(C=C3)C2C1=O)C(=O)c1ccc(C)cc1 |r,c:17,TLB:10:12:14:16.17,THB:19:18:14:16.17|
[H][C@]12CC=C[C@@H](C)[C@]1([H])C(=O)N(C2=O)c1cccc(O[C@@H](C)C(=O)c2ccc(C)cc2)c1 |r,c:3|
COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)NCc3ccccn3)c2c1
O=C(N1CCN(Cc2csc(n2)-c2ccco2)CC1)c1ccccc1Cc1ccccc1
O=C(N1CCN(Cc2cc(=O)n3ccsc3n2)CC1)c1cc2CCc3ccccc3-c2s1
O=C(N(CCc1ccccc1)c1nc2ccccc2s1)C1=NN([C@H]2CCS(=O)(=O)C2)C(=O)CC1 |r,t:23|
Cc1ccccc1OC[C@@H]1CCCN(C1)C(=O)CCc1nc(no1)-c1ccccn1 |r|
O=C(CCc1nc(no1)-c1ccco1)N1CCC[C@@H](C1)C(=O)c1ccccc1 |r|
O=C(Nc1cccc(\C=C\c2ccccn2)c1)c1occc1COc1ccccc1
C[C@H](N(C)C(=O)Cc1csc(n1)-c1ccc(C)o1)c1ccc(F)cc1 |r|
CN(Cc1ccccc1C)C(=O)Cc1csc(n1)-c1cccc(F)c1
Fc1cc(F)cc(c1)S(=O)(=O)N1CCN(Cc2csc(n2)-c2ccco2)CC1
C[C@H](Sc1nc(nc2ccccc12)-c1ccco1)C(=O)N1CCc2ccccc2C1 |r|
O=C(N(Cc1ccco1)Cc1ccco1)c1ccc(o1)-c1nc2ccccc2s1
Cc1nc(\C=C\C(=O)Oc2ccc3c(c2)oc(C)c(-c2c(F)cccc2Cl)c3=O)cs1 |(30.51,-27.54,;30,-26.41,;28.49,-26.09,;28.36,-24.57,;27.02,-23.8,;27.02,-22.26,;25.69,-21.48,;24.62,-22.1,;25.69,-19.94,;24.35,-19.17,;24.35,-17.63,;23.02,-16.86,;21.69,-17.63,;21.69,-19.17,;23.02,-19.94,;20.36,-19.94,;19.02,-19.17,;17.95,-19.78,;19.02,-17.63,;17.69,-16.85,;16.35,-17.62,;16.35,-18.86,;15.02,-16.85,;15.02,-15.31,;16.35,-14.54,;17.69,-15.31,;18.76,-14.7,;20.36,-16.86,;20.36,-15.62,;29.74,-23.93,;30.77,-25.08,)|
COc1ccc(cc1)C(=O)Oc1cc(=O)n(c2CCCCc12)-c1ccccc1
Cc1ccc(Oc2ncccc2NC(=O)c2ccc3OCCCOc3c2)c2CCCc12
O=C(CCC(=O)c1ccc2OCCOc2c1)Nc1cccc(c1)C#Cc1ccccn1
[H][C@@]12CCCCN1c1ccc(cc1NC2=O)C(=O)N1CCN(Cc2ccc3OCOc3c2)CC1 |r|
Cc1cc(no1)[C@@H]1CCCCN1C(=O)c1ccc(cc1)-c1cc[nH]n1 |r|
O=C(N1CCC[C@H]1c1ccncc1)c1cnc(s1)-c1ccccc1 |r|
COc1cccc(c1)-c1nc(C(=O)OCc2cccnc2)c(C)[nH]1
Fc1ccccc1COc1cccc(CNCc2ccccn2)c1
Cc1ccc(cc1)[C@H](CCO)n1cc(nn1)-c1ccnc2ccccc12 |r|
Cc1[nH]c2ccc(C)cc2c1CC(=O)N(Cc1cccnc1)C1CC1
CC(=O)N1N=C(O[C@@H]1c1cccnc1)c1cn(C(C)=O)c2ccccc12 |r,c:4|
O=C(CCCn1nnc2ccccc2c1=O)NC1Cc2ccccc2C1
Cc1cccc(C)c1NC(=O)CCCN1C(=O)c2cccnc2C1=O
COc1cccc(c1)-c1nc(no1)[C@H]1CN(Cc2ccccc2)C(=O)C1 |r|
C(c1ccncc1)n1ncc2[nH]c(nc12)-c1c[nH]nc1-c1ccccc1
COc1ccc(C[C@@H]2N(CCc3cc(OC)c(OC)cc23)[C@@H](C(=O)NC(C)C)c2ccccc2)cc1OC |r|
FC1(F)CCN(C[C@@H]1Oc1ccc2ccccc2n1)C(=O)c1nccc2[nH]cnc12 |r|
FC1(F)CCN(C[C@@H]1Oc1ccc2ccccc2n1)C(=O)c1cccn2ccnc12 |r|
[H][C@@]12CC[C@@]([H])([C@@H](C1)Nc1cnc(cn1)C(F)(F)F)N2C(=O)c1ccccc1-c1ncccn1 |r,TLB:8:6:2.3:19|
[H][C@@]12CC[C@@]([H])([C@@H](C1)Nc1cnc(cn1)C(F)(F)F)N2C(=O)c1c(F)cccc1-c1ncccn1 |r,TLB:8:6:2.3:19|
[H][C@@]12CC[C@@]([H])([C@@H](C1)Nc1cnc(cn1)C(F)(F)F)N2C(=O)c1cc(F)ccc1-c1ncccn1 |r,TLB:8:6:2.3:19|
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CC(C)C[C@H](NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CO)NC(=O)[C@@H](N)CCCNC(N)=N)C(=O)N[C@@H](CCC(N)=O)C(=O)NCC(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)CN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCSC)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NCCCCCC(=O)[C@H](CC(O)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCC(=O)N1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)CN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCSC)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(CCN)C(=O)[C@H](CO)NC(=O)[C@H](CS)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCNC(N)=N)NC(CCN)C(=O)[C@H](CS)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCC(=O)N1)[C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)CN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCSC)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)CN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCSC)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)CN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCSC)C(O)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)CN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCSC)C(O)=O
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(=O)N(C)C
CCN(CC)C(=O)c1cccc(c1)-c1ccc(OC)c(c1)S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(=O)N1CCCCC1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(=O)N1CCCC1
CCCNC(=O)c1cccc(c1)-c1ccc(OC)c(c1)S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(CN(C)C)c1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(C)C
CCN(CC)c1cccc(c1)-c1ccc(OC)c(c1)S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1
CCCN(CCC)c1cccc(c1)-c1ccc(OC)c(c1)S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(C)(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(F)(F)F
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCCNC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCC(C)NC(=O)c2ccccc2N(C)C)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCC(C)NC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(c1)N1CCN(CC1)C(=O)c1ccccc1N(C)C)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(c1)N1CCN(CC1)C(=O)c1cccc(C)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cc(ccn1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cncc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1ccnc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(n1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1csc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cc(cs1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1csc(n1)C(=O)N(C)C
COc1ccc(\C=C\C(=O)N(C)C)cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1
COc1ccc(CCC(=O)N(C)C)cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)CCN(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)NCCN(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)c1ccccn1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)Cc1ccccc1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)Cc1ccccn1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)NCc1ccccn1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)Cc1cccnc1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)Cc1ccncc1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)CCc1ccccn1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)CCc1ccncc1
COc1ccc(cc1C(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1C(=O)Nc1cccc(NCCNC(=O)c2cccc(C)c2)c1)-c1cccc(c1)C(=O)N(C)Cc1ccncc1
Cc1ccc(Cn2c3ccccc3n(CC(O)c3ccc(Cl)c(Cl)c3)c2=N)cc1
COC(=O)N1CCC[C@@H]([C@@H]1COC2CCC(CC2)c3ccccc3)NS(=O)(=O)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(CCNC(=O)c2ccccc2-n2nccn2)c1)-c1cccc(c1)C(=O)N(C)C
CCS(=O)(=O)N[C@@H]1CCCN([C@H]1CO[C@H]1CC[C@H](CC1)C(C)C)C(C)=O |r,wU:11.12,14.14,17.21,wD:6.5,(6.67,1.54,;5.33,.77,;4,1.54,;4.77,2.88,;3.23,2.88,;2.67,.77,;2.67,-.77,;4,-1.54,;4,-3.08,;2.67,-3.85,;1.33,-3.08,;1.33,-1.54,;-0,-.77,;-0,.77,;-1.33,1.54,;-2.67,.77,;-4,1.54,;-4,3.08,;-2.67,3.85,;-1.33,3.08,;-5.33,3.85,;-6.67,3.08,;-5.33,5.39,;-0,-3.85,;-1.33,-3.08,;-0,-5.39,)|
CCS(=O)(=O)N[C@H]1CCCN([C@H]1CO[C@H]1CC[C@@H](CC1)C(C)C)C(C)=O |r,wU:6.5,11.12,14.14,wD:17.21,(6.67,1.54,;5.33,.77,;4,1.54,;4.77,2.88,;3.23,2.88,;2.67,.77,;2.67,-.77,;4,-1.54,;4,-3.08,;2.67,-3.85,;1.33,-3.08,;1.33,-1.54,;-0,-.77,;-0,.77,;-1.33,1.54,;-2.67,.77,;-4,1.54,;-4,3.08,;-2.67,3.85,;-1.33,3.08,;-5.33,3.85,;-6.67,3.08,;-5.33,5.39,;-0,-3.85,;-1.33,-3.08,;-0,-5.39,)|
CCS(=O)(=O)N[C@H]1CCCN([C@H]1CO[C@H]1CC[C@H](CC1)C(C)C)C(C)=O |r,wU:14.14,11.12,6.5,17.21,(6.67,1.54,;5.33,.77,;4,1.54,;3.23,2.87,;4.77,2.87,;2.67,.77,;2.67,-.77,;4,-1.54,;4,-3.08,;2.67,-3.85,;1.33,-3.08,;1.33,-1.54,;,-.77,;,.77,;-1.33,1.54,;-2.67,.77,;-4,1.54,;-4,3.08,;-2.67,3.85,;-1.33,3.08,;-5.33,3.85,;-5.33,5.39,;-6.67,3.08,;,-3.85,;-1.33,-3.08,;,-5.39,)|
CCS(=O)(=O)N[C@@H]1CCCN([C@H]1CO[C@H]1CC[C@@H](CC1)C(C)C)C(C)=O |r,wU:11.12,14.14,wD:6.5,17.21,(6.67,1.54,;5.33,.77,;4,1.54,;4.77,2.88,;3.23,2.88,;2.67,.77,;2.67,-.77,;4,-1.54,;4,-3.08,;2.67,-3.85,;1.33,-3.08,;1.33,-1.54,;-0,-.77,;-0,.77,;-1.33,1.54,;-2.67,.77,;-4,1.54,;-4,3.08,;-2.67,3.85,;-1.33,3.08,;-5.34,3.85,;-6.67,3.08,;-5.34,5.39,;-0,-3.85,;-1.33,-3.08,;-0,-5.39,)|
CC(C)[C@@H]1CC[C@@H](CC1)OC[C@H]1[C@H](CCCN1C(C)=O)NS(C)(=O)=O |r,wU:3.2,6.9,11.11,12.21,(-6,3.08,;-4.67,3.85,;-4.67,5.39,;-3.33,3.08,;-3.33,1.54,;-2,.77,;-.67,1.54,;-.67,3.08,;-2,3.85,;.67,.77,;.67,-.77,;2,-1.54,;3.33,-.77,;4.67,-1.54,;4.67,-3.08,;3.33,-3.85,;2,-3.08,;.67,-3.85,;-.67,-3.08,;.67,-5.39,;3.33,.77,;4.67,1.54,;6,.77,;3.9,2.87,;5.44,2.87,)|
CC(C)[C@@H]1CC[C@@H](CC1)OC[C@H]1[C@H](CCCN1C(C)=O)NS(=O)(=O)C(C)C |r,wU:3.2,6.9,11.11,12.21,(-6.67,3.08,;-5.33,3.85,;-5.33,5.39,;-4,3.08,;-4,1.54,;-2.67,.77,;-1.33,1.54,;-1.33,3.08,;-2.67,3.85,;,.77,;,-.77,;1.33,-1.54,;2.67,-.77,;4,-1.54,;4,-3.08,;2.67,-3.85,;1.33,-3.08,;,-3.85,;-1.33,-3.08,;,-5.39,;2.67,.77,;4,1.54,;3.23,2.87,;4.77,2.87,;5.33,.77,;6.67,1.54,;5.33,-.77,)|
CCCS(=O)(=O)N[C@H]1CCCN([C@H]1CO[C@H]1CC[C@H](CC1)C(C)C)C(C)=O |r,wU:18.22,15.15,12.13,7.6,(7.34,.77,;6,1.54,;4.67,.77,;3.33,1.54,;2.56,2.87,;4.1,2.87,;2,.77,;2,-.77,;3.33,-1.54,;3.33,-3.08,;2,-3.85,;.67,-3.08,;.67,-1.54,;-.67,-.77,;-.67,.77,;-2,1.54,;-3.33,.77,;-4.67,1.54,;-4.67,3.08,;-3.33,3.85,;-2,3.08,;-6,3.85,;-7.34,3.08,;-6,5.39,;-.67,-3.85,;-2,-3.08,;-.67,-5.39,)|
CC(C)[C@@H]1CC[C@@H](CC1)OC[C@H]1[C@H](CCCN1C(C)=O)N(C)S(C)(=O)=O |r,wU:12.21,11.11,6.9,3.2,(-6,3.08,;-4.67,3.85,;-4.67,5.39,;-3.33,3.08,;-3.33,1.54,;-2,.77,;-.67,1.54,;-.67,3.08,;-2,3.85,;.67,.77,;.67,-.77,;2,-1.54,;3.33,-.77,;4.67,-1.54,;4.67,-3.08,;3.33,-3.85,;2,-3.08,;.67,-3.85,;-.67,-3.08,;.67,-5.39,;3.33,.77,;2,1.54,;4.67,1.54,;6,.77,;5.44,2.88,;3.9,2.88,)|
CC(C)[C@@H]1CC[C@@H](CC1)OC[C@H]1[C@H](CCCN1C(C)=O)NC(O)=O |r,wU:12.21,11.11,6.9,3.2,(-6,3.08,;-4.67,3.85,;-4.67,5.39,;-3.33,3.08,;-3.33,1.54,;-2,.77,;-.67,1.54,;-.67,3.08,;-2,3.85,;.67,.77,;.67,-.77,;2,-1.54,;3.33,-.77,;4.67,-1.54,;4.67,-3.08,;3.33,-3.85,;2,-3.08,;.67,-3.85,;-.67,-3.08,;.67,-5.39,;3.33,.77,;4.67,1.54,;6,.77,;4.67,3.08,)|
C[C@H]1CC[C@H](CC1)OC[C@H]1[C@H](CCCN1C(C)=O)NS(C)(=O)=O |r,wU:1.0,4.7,9.9,10.19,(-5.33,4.62,;-4,3.85,;-2.67,4.62,;-1.33,3.85,;-1.33,2.31,;-2.67,1.54,;-4,2.31,;,1.54,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;,-4.62,;2.67,1.54,;4,2.31,;5.33,1.54,;3.23,3.64,;4.77,3.64,)|
CC(=O)N1CCC[C@H](NS(C)(=O)=O)[C@@H]1CO[C@H]1CC[C@H](CC1)c1ccccc1 |r,wU:19.23,16.16,13.14,7.7,(,-3.47,;1.33,-4.23,;1.33,-5.78,;2.67,-3.47,;4,-4.24,;5.33,-3.47,;5.33,-1.93,;4,-1.16,;4,.38,;5.33,1.15,;6.67,.38,;4.56,2.49,;6.1,2.49,;2.67,-1.93,;1.33,-1.16,;1.33,.38,;,1.15,;-1.33,.38,;-2.67,1.15,;-2.67,2.69,;-1.33,3.46,;,2.69,;-4,3.46,;-4,5,;-5.33,5.78,;-6.67,5,;-6.67,3.46,;-5.33,2.69,)|
CS(=O)(=O)N[C@H]1CCCN[C@H]1CO[C@H]1CC[C@H](CC1)c1ccccc1 |r,wU:16.20,13.13,10.11,5.4,(6.99,-1.33,;5.9,-.24,;5.5,1.25,;6.99,.85,;4.41,-.64,;4.01,-2.12,;5.1,-3.21,;4.7,-4.7,;3.21,-5.1,;2.12,-4.01,;2.52,-2.52,;1.43,-1.43,;-.05,-1.83,;-1.14,-.74,;-2.63,-1.14,;-3.72,-.05,;-3.32,1.43,;-1.83,1.83,;-.74,.74,;-4.41,2.52,;-4.01,4.01,;-5.1,5.1,;-6.59,4.7,;-6.99,3.21,;-5.9,2.12,)|
CCC(=O)N1CCC[C@H](NS(C)(=O)=O)[C@@H]1CO[C@H]1CC[C@H](CC1)c1ccccc1 |r,wU:20.24,17.17,14.15,8.8,(-1.33,-4.24,;,-3.47,;1.33,-4.24,;1.33,-5.78,;2.67,-3.47,;4,-4.24,;5.33,-3.47,;5.33,-1.93,;4,-1.16,;4,.38,;5.33,1.16,;6.67,.38,;4.56,2.49,;6.1,2.49,;2.67,-1.93,;1.33,-1.16,;1.33,.38,;,1.16,;-1.33,.39,;-2.67,1.16,;-2.67,2.7,;-1.33,3.47,;,2.7,;-4,3.47,;-4,5.01,;-5.33,5.78,;-6.67,5.01,;-6.67,3.47,;-5.33,2.7,)|
CCOC(=O)N1CCC[C@H](NS(C)(=O)=O)[C@@H]1CO[C@H]1CC[C@H](CC1)c1ccccc1 |r,wU:21.25,18.18,15.16,9.9,(-3.03,-2.23,;-1.94,-3.32,;-.45,-2.92,;.64,-4.01,;.24,-5.5,;2.12,-3.61,;3.21,-4.7,;4.7,-4.3,;5.1,-2.81,;4.01,-1.73,;4.41,-.24,;5.9,.16,;6.99,-.93,;5.5,1.65,;6.99,1.25,;2.52,-2.12,;1.43,-1.04,;-.05,-1.43,;-1.14,-.35,;-2.63,-.74,;-3.72,.35,;-3.32,1.83,;-1.83,2.23,;-.74,1.14,;-4.41,2.92,;-4.01,4.41,;-5.1,5.5,;-6.59,5.1,;-6.99,3.61,;-5.9,2.52,)|
CCNC(=O)N1CCC[C@H](NS(C)(=O)=O)[C@@H]1CO[C@H]1CC[C@H](CC1)c1ccccc1 |r,wU:21.25,18.18,15.16,9.9,(.93,-6.79,;1.33,-5.3,;.24,-4.21,;.64,-2.72,;-.45,-1.63,;2.12,-2.32,;3.21,-3.41,;4.7,-3.01,;5.1,-1.53,;4.01,-.44,;4.41,1.05,;5.9,1.45,;6.99,.36,;5.5,2.94,;6.99,2.54,;2.52,-.84,;1.43,.25,;-.05,-.15,;-1.14,.94,;-2.63,.54,;-3.72,1.63,;-3.32,3.12,;-1.83,3.52,;-.74,2.43,;-4.41,4.21,;-4.01,5.7,;-5.1,6.79,;-6.59,6.39,;-6.99,4.9,;-5.9,3.81,)|
CCS(=O)(=O)NC1CCCN(C1COC1CCC(CC1)C(C)C)C(C)=O |(6.67,1.54,;5.33,.77,;4,1.54,;4.77,2.88,;3.23,2.88,;2.67,.77,;2.67,-.77,;4,-1.54,;4,-3.08,;2.67,-3.85,;1.33,-3.08,;1.33,-1.54,;-0,-.77,;-0,.77,;-1.33,1.54,;-2.67,.77,;-4,1.54,;-4,3.08,;-2.67,3.85,;-1.33,3.08,;-5.33,3.85,;-6.67,3.08,;-5.33,5.39,;-0,-3.85,;-1.33,-3.08,;-0,-5.39,)|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CS)NC(=O)[C@H](CO)NC(=O)[C@H](CS)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CS)NC(=O)[C@H](CS)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCC(=O)N1)[C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(O)=O |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(c1)N(C)C)[C@@](C)(O2)c1cccc(c1)N(C)C |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)OC(C)(C)C)c1)[C@@](C)(O2)c1cccc(NC(=O)OC(C)(C)C)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccccc3)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccccc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccccc3)c1)[C@](C)(O2)c1cccc(NC(=O)c2ccccc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1ccc(NS(=O)(=O)c3ccccc3)cc1)[C@@](C)(O2)c1cccc(NS(=O)(=O)c2ccccc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccccc3OC)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccccc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3cccc(OC)c3)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccccc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccccc3OC)c1)[C@](C)(O2)c1cccc(NC(=O)c2cccc(OC)c2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3cccc(OC)c3)c1)[C@](C)(O2)c1cccc(NC(=O)c2cccc(OC)c2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccccc3N(C)C)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccccc2N(C)C)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3cccc(c3)N(C)C)c1)[C@@](C)(O2)c1cccc(NC(=O)c2cccc(c2)N(C)C)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccc(cc3)N(C)C)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccc(cc2)N(C)C)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccccc3N(C)C)c1)[C@](C)(O2)c1cccc(NC(=O)c2ccccc2N(C)C)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3cccc(c3)N(C)C)c1)[C@](C)(O2)c1cccc(NC(=O)c2cccc(c2)N(C)C)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccc(cc3)N(C)C)c1)[C@](C)(O2)c1cccc(NC(=O)c2ccc(cc2)N(C)C)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccccn3)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccccn2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3cccnc3)c1)[C@@](C)(O2)c1cccc(NC(=O)c2cccnc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccncc3)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccncc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccccn3)c1)[C@](C)(O2)c1cccc(NC(=O)c2ccccn2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3cccnc3)c1)[C@](C)(O2)c1cccc(NC(=O)c2cccnc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccncc3)c1)[C@](C)(O2)c1cccc(NC(=O)c2ccncc2)c1 |r|
COc1ccc(cc1)C(=O)Nc1cccc(c1)C1(C)OC2COC3N2C1OC3(C)c1cccc(NC(=O)c2ccc(OC)cc2)c1
[H][C@@]12CO[C@@]3([H])N1[C@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccc(OC)cc3)c1)[C@](C)(O2)c1cccc(NC(=O)c2ccc(OC)cc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccc(OC)cc3)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccc(OC)cc2)c1 |r|
[H][C@@]12CO[C@@]3([H])N1[C@]([H])(O[C@@]3(C)c1cccc(NC(=O)c3ccc(OC)cc3)c1)[C@@](C)(O2)c1cccc(NC(=O)c2ccc(OC)cc2)c1 |r|
[H][C@]12CO[C@]3([H])N1[C@@]([H])(O[C@]3(C)c1cccc(NC(=O)c3ccc(OC)cc3)c1)[C@](C)(O2)c1cccc(NC(=O)c2ccc(OC)cc2)c1 |r|
[H][C@]12Oc3c4c(C[C@]5([H])C(CC[C@H]1N(C)C(=O)\C=C\c1ccoc1)[C@]24CCN5CC1CC1)ccc3OC |r,THB:28:27:9:4.5.6|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC6CC6)CC[C@@]14C5=CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)ccc3OC |r,t:21,THB:10:9:5.6.4:17|
[H][C@]12Oc3c4c(C[C@]5([H])C(CC[C@H]1N(C)C(=O)\C=C\c1ccoc1)[C@]24CCN5CC1CC1)ccc3O |r,THB:28:27:9:4.5.6|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC6CC6)CC[C@@]14C5=CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)ccc3O |r,t:21,THB:10:9:17:4.5.6|
[H][C@@]12Cc3ccc(OC)c4O[C@@]5([H])[C@@H](CCC1[C@@]5(CN2CC1CC1)c34)N(C)C(=O)\C=C\c1ccoc1 |r,THB:20:19:16:2.3.24|
[H][C@@]12Cc3ccc(OC)c4O[C@@]5([H])[C@@H](CC=C1[C@@]5(CN2CC1CC1)c34)N(C)C(=O)\C=C\c1ccoc1 |r,t:15,THB:20:19:16:2.3.24|
[H][C@@]12Cc3ccc(O)c4O[C@@]5([H])[C@@H](CCC1[C@@]5(CN2CC1CC1)c34)N(C)C(=O)\C=C\c1ccoc1 |r,THB:19:18:15:2.3.23|
[H][C@@]12Cc3ccc(O)c4O[C@@]5([H])[C@@H](CC=C1[C@@]5(CN2CC1CC1)c34)N(C)C(=O)\C=C\c1ccoc1 |r,t:14,THB:19:18:15:2.3.23|
COc1ccc(cc1S(=O)(=O)Nc1ccc2ccc(NC(=O)c3ccccc3)cc2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2ccc(cc2c1)N(C)C(=O)c1ccccc1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2cccc(NC(=O)c3ccccc3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2cccc(N(C)C(=O)c3ccccc3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccccc1C(=O)N(C)c1cccc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
COc1cccc(c1)C(=O)N(C)c1cccc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
COc1ccc(cc1)C(=O)N(C)c1cccc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
COc1cccc(c1)C(=O)Nc1cccc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
COc1cccc(c1)C(=O)Nc1c(C)ccc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
COc1cccc(c1)C(=O)N(C)c1c(C)ccc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1N(C)C)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14C5=CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1N(C)C)ccc3OC |r,t:16,THB:28:9:13:6.5.4|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5([H])CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1N(C)C)ccc3OC |r,THB:29:9:13:6.5.4|
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)c3ccccc3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)Cc3ccccc3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)CCc3ccccc3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)Nc3ccccc3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)C3CCCCC3)c2c1)-c1cccc(c1)C(=O)N(C)C
CCCCC(=O)N(C)C1CCCc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
COc1ccccc1CC(=O)N(C)C1CCCc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12
COc1ccc(CC(=O)N(C)C2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)cc1
COc1cccc(CC(=O)N(C)C2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)Cc3cccc(O)c3)c2c1)-c1cccc(c1)C(=O)N(C)C
CCOc1cccc(CC(=O)N(C)C2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)Cc3cccc(c3)N(C)C)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)Cc3cccc(F)c3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1ccc2CCCC(N(C)C(=O)Cc3cccnc3)c2c1)-c1cccc(c1)C(=O)N(C)C
COc1cccc(CC(=O)OC2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1
COc1cccc(CC(=O)NC2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1
CCN(C1CCCc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12)C(=O)Cc1cccc(OC)c1
CCCN(C1CCCc2ccc(NS(=O)(=O)c3cc(ccc3OC)-c3cccc(c3)C(=O)N(C)C)cc12)C(=O)Cc1cccc(OC)c1
COc1cccc(CC(=O)N(CC2CC2)C2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1
COc1ccc(CN(C)C2CCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)cc1
COc1cccc(CC(=O)N(C)c2cccc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1
COc1cccc(CC(=O)N(C)c2cccc3CCC(Cc23)NS(=O)(=O)c2cc(ccc2OC)-c2cccc(c2)C(=O)N(C)C)c1
COc1cccc(CC(=O)N(C)[C@H]2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1 |r|
COc1cccc(CC(=O)N(C)[C@@H]2CCCc3ccc(NS(=O)(=O)c4cc(ccc4OC)-c4cccc(c4)C(=O)N(C)C)cc23)c1 |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H]1CSSC[C@@H]2NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCN=C(N)N)NC2=O)[C@@H](C)O)C(=O)N[C@@H](CO)C(=O)N1)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCC(=O)N1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O
COc1cccc(OC)c1C(=O)N1CCCN(CC1)c1nc2ccc(Cl)cc2s1
Cc1ccc(c(c1)C(=O)N1CCC[C@@H](COc2ccc(F)cn2)C1)-n1nccn1 |r|
Fc1ccc(cc1)S(=O)(=O)N(Cc1ncc[nH]1)c1ccccc1-c1ccccc1
Cc1ccc(c(c1)C(=O)N1CCCN(CC1)c1ncc2ccccc2n1)-n1nccn1
O=C1N2CCCN(CC2)c2ccc3cc(CCCCc4ccc(c1c4)-n1nccn1)ccc3c2
C=CCCCc1ccc2cc(ccc2c1)N1CCCN(CC1)C(=O)c1cc(CC=C)ccc1-n1nccn1
Cc1ccc(c(CN2CCCN(CC2)c2ncc3ccccc3n2)c1)-n1nccn1
O=C(C1CCCCC1)N1CCCN(CC1)c1ncc2ccccc2n1
Cc1ccc(c(c1)C(=O)N1CCCN(CC1)c1ccc2ccccc2c1)-n1nccn1
CNC1CCCC1CN[C@H](C(=O)N1CCc2cc(OC)c(OC)cc2C1)C(C)(C)C |r|
COc1cc2CCN(Cc2cc1OC)C(=O)C(Cc1ccccc1)C(=O)c1cc(Cl)cc(Cl)c1
COc1ccc(CC2N(CC(=O)NCc3ccccc3)CCc3cc(OC)c(OC)cc23)cc1OC
CNC(=O)[C@H](N1CCc2cc(OC)c(OC)cc2[C@@H]1CCc1ccc(cc1)C(F)(F)F)c1ccccc1 |r|
COc1cc2CCN(C(C(=O)NCC3CC3)c3ccccc3)C(CCc3ccc(F)c(F)c3)c2cc1OC
CCCCNC(=O)C(N1CCc2cc(OC)c(OC)cc2C1CCc1ccc(F)c(F)c1)c1ccccc1
CCCCNC(=O)C(N1CCc2cc(OC)c(OC)cc2C1Cc1ccc(cc1)N(C)C)c1ccccc1
COc1cc2CCN(C(C(=O)NC3CC3)c3ccccc3)C(Cc3ccc4ccccc4c3)c2cc1OC
COCCNC(=O)C(N1CCc2cc(OC)c(OC)cc2C1Cc1ccc2ccccc2c1)c1ccccc1
CCCCNC(=O)C(N1CCc2cc(OC)c(OC)cc2C1Cc1ccc(OC)c(OC)c1)c1ccccc1
COc1ccc(CC2N(CCc3cc(OC)c(OC)cc23)C(C(=O)Nc2ccc3OCOc3c2)c2ccccc2)cc1OC
COc1cc2CCN(CC(=O)NCc3ccccc3)C(Cc3ccc(Oc4ncccn4)c(OC)c3)c2cc1OC
COc1cc2CCN(CC(=O)NCc3ccccc3)C(Cc3ccc(C)c(C)c3)c2cc1OC
COc1cc2CCN(CC(=O)NCc3ccccc3)C(Cc3ccc(Cl)c(Cl)c3)c2cc1OC
COc1cc2CCN(CC(=O)NCc3ccccc3)C(Cc3ccc(F)c(F)c3)c2cc1OC
COc1cc2CCN(CC(=O)NCc3ccccc3)C(Cc3ccc4OCOc4c3)c2cc1OC
COc1ccc(CC2N(CC(=O)NCc3ccccc3)CCc3cc(OC)c(OC)cc23)cc1
COc1cccc(CC2N(CC(=O)NCc3ccccc3)CCc3cc(OC)c(OC)cc23)c1
COc1cc2CCN(CC(=O)NCc3ccccc3)C(Cc3ccccc3)c2cc1OC
COc1cc2CCN(CC(=O)NC3CCc4ccccc34)C(Cc3ccc(C)c(C)c3)c2cc1OC
COc1cc2CCN(CC(=O)NC3CCc4ccccc34)C(Cc3ccc(F)c(F)c3)c2cc1OC
COc1ccc(CC2N(CC(=O)NC3CCc4ccccc34)CCc3cc(OC)c(OC)cc23)cc1F
COc1cc2CCN(CC(=O)NC3CCc4ccccc34)C(Cc3ccc4OCOc4c3)c2cc1OC
COc1ccc(CC2N(CC(=O)NC3CCc4ccccc34)CCc3cc(OC)c(OC)cc23)cc1
COc1cccc(CC2N(CC(=O)NC3CCc4ccccc34)CCc3cc(OC)c(OC)cc23)c1
COc1cc2CCN(CC(=O)NC3CCc4ccccc34)C(Cc3ccccc3)c2cc1OC
COc1ccc2CCC(NC(=O)CN3CCc4cc(OC)c(OC)cc4C3Cc3ccc(OC)c(OC)c3)c2c1
COc1ccc(CC2N(CC(=O)NC3Cc4ccccc4C3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)NC3CCc4ccccc34)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)N(C)C3CCCCC3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)NCc3ccno3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)NCc3ccncc3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)NCc3cccnc3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)NCc3ccccn3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)N3CCc4ccccc4C3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)N(C)Cc3ccccc3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(CC2N(CC(=O)NC(C)c3ccccc3)CCc3cc(OC)c(OC)cc23)cc1OC
COc1ccc(C[C@@H]2N(CC(=O)NCCc3ccccc3)CCc3cc(OC)c(OC)cc23)cc1OC |r|
COc1ccc(CC2N(CC(=O)Nc3ccccc3)CCc3cc(OC)c(OC)cc23)cc1OC
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(cc1)C(C)(C)C
CCc1nc(OC)c2[C@H](CCc3ccc(C)c(F)c3)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCn1nc(C)c2[C@H](CCc3cc(F)c(C)c(F)c3)N(CCCc12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(OC)c2C(CCc3ccc(C)c(C)c3)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
Cc1nc(C(=O)N2CCC[C@H](C2)NC(=O)c2c(C)nc3sccn23)c(s1)-c1cccc(C)c1 |r|
Cc1cccc(c1)-c1sc(N)nc1C(=O)N1CC[C@H]1CNC(=O)c1c(Cl)nc2sccn12 |r|
Cc1nc2sccn2c1C(=O)NC[C@@H]1[C@@H]2C[C@@H]2CN1C(=O)c1nc(CCCO)sc1-c1cccc(C)c1 |r|
Cc1nc(C(=O)N2[C@H]3C[C@H]3C[C@H]2CNC(=O)c2c(C)nc3sccn23)c(s1)-c1cccc(C)c1 |r|
CCN(Cc1cc(C)n(C)n1)C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(Cc1ccn(C)n1)C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(Cc1cccc(C)n1)C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(OC)c(OC)c1
O=C(CSc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1ccccc1-n1cccc1 |r|
O=C(CSc1nc2ccccc2[nH]1)N1CCC[C@@H]1C(=O)Nc1ccccc1-n1cccc1 |r|
CN(C)c1ccc(NC(=O)Nc2ccnc3c(F)ccc(F)c23)cc1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(CC)cc1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(C)cc1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(OC)cc1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(Br)cc1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(F)cc1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(cc1)C#N
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccc(OC(F)(F)F)cc1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccccc1C
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccccc1Cl
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1ccccc1F
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1cccc(C)c1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1cccc(Cl)c1
CCN(CC)C(=O)CN(c1ccc(C)cc1)S(=O)(=O)c1cccc(F)c1
CCN(CC)C(=O)CN(c1cc(ccc1C#N)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1Cl)C#N)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1Cl)C(F)(F)F)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1OC)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cccc(N(C)C)c1C#N)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1ccc(Cl)c(c1)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1ccc(C)cc1C#N)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(Cl)ccc1N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(C)ccc1Cl)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1Cl)C(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1Cl)N(CC)CC)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(C)c1ccc(Cl)c(c1)N(CC(=O)N(CC)CC)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1Cl)N1CCCC1)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc(ccc1Cl)-n1cccc1)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(CC)C(=O)CN(c1cc2c(C)nsc2cc1Cl)S(=O)(=O)c1ccc(OC)c(OC)c1
CCN(C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1)c1cccc(C)n1
CCN(C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1)c1cnc(C)cn1
CCN(C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1)c1ccn(C)n1
CCN(C(=O)CN(c1cc(ccc1Cl)N(C)C)S(=O)(=O)c1ccc(OC)c(OC)c1)c1cc(C)n(C)n1
CCN(C(=O)CN(c1cc2c(C)nsc2cc1Cl)S(=O)(=O)c1ccc(OC)c(OC)c1)c1ccccn1
CCN(C(=O)CN(c1cc2c(C)nsc2cc1Cl)S(=O)(=O)c1ccc(OC)c(OC)c1)c1cccc(C)n1
CCn1nc(C)c2C(CCc3ccccc3C)N(CCc12)C(C(=O)NC)c1ccccc1
CCn1nc(C)c2C(CCc3cccc(C)c3)N(CCc12)C(C(=O)NC)c1ccccc1
CCn1nc(C)c2C(CCc3ccc(C)cc3)N(CCc12)C(C(=O)NC)c1ccccc1
CCn1nc(C)c2C(CCc3ccc(OC)cc3)N(CCc12)C(C(=O)NC)c1ccccc1
CCc1ccc(CC[C@@H]2N(CCc3c2c(C)nn3CC)[C@@H](C(=O)NC)c2ccccc2)cc1 |r|
CCc1ccc(CC[C@H]2N(CCc3c2c(C)nn3CC)[C@@H](C(=O)NC)c2ccccc2)cc1 |r|
CCn1nc(C)c2[C@H](CCc3ccc(cc3)C(C)C)N(CCc12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCn1nc(C)c2[C@@H](CCc3ccc(cc3)C(C)C)N(CCc12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCn1nc(C)c2C(CCc3ccccc3F)N(CCc12)C(C(=O)NC)c1ccccc1
CCn1nc(C)c2C(CCc3cccc(F)c3)N(CCc12)C(C(=O)NC)c1ccccc1
CCn1nc(C)c2C(CCc3cccc(c3)C(F)(F)F)N(CCc12)C(C(=O)NC)c1ccccc1
CCn1nc(C)c2[C@H](CCc3ccc(cc3)C(F)(F)F)N(CCc12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCn1nc(C)c2C(CCc3ccc(Cl)cc3)N(CCc12)C(C(=O)NC)c1ccccc1
CCn1nc(C)c2[C@H](COc3ccc(C)cc3)N(CCc12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCn1nc(C)c2C(Cc3ccc(cc3)C(F)(F)F)N(CCc12)C(C(=O)NC)c1ccccc1
Cc1ccc(c(c1)C(=O)N1CCCN(CC1)c1ncc2cc(F)ccc2n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CC(C1)N(C2)c1ncc2ccccc2n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CC1CN(C2)c1ncc2ccccc2n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC2CC1CN2c1ncc2cc(F)ccc2n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CC1CCN2c1ncc2cc(F)ccc2n1)-n1nccn1
Fc1ccc2nc(ncc2c1)N1CC2CC1CN(C2)C(=O)c1cc(Cl)ccc1-n1nccn1
CC(=O)c1cccc(NC(=O)CSc2nnc(-c3ccoc3C)n2Cc2ccco2)c1
COc1ccc(C)cc1NC(=O)CSc1nnc(-c2ccoc2C)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2cccc(C)c2)n1Cc1ccco1
CC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccoc3C)n2Cc2ccco2)cc1
Cc1occc1-c1nnc(SCC(=O)Nc2ccc(Cl)cc2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2cccc(Cl)c2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2ccc(F)c(Cl)c2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2cc(C)cc(C)c2)n1Cc1ccco1
CN(C)c1ccc(NC(=O)CSc2nnc(-c3ccoc3C)n2Cc2ccco2)cc1
Cc1occc1-c1nnc(SCC(=O)Nc2ccc(C)c(C)c2)n1Cc1ccco1
Cc1nc(C(=O)N2CCCC[C@H]2CNC(=O)c2cccc3occc23)c(s1)-c1ccc(F)cc1 |r|
Cc1occc1-c1nnc(SCC(=O)Nc2cc(C)ccc2C)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2c(C)cccc2C)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2cccc(C)c2C)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2ccccc2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2ccc(C)cc2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2ccc(F)cc2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2ccccc2F)n1Cc1ccco1
COc1ccccc1NC(=O)CSc1nnc(-c2ccoc2C)n1Cc1ccco1
COc1ccc(NC(=O)CSc2nnc(-c3ccoc3C)n2Cc2ccco2)cc1
Cc1occc1-c1nnc(SCC(=O)Nc2cccc(c2)-c2ccc3OCOc3c2)n1Cc1ccco1
Cc1csc(NC(=O)CSc2nnc(-c3ccoc3C)n2Cc2ccco2)n1
Cc1nnc(NC(=O)CSc2nnc(-c3ccoc3C)n2Cc2ccco2)s1
Cc1occc1-c1nnc(SCC(=O)NCCc2ccccc2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)NN2CCc3ccccc23)n1Cc1ccco1
CCC(C)NC(=O)CSc1nnc(-c2ccoc2C)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(N)=O)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)N(c2cccnc2)c2cc(C)cc(C)c2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)N(C2CNCCN2)c2cc(C)cc(C)c2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2ccccc2C)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2cccc(F)c2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)N(c2cc(C)cc(C)c2)c2ccccn2)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2ccc(C)cc2C)n1Cc1ccco1
Cc1occc1-c1nnc(SCC(=O)Nc2nccs2)n1Cc1ccco1
COc1ccc2OC[C@@H](C)N([C@@H](C)c2c1)C(=O)c1ccc(Cl)cc1 |r|
C[C@@H]1COc2ccc(OC(F)F)cc2[C@H](C)N1C(=O)c1ccc(Cl)cc1 |r|
O=S(=O)(N1CCOC11CCN(CC1)c1cnc2ccccc2n1)c1ccccc1
O=C(Nc1ccccc1)N1CCC2(CC1)OCCN2S(=O)(=O)c1ccccc1
FC1(F)CN(CCC11OCCN1S(=O)(=O)c1ccccc1)C(=O)Nc1ccccc1
COc1cccc(c1)S(=O)(=O)N1CCOC11CCN(CC1F)C(=O)Nc1ccccc1
COc1ccc(cc1)S(=O)(=O)N1CCOC11CCN(CC1F)C(=O)Nc1ccccc1
COc1ccc(cc1OC)S(=O)(=O)N1CCOC11CCN(CC1F)C(=O)Nc1ccccc1
F[C@@H]1CN(CCC11OCCN1S(=O)(=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
F[C@H]1CN(CCC11OCCN1S(=O)(=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
Cn1c(SCC(=O)N2CCC[C@H]2C(=O)Nc2ccccc2-c2ccccc2)nc2ccccc12
Cc1ccc2nc(SCC(=O)N3CCC[C@H]3C(=O)Nc3ccccc3-n3cccc3)n(C)c2c1
Cc1ccc2n(C)c(SCC(=O)N3CCC[C@H]3C(=O)Nc3ccccc3-n3cccc3)nc2c1
O=C(CSc1nc2ccccc2o1)N1CCC[C@H]1C(=O)Nc1ccccc1-n1cccc1
O=C(CSc1nc2ccccc2s1)N1CCC[C@H]1C(=O)Nc1ccccc1-n1cccc1
Cn1c(SCC(=O)N2CCC[C@H]2C(=O)Nc2ccccc2-n2cccc2)nc2ccccc12
O=C(CCc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1ccccc1-n1cccc1
COc1ccccc1-c1ccccc1NC(=O)[C@@H]1CCCN1C(=O)CCc1nc2ccccc2[nH]1
O=C(CCc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1ccccc1-c1ccccc1
O=C(CSc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1ccccc1Oc1ccccc1
O=C(CSc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1cccc(c1)-c1ccccc1
O=C(CSc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1ccccc1-c1ccccc1
Cn1c(CCC(=O)N2CCC[C@H]2C(=O)Nc2ccccc2-c2ccccc2)nc2ccccc12
Cc1ccc2nc(SCC(=O)N3CCC[C@H]3C(=O)Nc3ccccc3-n3cccc3)[nH]c2c1
Cn1c(CCC(=O)N2CCC[C@H]2C(=O)Nc2ccccc2-n2cccc2)nc2ccccc12
Fc1ccccc1-c1ccccc1NC(=O)[C@@H]1CCCN1C(=O)CCc1nc2ccccc2[nH]1
O=C(CSc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1ccc(cc1)-c1ccccc1
O=C(CSc1nc2ccccc2[nH]1)N1CCC[C@H]1C(=O)Nc1ccccc1
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1ncc2ccccc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1ncc2ccccc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1ncc2cc(F)ccc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1cnc2cc(F)c(F)cc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1ncc2CCCCc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1nc2ccccc2o1 |r|
C[C@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1ncc2ccccc2n1 |r|
Fc1ccc2nc(ncc2c1)N1C[C@H]2C[C@@H]1CN(C2)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1C2CCC1CN(CC2)c1ncc2ccc(F)cc2n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC2CCC(C1)N2c1ncc2ccc(F)cc2n1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1C[C@H]2CC[C@@H]1CN(C2)c1ncc2ccc(F)cc2n1)-n1nccn1 |r,THB:7:9:15.16.17:13.12|
Cc1ccc(c(c1)C(=O)N1C[C@@H]2CC[C@H]1CN(C2)c1ncc2ccc(F)cc2n1)-n1nccn1 |r,THB:7:9:15.16.17:13.12|
Cc1ccc(c(c1)C(=O)N1CC[C@@H]2CC[C@H]1CN2c1ncc2ccc(F)cc2n1)-n1nccn1 |r,THB:18:17:9.10.11:14.13|
Cc1ccc(c(c1)C(=O)N1CC[C@H]2CC[C@@H]1CN2c1ncc2ccc(F)cc2n1)-n1nccn1 |r,THB:18:17:9.10.11:14.13|
Cc1ccc(c(c1)C(=O)N1C[C@H]2CC[C@@H]1CCN2c1ncc2ccc(F)cc2n1)-n1nccn1 |r,THB:7:9:17.15.16:13.12|
Cc1ccc(c(c1)C(=O)N1C[C@@H]2CC[C@H]1CCN2c1ncc2ccc(F)cc2n1)-n1nccn1 |r,THB:7:9:17.15.16:13.12|
FC1(F)CC[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
O=C(NCC1CCCCN1C(=O)c1ccccc1-c1ccccc1)c1cccc2cccnc12
Cc1nc(C(=O)N2CCCCC2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccc(F)cc1
Cc1nc(c(s1)C(=O)N1CCCCC1CNC(=O)c1cccc2occc12)-c1ccccc1
Cc1nc(c(s1)C(=O)N1CCCCC1CNC(=O)c1cccc2cccnc12)-c1ccccc1
Cc1nc(c(s1)C(=O)N1CCCCC1CNc1ccc(cn1)C(F)(F)F)-c1ccccc1
COc1cccc(C(=O)NC[C@@H]2[C@H](C)CCCN2C(=O)c2nc(C)sc2-c2ccccc2)c1C |r|
O[C@@H]1CCN([C@H](CNC(=O)c2cccc3cccnc23)C1)C(=O)c1ccccc1-c1ccccc1 |r|
F[C@H]1CCN([C@H](CNC(=O)c2cccc3cccnc23)C1)C(=O)c1ccccc1-c1ccccc1 |r|
CO[C@@H]1CCN([C@H](CNC(=O)c2cccc3cccnc23)C1)C(=O)c1sc(C)nc1-c1ccccc1 |r|
OCCNC1CC[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
OC1CC[C@@H](CNC(=O)c2cccc3cccnc23)N(C1)C(=O)c1ccccc1-c1ccccc1 |r|
Cc1nc(C(=O)N2CC(F)CC[C@H]2CNC(=O)c2cccc3occc23)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2CC(N)CC[C@H]2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2CC(F)CC[C@H]2CNc2ccc(cn2)C(F)(F)F)c(s1)-c1ccccc1 |r|
C[C@H]1CCC[C@@H](CNC(=O)c2cccc3occc23)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCC[C@@H](CNC(=O)c2cccc3cccnc23)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCC[C@@H](CNc2ccc(cn2)C(F)(F)F)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
C[C@H]1CCC[C@@H](CNc2nc3ccccc3o2)N1C(=O)c1nc(C)sc1-c1ccc(F)cc1 |r|
CC(=O)Nc1ccc(NC(=O)Nc2ccnc3cccnc23)cc1O
COc1cccc(c1)C(=O)N1CCCCC1CCOc1ccc(Cl)c(Cl)c1
O=C(NC[C@@H]1CCCCN1C(=O)c1ccccc1-c1ccccc1)Nc1ccccc1 |r|
Clc1ccc(OCCC2CCCCN2C(=O)c2cccc(c2)C#N)cc1Cl
O=C(C[C@@H]1CCCCN1C(=O)c1ccccc1-c1ccccc1)Nc1ccccc1 |r|
CN(C[C@@H]1CCCCN1C(=O)c1ccccc1-c1ccccc1)C(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)C(=O)NC[C@H]1CCCCN1C(=O)c1ccccc1-c1ccccc1 |r|
O=C(NC[C@@H]1CCCCN1C(=O)c1ccccc1-c1ccccc1)c1ccccc1 |r|
Fc1ccc(OCC[C@@H]2CCCCN2C(=O)c2ccccc2-c2ccccc2)c(F)c1 |r|
Fc1ccc(OCC[C@@H]2CCCCN2C(=O)c2cccc3ccccc23)cc1 |r|
Fc1ccc(OCCC2CCCCN2C(=O)c2ccccc2-c2ccccc2)cc1
O=C(CC[C@@H]1CCCCN1C(=O)c1ccccc1-c1ccccc1)c1ccccc1 |r|
Fc1ccc(cc1)C(=O)NC[C@@H]1CCCCN1C(=O)c1ccccc1-c1ccccc1 |r|
Clc1ccc(OCCC2CCCCN2C(=O)c2ccc(Cl)c(Cl)c2)cc1Cl
CNC(=O)[C@H](N1CCn2c(nc(Cl)c2[C@@H]1CCc1ccc(cc1)C(F)(F)F)C1CC1)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(nc(Cl)c2[C@@H]1CCc1ccc(cc1)C(F)(F)F)C(C)C)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(COC)nc(Cl)c2[C@@H]1CCc1ccc(cc1)C(F)(F)F)c1ccccc1 |r|
CCCc1nc(Cl)c2[C@H](CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(C)nc(Cl)c2[C@@H]1CCc1ccc(cc1)C(F)(F)F)c1ccccc1 |r|
CCc1nc(C(=O)N(C)C)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(C(=O)NC)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(C(N)=O)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(C#N)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(c2[C@H](CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1)S(C)(=O)=O |r|
CCc1nc(SC)c2[C@H](CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCOc1nc(CC)n2CCN([C@@H](C(=O)NC)c3ccccc3)C(CCc3ccc(cc3)C(F)(F)F)c12 |r|
CCc1nc(OC)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(c2[C@H](CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1)C(F)(F)F |r|
CCc1nc(Cl)c2[C@@H](CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(I)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(C=C)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(C2CC2)c2[C@H](CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(C(C)C)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCCc1nc(CC)n2CCN([C@@H](C(=O)NC)c3ccccc3)C(CCc3ccc(cc3)C(F)(F)F)c12 |r|
CCc1nc(CC)n2CCN([C@@H](C(=O)NC)c3ccccc3)C(CCc3ccc(cc3)C(F)(F)F)c12 |r|
CCc1nc(C)c2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1ncc2C(CCc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(CC3CC3)nc(Cl)c2[C@@H]1CCc1ccc(cc1)C(F)(F)F)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(nc(Cl)c2[C@@H]1CCc1ccc(OC(F)F)c(F)c1)C1CC1)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(nc(Cl)c2[C@@H]1CCc1ccc(cc1F)C(F)(F)F)C1CC1)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(nc(Cl)c2[C@@H]1CCc1ccc(c(F)c1)C(F)(F)F)C1CC1)c1ccccc1 |r|
CNC(=O)[C@H](N1CCn2c(nc(Cl)c2[C@@H]1CCc1cccc(c1)C(F)(F)F)C1CC1)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3cccc(c3F)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(F)c(c3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(F)c(F)c3F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3cc(F)c(c(F)c3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3cc(F)c(cc3F)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(c(F)c3F)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(cc3F)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(c(Cl)c3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@@H](CCc3ccc(c(F)c3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(c(F)c3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(OC(F)(F)F)cc3)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(OC(F)F)cc3)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3ccc(cc3)C#N)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](COc3cccc(c3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](COc3ccc(cc3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
CCc1nc(Cl)c2[C@H](CCc3cccc(c3)C(F)(F)F)N(CCn12)[C@@H](C(=O)NC)c1ccccc1 |r|
COC(=O)c1ccc2[nH]cc(CN3CCCC4(CCN(CC4)c4nc(C)cc(C)n4)C3=O)c2c1
Cc1noc(n1)-c1ccccc1CN1CCCC2(CCN(CC2)c2nc(C)cc(C)n2)C1=O
Cc1nc(C(=O)N2CCCC[C@H]2CNC(=O)c2cccc3cccnc23)c(s1)-c1ccc(F)cc1 |r|
CN(Cc1ccc(F)cc1)C(=O)Cc1c(C)c(c2ccccn12)S(=O)(=O)Cc1ccc(F)cc1
CCN(CC)c1ccc(NC(=O)c2oc3ccccc3c2C)cc1
CCn1nc(C)cc1C(=O)NCC[C@H](Cc1ccccc1)N(C)C(=O)c1cc(C)ccc1-n1nccn1 |r|
CCOc1cccc(c1)C(=O)N(C)[C@H](CCNC(=O)c1cccn1C)Cc1ccccc1 |r|
Cc1cc(C)nc(n1)N1CC[C@@H]2CN([C@H]2C1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
Cc1cc(C)nc(n1)N1C[C@@H]2CCN(C[C@H]12)C(=O)c1cc(F)ccc1-n1nccn1 |r|
C[C@@H]1CO[C@@H](COc2nccc3ccccc23)CN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CO[C@@H](COc2ncccc2C)CN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
CN(Cc1ccccc1)C(=O)Cn1nc(c2ccccc12)S(=O)(=O)Cc1ccccc1
CN(Cc1ccccc1)C(=O)Cn1cc(c2ccccc12)S(=O)(=O)Cc1ccccc1
Fc1ccc(CNC(=O)Cn2cc(c3ccccc23)S(=O)(=O)Cc2ccc(F)cc2)cc1
CN(Cc1ccc(F)cc1)C(=O)Cn1cc(c2ccccc12)S(=O)(=O)Cc1ccc(F)cc1
CN(Cc1ccc(F)cc1)C(=O)Cc1nc(c2ccccn12)S(=O)(=O)Cc1ccccc1
CN(Cc1ccc(F)cc1)C(=O)Cc1c(C)c(c2ccccn12)S(=O)(=O)Cc1ccccc1
CN(Cc1ccccc1)C(=O)Cc1c(C)c(c2ccccn12)S(=O)(=O)Cc1ccccc1
Cc1nc(C(=O)N2CCC2CNC(=O)c2c(N)nc3sccn23)c(s1)-c1cccc(C)c1
CN1CCOc2c1cccc2C(=O)NCC1CCN1C(=O)c1nc(C)sc1-c1cccc(C)c1
C[C@H]1[C@H](COc2ccccn2)CCCN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@H]1[C@H](COc2nccc3ccccc23)CCCN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
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CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H]1CCCN1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCSC)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O
COc1cccc(OC)c1C1CCCC(=O)N1CCc1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1c1ccccc1
COc1cccc(OC)c1C1CCCC(=O)N1Cc1ccccc1
COc1cc(OC)c(C2CCCCN2Cc2ccc(OC(F)(F)F)cc2)c(OC)c1
COc1cccc(OC)c1C1SCC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1C2CC2C(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1C1N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c2ccccc12
COc1cccc(OC)c1C1COC(=O)N1Cc1ccc(OC(F)(F)F)cc1
COc1cccc(OC)c1[C@H]1C[C@H](C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1ccnc(CO)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1cccc(CO)c1 |r|
C[C@@H]1CC[C@@H](CCc2ccc(F)cn2)CN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)\C=C\c1ccc(F)cn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)\C=C/c1ccc(F)cn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1ccc(F)cn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1ccccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1cccnc1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1ccncc1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1cccnc1O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1cnccc1O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1ccc(CO)cn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1cccc(CO)n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1cc(CO)ccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1ccc(CO)nc1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)C#Cc1cncc(CO)c1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1ncc2cnn(C)c2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1ncc2c(C)nn(C)c2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1ncc2c(C)nn(C)c2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1ncc2c(C)coc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1ncc2c(C)c(C)oc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1ncc2c(C)csc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1nc(N)c2c(C)coc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1nc(N)c2c(C)coc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1nc(N)c2ccsc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1nc(N)c2ccsc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1nc(N)c2cc(C)sc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1nc(N)c2cc(C)sc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1cc(C)ccc1-n1nccn1)c1nc(N)c2c(C)csc2n1 |r|
C[C@@H]1CCN(CCN1C(=O)c1ccccc1-n1nccn1)c1nc(N)c2c(C)csc2n1 |r|
COc1ccc(CNC(=O)c2cc(ncc2N2CCCC2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2N2CCC2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2cnn(C)c2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2nccs2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(cnc2-c2ccccc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2nc(ccc2-c2ccccc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2ccccc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2nc(cnc2-c2ccccc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2nc(ncc2-c2ccccc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(nnc2-c2ccccc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ccc2-c2ccccc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(nc3onc(-c4ccccc4)c23)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2sc(nc2-c2cccc(F)c2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2ccccc2F)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2cccc(F)c2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2ccccn2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2cnccn2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2ccnnc2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2-c2cncc(F)c2)-c2cncc(C)c2)nc1OC
COc1ccc(CNC(=O)c2cc(ncc2N2CCOCC2)-c2cncc(C)c2)nc1OC
COc1ccc(OC[C@]2(C[C@H]2C(=O)c2ccccc2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Cc2ccccc2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2CNc2ccccc2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2ccccc2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)NC2CCCCC2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)N(C)c2ccccc2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)N2CCCc3ccccc23)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2ccccn2)c2ccccc2)cc1OC |r|
O=C(Nc1ccccn1)[C@@H]1C[C@@]1(COc1ccccc1)c1ccccc1 |r|
COc1ccc(cc1OC)[C@]1(COc2ccccc2)C[C@H]1C(=O)Nc1ccccn1 |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2ccccn2)c2ccccc2)cc1 |r|
COc1cccc(OC[C@]2(C[C@H]2C(=O)Nc2ccccn2)c2ccccc2)c1 |r|
COCc1cc(OC[C@]2(C[C@H]2C(=O)Nc2ccccn2)c2ccccc2)ccc1OC |r|
COCc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2ccccn2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2cccnc2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2ccncc2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2ncc(C)s2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2nc(C)cs2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2cc(C)on2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)c2nc3cc(F)ccc3[nH]2)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2cc(ccn2)C#N)c2ccccc2)cc1OC |r|
COc1ccc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)cc1OC |r|
COc1ccc(OCC2(CC2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)cc1OC
Cc1ccc(c(c1)C(=O)N1CCCC(C1)Oc1ccc(F)c(C)c1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCC(C1)Oc1cccc2ccccc12)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCCC(COc2ccc(F)c(C)c2)C1)-n1nccn1
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1ccnc2ccc(Br)cc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(C)nc2ccccc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2ncccc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2cccnc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2ccncc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1ccnc2ccccc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc2cnccc12
C[C@@H]1CC[C@H](CN1C(=O)c1cc(C)ccc1-n1nccn1)Oc1cccc2ccccc12 |r|
FC1(F)CCN(C[C@@H]1Oc1ccc2ccccc2n1)C(=O)c1ccccc1-n1nccn1 |r|
COc1cnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c2ccccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1cnn[nH]1)Oc1ccnc2c(F)cccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1ccccn1)Oc1ccnc2c(F)cccc12 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-c1cccnc1)Oc1ccnc2c(F)cccc12 |r|
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1ccnc2c(Cl)cccc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1ccnc2c(F)cccc12
CC1CCC(CN1C(=O)c1ccccc1-n1nccn1)Oc1ccnc2c(Br)cccc12
COc1cccc(F)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
COc1cccc(F)c1C1C[C@@H](O)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
COc1cccc(F)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
COc1cccc(F)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
COc1cccc(OC)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
COc1cccc(OC)c1[C@@H]1C[C@@H](N(C)C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](N(C)C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
CN[C@@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |r|
CN[C@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |r|
COc1cccc(OC)c1[C@@H]1C[C@@H](N)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](N)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
CO[C@@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |r|
CCO[C@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |r|
CO[C@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |r|
COc1cccc(OC)c1[C@@H]1C[C@@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](O)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](F)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(OC)c1[C@@H]1C[C@H](Cl)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
CC[C@H]1C[C@H](N(Cc2ccc(OC(F)(F)F)cc2)C1=O)c1c(OC)cccc1OC |r|
COc1cccc(OC)c1[C@@H]1C[C@@H](C)C(=O)N1Cc1ccc(OC(F)(F)F)cc1 |r|
COc1cccc(F)c1[C@H]1C[C@H](O)C(=O)N1Cc1ccc2oc3ccccc3c2c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(F)ccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C(=O)N(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C#C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)C(F)(F)F |r|
CCc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ncccc1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(C)ccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1ccc(C)cn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cccc(C)n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1OC(F)F)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1CC(F)(F)F)Oc1cc(ccn1)C#N |r|
CC(C)OC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1cc(ccn1)C#N |r|
CCOC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1cc(ccn1)C#N |r|
COC(=O)c1ccccc1C(=O)N1C[C@@H](CC[C@H]1C)Oc1cc(ccn1)C#N |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)-c1ccccc1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)N(C)C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(ccn1)S(C)(=O)=O |r|
CSc1ccnc(O[C@@H]2CC[C@@H](C)N(C2)C(=O)c2ccccc2-n2nccn2)c1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(I)ccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(Br)ccn1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)Oc1cc(Cl)ccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(OC)cc(OC)n1)C(=O)c1ccccc1-c1cccs1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1ccccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1cccc(F)c1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1ccc(F)cc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1ccccc1-c1ncn[nH]1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1cccc(C)c1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1c(C)cccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nccc(n1)-c1ccccc1)C(=O)c1ccccc1-c1ccccc1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1cnc2ccccc2n1)C(=O)c1ccccc1-c1ccccc1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nccc(C)n1)C(=O)c1ccccc1-c1ccccc1 |r|
COc1ccc(CNC(=O)c2cc(cnc2-c2ccccn2)-c2cncc(Cl)c2)nc1OC
[H][C@@]12CN(C[C@]1([H])CN(C2)c1cnc2ccccc2n1)C(=O)c1ccccc1-n1cccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1cnc2ccccc2n1)C(=O)c1ccccc1-c1cccs1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1ccccc1-c1cccs1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1c(C)ccc2ccccc12 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nccc(OC)n1)C(=O)c1c(C)ccc2ccccc12 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1ccccc1-c1cccc(F)c1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1c(OCC)ccc2ccccc12 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccc(Cl)cc2s1)C(=O)c1c(OC)cccc1OC |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccc(Cl)cc2s1)C(=O)c1ccc(OC)cc1OC |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccc(C)cc2s1)C(=O)c1ccc(OC)cc1OC |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccc(OC)cc2s1)C(=O)c1ccc(OC)cc1OC |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccc(F)cc2s1)C(=O)c1ccc(OC)cc1OC |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccccc2s1)C(=O)c1ccccc1-c1ccccc1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccc(F)cc2s1)C(=O)c1ccccc1-c1ccccc1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccc(F)cc2s1)C(=O)c1ccccc1-c1cccs1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1cc(OC)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)cc(C)n1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
CCn1cc(OCC2(CC2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)c(C)n1
Cc1nn(C)cc1OCC1(CC1C(=O)Nc1ccc(cn1)C#N)c1ccccc1
Cc1cc(OCC2(CC2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)cc(C)n1
Cc1ccc(OCC2(CC2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)c(C)n1
Cc1ccc(NC(=O)[C@@H]2C[C@@]2(COc2cnc(C)nc2C)c2ccccc2)nc1 |r|
Cc1ccnc(NC(=O)[C@@H]2C[C@@]2(COc2cnc(C)nc2C)c2ccccc2)c1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2cc(C)c(F)cn2)c2ccccc2)c(C)n1 |r|
COc1cc(NC(=O)[C@@H]2C[C@@]2(COc2cnc(C)nc2C)c2ccccc2)ncc1F |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(F)cn2)c2ccccc2F)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(F)cn2)c2ccc(F)cc2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(F)cn2)c2cc(F)cc(F)c2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(F)cn2)c2ccc(F)c(F)c2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2cc(C)c(F)cn2)c2cccc(F)c2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(Cl)cn2)c2ccccc2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2cccc(F)n2)c2ccccc2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(F)cn2)c2ccccc2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccncc2)c2ccccc2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2cccnc2)c2ccccc2)c(C)n1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccccn2)c2ccccc2)c(C)n1 |r|
COCc1nc(C)ncc1OC[C@]1(C[C@H]1C(=O)Nc1ccc(cn1)C#N)c1ccccc1 |r|
Cc1cnc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)c(C)n1 |r|
CCc1nc(C)ncc1OC[C@]1(C[C@H]1C(=O)Nc1ccc(cn1)C#N)c1ccccc1 |r|
Cc1ncc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)c(C)n1 |r|
CCn1cc(OC[C@]2(C[C@H]2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)c(C)n1 |r|
CCn1cc(OC[C@@]2(C[C@@H]2C(=O)Nc2ccc(cn2)C#N)c2ccccc2)c(C)n1 |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1cc(ccn1)C(F)(F)F |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccsc1-n1nccn1)Oc1ncccc1C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1ncnn1)Oc1nccc(c1F)C(C)(C)O |r|
C[C@@H]1CC[C@H](CN1C(=O)c1ccccc1-n1nccn1)c1nc(c(o1)C1CC1)C(C)(C)O |r|
CCN(CCCOc1ccc(F)cc1)C(=O)c1nc(C)sc1-c1ccccc1
Cc1nc(C(=O)N2CCC[C@@H](COc3ccc(F)cc3)C2)c(s1)-c1ccccc1 |r|
Cc1nc(C(=O)N2CCCC[C@H]2CCOc2ccc(F)cc2)c(s1)-c1ccccc1 |r|
FC(F)(F)c1cnc(N[C@@H]2CC3CCC2N3C(=O)c2ccccc2-c2ncccn2)cn1 |r,TLB:8:9:13.12:15|
Fc1ccc(OC[C@@H]2CC3CCC2N3C(=O)c2ccccc2-c2cccs2)nc1 |r,TLB:6:7:11.10:13|
Fc1ccc(O[C@@H]2CC3CC2N(C3)C(=O)c2ccccc2-n2nccn2)nc1 |r,TLB:13:11:6.7:9,THB:5:6:9:12.11|
FC(F)(F)c1cnc(N[C@@H]2CC3CCC2N(C3)C(=O)c2ccccc2-c2ncccn2)cn1 |r,TLB:17:15:9.10:13.12,THB:8:9:15.16:13.12|
COc1ccccc1C(=O)NCCNc1cccc(NS(=O)(=O)c2cc(ccc2OC)-c2cccc(c2)C(=O)N(C)C)c1
COc1cccc(c1)C(=O)NCCNc1cccc(NS(=O)(=O)c2cc(ccc2OC)-c2cccc(c2)C(=O)N(C)C)c1
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2ccccc2Cl)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1S(=O)(=O)Nc1cccc(NCCNC(=O)c2cccc(Cl)c2)c1)-c1cccc(c1)C(=O)N(C)C
COc1ccc(cc1)[C@@H](C)NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F |r|
C[C@@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1c(C)n[nH]c1C |r|
C[C@H](NC(=O)CNc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1c(C)nn(C)c1C |r|
C[C@H](NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccn1)C(F)(F)F)c1ccccc1 |r|
Cc1cc2CC[C@H](NC(=O)COc3cc(C)c4c(nn(C)c4n3)C3CC3)c2cn1 |r|
CC(NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)C1CC1)c1c(C)nn(C)c1C
CC(NC(=O)COc1cc(C(F)F)c2c(nn(C)c2n1)-c1ccccc1)c1c(C)nn(C)c1C
COc1ccccc1C(C)NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F
CC(NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1ccccn1
CC(NC(=O)COc1cc(c2c(nn(C)c2n1)-c1ccccc1)C(F)(F)F)c1cccnc1
CCN(CCN(C)c1nc2ccccc2o1)C(=O)c1cc(C)ccc1-n1nccn1
Cc1nc(C(=O)N2CCCCC2CCOc2ccc(F)cc2)c(s1)-c1ccccc1
C[C@@H]1CC[C@H](COc2ccc(F)c(C)c2)CN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
C[C@@H]1CC[C@@H](COc2ccc(F)c(C)c2)CN1C(=O)c1cc(C)ccc1-n1nccn1 |r|
COc1ccc(CC2N(CC(=O)NCc3ccccc3)CCc3cc(OC)c(OC(C)C)cc23)cc1OC
FC1(F)CCN(C[C@@H]1Oc1ccc2ccccc2n1)C(=O)c1cccn2cncc12 |r|
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(cc1)N(C)C)ccc3O |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccccn1)S(=O)(=O)c1ccccc1N(C)C)ccc3OC |r,THB:30:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1cccnc1)S(=O)(=O)c1ccccc1N(C)C)ccc3OC |r,THB:30:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC6CC6)CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)ccc3OC |r,THB:10:9:17:4.5.6|
CN([C@@H]1CC[C@@]2(O)[C@H]3Cc4cccc5O[C@@H]1[C@]2(CCN3CC1CC1)c45)C(=O)\C=C\c1ccoc1 |r,TLB:4:5:9.24.8:17.19.18,THB:6:5:9.24.8:17.19.18|
CN([C@@H]1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5O[C@@H]1[C@]2(CCN3CC1CC1)c45)C(=O)\C=C\c1ccccc1 |r,TLB:4:5:9.25.8:18.20.19,THB:6:5:9.25.8:18.20.19|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)C(=O)OC(C)(C)C)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)C(C)=O)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)C(=O)\C=C\c1ccccc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1F)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(c1)C#N)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(Br)cc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1Cl)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccccc1OC)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(cc1)[N+]([O-])=O)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(OC)c1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(c1)[N+]([O-])=O)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1cccc(c1)C(F)(F)F)ccc3OC |r,THB:29:9:5.4.6:13|
CN([C@@H]1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5O[C@@H]1[C@]2(CCN3CC1CC1)c45)C(=O)\C=C\c1ccco1 |r,TLB:4:5:9.25.8:18.20.19,THB:6:5:9.25.8:18.20.19|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(cc1)C(F)(F)F)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(Cl)cc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)C=Cc1ccoc1)S(=O)(=O)c1ccc(cc1)N(C)C)ccc3OC
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(F)cc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)C=Cc1ccoc1)S(=O)(=O)c1cccc(c1)N(C)C)ccc3OC
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(OC)cc1)ccc3OC |r,THB:29:9:5.4.6:13|
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)C=Cc1ccoc1)S(=O)(=O)c1ccccc1N(C)C)ccc3OC
[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC[C@@]14[C@@]5(O)CC[C@H]2N(C)C(=O)\C=C\c1ccoc1)S(=O)(=O)c1ccc(cc1)C#N)ccc3OC |r,THB:29:9:5.4.6:13|
C[C@@H]1CC[C@H](CN1C(=O)c1cc(NC(C)=O)ncc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
C[C@@H]1CC[C@H](CN1C(=O)c1nc(NC(C)=O)ccc1-c1ccccc1)Oc1nccc(C#N)c1C |r|
COC(=O)c1cccnc1O[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
COC(=O)c1cccnc1N[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
COC(=O)c1cccnc1S[C@@H]1CC[C@@H](C)N(C1)C(=O)c1ccccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CC2CN(CC2(C)C1)c1nc2cc(Cl)ccc2o1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CCN(C2C1)c1nc2cc(Cl)ccc2o1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CCC2CN(CC12)c1nc2cc(Cl)ccc2o1)-n1nccn1
Cc1ccc(c(c1)C(=O)N1CC2CCCN(C2C1)c1nc2cc(Cl)ccc2o1)-n1nccn1
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2o1)C(=O)c1cc(Cl)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2o1)C(=O)c1cc(F)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2o1)C(=O)c1ccccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2o1)C(=O)c1cc(OC)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2o1)C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccccc2n1C)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(C)c(C)c(C)n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1ncnc2ccccc12)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(Cc3nc4cc(Cl)ccc4o3)C[C@]1([H])CN(C2)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1ncc2cc(F)ccc2n1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(F)ccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(OC(F)(F)F)ccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(C)ccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2ccccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(ccc2o1)C(F)(F)F)C(=O)c1cc(C)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1C[C@]2(F)CN(C[C@]2(F)C1)c1nc2ccccc2o1)-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2s1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1C[C@]2(C)CN(C[C@]2(C)C1)c1nc2cc(Cl)ccc2o1)-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(co1)-c1cccc(Cl)c1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(Cl)ccc2o1)C(=O)c1cc(OC(F)(F)F)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1C[C@]2(F)CN(C[C@]2(F)C1)c1nc2cc(Cl)ccc2o1)-n1nccn1 |r|
[H][C@@]12CN(C[C@]1([H])CN(C2)c1nc2cc(OC)ccc2o1)C(=O)c1cc(C)ccc1-n1nccn1 |r|
Cc1ccc(c(c1)C(=O)N1CCCC2CN(CC12)c1nc2cc(Cl)ccc2o1)-n1nccn1