9827 SMILES Strings for Sodium channel protein type 9 subunit alpha

Compound Name
SMILES String
Fc1cc(O[C@@H]2CCCN(Cc3ccccc3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(O[C@H]2CCCN(Cc3ccccc3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)c(Cl)c1 |r|
Fc1cc(OCC2CC3CCC(C2)N3C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
C[C@@H](c1cc(cc(c1)Cl)Cl)N2CCC(CC2)COc3cc(c(cc3C4CC4)C(=O)NS(=O)(=O)C)F
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](COC)c2cc(Cl)cc(Cl)c2)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](COC)c2cc(Cl)cc(Cl)c2)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](c2cc(Cl)cc(Cl)c2)C(C)(C)OC)cc1F |r|
CC(C)(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1
CC(C)Oc1ncc(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)CC2)cc1Cl
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(F)cc(c3)C(F)(F)F)CC2)cc1F
Fc1cc(OCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(F)cc(Cl)c3)CC2)cc1F
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O)c1ccc(Cl)c(n1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(F)cc3Cl)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(F)CCN(Cc3cc(cc(Cl)c3F)C(F)(F)F)CC2)cc1F
COc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)c(C)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCO[C@H](Cc3cc(Cl)cc(Cl)c3)C2)cc1F |r|
Fc1cc(CN2CCO[C@H](Cc3cc(Cl)cc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(CN2CCC(CC2)Oc2ncc(cc2Cl)C2CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(CN2[C@H]3CC[C@@H]2CC(C3)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,TLB:4:5:7.8:10.12.11|
CC(C)(N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1)c1cc(Cl)cc(Cl)c1 |r|
CC1(COc2cc(F)c(cc2C2CC2)C(N)=O)CN(C1)c1cc(c(Cl)cn1)C(F)(F)F
COC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(Cl)c3C#N)CC2)cc1F
FC(F)(F)c1ccc(CN2C(=O)C3(COc4cc5OCOc5cc34)c3ccccc23)o1
FC(F)(F)c1ccc(CN2C(=O)[C@]3(COc4cc5OCOc5cc34)c3ccccc23)o1
FC(F)(F)c1ccc(CN2C(=O)[C@@]3(COc4cc5OCOc5cc34)c3ccccc23)o1
FC(F)(F)c1cccnc1CN1C(=O)C2(COc3cc4OCCOc4cc23)c2ccccc12
FC(F)(F)c1cccnc1CN1C(=O)[C@@]2(COc3cc4OCCOc4cc23)c2ccccc12
Fc1cc(O[C@@H]2CCCN(Cc3cccc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(CN2C3CCC2CC(C3)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(Cl)c3C#N)CC2)cc1F
FC(F)(F)c1ccc(Oc2ccc3c(CN(c4nccs4)S3(=O)=O)c2)c(c1)-c1ccnnc1
O=S1(=O)N(Cc2cc(Oc3ccccc3-c3ccccc3)ccc12)c1nccs1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc2c(CN(c3nccs3)S2(=O)=O)c1
O=S1(=O)N(Cc2cc(ccc12)N1CCC2(CC1)OCc1ccccc21)c1nccs1
O=S1(=O)N(CCc2cc(ccc12)N1CCC2(CC1)OCc1ccccc21)c1nccs1
O=S1(=O)N(CCc2cc(Oc3ccccc3-c3ccccc3)ccc12)c1nccs1
FC(F)(F)c1ccc(Oc2ccc(cc2)-c2ccc3c(CCN(c4nccs4)S3(=O)=O)c2)cc1
OC[C@@H](O)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OC[C@@H](O)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(C#N)c(c2)C(F)(F)F)cc1 |r|
OC[C@@H](O)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1 |r|
OC[C@@H](O)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1 |r|
OC[C@@H](O)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1 |r|
NC(=O)C(O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)C1CC1 |TLB:21:12:19:15.17.16,11:12:19:15.17.16,THB:17:18:13:15.16.21,17:16:13:19.18.20,21:16:19:12.13.20|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(Br)cn12 |TLB:22:13:20:16.17.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14,12:13:20:16.17.18|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:22:13:20:16.18.17,16:17:21:15.20.14,THB:22:17:20:21.13.14,16:15:21:22.18.17,12:13:20:16.18.17|
O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)N1CCCC1 |TLB:21:12:19:15.17.16,15:16:20:14.19.13,THB:21:16:19:20.12.13,15:14:20:21.17.16,11:12:19:15.17.16|
CCc1cn2c(NS(=O)(=O)C3CC3)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:29:20:27:23.24.25,23:24:28:22.27.21,THB:29:24:27:28.20.21,23:22:28:29.24.25,19:20:27:23.24.25|
CS(=O)(=O)Nc1nnc2cc(OCC3CCCCC3)c(Br)cn12
CC1(COc2cc3nnc(NS(C)(=O)=O)n3cc2C=C)CCCCC1
CC(=C)c1cn2c(NS(C)(=O)=O)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:28:19:26:22.23.24,THB:18:19:26:22.23.24,28:23:26:19.27.20,27:19:22:26.25.24,27:25:22:19.28.20|
Brc1cn2c(NS(=O)(=O)N3CCOCC3)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:31:22:29:25.26.27,THB:21:22:29:25.26.27,31:26:29:22.30.23,30:22:25:29.28.27,30:28:25:22.31.23|
COc1ncccc1-c1cn2c(NS(C)(=O)=O)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:33:24:31:27.28.29,THB:23:24:31:27.28.29,33:28:31:24.32.25,32:24:27:31.30.29,32:30:27:24.33.25|
CC(C)c1cn2c(N)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:24:15:22:18.19.20,THB:14:15:22:18.19.20,24:19:22:15.23.16,23:15:18:22.21.20,23:21:18:15.24.16|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1=CCCC1 |t:31,TLB:22:13:20:16.17.18,THB:12:13:20:16.17.18,22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)Nc1nnc2cc(OC[C@H]3CC[C@@H](CC3)C(F)(F)F)c(cn12)C1CC1 |r,wU:16.19,wD:13.12,(8.42,3.92,;6.93,3.52,;6.53,5,;7.33,2.03,;5.45,3.12,;5.05,1.63,;5.95,.39,;5.05,-.86,;3.58,-.38,;2.25,-1.15,;.92,-.38,;-.42,-1.15,;-1.75,-.38,;-3.09,-1.15,;-4.42,-.38,;-5.75,-1.15,;-5.75,-2.69,;-4.42,-3.46,;-3.09,-2.69,;-7.09,-3.46,;-8.42,-2.69,;-7.09,-5,;-8.42,-4.23,;.92,1.16,;2.25,1.93,;3.58,1.16,;-.42,1.93,;-1.19,3.26,;-1.96,1.93,)|
CC1(COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CCCCC1
CCc1cn2c(NS(=O)(=O)N3CC(F)C3)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:25:26:30:24.29.23,29:28:31:25.24.23,29:24:31:28.30.27,THB:25:24:30:31.27.26|
O=S(=O)(Nc1nnc2cc(OCC3CCC4(CC4)CC3)c(cn12)C1CC1)C1CC1
CCS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:23:14:21:17.18.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15,13:14:21:17.18.19|
CNS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:23:14:21:17.18.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15,13:14:21:17.18.19|
CC1(CC1)S(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:25:16:23:19.20.21,THB:25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17,15:16:23:19.20.21|
O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)C1CCC1 |TLB:21:12:19:15.16.17,THB:21:16:19:12.20.13,20:12:15:19.18.17,20:18:15:12.21.13,11:12:19:15.16.17|
CS(=O)(=O)Nc1nnc2cc(OCCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:23:14:21:17.18.19,13:14:17:21.20.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15|
O=S(=O)(Nc1nnc2cc(OCCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)C1CC1 |TLB:22:13:20:16.17.18,12:13:16:20.19.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)Nc1nnc2cc(OC3C4CC5CC(C4)CC3C5)c(cn12)C1CC1 |TLB:11:12:14:16.17.18,THB:12:20:16:14.13.18,12:13:16:20.19.21,19:20:14:16.17.18,19:17:14:20.12.21,(7.1,-2.22,;5.61,-2.62,;4.52,-3.71,;6.01,-4.11,;4.52,-1.53,;3.03,-1.93,;2.56,-3.39,;1.02,-3.39,;.54,-1.93,;-.86,-1.3,;-1.03,.23,;-2.51,.63,;-3.6,-.46,;-4.93,.31,;-6.26,-.46,;-6.26,-2,;-7.1,-3.9,;-5.7,-3.26,;-5.69,-.86,;-4.5,-3.93,;-3.6,-2,;-4.93,-2.77,;.22,1.13,;1.63,.51,;1.79,-1.02,;-.18,2.62,;.22,4.11,;-1.27,3.71,)|
O=S(=O)(Nc1nnc2cc(OC3C4CC5CC(C4)CC3C5)c(cn12)C1CC1)C1CC1 |TLB:17:16:20:13.12.11,17:12:20:15.16.18,THB:11:19:15:13.17.12,11:12:15:19.20.18,10:11:20:15.16.18,(5.44,-4.2,;5.04,-2.71,;3.95,-3.8,;3.95,-1.62,;2.46,-2.02,;1.84,-3.42,;.31,-3.26,;-.01,-1.76,;-1.35,-.99,;-1.35,.55,;-2.68,1.32,;-4.01,.55,;-4.01,-.99,;-6.32,-.37,;-8.02,1.32,;-8.02,-.22,;-6.68,-.99,;-5.35,-1.76,;-6.68,1.32,;-5.35,1.32,;-6.68,2.09,;-.01,1.32,;1.32,.55,;1.32,-.99,;-.01,2.86,;.76,4.2,;-.78,4.2,;6.53,-2.31,;8.02,-2.71,;7.62,-1.22,)|
CS(=O)(=O)Nc1nnc2cc(OCC3CC4C5CCC(C5)C4C3)c(cn12)C1CC1 |TLB:14:15:17.18:20|
O=S(=O)(Nc1nnc2cc(OCC3CC4C5CCC(C5)C4C3)c(cn12)C1CC1)C1CC1 |TLB:13:14:16.17:19|
O=S(=O)(Nc1nnc2cc(OCC3CC4C5CCC(C5)C4C3)c(cn12)C1CC1)N1CCC1 |TLB:13:14:16.17:19|
CC1(C)[C@@H]2C[C@H]1[C@@H](COc1cc3nnc(NS(C)(=O)=O)n3cc1C1CC1)CC2 |r|
CC1(C)[C@@H]2C[C@H]1[C@@H](COc1cc3nnc(NS(=O)(=O)C4CC4)n3cc1C1CC1)CC2 |r|
CC1(C)[C@@H]2C[C@H]1[C@@H](COc1cc3nnc(NS(=O)(=O)N4CCC4)n3cc1C1CC1)CC2 |r|
CC1(C)[C@H]2CC[C@@]1(C)[C@@H](C2)Oc1cc2nnc(NS(C)(=O)=O)n2cc1C1CC1 |r|
C[C@H]1CC[C@H](COc2cc3nnc(NS(C)(=O)=O)n3cc2Br)CC1 |r,wU:4.4,wD:1.0,(-8.36,-1.24,;-6.82,-1.24,;-6.05,-2.57,;-4.51,-2.57,;-3.74,-1.24,;-2.2,-1.24,;-1.43,.09,;.11,.09,;.88,1.43,;2.42,1.43,;3.45,2.57,;4.86,1.95,;4.7,.41,;5.78,-.67,;7.27,-.28,;8.36,-1.36,;8.36,.81,;6.87,1.21,;3.19,.09,;2.42,-1.24,;.88,-1.24,;.11,-2.57,;-4.51,.09,;-6.05,.09,)|
C[C@H]1CC[C@H](COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CC1 |r,wU:4.4,wD:1.0,(-8.36,-.47,;-6.82,-.47,;-6.05,-1.8,;-4.51,-1.8,;-3.74,-.47,;-2.2,-.47,;-1.43,.86,;.11,.86,;.88,2.2,;2.42,2.2,;3.45,3.34,;4.86,2.72,;4.7,1.18,;5.78,.1,;7.27,.49,;8.36,-.59,;8.36,1.58,;6.87,1.98,;3.19,.86,;2.42,-.47,;.88,-.47,;.11,-1.8,;-1.22,-2.57,;.11,-3.34,;-4.51,.86,;-6.05,.86,)|
COc1ncccc1-c1cn2c(NS(C)(=O)=O)nnc2cc1OC[C@H]1CC[C@H](C)CC1 |r,wU:24.26,wD:27.30,(3.19,-3.91,;2.42,-2.57,;.88,-2.57,;.11,-3.91,;-1.43,-3.91,;-2.2,-2.57,;-1.43,-1.24,;.11,-1.24,;.88,.09,;2.42,.09,;3.19,1.43,;4.7,1.75,;5.78,.66,;7.27,1.06,;8.36,-.03,;8.36,2.15,;6.87,2.55,;4.86,3.28,;3.45,3.91,;2.42,2.76,;.88,2.76,;.11,1.43,;-1.43,1.43,;-2.2,.09,;-3.74,.09,;-4.51,-1.24,;-6.05,-1.24,;-6.82,.09,;-8.36,.09,;-6.05,1.43,;-4.51,1.43,)|
O=S(=O)(Nc1nnc2cc(OC3CCC4(CCCCC4)CC3)c(cn12)C1CC1)C1CC1
FC(F)S(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:14:15:18:22.21.20,14:15:22:18.19.20,24:15:22:18.19.20,THB:24:19:22:15.23.16,23:15:18:22.21.20,23:21:18:15.24.16|
CS(=O)(=O)Nc1nnc2cc(OCC3(CCCC3)C(F)(F)F)c(cn12)C1CC1
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)ccn12 |TLB:12:13:16:20.19.18,12:13:20:16.17.18,22:13:20:16.17.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CCC1 |TLB:12:13:16:20.19.18,12:13:20:16.17.18,22:13:20:16.17.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
Clc1ccc(OCc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)cc1Cl
CS(=O)(=O)Nc1nnc2cc(COc3ccc(Cl)c(Cl)c3)c(cn12)C1CC1
Clc1ccc(OCc2cc3nnc(NS(=O)(=O)N4CCC4)n3cc2C2CC2)cc1Cl
FC(F)(F)Oc1cc(Cl)cc(OCc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)c1
CS(=O)(=O)Nc1nnc2cc(COc3cc(Cl)cc(OC(F)(F)F)c3)c(cn12)C1CC1
FC(F)(F)Oc1cc(Cl)cc(OCc2cc3nnc(NS(=O)(=O)N4CCC4)n3cc2C2CC2)c1
CS(=O)(=O)Nc1nnc2cc(COc3ccc(Cl)c(c3)C(F)(F)F)c(cn12)C1CC1
FC(F)(F)c1cc(OCc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)ccc1Cl
Cc1cc(Cl)cc(OCc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)c1
Cc1cc(Cl)cc(OCc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)c1
CC1(CC1)S(=O)(=O)Nc1nnc2cc(COc3cc(Cl)cc(OC(F)(F)F)c3)c(cn12)C1CC1
CC1(CC1)S(=O)(=O)Nc1nnc2cc(COc3cc(Cl)cc(Cl)c3)c(cn12)C1CC1
CS(=O)(=O)Nc1nnc2cc(COc3cc(Cl)cc(Cl)c3)c(cn12)C1CC1
Clc1cc(Cl)cc(OCc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)c1
CC1(COc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)CCC(F)(F)CC1
CS(=O)(=O)Nc1nnc2cc(OCC3CCCCC3)c(cn12)C1CC1
CS(=O)(=O)Nc1nnc2cc(COc3ccc(Cl)c(Cl)c3)c(Br)cn12
O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)C1CC1 |TLB:21:12:19:15.16.17,THB:21:16:19:12.20.13,20:12:15:19.18.17,20:18:15:12.21.13,11:12:19:15.16.17|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(Br)cn12 |TLB:12:13:15.16.20:18,THB:21:19:16:22.13.14,21:13:16:20.18.19,14:15:18:22.21.13,14:13:15.16.20:18|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:12:13:15.16.20:18,THB:21:19:16:22.13.14,21:13:16:20.18.19,14:15:18:22.21.13,14:13:15.16.20:18|
O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)N1CCCC1 |TLB:11:12:14.15.19:17,THB:20:18:15:21.12.13,20:12:15:19.17.18,13:14:17:21.20.12,13:12:14.15.19:17|
CCc1cn2c(NS(=O)(=O)C3CC3)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:19:20:22.23.27:25,THB:28:26:23:29.20.21,28:20:23:27.25.26,21:22:25:29.28.20,21:20:22.23.27:25|
CS(=O)(=O)Nc1nnc2cc(OC[C@H]3CC[C@@H](CC3)C(F)(F)F)c(cn12)C1CC1 |r,wU:16.19,wD:13.12,(8.61,3.84,;7.12,3.44,;6.72,4.93,;7.52,1.95,;5.63,3.04,;4.86,1.71,;5.77,.46,;4.86,-.78,;3.4,-.31,;2.06,-1.08,;.73,-.31,;-.6,-1.08,;-1.94,-.31,;-3.27,-1.08,;-4.61,-.31,;-5.94,-1.08,;-5.94,-2.62,;-4.61,-3.39,;-3.27,-2.62,;-7.27,-3.39,;-8.61,-2.62,;-7.27,-4.93,;-8.61,-4.16,;.73,1.23,;2.06,2,;3.4,1.23,;-.6,2,;-1.37,3.34,;-2.14,2,)|
CCc1cn2c(NS(=O)(=O)N3CC(F)C3)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:31:22:29:25.26.27,THB:31:26:29:22.30.23,21:22:29:25.26.27,30:22:25:29.28.27,30:28:25:22.31.23|
CCS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:23:14:21:17.18.19,THB:23:18:21:22.15.14,22:20:17:23.15.14,22:14:17:21.20.19,13:14:21:17.18.19|
CNS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:23:14:21:17.18.19,THB:23:18:21:22.15.14,22:20:17:23.15.14,22:14:17:21.20.19,13:14:21:17.18.19|
CC1(CC1)S(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:25:16:23:19.20.21,THB:25:20:23:24.17.16,24:22:19:25.17.16,24:16:19:23.22.21,15:16:23:19.20.21|
O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)C1CCC1 |TLB:21:12:19:15.16.17,THB:21:16:19:20.13.12,20:18:15:21.13.12,20:12:15:19.18.17,11:12:19:15.16.17|
CS(=O)(=O)Nc1nnc2cc(OCCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:23:14:21:17.18.19,13:14:17:21.20.19,THB:23:18:21:22.15.14,22:20:17:23.15.14,22:14:17:21.20.19|
O=S(=O)(Nc1nnc2cc(OCCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)C1CC1 |TLB:22:13:20:16.17.18,12:13:16:20.19.18,THB:22:17:20:21.14.13,21:19:16:22.14.13,21:13:16:20.19.18|
CS(=O)(=O)Nc1nnc2cc(OC3C4CC5CC(C4)CC3C5)c(cn12)C1CC1 |TLB:11:12:14:16.17.18,THB:12:13:16:19.21.20,12:20:16:14.13.18,19:17:14:12.21.20,19:20:14:16.17.18,(7.1,-2.22,;5.61,-2.62,;6.01,-4.11,;4.52,-3.71,;4.52,-1.53,;3.03,-1.93,;2.56,-3.39,;1.02,-3.39,;.54,-1.93,;-.86,-1.3,;-1.03,.23,;-2.51,.63,;-3.6,-.46,;-4.93,.31,;-6.26,-.46,;-6.26,-2,;-7.1,-3.9,;-5.7,-3.26,;-5.69,-.86,;-4.5,-3.93,;-3.6,-2,;-4.93,-2.77,;.22,1.13,;1.63,.51,;1.79,-1.02,;-.18,2.62,;.22,4.11,;-1.27,3.71,)|
C[C@H]1CC[C@H](COc2cc3nnc(NS(C)(=O)=O)n3cc2Br)CC1 |r,wU:4.4,wD:1.0,(-8.36,-1.24,;-6.82,-1.24,;-6.05,-2.57,;-4.51,-2.57,;-3.74,-1.24,;-2.2,-1.24,;-1.43,.09,;.11,.09,;.88,1.43,;2.42,1.43,;3.45,2.57,;4.86,1.95,;4.7,.41,;5.78,-.67,;7.27,-.28,;8.36,-1.36,;6.87,1.21,;8.36,.81,;3.19,.09,;2.42,-1.24,;.88,-1.24,;.11,-2.57,;-4.51,.09,;-6.05,.09,)|
C[C@H]1CC[C@H](COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CC1 |r,wU:4.4,wD:1.0,(-8.36,-.47,;-6.82,-.47,;-6.05,-1.8,;-4.51,-1.8,;-3.74,-.47,;-2.2,-.47,;-1.43,.86,;.11,.86,;.88,2.2,;2.42,2.2,;3.45,3.34,;4.86,2.72,;4.7,1.18,;5.78,.1,;7.27,.49,;8.36,-.59,;6.87,1.98,;8.36,1.58,;3.19,.86,;2.42,-.47,;.88,-.47,;.11,-1.8,;-1.22,-2.57,;.11,-3.34,;-4.51,.86,;-6.05,.86,)|
COc1ncccc1-c1cn2c(NS(C)(=O)=O)nnc2cc1OC[C@H]1CC[C@H](C)CC1 |r,wU:24.26,wD:27.30,(3.19,-3.91,;2.42,-2.57,;.88,-2.57,;.11,-3.91,;-1.43,-3.91,;-2.2,-2.57,;-1.43,-1.24,;.11,-1.24,;.88,.09,;2.42,.09,;3.19,1.43,;4.7,1.75,;5.78,.66,;7.27,1.06,;8.36,-.03,;6.87,2.55,;8.36,2.15,;4.86,3.28,;3.45,3.91,;2.42,2.76,;.88,2.76,;.11,1.43,;-1.43,1.43,;-2.2,.09,;-3.74,.09,;-4.51,-1.24,;-6.05,-1.24,;-6.82,.09,;-8.36,.09,;-6.05,1.43,;-4.51,1.43,)|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)ccn12 |TLB:22:13:20:16.17.18,12:13:16:20.19.18,12:13:20:16.17.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CCC1 |TLB:22:13:20:16.17.18,12:13:16:20.19.18,12:13:20:16.17.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
Clc1ccc(COc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)cc1Cl
CC1(COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CCN(Cc2cc(Cl)cc(Cl)c2)CC1
CC1(COc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)CCN(Cc2cc(Cl)cc(Cl)c2)CC1
CS(=O)(=O)Nc1nnc2cc(O[C@@H]3CCCN(Cc4ccc(F)cc4Cl)C3)c(cn12)C1CC1 |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)c(Cl)c1 |r|
CC1(COc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)CCC2(CC2)CC1
FC12CCC(COc3cc4nnc(NS(=O)(=O)C5CC5)n4cc3C3CC3)(CC1)CC2
CC1(COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CCN(CC1)C(c1ccccc1)c1ccccc1
C[C@H](N1CCC(C)(COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCC(C)(COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCC(COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc3nnc(NS(C)(=O)=O)n3cc2C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc3nnc(NS(=O)(=O)C4CC4)n3cc2C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
CC12CC3(C)CC(C)(C1)CC(COc1cc4nnc(NS(C)(=O)=O)n4cc1C1CC1)(C2)C3 |TLB:11:10:5:2.1.8,7:6:2:10.30.31,THB:30:10:5:2.1.8,30:1:5:10.9.31,9:10:2:5.6.8,9:6:2:10.30.31|
CS(=O)(=O)Nc1nnc2cc(OC[C@H]3C[C@@H]4CC[C@H](C3)N4C(c3ccccc3)c3ccccc3)c(cn12)C1CC1 |r,THB:21:20:13.14.19:17.16|
Clc1cc(Cl)cc(OC2CCN(Cc3cc4nnc(NS(=O)(=O)C5CC5)n4cc3C3CC3)CC2)c1
CCc1cn2c(NS(C)(=O)=O)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:27:18:25:21.22.23,17:18:21:25.24.23,THB:27:22:25:18.26.19,26:18:21:25.24.23,26:24:21:18.27.19|
CCc1cn2c(NS(=O)(=O)N3CCC3)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:20:21:24:28.27.26,20:21:28:24.25.26,30:21:28:24.25.26,THB:30:25:28:21.29.22,29:21:24:28.27.26,29:27:24:21.30.22|
O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)N1CCC1 |TLB:11:12:15:19.18.17,11:12:19:15.16.17,21:12:19:15.16.17,THB:21:16:19:12.20.13,20:12:15:19.18.17,20:18:15:12.21.13|
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(C=C)cn12 |TLB:22:13:20:16.17.18,12:13:16:20.19.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(Cl)c(c2)C(F)(F)F)cc1F
CN(C)S(=O)(=O)NC(=O)c1ccc(COc2ccc(Cl)c(Cl)c2)cc1
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N(C)C)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(N)(=O)=O)cc1Cl
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc(Cl)c(Cl)c2)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(OCC(C)C)c(Cl)c2)cc1F
NS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(Cl)c(c2)C(F)(F)F)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(Cl)c(c2)C(F)(F)F)cc1F
Fc1cc(Oc2ccc(Cl)c(c2)C(F)(F)F)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
NS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(OC(F)(F)F)c(Cl)c2)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(OC(F)(F)F)c(Cl)c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(OC(F)(F)F)c(Cl)c2)cc1F
CCCCN(CCCC)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(OCC(C)C)c(Cl)c2)cc1F
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCCC2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCCCC2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCCCCC2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N(C)C(C)C)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)NCc2ccccc2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N(C)Cc2ccccc2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)NCc2ccccn2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)Nc2ccc(cc2)C#N)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)NCc2cccnc2)cc1Cl
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCc2ccc(Cl)c(Cl)c2)cc1F
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)c2cn(C)cn2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCc3ccccc23)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)c2c[nH]cn2)cc1Cl
COC(=O)C1CCN(CC1)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(OCC(C)C)c(Cl)c2)cc1F
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)c2cccnc2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)NC(=O)OC(C)(C)C)cc1Cl
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(OCC(F)(F)C(F)F)c(Cl)c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(F)c(Oc2ccc(OC(F)(F)F)c(Cl)c2)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(OCC(F)(F)C(F)F)c(Cl)c2)cc1F
NS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(Cl)c(Cl)c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(Cl)c(Cl)c2)cc1F
NS(=O)(=O)NC(=O)c1cc(Cl)c(COc2cnc(OCC(F)(F)C(F)F)c(Cl)c2)cc1F
NS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(OCC(F)(F)C(F)F)c(Cl)c2)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(Cl)c(Cl)c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(COc2cnc(OCC(F)(F)C(F)F)c(Cl)c2)cc1F
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N(C)C)cc1C(F)(F)F
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCN(CC2)C(=O)OC(C)(C)C)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCNCC2)cc1Cl
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(cc2)C#N)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(cc2)-c2nccs2)cc1F
Fc1cc(Oc2ccc(OC(F)(F)F)c(Cl)c2)c(Cl)cc1C(=O)NS(=O)(=O)NC1CCC1
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3ccccc3c2)cc1F
NS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3ccccc3c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(F)c(F)c2)cc1F
NS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(F)c(F)c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCOc2ccccc2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cccc3ccccc23)cc1F
NS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cccc3ccccc23)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cccc3[nH]ccc23)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3cc[nH]c3c2)cc1F
COc1ccc(CCOc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N(C)C)cc1
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCc2ccccc2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3[nH]c(C)cc3c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cccc3cnccc23)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc(cc2)S(C)(=O)=O)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3cnn(C)c3c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(N3CCCCC3)c(Cl)c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3nc(C)sc3c2)cc1F
CC(C)COc1ncc(Oc2cc(F)c(cc2C#N)C(=O)NS(=O)(=O)N(C)C)cc1Cl
FC(F)C(F)(F)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCCC2)cc1Cl
FC(F)C(F)(F)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCOCC2)cc1Cl
CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCOCC2)cc1Cl
FC(F)C(F)(F)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)c2cccnc2)cc1Cl
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cc(OC(F)(F)F)ccc2F)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cccc3ncccc23)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3ncccc3c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3ccncc3c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cc(C)c(C#N)c(C)c2)cc1F
CC(C)COc1ncc(Oc2cc(F)c(cc2C#N)C(=O)NS(N)(=O)=O)cc1Cl
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2cnc(OC(C)C)c(Cl)c2)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc(Cl)c(c2)C(F)(F)F)cc1F
Fc1cc(COc2ccc(OC(F)(F)F)c(Cl)c2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc(Cl)c(Cl)c2)cc1F
OC1(COC1)c1cc(ccc1Oc1ccc(OC(F)(F)F)c(Cl)c1)C(=O)NS(=O)(=O)N1CCC1
CC(C)Oc1ncc(OCc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
CNS(=O)(=O)NC(=O)c1ccc(Oc2cnc(OC(C)C)c(Cl)c2)c(c1)-c1cccnc1OC
CC(C)Oc1ncc(Oc2ccc(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
Fc1cc(COc2ccc(Cl)c(c2)C(F)(F)F)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
COc1ncccc1-c1cc(ccc1Oc1cnc(OC(C)C)c(Cl)c1)C(=O)NS(=O)(=O)N1CCC1
CC(C)Oc1ncc(Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
CC(C)Oc1ncc(Oc2cc(F)c(cc2C2(F)COC2)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
CC(C)Oc1ncc(Oc2cc(F)c(cc2C2(O)COC2)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(Oc2cnc(OC(C)C)c(Cl)c2)cc1F
CC(C)Oc1ncc(Oc2cc(F)c(cc2C=C)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
Fc1cc(Oc2cnc(OCC(F)(F)F)c(Cl)c2)c(C=C)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(Oc2cnc(OCC(F)(F)F)c(Cl)c2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(Oc2cnc(OCC(F)(F)F)c(Cl)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(COc2cc(Cl)cc(OC(F)(F)F)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(COc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
COc1ncccc1-c1cc(ccc1Oc1ccc(OC(F)(F)F)c(Cl)c1)C(=O)NS(=O)(=O)N1CCC1
Fc1cc(COc2ccc(Cl)c(Cl)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(COc2ccc(Cl)c(Cl)c2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc(OC(F)(F)F)c(Cl)c2)cc1F
FC(F)C(F)(F)COc1ncc(OCc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)N1CCC2(CC1)OCc1ccccc21 |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)N1CCC2(CC1)C=Cc1ccccc21 |r,c:25|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)N1CCC2(CC1)OC(=O)c1ccccc21 |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)N1CCC2(CC1)N(CNC2=O)c1ccccc1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
CC1C=CC=C1[C@H]1CCCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r,c:2,4|
Cc1cc(c(F)cc1O[C@H]1CCC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC(F)(F)C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(ccc1O[C@H]1CCC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(ccc1O[C@H]1CCCC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(ccc1O[C@H]1CCCCC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCCC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(C)(C)CC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC(C)(C)C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1ccc(c(F)c1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(c(F)c1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cc1c(O[C@H]2CC(F)(F)CC[C@@H]2c2ccnn2C)ccc(c1F)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CC(F)(F)CC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(C)(C)C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CCCC[C@@H]2c2cn[nH]c2)cc(F)c1S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(F)(F)C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC(F)(F)C[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CCC(F)(F)C[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CC(F)(F)CC[C@@H]1c1cn[nH]c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(F)(F)CC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(F)(F)CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CC(F)(F)C[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(F)(F)C[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CCC[C@@H]1c1ccn[nH]1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CCC[C@@H]2c2ccn[nH]2)cc(F)c1S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CCC[C@@H]2c2ccn[nH]2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC(F)(F)C[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(F)(F)C[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CC(F)(F)CC[C@@H]2c2cn[nH]c2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1C[C@H](O)CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CC(F)(F)CC[C@@H]1c1ccn[nH]1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CC(F)(F)CC[C@@H]2c2ccn[nH]2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CCC(F)(F)C[C@@H]1c1ccn[nH]1)S(=O)(=O)Nc1ccncn1 |r|
CC(=O)O[C@@H]1CC[C@H](Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ccncn2)[C@H](C1)c1ccnn1C |r|
Fc1cc(O[C@H]2CCCC[C@@H]2c2ccn[nH]2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1cn[nH]c1)S(=O)(=O)Nc1ccncn1 |r|
CC(C)C[C@H](NC(C)=O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(=O)c1ccccn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(=O)C1CC1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
COCCOCC(=O)N[C@@H](CC(C)C)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(=O)c1cccnc1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(=O)NC(C)C)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(N)=O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(=O)NC(C)(C)C)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CS(=O)(=O)Nc1cc(Cl)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
CS(=O)(=O)N(C[C@H](O)CO)c1cc(Cl)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NS(=O)(=O)Nc1cc(Cl)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
CS(=O)(=O)Nc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO |r|
Cn1cnc(c1)S(=O)(=O)Nc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO |r|
CS(=O)(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(NS(=O)(=O)C3CC3)n2)cc1
Cn1cnc(c1)S(=O)(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
N[C@@H](Cc1c[nH]cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Fc1ccc(Oc2ccc(cc2)-c2cccc(NC(=O)[C@H](Cc3c[nH]cn3)NC(=O)C3CC3)n2)cc1 |r|
CC(=O)N1CCC(CC1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
COCC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OCC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)(O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CS(=O)(=O)N[C@@H](Cc1c[nH]cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)(C)OC(=O)N[C@@H](CC(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
CC(C)(C)OC(=O)N[C@@H](CC(N)=O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(=O)C1CC1)C(=O)Nc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO |r|
CC(C)C[C@H](NC(=O)c1ccccn1)C(=O)Nc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO |r|
OC(=O)CN1CCC(CC1)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
OC(=O)C1CCN(CC1)c1cc(Cl)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
OC[C@H](NC(=O)c1ccccn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OC[C@H](NC(=O)C1CC1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OC[C@H](NC(=O)c1cccnc1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OC[C@H](NC(=O)c1ccncc1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Cc1cc(no1)C(=O)N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)(C)OC(=O)N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OC[C@H](NC(=O)CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
O[C@@H]1C[C@H](N(C1)c1ncc(cc1Cl)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O |r|
O[C@@H]1C[C@H](N(C1)c1cc(Cl)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O |r|
Fc1ccc(Oc2ccc(cc2)-c2cc(Cl)cc(NCCN3CCNC3=O)n2)cc1
Nc1nc(O)cc(n1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
OC[C@@H](O)c1cc(NCCN2CCNC2=O)nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OCC(O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
OCC(O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1
OCC(O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
OCC(O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(C#N)c(c2)C(F)(F)F)cc1
OCC(O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1
CC(=O)N[C@@H](Cc1cn(C)cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Cn1cnc(C[C@@H](NC(=O)C(C)(C)O)C(=O)Nc2cccc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)c1 |r|
C[C@H](Nc1cc(Cl)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
C[C@H](Nc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
CCC(=O)N[C@@H](Cc1cn(C)cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C(=O)N[C@@H](Cc1cn(C)cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Cn1cnc(C[C@H](NC(=O)C(C)(C)C)C(=O)Nc2cccc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)c1 |r|
CC(=O)N[C@@H](Cc1cn(C)cn1)C(=O)Nc1cc(ccn1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Cn1cnc(C[C@H](NC(=O)C2CC2)C(=O)Nc2cccc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)c1 |r|
Cn1cnc(C[C@H](NC(=O)CC(F)(F)F)C(=O)Nc2cccc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)c1 |r|
CC(=O)N[C@@H](Cc1cn(C)cn1)C(=O)Nc4cccc(c3ccc(Oc2ccc(F)cc2)cc3)n4
Cn1cnc(C[C@@H](NC(=O)c2ccc(cc2)C(F)(F)F)C(=O)Nc2cccc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)c1 |r|
CC(C)(C)NC(=O)N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)C[C@H](NC(=O)CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)NC(=O)N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)(O)C(=O)N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
COCC(=O)N[C@@H](CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(=O)N[C@H](Cc1cn(C)cn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
CC(O)[C@H](NC(=O)CO)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OCC(O)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(NS(=O)(=O)\C=C\c3ccccc3)n2)cc1
Cn1cnc2ccc(cc12)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
Cn1cnc(C[C@H](NC(=O)Nc2cccc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)C(N)=O)c1 |r|
COC(=O)[C@H](Cc1cn(C)cn1)NC(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)[C@@H](Cc1cc2ccccc2[nH]1)NC(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)C[C@@H](NC(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)[C@@H](Cc1cnc[nH]1)NC(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
NC(=O)CNc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
CC(C)C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
NC(=O)[C@H](CO)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
Cn1cnc(C[C@H](Nc2cc(nc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)C(N)=O)C(N)=O)c1 |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)c1cc(NC2(CC2)C(N)=O)nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NC2(CCC2)C(N)=O)nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
CC(C)(Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(C#N)c(c2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
COC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
CCOC(=O)[C@@H]1Cc2ccccc2N1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
CCOC(=O)C1(CC1)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
COC(=O)C(C)(C)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)CCNc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
C[C@H](N(C)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
C[C@@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
CC(Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O
CC(CC(N)=O)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)C1CCCN(C1)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)C1COCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)C1CN(CCO1)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)C1CNCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(O)=O |r|
OC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCC[C@H]1C(O)=O |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1[C@@H](Cc2ccccc12)C(O)=O |r|
COC(=O)[C@H](C)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)OC(C)(C)C |r|
COC(=O)[C@H](C)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)OC(C)(C)C)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O)C(N)=O |r|
NC(=O)[C@@H]1Cc2ccccc2N1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(cn2)C#N)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2cc(Cl)ccc2F)cc1)C(N)=O)C(N)=O |r|
COC(=O)[C@H](C)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)OC |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCOCC1CO
C[C@@H](CO)Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCC[C@H]1CO |r|
CC(C)(O)CNc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(NCC2(O)CCCCC2)nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NC[C@H](O)CO)nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)c1cc(NC(CO)CO)nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCNCC1CO
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CC(O)C(O)C1 |w:25.28,27.30|
NC(=O)[C@@H](O)CNc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)c1cc(NC[C@H](O)C(O)=O)nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC1(C)OCC(CN(c2cc(nc(n2)-c2ccc(Oc3ccc(F)cc3)cc2)C(N)=O)S(C)(=O)=O)O1
CS(=O)(=O)N(CC(O)CO)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
C[C@H](Nc1nc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)C(N)=O)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
C[C@H](Oc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2cc(ccn2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ncccc2C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2cccc(n2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(nc2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2cccc(F)n2)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cn2)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(Cl)cn2)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(O)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)[N+]#[C-])cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(Oc2ccc(Cl)cc2-c2ccnc(N)c2)n1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccnc(Oc2ccc(F)cc2)c1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)nc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCN(CC1)c1ccc(F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCN(CC1)C(c1ccc(F)cc1)c1ccc(F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(Oc2ccc(cc2-c2ccnnc2)C(F)(F)F)n1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCC(CC1)C1Cc2ccccc2C1)C(N)=O)C(N)=O |r|
NC(=O)C1CN(CCN1)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1 |r|
C[C@H](Oc1cc(nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)C(N)=O)C(N)=O |r|
C[C@H](Oc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1)C(N)=O)C(N)=O |r|
NC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)C(N)=O |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1C[C@H](O)[C@@H](O)C1 |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1C[C@@H](O)[C@H](O)C1 |r|
CN1CCN(C(C1)C(N)=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O
CN1CCN(C(C1)C(N)=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
CN1CCN(C(C1)C(N)=O)c1cc(nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)C(N)=O
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc3OCOc3c2)cc1)C(N)=O)C(N)=O |r|
NC(=O)C1CNCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O
NC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2cc(Cl)ccc2F)cc1)C(N)=O |r|
NC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1)C(N)=O |r|
NC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1)C(N)=O |r|
NC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc3OCOc3c2)cc1)C(N)=O |r|
NC(=O)[C@@H]1CCCN1c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O |r|
C[C@H](Oc1cc(nc(n1)-c1ccc(Oc2cc(Cl)ccc2F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Oc1cc(nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(=O)NCCO |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(=O)N1CCOCC1 |r|
COC(=O)c1cc(ccc1Oc1ccc(F)cc1)-c1nc(N[C@@H](C)C(N)=O)cc(n1)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)c(CO)c1)C(N)=O)C(N)=O |r|
C[C@H](Oc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
C[C@H](Nc1cc(nc(n1)N1CCC(CC1)Oc1ccc(cc1)C#N)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CC(C1)Oc1ccc(OC(F)(F)F)cc1)C(N)=O)C(N)=O |r|
NC(=O)c1cc(O[C@H]2CCNC2=O)nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F |r,t:18|
C[C@H](Nc1cc(nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F)C(N)=O)C(N)=O |r,t:10|
Cn1ncc2c(Oc3ccc(cc3)-c3nc(N[C@H]4CCNC4=O)cc(n3)C(N)=O)ccc(Cl)c12 |r|
Cn1ncc2c(Oc3ccc(cc3)-c3nccc(n3)C(N)=O)ccc(Cl)c12
Cn1ncc2c(Oc3ccc(cc3)-c3cccc(n3)C(N)=O)ccc(Cl)c12
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)c3n(C)ncc23)cc1)C(N)=O)C(N)=O |r|
Cn1ncc2c(Oc3ccc(cc3)-c3nc(N[C@H]4CCNC4=O)cc(n3)C(N)=O)ccc(F)c12 |r|
Cn1ncc2c(Oc3ccc(cc3)-c3nc(N[C@H]4CCNC4=O)cc(n3)C(N)=O)cccc12 |r|
Cn1ncc2c(Oc3ccc(cc3)-c3nc(cc(n3)C(N)=O)[C@H](O)CO)ccc(Cl)c12 |r|
Cn1ncc2c(Oc3ccc(cc3)-c3cc(cc(n3)C(N)=O)[C@H](O)CO)ccc(Cl)c12 |r|
Cn1ncc2c(Oc3ccc(cc3)-c3cc(cc(n3)C(N)=O)[C@H](O)CO)ccc(F)c12 |r|
Cn1ncc2c(Oc3ccc(cc3)-c3cc(cc(n3)C(N)=O)[C@@H](O)CO)ccc(F)c12 |r|
Cn1ncc2c(Oc3cc(F)c(cc3Cl)S(=O)(=O)Nc3nncs3)ccc(Cl)c12
Cn1ncc2c(Oc3ccc(cc3)S(=O)(=O)Nc3nncs3)ccc(Cl)c12
OCC(O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1 |r|
OC[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1 |r|
CC(C)NC(=O)N1CCN(CC1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@@H](O)CO |r|
OCC(O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1
OCC(O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(F)(F)F)C#N)cc1
OCC(O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C#N)C(F)(F)F)cc1
OC[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(F)(F)F)C#N)cc1 |r|
OCC(O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
OC[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1 |r|
OC[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1 |r|
OCC(O)c1cccc(n1)-c1ccc(Oc2ncc(cc2Cl)C(F)(F)F)cc1
OCC(O)c1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1
OCC(O)c1cccc(n1)-c1ccc(Oc2ccc(nc2)C(F)(F)F)cc1
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1 |r|
CC(=O)c1ccc(Oc2ccc(cc2)-c2cccc(n2)C(O)CO)c(c1)C(F)(F)F
OC[C@H](O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCNCC1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(F)(F)F)C#N)cc1 |r|
OC[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
Cc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(O)CO)cn1
OCC(O)c1cccc(n1)-c1ccc(Oc2ncccc2C(F)(F)F)cc1
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(C#N)c(c2)C(F)(F)F)cc1)[C@H](O)CO |r|
NC(=O)c1ccc(Oc2ccc(cc2)-c2cc(cc(n2)C(N)=O)[C@H](O)CO)c(c1)C(F)(F)F |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(cc2C(F)(F)F)C#N)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(cc2C(F)(F)F)C#N)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2cc(Cl)ccc2F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO |r|
OC[C@@H](O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCCN1CCCCC1 |r|
CN(c1ccccc1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N(CCC#N)c1ccccc1
NC(=O)c1cc(NCc2cccnc2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NCc2ccncc2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NCc2ccccn2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NCCN2CCS(=O)(=O)CC2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NCc2ncccn2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
CS(=O)(=O)NCc1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(CN2CCNCC2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)CN1CCC(CNc2cc(nc(c2)-c2ccc(Oc3ccc(F)cc3)cc2)C(N)=O)CC1
NC(=O)c1cc(NCCN2CCOCC2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NCCCn2ccnc2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCNCC1
NC(=O)C1CCN(CC1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(NCC2CCNCC2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(NCCN2CCNC2=O)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCC(CC1)C(O)=O
NC(=O)c1cc(CNCCN2CCNC2=O)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
FC(F)(F)c1ccc(Oc2ccc(cc2)-c2cccc(CNCCN3CCNC3=O)n2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(CNCCN3CCNC3=O)n2)cc1
FC(F)(F)c1ccc(Oc2ccc(cc2)-c2cccc(CNCCN3CCNC3=O)n2)c(c1)C#N
Fc1ccc(Oc2ccc(cc2)-c2cccc(CCNCCN3CCNC3=O)n2)cc1
FC(F)(F)c1cc(ccc1Oc1ccc(cc1)-c1cccc(CNCCN2CCNC2=O)n1)C#N
FC(F)(F)c1cnc(Oc2ccc(cc2)-c2cccc(CNCCN3CCNC3=O)n2)c(Cl)c1
O=C1NCCN1CCNCc1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1
FC(F)(F)c1ccc(Oc2ccc(cc2)-c2cccc(CNCCN3CCNC3=O)n2)nc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(CN(CCN3CCNC3=O)CC#N)n2)cc1
FC(F)(F)c1ccc(Oc2ccc(cc2)-c2cccc(CNCCN3CCNC3=O)n2)cc1C#N
CS(=O)(=O)c1ccc(Oc2ccc(cc2)-c2cccc(CNCCN3CCNC3=O)n2)cc1
NC(=O)CN(CCN1CCNC1=O)Cc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
CC(C)NC(=O)N1CCN(CC1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCN(CC1)c1ncccn1
NC(=O)N1CCN(CC1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N1CCN(CC1)C1=NCCCN1 |t:33|
Fc1ccc(Oc2ccc(cc2)-c2cc(cc(n2)C(=O)N2CCNCC2)N2CCNCC2)cc1
OCc1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCCN1CCCCC1
NC(=N)N1CCN(CC1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCCN1CCCCC1
CC(C)NC(=O)N1CCN(CC1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C#N
NC(=N)N1CCN(CC1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C#N
NC(=O)c1cc(NC(=O)Nc2ccccc2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
OC(=O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCCN1CCCCC1
Fc1ccc(Oc2ccc(cc2)-c2cc(cc(n2)C(=O)NCCN2CCCCC2)-c2nnn[nH]2)cc1
NC(=O)c1cc(NC(=O)NCC(O)=O)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
C[C@H](NCc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@@H](O)CO |r|
CN(c1ccc(cc1)C(O)=O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N(CC(O)=O)c1ccccc1
OC(=O)c1cn(-c2cc(nc(c2)-c2ccc(Oc3ccc(F)cc3)cc2)C(O)=O)c2ccccc12
OC(=O)c1cc(cc(n1)N(CCC#N)c1ccccc1)-c1ccc(Oc2ccc(F)cc2)cc1
OC[C@@H](O)c1cc(cc(n1)C(O)=O)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)c1cc(cc(n1)[C@@H](O)CO)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)CN(c1ccccc1)c1cc(cc(n1)C(O)=O)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)-n1ccc2c(cccc12)C#N
NC(=O)c1cc(cc(n1)-n1ccc2c(cccc12)C#N)-c1ccc(Oc2ccc(F)cc2)cc1
OC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)-n1ccc2c(cccc12)C#N
NC(=O)c1cc(CN2CCN(CC(O)=O)CC2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cc(CNCCN3CCNC3=O)ccn2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cc(CNCCN3CCNC3=O)cc(n2)C#N)cc1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCCN1CCCCC1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)-c1nnn(CC(N)=O)n1
NC(=O)CN1CCN(CC1)c1cc(Cl)nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cc(NCCCn3ccnc3)cc(n2)C#N)cc1
OC[C@H](O)c1cc(NCCN2CCOCC2)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
OC[C@@H](O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C#N |r|
CN(c1ccccc1)c1cc(cc(n1)C(N)=O)-c1ccc(Oc2ccc(F)cc2)cc1
CN(c1ccccc1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O
NC(=O)c1cc(cc(n1)N(CCC#N)c1ccccc1)-c1ccc(Oc2ccc(F)cc2)cc1
CN(c1ccc(cc1)C(O)=O)c1cc(cc(n1)C(N)=O)-c1ccc(Oc2ccc(F)cc2)cc1
CN(c1ccc(cc1)C(O)=O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O
CN(c1ccccc1)c1cc(cc(n1)C(O)=O)-c1ccc(Oc2ccc(F)cc2)cc1
CN(c1ccc(cc1)C(O)=O)c1cc(cc(n1)C(O)=O)-c1ccc(Oc2ccc(F)cc2)cc1
OC(=O)CN(c1ccccc1)c1cc(cc(n1)C(O)=O)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C1=CCNCC1 |t:26|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2cc(Cl)ccc2F)cc1)[C@@H](O)CO |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(cc1)S(=O)(=O)Nc1ccc(F)cc1 |r|
OCC(CO)NC(=O)c1cc(cc(Cl)n1)-c1ccc(Oc2ccc(F)cc2)cc1
OC(=O)c1cc(cc(n1)-n1ccc2c(cccc12)C#N)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(C#N)c(c2)C(F)(F)F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(NC(CO)CO)n1)-c1ccc(Oc2ccc(F)cc2)cc1
C[C@H](O)[C@@H](O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
OC(=O)c1ccc2ccn(-c3cc(nc(c3)-c3ccc(Oc4ccc(F)cc4)cc3)C(O)=O)c2c1
C[C@@H](O)[C@H](O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(NC(CO)CO)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(C[C@@H](O)CO)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)c1cc(C[C@H](O)CO)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)c1cc(O)cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
OC[C@@H](O)c1cccc(n1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1cccc(Oc2ccc(F)cc2)c1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)N(CC(O)=O)c1ccccc1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)N(CCC(O)=O)c1ccccc1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N(CCC(O)=O)c1ccccc1
CN(c1ccccc1)c1cc(cc(n1)C(N)=O)-c1ccc(Oc2ccc(cc2)C#N)cc1
CN(c1ccccc1)c1cc(nc(c1)-c1ccc(Oc2ccc(cc2)C#N)cc1)C(N)=O
CN(c1ccccc1)c1cc(cc(n1)C(N)=O)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1
CN(c1ccccc1)c1cc(nc(c1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N(CCc1nn[nH]n1)c1ccccc1
NC(=O)c1cc(cc(n1)N(CCc1nn[nH]n1)c1ccccc1)-c1ccc(Oc2ccc(F)cc2)cc1
OC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N(CCc1nn[nH]n1)c1ccccc1
OC(=O)c1cc(cc(n1)N(CCc1nn[nH]n1)c1ccccc1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1cc(cc(n1)-c1ccc(cc1)-c1ccc(F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(cc1)-c1ccc(F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)[C@H](O)CO)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1 |r|
NC(=O)c1cc(cc(n1)[C@@H](O)CO)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1 |r|
NC(=O)c1cc(cc(n1)[C@H](O)CO)-c1ccc(Oc2cccc(OC(F)(F)F)c2)cc1 |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)[C@H](O)CO)-c1ccc(cc1)-c1ccc(F)cc1 |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2cccc(OC(F)(F)F)c2)cc1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2cccc(OC(F)(F)F)c2)cc1)[C@@H](O)CO |r|
C[C@H](Nc1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C#N)C(N)=O |r|
C[C@H](Nc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C#N)C(N)=O |r|
C[C@H](Nc1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O)C(N)=O |r|
CCOC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
NC(=O)[C@H](O)[C@@H](O)c1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
CCOC(=O)[C@@H](O)[C@H](O)c1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
CNC(=O)[C@@H](O)[C@H](O)c1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
NC(=O)[C@@H](O)[C@H](O)c1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
NC(=O)[C@H](O)[C@@H](O)c1ccnc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1 |r|
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(Cl)cn2)cc1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(Cl)cn2)cc1 |r|
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(C#N)c(c2)C(F)(F)F)cc1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(C#N)c(c2)C(F)(F)F)cc1 |r|
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(Cl)nc2)cc1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(Cl)nc2)cc1 |r|
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2)C#N)cc1 |r|
COc1ccc(OCC(F)(F)C(F)(F)F)c(c1)-c1ccc2c(N)nn(C)c2c1
Cn1nc(N)c2ccc(cc12)-c1ccccc1OCC(F)(F)F
Cn1nc(NCCO)c2ccc(cc12)-c1ccccc1OCC(F)(F)C(F)(F)F
Nc1n[nH]c2cc(ccc12)-c1ccccc1OCC(F)(F)C(F)(F)F
Cn1nc(N)c2ccc(cc12)-c1cccc(F)c1OCC(F)(F)C(F)(F)F
Cn1nc(N)c2ccc(cc12)-c1c(F)cccc1OCC(F)(F)C(F)(F)F
Cn1nc(NCCCO)c2ccc(cc12)-c1ccccc1OCC(F)(F)C(F)(F)F
NC(=O)Cn1nc(N)c2ccc(cc12)-c1cccc(F)c1OCC(F)(F)C(F)(F)F
COc1cccc(-c2ccc3c(N)nn(C)c3c2)c1OCC(F)(F)F
COc1cccc(-c2ccc3c(N)nn(C)c3c2)c1OCC(F)F
Cn1nc(N)c2ccc(cc12)-c1cccc(F)c1OCC(F)F
CN1CCC(CNc2nn(C)c3cc(ccc23)-c2cccc(F)c2OCC(F)(F)F)CC1
Cn1nc(N)c2ccc(cc12)-c1cccnc1OCC(F)(F)F
CNc1nn(C)c2cc(ccc12)-c1cccc(F)c1OCC(F)F
Cn1nc(N)c2ccc(cc12)-c1cccc(F)c1OC(F)F
Nc1nn(CCCO)c2cc(ccc12)-c1ccccc1C(F)(F)F
Nc1nn(CCCO)c2cc(ccc12)-c1ccccc1OC(F)(F)F
COCCn1nc(N)c2ccc(cc12)-c1ccccc1OC(F)(F)F
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)[C@@H]1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)C1CCNCC1(F)COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1ccc(cc1F)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncccn1 |r|
Fc1ccc(cc1)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncccn1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1nncs1 |r|
Cc1nsc(NS(=O)(=O)c2cc(F)c(OC[C@@H]3CNCCC3c3ccc(Cl)cc3)cc2F)n1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
Cc1cc(NS(=O)(=O)c2cc(F)c(OC[C@@H]3CNCCC3c3ccc(Cl)cc3)cc2F)no1 |r|
Cc1cnc(NS(=O)(=O)c2cc(F)c(OC[C@@H]3CNCCC3c3ccc(Cl)cc3)cc2F)o1 |r|
Clc1ccc(cc1)C1CCNC[C@H]1COc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(ccc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ccncn1 |r|
Fc1ccc(cc1F)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncc(Cl)s1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncc(Cl)s1 |r|
Fc1ccc(NS(=O)(=O)c2cc(F)c(OC[C@@H]3CNCCC3c3ccc(Cl)cc3)cc2F)nc1 |r|
Fc1cnc(NS(=O)(=O)c2cc(F)c(OC[C@@H]3CNCCC3c3ccc(Cl)cc3)cc2F)nc1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1cccnn1 |r|
Fc1cc(c(F)cc1OC[C@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)C1CCCC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
CC(C)(C)OC(=O)N1CCC([C@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C1)c1ccc(Cl)cc1 |r|
CN1CCC([C@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C1)c1ccc(Cl)cc1 |r|
Fc1cc(c(F)cc1OC[C@H]1CNCC[C@@H]1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
Cn1cns\c1=N\S(=O)(=O)c1cc(F)c(OC[C@@H]2CNCCC2c2ccc(Cl)cc2)cc1F |r|
CN(c1ncns1)S(=O)(=O)c1cc(F)c(OC[C@@H]2CNCCC2c2ccc(Cl)cc2)cc1F |r|
FCCN1CCC([C@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C1)c1ccc(Cl)cc1 |r|
Fc1cc(cc(F)c1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)C1CNCC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
FC(F)CN1CCC([C@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C1)c1ccc(Cl)cc1 |r|
CN1CC[C@@H]([C@@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C1)c1ccc(Cl)cc1 |r|
CN1CC[C@H]([C@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C1)c1ccc(Cl)cc1 |r|
Fc1ccc(cc1)C1CC(=O)NC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CN(CC(F)(F)F)CCC1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
NC(=O)N1CCC([C@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncc(Cl)s2)C1)c1ccc(F)c(F)c1 |r|
CC(C)NS(=O)(=O)c1ccc(OC[C@@H]2CNCCC2c2ccc(Cl)cc2)c(c1)C#N |r|
Clc1ccc(cc1)C1CCNC[C@H]1COc1ccc(cc1C#N)S(=O)(=O)NC1(CC1)C#N |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)c(Cl)c1)S(=O)(=O)Nc1ncns1 |r|
FC(F)(F)CNS(=O)(=O)c1ccc(OC[C@@H]2CNCCC2c2ccc(Cl)cc2)c(c1)C#N |r|
COc1ccc(cc1)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
NS(=O)(=O)c1cc(F)c(OC[C@@H]2CNCCC2c2ccc(Cl)cc2)cc1F |r|
CC(C)CNS(=O)(=O)c1cc(F)c(OC[C@@H]2CNCC[C@H]2c2ccc(Cl)cc2)cc1F |r|
Fc1cc(ccc1Cl)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)n1cccn1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)NC(=O)c1ccccn1 |r|
Cc1ccc(cc1)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(F)c(cc1F)C1CC(=O)NC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
CC(=O)NS(=O)(=O)c1cc(F)c(OC[C@@H]2CNCCC2c2ccc(Cl)cc2)cc1F |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)NC(=O)c1cccnc1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(Cl)cc1)S(=O)(=O)NC(=O)c1ccccc1 |r|
CC(C)NC(=O)NS(=O)(=O)c1cc(F)c(OC[C@@H]2CNCCC2c2ccc(Cl)cc2)cc1F |r|
Fc1cc(F)c(cc1F)C1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CNCCC1c1ccc(F)c(c1)C(F)(F)F)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1OC[C@@H]1CC(=O)CC[C@H]1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
O[C@@H]1CCC([C@H](COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C1)c1ccc(Cl)cc1 |r|
Fc1cc(c(F)cc1OCC1CNCCN1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1cnc(Oc2c(C)cccc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(C)c(Cl)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(C)cc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(Cl)cc2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(N2CCC[C@H]2C(C)C)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(F)c(F)c2F)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(F)cc2C)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2c(F)ccc(F)c2F)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(F)ccc2F)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(C)c(Cl)c(C)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1ccc(Oc2ncc(cc2Cl)-c2ccc(cc2OC)C(=O)NS(C)(=O)=O)c(Cl)c1
CCc1cc(Oc2ncc(cc2Cl)-c2ccc(cc2OC)C(=O)NS(C)(=O)=O)ccc1Cl
COc1ccc(Cl)c(Oc2ncc(cc2Cl)-c2ccc(cc2OC)C(=O)NS(C)(=O)=O)c1
COc1cc(ccc1-c1cnc(Oc2ccc(Cl)c(c2)C(F)(F)F)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(F)ccc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(OC(F)(F)F)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(Cl)c(OC(F)(F)F)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(c2)C(F)(F)F)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(Cl)cc2F)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(F)cc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)ccc2C)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(c1)C(F)F)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cccc(F)c2F)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1ncc(Oc2ncc(cc2Cl)-c2ccc(cc2OC2COC2)C(=O)NS(C)(=O)=O)cc1Cl
Cc1cc(Oc2ncc(cc2Cl)-c2ccc(cc2OC2COC2)C(=O)NS(C)(=O)=O)ccc1Cl
CS(=O)(=O)NC(=O)c1ccc(c(OC2COC2)c1)-c1cnc(Oc2cccc3ccccc23)c(Cl)c1
CS(=O)(=O)NC(=O)c1ccc(c(OC2COC2)c1)-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1
Cc1ccc(Cl)c(Oc2ncc(cc2Cl)-c2ccc(cc2OC2COC2)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(c(OC2COC2)c1)-c1cnc(Oc2ccc3ccccc3c2)c(Cl)c1
Cc1ccc(Oc2ncc(cc2Cl)-c2ccc(cc2OC2COC2)C(=O)NS(C)(=O)=O)cc1Cl
Cc1cccc(Cl)c1Oc1ncc(cc1Cl)-c1ccc(cc1OC1COC1)C(=O)NS(C)(=O)=O
COc1ncc(Oc2ncc(cc2Cl)-c2ccc(cc2OC(F)F)C(=O)NS(C)(=O)=O)cc1Cl
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(Oc2ccc3ccccc3c2)c(Cl)c1
Cc1ccc(Oc2ncc(cc2Cl)-c2ccc(cc2OC(F)F)C(=O)NS(C)(=O)=O)cc1Cl
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(Oc2cccc3ccccc23)c(Cl)c1
Cc1cc(Oc2ncc(cc2Cl)-c2ccc(cc2OC(F)F)C(=O)NS(C)(=O)=O)ccc1Cl
C[C@@H](Oc1ncc(cc1Cl)-c1ccc(cc1OC(F)F)C(=O)NS(C)(=O)=O)c1ccccc1
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(Oc2cccc(c2)C(F)(F)F)c(Cl)c1
C[C@H](Oc1ncc(cc1Cl)-c1ccc(cc1OC(F)F)C(=O)NS(C)(=O)=O)c1ccccc1
Cc1ccc(Oc2ncc(cc2Cl)-c2ccc(cc2OC(F)F)C(=O)NS(C)(=O)=O)cc1C
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(Oc2ccc(Cl)c(F)c2)c(Cl)c1
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1
Cc1ccc(Cl)c(Oc2ncc(cc2Cl)-c2ccc(cc2OC(F)F)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(Oc2ccccc2C(F)(F)F)c(Cl)c1
Cc1ccc(Oc2ncc(cc2Cl)-c2ccc(cc2OC(F)F)C(=O)NS(C)(=O)=O)c(Cl)c1
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(Oc2ccc(Cl)cc2)c(Cl)c1
CS(=O)(=O)NC(=O)c1ccc(c(OC(F)F)c1)-c1cnc(OCCc2ccccc2)c(Cl)c1
Cc1cccc(Cl)c1Oc1ncc(cc1Cl)-c1ccc(cc1OC(F)F)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(OCCc2ccccc2)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(C)c(Cl)c2)c(c1)C#N)C(=O)NS(C)(=O)=O
C[C@@](Oc1ncc(cc1Cl)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O)(c1ccccc1)C(F)(F)F
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(F)c(cc1F)-c1cnc(Oc2c(Cl)cc(Cl)cc2Cl)c(Cl)c1
Cc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2F)C(=O)NS(C)(=O)=O)c(F)c1F
CS(=O)(=O)NC(=O)c1cc(F)c(cc1F)-c1cnc(Oc2ccc(Cl)c(Cl)c2)c(Cl)c1
Cc1ccc(Cl)cc1Oc1ncc(cc1Cl)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(F)c(cc1F)-c1cnc(Oc2c(Cl)cc(F)cc2Cl)c(Cl)c1
CS(=O)(=O)NC(=O)c1cc(F)c(cc1F)-c1cnc(Oc2ccc(F)c3CCCc23)c(Cl)c1
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O)c1ccc(F)cc1F
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Br)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(OCc2ccc(Cl)cc2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(OCc2ccccc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2c(C)cc(Cl)cc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cccc(Cl)c2C)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc3CCCc3c2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2c(Cl)cccc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)ccc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cccc(Cl)c2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1ccc(cc1OC1COC1)C(=O)NS(C)(=O)=O
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1ccc(cc1OC(F)F)C(=O)NS(C)(=O)=O
Cc1c(Cl)cccc1Oc1ncc(cc1Cl)-c1ccc(cc1OC(F)F)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@](C)(c2ccccc2)C(F)(F)F)c(Cl)c1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-c1cnc(Oc2ccc(F)c(F)c2F)c(Cl)c1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-c1cnc(Oc2cc(F)cc(F)c2F)c(Cl)c1
Cc1ccc(Cl)cc1Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
Cc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2Cl)C(=O)NS(C)(=O)=O)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-c1cnc(Oc2c(Cl)cccc2Cl)c(Cl)c1
CC[C@H](Cc1ccccc1)Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CC(C)[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)c1ccccc1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-c1cnc(Oc2cc(F)ccc2Cl)c(Cl)c1
CC[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)c1ccc(F)cc1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-c1cnc(Oc2cc(F)ccc2F)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-c1cnc(Oc2cc(F)cc(F)c2Cl)c(Cl)c1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-c1cnc(OCC2CCCC2)c(Cl)c1
CCC(CC)Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CC1(CCC1)Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)cc2F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(F)c2F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)ccc2F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)c(Br)cc2Cl)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(Br)c2)c(Cl)c1
Cc1ccc2ccccc2c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Br)cc2)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc3CCCCc23)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(cc2Cl)C(C)(C)C)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccccc2-c2ccccc2)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Cl)c3ccccc23)c(Cl)c1
Cc1cc(Br)ccc1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)c(F)c2F)c(Cl)c1
Cc1ccc(Cl)cc1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)ccc2F)c(Cl)c1
Cc1cccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c1F
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(Cl)c2F)c(Cl)c1
Cc1cc(Cl)ccc1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(F)cc(F)cc2F)c(Cl)c1
Cc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)cc1F
Cc1ccc(c(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c1)C(C)(C)C
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(F)ccc(Cl)c2F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)c(Cl)c2)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(Cl)cccc2Cl)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)cc(F)c2F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)cc(F)c2)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)cc(F)c2Cl)c(Cl)c1
Cc1cc(Cl)c(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)cc1C
Cc1cccc(c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)C(C)(C)C
Cc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c(c1)C(C)(C)C
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H]2C[C@H]3CC[C@@H]2C3)c(Cl)c1 |THB:19:20:23.24:26|
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCc2nc3ccccc3s2)c(Cl)c1
CC(C)CCOc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
C[C@H](CCc1ccccc1)Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
CC[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1ccc(F)cc1
CC[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1ccc(Cl)cc1
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)C1CCC1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(ccc2Cl)C(F)(F)F)c(Cl)c1
Cc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c(F)c1F
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(Cl)cc(F)cc2Cl)c(Cl)c1
CCOc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)cc1F
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N2CCC[C@H]2c2ccccc2)c(Cl)c1
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1nc2ccccc2s1
COc1ccccc1C[C@@H](C)Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
CC[C@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1ccc(F)cc1
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1ccc(F)cc1Cl
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1nc2cc(Cl)ccc2s1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCc2cccc3ncccc23)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N2CCC[C@@H]2c2cccc(c2)C(F)(F)F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N2CCC[C@@H]2c2cccc(Cl)c2)c(Cl)c1
Cc1ccc(cc1)[C@H]1CCCN1c1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N2CCC[C@@H]2c2ccc(Cl)c(Cl)c2)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N2CCC[C@@H]2c2ccccc2C(F)(F)F)c(Cl)c1
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1cc(F)c(F)cc1F
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1c(F)cc(F)cc1F
Cc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c2CCCc12
CC(C)Oc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)cc1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Cl)c(Cl)c2)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Cl)cc2Cl)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(F)cc(F)cc2Cl)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)c(Cl)cc2Cl)c(Cl)c1
Cc1cc(Cl)cc(C)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1ccc(Cl)c(Oc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c1F
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(c(F)c2)C(F)(F)F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)c3CCCc23)c(Cl)c1
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1cc(Cl)ccc1Cl
C[C@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1cc(Cl)ccc1Cl
CC[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1ccc(F)c(C)c1
CC[C@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1cccc(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(c2C)C(F)(F)F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)cc2C(F)(F)F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Cl)cc2C(F)(F)F)c(Cl)c1
CCc1ccc(C)cc1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(Cl)ccc1COc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
C[C@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1cccc2ccccc12
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCCC2CC2)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H](c2ccccc2)C(F)(F)F)c(Cl)c1
CC[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1ccc(C)cc1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OC(C(F)(F)F)C(F)(F)F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H]2CCCC(C)(C)C2)c(Cl)c1
C[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1ccccc1C(F)(F)F
COc1cc(ccc1-c1cnc(Oc2c(C)cc(Cl)cc2Cl)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cccc(Cl)c2C)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(Cl)cc2Cl)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2ccc(Cl)c(Cl)c2)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2c(Cl)cc(C)cc2Cl)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2c(Cl)ccc(Cl)c2C)c(c1)C#N)C(=O)NS(C)(=O)=O
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H](C)c2ccccc2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N(C)C2CCC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(C)c(F)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)ccc2C)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)cc(F)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)c(F)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OC2CCC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H]2C[C@H]3CC[C@@H]2C3)c(Cl)c1 |THB:20:21:24.25:27|
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(Cl)c2C)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)ccc2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H](C)Cc2ccccc2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)cc(F)c2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCc2nc3ccccc3s2)c(Cl)c1
C[C@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O)c1nc2ccccc2s1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(C)cc(Cl)cc2Cl)c(Cl)c1
CC[C@H](Cc1ccccc1)Oc1ncc(cc1Cl)-c1cc(F)c(cc1OC)C(=O)NS(C)(=O)=O
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCC2(C)CCCCC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc3ccccc3cc2Cl)c(Cl)c1
COc1cc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2OC)C(=O)NS(C)(=O)=O)c(Cl)cc1Cl
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc3ccccc3c2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCC2C(C)(C)C2(C)C)c(Cl)c1
CC[C@@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1OC)C(=O)NS(C)(=O)=O)C(F)(F)F
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N[C@@H]2CC22CCCC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(NCC2CCC(C)(C)CC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N[C@@H]2CCC22CCC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(NCC2CC(C)(C)C2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(NC2CCC(C)(C)CC2)c(Cl)c1
CCC(CC)Nc1ncc(cc1Cl)-c1cc(F)c(cc1OC)C(=O)NS(C)(=O)=O
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H](C)CC(C)C)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H]2CCC[C@H]2C)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Sc2ccc(C)cc2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Sc2cc(C)cc(C)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(SCc2cc(F)ccc2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(NCCC2CCCC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H](C)C2CCC2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H]2CC[C@H]2C)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OC2(CCC2)C(F)(F)F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H]2C[C@H](C)C2)c(Cl)c1 |r,wU:23.24,wD:21.21,(8.95,-5.62,;10.28,-4.85,;10.28,-3.31,;11.61,-2.54,;11.61,-1,;12.95,-.23,;12.95,1.31,;14.28,-1,;15.61,-.23,;14.84,1.11,;16.95,.54,;16.38,-1.56,;10.28,-.23,;10.28,1.31,;8.95,-1,;8.95,-2.54,;7.61,-3.31,;7.61,-4.85,;6.28,-5.62,;4.94,-4.85,;3.61,-5.62,;3.61,-7.16,;2.52,-8.24,;3.61,-9.33,;3.61,-10.87,;4.7,-8.24,;4.94,-3.31,;3.61,-2.54,;6.28,-2.54,)|
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(Cl)cc(F)cc2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Cl)cc2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)c(Cl)cc2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)cc(F)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)c(Cl)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)cc2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)ccc2C)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(F)ccc(Cl)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(Cl)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(C)c(F)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)ccc2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(C)cccc2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCc2ccc(Cl)cc2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(C)c(Cl)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(C)ccc2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Cl)cc2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)c(C)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(Cl)c(Cl)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2ccc(F)c3CCCc23)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H](C)Cc2ccccc2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(F)ccc(C)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(C)c2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H](C)c2ccc(F)cc2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(Cl)ccc(C)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)c(Cl)c(F)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(Cl)cccc2Cl)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(Cl)c2)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2c(F)ccc(F)c2F)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H](C)C2CCC2)c(Cl)c1
CC[C@H](Oc1ncc(cc1Cl)-c1cc(F)c(cc1OC)C(=O)NS(C)(=O)=O)C(F)(F)F
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@@H]2CC[C@@H]2C)c(Cl)c1
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(N[C@H]2CC22CCCC2)c(Cl)c1
CNS(=O)(=O)NC(=O)c1ccc(c(OC)c1)-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1)C(=O)NS(=O)(=O)N1CCC1
COc1cc(ccc1-c1cnc(COc2ccc(Cl)c(Cl)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1ccc(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1ccc(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1ccc(c(Cl)c1)-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1
CS(=O)(=O)NC(=O)c1ccc(c(Cl)c1)-c1cnc(Oc2c(F)ccc(F)c2F)c(Cl)c1
CCOc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cccc(Cl)c2C)c(Cl)c1
Cc1c(Cl)cccc1Oc1ncc(cc1Cl)-c1cc(F)c(cc1OC(F)F)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(OC(F)F)c(cc1F)-c1cnc(OC2CCC2)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1OC(F)F)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(OC(F)F)c(cc1F)-c1cnc(O[C@@H]2C[C@H]3CC[C@H]2C3)c(Cl)c1 |THB:22:23:26.27:29|
NC(=O)c1cc(OC(F)F)c(cc1S(=O)(=O)CF)-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(Cl)c1
CS(=O)(=O)NC(=O)c1cc(OC(F)F)c(cc1F)-c1cnc(Oc2c(F)ccc(F)c2F)c(Cl)c1
CS(=O)(=O)NC(=O)c1cc(OC(F)F)c(cc1F)-c1cnc(OCc2ccc(Cl)cc2)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1C#N)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
CCS(=O)(=O)NC(=O)c1ccc(c(OC)c1)-c1cnc(Oc2c(C)cc(Cl)cc2Cl)c(Cl)c1
CCS(=O)(=O)NC(=O)c1ccc(c(OC)c1)-c1cnc(Oc2cccc(Cl)c2C)c(Cl)c1
CCS(=O)(=O)NC(=O)c1ccc(c(OC)c1)-c1cnc(OC2CCC2)c(Cl)c1
CCS(=O)(=O)NC(=O)c1ccc(c(OC)c1)-c1cnc(Oc2c(F)ccc(F)c2F)c(Cl)c1
CCS(=O)(=O)NC(=O)c1ccc(c(OC)c1)-c1cnc(O[C@H]2C[C@H]3CC[C@@H]2C3)c(Cl)c1 |THB:20:21:24.25:27|
COc1cc(ccc1-c1cnc(Cc2ccc(Cl)c(Cl)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1ccc(cc1Br)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(=O)(=O)c2nccs2)c(F)cc1-c1cnc(OC2CCC2)c(Cl)c1
CCCS(=O)(=O)NC(=O)c1cc(C)c(cc1F)-c1cnc(OC2CCC2)c(Cl)c1
Cc1cc(C(=O)NS(=O)(=O)C2CC2)c(F)cc1-c1cnc(OC2CCC2)c(Cl)c1
Cc1cc(C(=O)NS(=O)(=O)C2CCC2)c(F)cc1-c1cnc(OC2CCC2)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(=O)(=O)c1nccs1
CCS(=O)(=O)NC(=O)c1cc(C)c(cc1F)-c1cnc(Oc2c(C)cc(Cl)cc2Cl)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(=O)(=O)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(cc1F)-c1cnc(OC2CCC2)c(Cl)c1
COc1cc(ccc1-c1cc(Cl)nc(Oc2cc(Cl)cc(Cl)c2)c1)C(=O)NS(C)(=O)=O
C[C@](Oc1ncc(cc1Cl)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O)(c1ccccc1)C(F)(F)F
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1ccc(Cl)c(c1)C(F)(F)F
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1ccc(c(Cl)c1)C(F)(F)F
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCC(F)F)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1ccc2OC(F)(F)Oc2c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1ccc(OCC(F)(F)F)cc1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1ccc(OC(F)(F)C(F)F)cc1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cccc(OC(F)(F)C(F)F)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1ccc(CC2CC2)c(Cl)c1
CCc1ccc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(NC(C)(C)C)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OC(C)(C)C)c(Cl)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(c1)C(F)(F)F
COc1cccc(CSc2ncc(cc2Cl)-c2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)c1
COc1cc(ccc1-c1cnc(COc2ccc(cc2)C#N)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1nccc(C)c1-c1cc(ccc1-c1cnc(OCC(C)C)c(Cl)c1)C(=O)NS(C)(=O)=O |(-.86,-4.93,;-2.36,-5.25,;-2.84,-6.72,;-1.81,-7.86,;-2.29,-9.33,;-3.79,-9.65,;-4.82,-8.5,;-6.33,-8.82,;-4.35,-7.04,;-5.38,-5.89,;-6.71,-6.66,;-8.04,-5.89,;-8.04,-4.35,;-6.71,-3.58,;-5.38,-4.35,;-4.04,-3.58,;-2.71,-4.35,;-1.38,-3.58,;-1.38,-2.04,;-.04,-1.27,;1.29,-2.04,;2.63,-1.27,;3.96,-2.04,;2.63,.27,;-2.71,-1.27,;-2.71,.27,;-4.04,-2.04,;-9.38,-6.66,;-9.38,-8.2,;-10.71,-5.89,;-12.05,-6.66,;-11.28,-8,;-13.38,-7.43,;-12.82,-5.33,)|
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(C=O)c1)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(c1)C(F)F
COc1cc(ccc1-c1cnc(Oc2ccnc(OC)c2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O
CC(C)[C@H]1CCCN1c1ncc(cc1Cl)-c1ccc(cc1OC(F)F)C(=O)NS(C)(=O)=O
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(c(Cl)c1)-c1cc(F)cc(F)c1
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(c(Cl)c1)-c1ccc(Cl)c(Cl)c1
CC(C)COc1ncc(cc1Br)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
COc1ncc(F)cc1-c1cc(cnc1OCC(C)C)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1-c1cc(F)cc(F)c1)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
COc1nccc(C)c1-c1ncc(cc1Cl)-c1cc(F)c(cc1C)C(=O)NS(C)(=O)=O |(2.67,1.54,;2.67,,;4,-.77,;5.33,,;6.67,-.77,;6.67,-2.31,;5.33,-3.08,;5.33,-4.62,;4,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-5.39,;,-4.62,;,-3.08,;1.33,-2.31,;1.33,-.77,;-1.33,-5.39,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-6.93,;-4,-5.39,;-2.67,-4.62,;-2.67,-3.08,;-5.33,-7.7,;-5.33,-9.24,;-6.67,-6.93,;-8,-7.7,;-8.77,-6.37,;-9.34,-8.47,;-7.23,-9.03,)|
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(C)c1)C(=O)NS(C)(=O)=O
COCCOCCOCCN1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl
COCCOCCOCCOCC(=O)N1CCN(CC1)C(=O)OC(C)(C)C
COCCOCCOCC(=O)N1CCN(CC1)C(=O)OC(C)(C)C
COCCOCCOCC(=O)N1CCN(CC1)c1nnc(c(N)n1)-c1cc(F)cc(Cl)c1Cl
COCCOCCOCCOc1ccc(c(Cl)c1Cl)-c1nnc(N)nc1N
Nc1nc(NC(CO)CO)nnc1-c1cccc(Cl)c1Cl
COCCOCCOCC(=O)N1CCC(CC1)NC(=O)OC(C)(C)C
COCCOCCOCCN1CCC(N)CC1
COCCOCCOCCN1CCC(CC1)Nc1nnc(c(N)n1)-c1cc(F)cc(Cl)c1Cl
Nc1nc(NC2CCNCC2)nnc1-c1cccc(Cl)c1Cl
COCC(COC)OCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCNCC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;1;2;3;4;5;6$|
Nc1nc(nnc1-c1cc(F)cc(Cl)c1Cl)N1CCNCC1
COCCOCCOCCN1C(C)CN(CC1C)c1nnc(Cl)c(N)n1
C[C@H]1CN(C[C@@H](C)N1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
C[C@H]1CN(C[C@@H](C)N1)c1nnc(c(N)n1)-c1cc(F)cc(Cl)c1Cl |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CC(O)CO)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;4;3;2;1;3;2;;1;;6;5$|
COCCOCCOCCN(C)C1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CC1)C1CCOCC1
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CC1)C1CCNCC1
Nc1nc(nnc1Cl)N1CCN[C@@H](CO)C1 |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN[C@H](CO)C1 |r|
Nc1nc(nnc1-c1cc(F)cc(Cl)c1Cl)N1CCN[C@H](CO)C1 |r|
Nc1nc(nnc1-c1cc(F)cc(Cl)c1Cl)N1CCN[C@@H](CO)C1 |r|
CC(CS(=O)(=O)CCO)Nc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:3;2;1;;;;2;1;;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COC[C@H](O)CN1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;3;2;;1;1;2;3;4;5;6;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COC[C@@H](O)CN1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;3;2;;1;1;2;3;4;5;6;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CC(F)(F)F)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;1;2;3;4;1;2;;;;5;6$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN2[C@@H](COC2=O)C1 |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN2[C@H](COC2=O)C1 |r|
NC1CN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl
CC(CO)N1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:3;2;1;;1;2;3;4;5;6;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CCOC(F)(F)F)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;1;2;3;4;1;2;;1;;;;5;6$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CC(O)C1
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN2[C@@H](COCC2=O)C1 |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN2CCOC[C@@H]2C1 |r|
CC(C)(CO)N1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:3;2;;1;;1;2;3;4;5;6;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CC(C)(C)OC(=O)N1CC(C1)Nc1nnc(c(N)n1)-c1cccc(Cl)c1Cl
CN(CCNC[C@H](O)C(F)(F)F)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
CN(CCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl)C[C@H](O)C(F)(F)F |$_AV:;;1;2;;3;2;1;6;5;;4;1;6;5;4;3;;2;;3;2;;1;;;$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CC(O)(C1)C(F)(F)F
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCC(O)(CC1)C(F)(F)F
COC[C@@H](O)CN1CCN(C[C@H]1CO)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
CC(C)(C)OC(=O)N1CCN([C@H](CO)C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
CC(C)(C)OCC(O)CN1CCN(C[C@H]1CO)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CC(O)CO)[C@H](CO)C1 |r|
COC[C@@H](O)CN1CCN([C@H](CO)C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
CC(C)(C)OCC(O)CN1CCN([C@H](CO)C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CC(O)CO)C[C@H]1CO |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;4;5;6;1;3;2;;1;;2;3;1;$|
CCOC[C@H](O)CN1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
CC(C)OC[C@H](O)CN1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
CC(C)(C)OC(=O)N1CCN(c2nnc(c(N)n2)-c2cccc(Cl)c2Cl)C2(CC2)C1
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CC(C1)OCC(F)(F)F |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;1;2;3;4;;1;2;;;$|
COC[C@H](O)CO[C@H]1CCN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
COC[C@@H](O)COC1CN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(C[C@H](O)COCC2CCC2)CC1 |r|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(C[C@H](O)COCC2CC2)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;4;3;2;1;1;2;;3;;1;1;2;3;6;5$|
COC[C@@H](O)CN(C)CC1CN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;3;2;;1;;;1;3;2;1;4;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COC[C@@H](O)CN1CCC11CCCN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;3;2;;1;1;2;3;4;9;8;7;6;5;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(C[C@H](O)COC2CCC2)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;4;3;2;1;1;2;;3;;1;2;3;4;6;5$|
COC[C@@H](O)CNC1(C)CCN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;3;2;;1;;3;;4;5;1;2;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COC[C@@H](O)CNC1CN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;3;2;;1;;3;2;1;4;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COC[C@@H](O)CN[C@@H]1CCN(C1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;3;2;;1;;3;4;5;1;2;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(C[C@H](O)CCl)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;4;3;2;1;1;2;;3;;6;5$|
CN1CCN(CCOCCNc2nnc(c(N)n2)-c2cccc(Cl)c2Cl)CC1 |$_AV:;4;3;2;1;2;1;;2;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;;6;5$|
CC(C)OCCOCCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;;;2;1;;2;1;;2;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COCCNCCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;2;1;;2;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CC(=O)NCCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:2;1;;;1;2;;1;2;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CS(=O)(=O)CCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;;;2;1;;2;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COCCOCCOCC(C)CNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;2;1;;3;2;;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
Nc1nc(NCCOCCNCC(O)=O)nnc1-c1cccc(Cl)c1Cl |$_AV:;5;4;3;;2;1;;2;1;;2;1;;;2;1;6;1;6;5;4;3;;2;$|
COCCOCCOCC(O)CNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl
COCCOCCOCC(COCCOCCOC)OCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:1;2;3;4;5;6;7;8;9;10;1;;1;2;;1;2;;;11;12;13;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CC(CO)Nc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:3;2;1;;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CN(CCO)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COCCS(=O)(=O)CCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;;;2;1;;2;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CS(=O)CCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;;2;1;;2;1;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COCCOCCOCC(C)Nc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;2;1;;1;2;3;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
Nc1nc(NCCOCCOCCOC(F)(F)F)nnc1-c1ccc(Cl)c(Cl)c1
COC(=O)COCCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;1;;2;;1;2;;1;2;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COCCOCC(=O)N(C)CCN(C)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;2;1;;;;1;2;;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COCCOCC(=O)NCC(O)CNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;2;1;;;1;2;;3;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CN(CCOCCNc1cnc(c(N)n1)-c1cccc(Cl)c1Cl)CC(N)=O |$_AV:;;1;2;;1;2;;2;3;4;5;6;;1;1;6;5;4;3;;2;;2;1;;$|
CN(CCN(C)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl)C(=O)COCC(N)=O |$_AV:;;1;2;;;3;2;1;6;5;;4;1;6;5;4;3;;2;;1;;2;;1;2;;$|
COCCOCCN(C)CCN(C)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;2;1;;2;1;;;2;1;;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
NC(=O)CNCCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;1;;2;;1;2;;1;2;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
COC(=O)CNCCOCCNc1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;1;;2;;1;2;;1;2;;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CCO)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;4;3;2;1;2;1;;6;5$|
Nc1nc(nnc1-c1cccc(Cl)c1Cl)N1CCN(CCOCCO)CC1 |$_AV:;5;4;3;2;1;6;1;6;5;4;3;;2;;4;3;2;1;2;1;;2;1;;6;5$|
CS(=O)(=O)CCN1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;;;2;1;4;3;2;1;6;5;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
CC(C)(C)OC(=O)COCCN1CCN(CC1)c1nnc(c(N)n1)-c1cccc(Cl)c1Cl |$_AV:;;;;;1;;2;;1;2;1;2;3;4;5;6;3;2;1;6;5;;4;1;6;5;4;3;;2;$|
NC(=O)c1cc(CNC2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(cn2)C2CC2)cc1
NC(=O)c1cc(CNC2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1
NC(=O)[C@@H]1CCCN1Cc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O |r|
NC(=O)c1cc(CNC2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1
C[C@H](NCc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
CC(C)[C@H](NCc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
NC(=O)[C@H](CO)NCc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O |r|
NC(=O)c1cc(CN2C[C@H](O)C[C@H]2NC=O)nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1 |r|
NC(=O)c1cc(CN[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
C[C@H](NCc1cc(nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F)C(N)=O)C(N)=O |r,t:11|
NC(=O)c1cc(CO)nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F |t:12|
NC(=O)[C@H](CO)NCc1cc(nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F)C(N)=O |r,t:15|
NC(=O)c1cc(CN2CCNC(=O)C2)nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1
NC(=O)c1cc(CN[C@@H]2CCNC2=O)nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F |r,t:19|
OC[C@@H](O)c1cc(CN[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1 |r|
OC[C@@H](O)c1cc(CN2CCNC(=O)C2)nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1 |r|
NC(=O)c1cc(CN2CCNC(=O)C2)nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1
NC(=O)c1cc(CN2CCNC(=O)C2)nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F |t:19|
CC1(C)N(Cc2cc(nc(n2)-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)C(N)=O)CCNC1=O
CC1(C)N(Cc2cc(nc(n2)-c2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)C(N)=O)CCNC1=O
NC(=O)c1cc(CN2CC(=O)NC(=O)C2)nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1
NC(=O)[C@@H]1[C@H](O)CCN1Cc1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)C(N)=O |r|
NC(CO)Cc1c[nH]c2c(cccc12)-c1ccc(Oc2ccccc2)cc1
NC(Cc1c([nH]c2ccccc12)-c1ccc(Oc2ccccc2)cc1)C(N)=O
NC(Cc1cn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12)C(N)=O
NC(CO)Cc1c[nH]c2ccc(cc12)-c1ccc(Oc2ccccc2)cc1
NC(Cc1cn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12)C(=O)NCCO
NC(CO)Cc1cn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12
NC(Cc1c[nH]c2ccc(cc12)-c1ccc(Oc2ccccc2)cc1)C(N)=O
CCOC(=O)C(N)Cc1c[nH]c2ccc(cc12)-c1ccc(Oc2ccccc2)cc1
CS(=O)(=O)NC(Cc1cn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12)C(N)=O
CC(C)(C)OC(=O)NC(Cc1c[nH]c2cc(ccc12)-c1ccc(Oc2ccccc2)cc1)C(O)=O
NC(Cc1c[nH]c2cc(ccc12)-c1ccc(Oc2ccccc2)cc1)C(N)=O
CCOC(=O)C(Cc1c[nH]c2cc(ccc12)-c1ccc(Oc2ccccc2)cc1)NC(=O)OC(C)(C)C
CCOC(=O)C(Cc1c[nH]c2ccc(cc12)-c1ccc(Oc2ccccc2)cc1)[N+]([O-])=O
NC(Cc1c[nH]c2ccc(cc12)-c1ccc(Oc2ccccc2)cc1)C(O)=O
N[C@H](CO)Cc1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
N[C@@H](CO)Cc1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
FC(F)(F)c1ccc(Oc2ccc(cc2)-n2cc(C[C@H]3COC(=O)N3)c3ccccc23)cc1C#N
CN(C)CCc1cn(-c2ccc(Oc3ccccc3)cc2)c2ccc(C[C@H]3COC(=O)N3)cc12
CN(C)CCc1cn(-c2ccc(Oc3ccccc3)cc2)c2ccc(C[C@H](N)CO)cc12
NCCc1cn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12
OCC(O)c1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
CCOC(=O)C(=O)c1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
N[C@H](CO)Cc1cn(-c2ccc(Oc3cccc(c3)C#N)cc2)c2ccccc12
NC(=O)C(=O)c1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
NC(=O)C(O)c1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
COC(=O)c1ccc2c(cn(-c3ccc(Oc4ccc(c(c4)C#N)C(F)(F)F)cc3)c2c1)C(O)C(N)=O
OC[C@@H](O)CNC(=O)C(=O)c1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
OC[C@@H](O)CNC(=O)C(O)c1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
OC[C@@H](O)Cc1cn(C[C@H](O)CO)c2ccc(cc12)-c1ccc(Oc2ccc(F)cc2)cc1
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(cc3)C#N)cc2)c2ccccc12
OC[C@H](O)Cc1cn(-c2ccc(Oc3ccc(cc3)C#N)cc2)c2ccccc12
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)c2ccccc12
CN(c1ccc(F)cc1)S(=O)(=O)c1ccc(cc1)-n1cc(C[C@H](O)CO)c2ccccc12
OC[C@@H](O)Cc1cn(-c2ccc(cc2)S(=O)(=O)Nc2ccc(F)cc2)c2ccccc12
OC[C@H](O)c1ccc2n(cc(C(=O)C(O)=O)c2c1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(F)cc3)cc2)c2cc(ccc12)C#N
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccc(cc12)C#N
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(F)cc3)cc2)c2c(cccc12)C#N
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(F)cc3)cc2)c2cccc(C#N)c12
NC(=O)c1cccc2n(cc(C[C@H](O)CO)c12)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)c1ccc2c(C[C@H](O)CO)cn(-c3ccc(Oc4ccc(F)cc4)cc3)c2c1
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(F)cc3)cc2)c2cccc(C(O)=O)c12
OC[C@H](O)Cc1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2cccc(C(O)CO)c12 |r|
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2cccc(C(O)CO)c12 |r|
OCCNC(=O)c1nn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12
NC(=O)c1nn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12
ONC(=O)c1nn(-c2ccc(Oc3ccccc3)cc2)c2ccccc12
NC(=O)c1nn(-c2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)c2ccc(F)cc12
NC(=O)c1nn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
NC(=O)c1nn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
OCC(O)CNC(=O)c1nn(-c2ccc(Oc3ccc(cc3)C#N)cc2)c2ccccc12
OCc1cn(-c2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)c2cnccc12
OC[C@H](O)c1nn(-c2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)c2cnccc12
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(F)cc3)cc2)c2cnccc12
OC[C@@H](O)Cc1cn(-c2ccc(Oc3ccc(cc3)C#N)cc2)c2cccnc12
CCN(CC)CCn1ccc2cc(ccc12)-c1ccc(Oc2ccc(F)cc2)cc1
CCN(CC)CCn1cc(C(=O)C(N)=O)c2cc(ccc12)-c1ccc(Oc2ccc(F)cc2)cc1
CCN(CC)CCn1cc(C(O)C(N)=O)c2cc(ccc12)-c1ccc(Oc2ccc(F)cc2)cc1
CCN(CC)CCn1cc(C[C@H](O)CO)c2cc(ccc12)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)Cn1cc(C[C@H](O)CO)c2cc(ccc12)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)C(O)(c1cn(-c2ccc(Oc3ccc(C#N)c(c3)C(F)(F)F)cc2)c2ccccc12)C(F)(F)F
NC(=O)C(O)c1cn(-c2ccc(Oc3ccc(C#N)c(c3)C(F)(F)F)cc2)c2ccccc12
NC(=O)C(O)c1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
N[C@H](CO)Cc1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
OCCn1cc(C[C@H](O)CO)c2cc(ccc12)-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)N2CCN(CC2)S(=O)(=O)c2ccc(OC(F)(F)F)cc2)cc1
CS(=O)(=O)c1cccc(c1)S(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)N2CCN(CC2)S(=O)(=O)c2cccc(c2)C#N)cc1
CN(C)S(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
CC1(C)C2CCC1(CS(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc3ccc(F)cc3)cc1)C(=O)C2 |TLB:40:39:4.5:1|
CS(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
Cc1noc(C)c1S(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)N2CCN(CC2)S(=O)(=O)c2cccnc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)N2CCN(CC2)S(=O)(=O)c2cccc(OC(F)(F)F)c2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)N2CCN(CC2)S(=O)(=O)c2ccc(cc2)C#N)cc1
OC(=O)c1cccc(c1)S(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
OC(=O)c1ccc(cc1)S(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
CS(=O)(=O)NCCNC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-c2ccc(cn2)S(=O)(=O)NCCNC(=O)c2ccccn2)cc1
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)NCCNS(=O)(=O)c2cccc(c2)C#N)cc1
NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
C[C@H](NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)C[C@H](NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)[C@@H](CO)NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)[C@@H]1CCCN1C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(O)[C@H](NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
CC(C)C[C@H](NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)[C@H](Cc1cccnc1)NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
CC(C)[C@H](NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)[C@H](CO)NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Fc1ccc(Oc2cccc(n2)C(=O)N2CCN(CC2)S(=O)(=O)c2cccc(c2)C#N)cc1
Fc1ccc(cc1)-c1cccc(n1)C(=O)N1CCN(CC1)S(=O)(=O)c1cccc(c1)C#N
OC[C@@H](O)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)N1CCN(CC1)S(=O)(=O)c1cccc(c1)C#N |r|
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)N2CCN(CC2)S(=O)(=O)c2ccc(F)c(c2)C#N)cc1
CN1CCOc2cc(ccc12)S(=O)(=O)N1CCN(CC1)C(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
C[C@H](NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1)C(N)=O |r|
CC(C)C[C@H](NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO)C(N)=O
NC(=O)C[C@H](NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO)C(N)=O |r|
CC(C)C[C@H](NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@@H](O)CO)C(N)=O |r|
CC(N)C[C@H](NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@@H](O)CO)C(N)=O
CS(=O)(=O)NC(=O)c1cc(F)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:21:16:23:19.20.22,21:20:15.16.17:23,THB:19:18:15:21.20.22,19:20:15:17.18.23|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:13:14:17:21.20.19,23:14:21:17.18.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15|
CC1(C)[C@@H]2C[C@H]1[C@@H](COc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)CC2 |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC2C3CC4CC(C3)CC2C4)cc1F |TLB:12:13:20:17.16.22,15:16:20:14.13.19,THB:15:14:20:17.16.22,13:14:17:20.21.22,13:21:17:14.15.19,(6.07,.01,;5.3,1.35,;4.53,2.68,;6.63,2.12,;3.97,.58,;2.63,1.35,;2.63,2.89,;1.3,.58,;1.3,-.96,;-.03,-1.73,;-.03,-3.27,;-1.37,-.96,;-2.7,-1.73,;-4.04,-.96,;-3.14,.96,;-3.14,2.5,;-4.47,3.27,;-5.8,2.5,;-5.8,.96,;-4.47,.19,;-6.63,-.94,;-5.24,-.29,;-5.22,2.11,;-1.37,.58,;-.03,1.35,;-.03,2.89,)|
C[C@@H]1[C@H]2C[C@@H](C[C@H]1Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)C2(C)C |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:14:15:18:22.21.20,24:15:22:18.19.20,THB:24:19:22:15.23.16,23:15:18:22.21.20,23:21:18:15.24.16|
CC1(C)C2CCC1(C)C(C2)Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O |THB:10:8:1:5.4|
C[C@H]1[C@@H]2C[C@H](C[C@@H]1Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)C2(C)C |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCCC2CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(F)(C4)C2)C3)cc1F |TLB:24:14:22:17.18.19,THB:13:14:22:17.18.19,24:18:22:14.23.15,23:14:17:22.20.19,23:20:17:14.24.15,21:20:17:14.24.15|
CS(=O)(=O)NC(=O)c1cc(Cl)c(NCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:23:14:21:17.18.19,THB:13:14:21:17.18.19,23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15|
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:20:19:22:16.15.14,20:15:22:19.21.18,THB:12:13:16:19.20.18,21:19:16:22.14.13,21:13:16:19.20.18|
CS(=O)(=O)NC(=O)c1ccc(OCCC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:13:14:17:21.20.19,23:14:21:17.18.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15|
CS(=O)(=O)NC(=O)c1cnc(OCC23CC4CC5(CC(C5)(C4)C2)C3)c(Cl)c1 |TLB:16:17:22:15.21.14,14:13:18:20,THB:16:15:22:18.23.17,20:17:22:15.21.14,12:13:18:20,(6.38,2.1,;5.61,3.43,;6.95,4.2,;4.84,4.77,;4.28,2.66,;2.94,3.43,;2.94,4.97,;1.61,2.66,;.28,3.43,;-1.06,2.66,;-1.06,1.12,;-2.39,.35,;-3.93,.35,;-4.7,-.98,;-6.17,-.57,;-6.94,-1.9,;-6.95,-3.44,;-5.46,-3.86,;-4.37,-4.95,;-4.39,-3.43,;-4.4,-4.97,;-5.87,-3.02,;-3.61,-2.07,;-4.7,-2.52,;.28,.35,;.28,-1.19,;1.61,1.12,)|
CS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2ccc3CCCCc3c2)cc1F
CC12CC3CC(C)(C1)CC(COc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)(C3)C2 |TLB:27:9:7:4.3.2,10:9:4:7.1.2,THB:27:3:7:9.28.8,28:9:4:7.1.2,28:1:4:9.27.8|
CC1(C)[C@@H]2CC[C@@]1(C)[C@H](C2)Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O |r|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:25:16:23:19.20.21,THB:15:16:23:19.20.21,25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17|
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)C(=O)NC12CC3CC(CC(C3)C1)C2 |TLB:27:18:25:21.22.23,THB:17:18:25:21.22.23,27:22:25:18.26.19,26:18:21:25.24.23,26:24:21:18.27.19|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(O)(C4)C2)C3)cc1F |TLB:24:14:22:19.18.17,THB:24:18:22:14.15.23,13:14:22:19.18.17,15:14:19:22.16.17,15:16:19:14.24.23|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCCCC2)cc1F
CC(Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)C12CC3CC(CC(C3)C1)C2 |TLB:27:18:25:21.22.23,THB:1:18:25:21.22.23,27:22:25:18.26.19,26:18:21:25.24.23,26:24:21:18.27.19|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC2C3CC4CC(C3)CC2C4)cc1F |TLB:14:15:17:19.20.21,THB:15:23:19:17.16.21,15:16:19:23.22.24,22:23:17:19.20.21,22:20:17:23.15.24,(7.75,-1.15,;6.42,-1.93,;6.42,-3.47,;5.08,-1.15,;4.31,-2.49,;5.85,.18,;3.75,-.38,;2.41,-1.15,;2.41,-2.7,;1.08,-.38,;1.08,1.16,;-.25,1.93,;-.25,3.47,;-1.59,1.15,;-2.92,1.93,;-4.25,1.15,;-5.58,1.92,;-6.92,1.15,;-6.92,-.38,;-7.75,-2.29,;-6.35,-1.64,;-6.34,.76,;-5.15,-2.31,;-4.25,-.38,;-5.58,-1.16,;-1.59,-.38,;-.25,-1.15,;-.25,-2.7,)|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC[C@H]2CC[C@H]3C[C@@H]2C3(C)C)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCCC2CCCCC2)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(O[C@H]2C3CC4CC2CC(Cl)(C4)C3)cc1F |r,TLB:12:13:15:22.20.23,13:14:22:18.19.17,THB:13:18:22:15.14.23,19:18:15:22.20.23,19:20:15:18.13.17|
CC1(C)CCc2cc(OCc3cc(F)c(cc3Cl)C(=O)NS(=O)(=O)N3CCC3)ccc2O1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:25:16:23:19.20.21,THB:15:16:23:19.20.21,25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17|
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:26:17:24:20.21.22,THB:16:17:24:20.21.22,26:21:24:17.25.18,25:17:20:24.23.22,25:23:20:17.26.18|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:5:6:9:13.12.11,15:6:13:9.10.11,THB:15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
CNS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:24:15:22:18.19.20,THB:14:15:22:18.19.20,24:19:22:15.23.16,23:15:18:22.21.20,23:21:18:15.24.16|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
COCCS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:26:17:24:20.21.22,THB:26:21:24:17.25.18,16:17:24:20.21.22,25:17:20:24.23.22,25:23:20:17.26.18|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC2CCC3(CCCCC3)CC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2(CCC2)C(F)(F)F)cc1F
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C1CC1 |TLB:12:13:16:20.19.18,22:13:20:16.17.18,THB:21:13:16:20.19.18,21:19:16:13.22.14,22:17:20:13.21.14|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2C3CC4CC(C3)CC2C4)cc1F |TLB:15:16:18:20.21.22,THB:16:24:20:18.17.22,16:17:20:24.23.25,23:24:18:20.21.22,23:21:18:24.16.25,(8.42,2.5,;7.08,1.73,;7.08,.19,;5.75,2.5,;4.98,3.84,;6.52,3.84,;4.42,1.73,;3.08,2.5,;3.08,4.04,;1.75,1.73,;1.75,.19,;.41,-.58,;.41,-2.12,;-.92,.19,;-2.25,-.58,;-3.59,.19,;-4.92,-.58,;-6.25,.19,;-7.58,-.58,;-7.58,-2.12,;-8.42,-4.02,;-7.02,-3.37,;-7,-.97,;-5.82,-4.04,;-4.92,-2.12,;-6.25,-2.89,;-.92,1.73,;.41,2.5,;.41,4.04,)|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC[C@H]2CC[C@@H](CC2)C(F)(F)F)cc1F |r,wU:14.13,wD:17.20,(8.67,3.36,;7.34,2.59,;6.57,3.93,;8.11,1.26,;6,1.82,;4.67,2.59,;4.67,4.13,;3.33,1.82,;3.33,.28,;2,-.49,;2,-2.03,;.67,.28,;-.67,-.49,;-2,.28,;-3.33,-.49,;-3.33,-2.03,;-4.67,-2.8,;-6,-2.03,;-6,-.49,;-4.67,.28,;-7.34,-2.8,;-8.67,-3.57,;-8.11,-1.46,;-6.57,-4.13,;.67,1.82,;2,2.59,;2,4.13,)|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC2CCC(CC2)C(F)(F)F)cc1F |(8,1.54,;6.67,.77,;5.9,2.1,;7.44,-.56,;5.33,,;4,.77,;4,2.31,;2.67,,;1.33,.77,;;-1.33,.77,;,-1.54,;-1.33,-2.31,;-2.67,-1.54,;-2.67,,;-4,.77,;-5.33,,;-5.33,-1.54,;-4,-2.31,;-6.67,.77,;-8,1.54,;-5.9,2.1,;-7.44,-.56,;1.33,-2.31,;2.67,-1.54,;4,-2.31,)|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC2CC3CC2C2CCCC32)cc1F |THB:14:15:18:24.20,23:24:15.16:18,21:20:15.16:18|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CC3C4CCC(C4)C3C2)cc1F |TLB:15:16:21:18.19,THB:23:22:21:18.19|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
O[C@H]1CCN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |r,TLB:30:21:28:24.25.26,THB:20:21:28:24.25.26,30:25:28:21.29.22,29:21:24:28.27.26,29:27:24:21.30.22|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
FC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:29:20:27:23.24.25,THB:19:20:27:23.24.25,29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.29.21|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(C2)C(F)(F)C(C4)C3)cc1F |TLB:13:14:20:17.16.24,THB:15:14:20:17.16.24,15:16:20:14.25.19,25:14:17:20.23.24,25:23:17:14.15.19|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC(F)(F)CC2)cc1F
OCCCNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:29:20:27:23.24.25,THB:19:20:27:23.24.25,29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.29.21|
COC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:30:21:28:24.25.26,THB:20:21:28:24.25.26,30:25:28:21.29.22,29:21:24:28.27.26,29:27:24:21.30.22|
Fc1cc(OCC23CC4CC(C2)C(F)(F)C(C4)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:5:6:9:12.15.16,THB:17:6:9:12.15.16,17:15:9:6.7.11,7:6:12:9.8.16,7:8:12:6.17.11|
Fc1cc(OCC23CC2CCCC3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
COc1cc(c(Cl)cc1-c1nccc2cc(c(F)cc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(ccc1-c1nccc2cc(c(F)cc12)S(=O)(=O)Nc1ncns1)-c1cccc(F)c1
COc1nc(Oc2ccc(F)cc2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)N(CC(C)C)CC(C)C
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccccc1
COc1nc(OC2CCCCC2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1ccccc1
COc1nc(OCC2CCCCC2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(OCC(C)(C)C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)N(C)CC(C)C
COc1nc(OCC2CCC(F)(F)CC2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(c(NCC(C)(C)C)n1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)N1CCC(F)(F)CC1
COc1nc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)N1CCCC1
COc1nc(NC2CCCCC2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(NC2CCC(F)(F)CC2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(NCC(C)(C)C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(OC2CCC(F)(F)CC2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(-c2ccc(Cl)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2cc(C)cc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2ccc(C)c(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N)-c1ccccc1C
COc1cc(-c2ccc(F)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2ccc(C)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2ccc(Cl)c(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N)-c1cc(F)cnc1OC
COc1cc(-c2ccc(F)c(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2ccc(F)c(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2cc(F)cc(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)c(C)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)c(C)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cc(F)cnc1OC
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(Cl)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccsn1)-c1cc(F)cnc1OC
COc1cc(c(F)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
Cn1nccc1-c1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC
COc1cc(-c2ccc(F)cc2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2cc(F)cc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C#N
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccsn1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(-c2cccc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C#N
COc1cc(Cl)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(-c2cccc(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2cccc(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(c(Cl)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(F)c1
COc1cc(-c2cc(C)cc(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(c(Cl)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1
COc1cc(Br)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncon1)C#N
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cccnn1)-c1cccc(F)c1
COc1cc(Cl)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncon1)-c1cccc(F)c1
COc1cc(Cl)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cc(F)cc(F)c1
COc1cc(NS(=O)(=O)c2ccc3c(nccc3c2)-c2ccc(cc2OC)-c2cc(F)cc(F)c2)ncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cc(C)on1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncon1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccno1)-c1cc(F)cc(F)c1
COc1nnc(NS(=O)(=O)c2ccc3c(nccc3c2)-c2ccc(cc2OC)-c2cc(F)cc(F)c2)s1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cnsn1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nc(C)ns1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cncc(C)n1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(s1)C#N)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nnc(C)s1)-c1cc(F)cc(F)c1
COc1nsc(NS(=O)(=O)c2ccc3c(nccc3c2)-c2ccc(cc2OC)-c2cc(F)cc(F)c2)n1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)NC(C)=O)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncco1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cccnn1)-c1cc(F)cc(F)c1
COc1cc(C#N)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cnccn1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccccn1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(o1)C(F)(F)F)-c1cc(F)cc(F)c1
OCc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(-c2cccc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
OCc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(C#N)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(F)cc(F)c1
OCc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
COc1cc(-c2ccc(cc2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(cc1)C(F)(F)F
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(NS(=O)(=O)c2ccc3c(nccc3c2)-c2ccc(cc2OC)-c2cc(F)cc(F)c2)no1
COc1cc(C#N)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
Cc1ccc(OCc2ccccc2)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-.11,-.1,;1.22,-.87,;2.55,-.1,;2.55,1.44,;3.89,2.21,;5.22,1.44,;6.55,2.21,;5.22,-.1,;3.89,-.87,;3.89,-2.41,;2.55,-3.18,;1.22,-2.41,;-.11,-3.18,;-.11,-4.72,;1.22,-5.49,;2.55,-4.72,;3.89,-5.49,;5.22,-4.72,;5.22,-3.18,;6.55,-2.41,;-1.45,-5.49,;-2.22,-4.16,;-.68,-6.83,;-2.78,-6.26,;-4.12,-5.49,;-5.52,-6.12,;-6.55,-4.98,;-5.78,-3.64,;-4.28,-3.96,;3.89,3.75,;5.22,4.52,;5.22,6.06,;3.89,6.83,;2.55,6.06,;1.22,6.83,;2.55,4.52,)|
Cc1ccc(Oc2ccccc2)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ncc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccccc1
Cc1ccc(Oc2ccccn2)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
Cc1ccc(OCC2CC2)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(-c2ccc(Cl)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(-c2ccc(F)c(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(-c2cccc(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N)-c1ccccc1C
COc1cc(-c2ccc(F)c(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(-c2ccc(C)c(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(-c2cc(C)cc(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(Oc2ccc(F)c(C)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(-c2ccc(Cl)c(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1ccc(F)cc1-c1cc(OC)c(cc1C#N)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(-c2ccc(C)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(-c2cc(C)cc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N)-c1cc(C)c(C)cc1C
COc1cc(-c2cc(F)cc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cnc1OC
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccnc1OC
COc1cc(c(C)cc1-c1cccc(F)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(C)cc1-c1ccc(Cl)c(C)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1ccc(F)cc1-c1cc(C)c(cc1OC)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(C(F)F)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(Oc2ccccc2C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1ccc(F)c(F)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
COc1ccc(C)c(c1)-c1cc(C)c(cc1OC)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(Oc2ccc(F)cc2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(c(C)cc1-c1ccc(Cl)c(C)c1)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(Oc2ccc(F)c(F)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2ccc(C)c(C)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2ccc(C)c(F)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2cc(F)cc(F)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2cc(C)cc(F)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2cc(C)cc(C)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2cccc(C)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(Oc2ccc(c(OC)c2)-c2nccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)cc1
COc1cccc(Oc2ccc(c(OC)c2)-c2nccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c1
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(-c2ccc(cc2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(-c2ccc(F)cc2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(Oc2cc(F)ccc2F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
FC(F)(F)c1ccc(c(c1)C1CC1)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(C)cnc1OC
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-n1ccc2ccccc12
COc1cc(c(F)cn1)-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(Oc2cc(C)ccc2F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1ccc(F)cc1-c1cc(OC)c(cc1C)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
FC(F)(F)c1ccc(c(c1)C1CC1)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccnc1OC(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)n1
COc1cc(Oc2ccc(C)c(F)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(Oc2ccc(F)cn2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(Oc2cc(C)cc(F)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1ccc(c(F)n1)-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(-c2ccc(F)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(F)c1
COc1cc(c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N)-c1cc(F)cnc1OC
COc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
COc1cc(c(Cl)cc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1cccnn1)-c1cccc(F)c1
COc1cc(-c2cc(F)cc(F)c2)c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2cccc(F)c2)c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(ccc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(Cl)c1
COc1cc(c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N)-c1cc(F)cnc1OC
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1cnsn1)-c1cccc(F)c1
Fc1cccc(c1)-c1ccc(c(OCC#N)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cnc1OC
COc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)n1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC
COc1cc(c(Cl)cc1-c1nn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(-c2cc(F)cc(F)c2)c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2cccc(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2ccc(C)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2ccc(cc2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2ccc(F)cc2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N)-c1ccccc1C
COc1cc(-c2ccc(F)c(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(c(Cl)cc1-c1ncc(O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(-c2cc(C)cc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N)-c1cc(F)cnc1OC
COc1cc(-c2ccc(Cl)c(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(N2CC(F)(F)C2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2cc(C)cc(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(N2CC(F)(F)C2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2ccc(Cl)c(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2ccc(C)c(Cl)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2ccc(F)c(C)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
Fc1cccc(c1)-c1ccc(c(OCC#N)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(Cl)cc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(c(F)cc1-c1nn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(c1)C(F)(F)F
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
COc1nc(N2CC(F)(F)C2)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1nc(N2CCC(F)(F)C2)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(c(F)cc1-c1nn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
Fc1cccc(c1)-c1ccc(c(OCC#N)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(c(Cl)cc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1ncc(C#N)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1nc(Cl)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(-c2cccc(F)c2)c(cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1nc(N(C)C)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(F)c1
COc1nc(N2CCC(F)(F)CC2)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1
COc1cc(ccc1[C@@H]1N(CCc2cc(ccc12)S(=O)(=O)Nc1nncs1)C(C)=O)-c1cccc(F)c1
COc1cc(ccc1C1N(CCc2cc(ccc12)S(=O)(=O)Oc1c(F)c(F)c(F)c(F)c1F)C(C)=O)-c1cccc(F)c1
COc1cc(ccc1[C@@H]1N(CCc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(C)=O)C(F)(F)F
COc1cc(c(Cl)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1
COc1cc(Cl)c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(Cl)c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C(F)(F)F
COc1cc(C(F)F)c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(C(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C1CC1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cscn1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nnc(OC)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccsn1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ccsn1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ccsn1)-c1cc(F)cc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncco1)-c1cccc(F)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C(F)(F)F
COc1cc(c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C1CC1)C(F)(F)F
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)C(F)(F)F
COc1cn(-c2cc(F)cc(F)c2)c(=O)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(F)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)c(C)cc1C
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
COc1ccc(Cl)cc1-c1cc(OC)c(cc1C)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(F)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(F)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)c(C)cc1C
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC
COc1ccc(F)cc1-c1cc(OC)c(cc1C)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1ccc(Cl)cc1-c1cc(OC)c(cc1C)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(Cl)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(Cl)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1
COc1cc(c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1
COc1cc(c(Cl)cc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(-c2cccc(F)c2)c(cc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)c(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(F)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)c(Cl)c(F)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1F
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(Cl)c1
COc1cc(c(Cl)cc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(Cl)cc(Cl)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(F)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(OCC(F)(F)F)nc1
COc1nc(-c2cc(F)cc(F)c2)c(cc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
CCOc1ccc(cc1C)-c1cc(OC)c(cc1F)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(F)cc(c1)-c1cc(OC)c(cc1F)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(c1)C1CC1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C1CC1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)ccc1F
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1F
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(Cl)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(Cl)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(C)c1
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1F)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(cc(F)c1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |(-.11,-.1,;1.22,-.87,;2.55,-.1,;2.55,1.44,;3.89,2.21,;5.22,1.44,;5.22,-.1,;6.55,-.87,;3.89,-.87,;3.89,-2.41,;5.22,-3.18,;5.22,-4.72,;3.89,-5.49,;2.55,-4.72,;1.22,-5.49,;-.11,-4.72,;-.11,-3.18,;1.22,-2.41,;2.55,-3.18,;-1.45,-5.49,;-2.22,-4.16,;-.68,-6.83,;-2.78,-6.26,;-4.12,-5.49,;-5.52,-6.12,;-6.55,-4.98,;-5.78,-3.64,;-4.28,-3.96,;3.89,3.75,;5.22,4.52,;5.22,6.06,;3.89,6.83,;2.55,6.06,;1.22,6.83,;2.55,4.52,)|
Cc1ncc2cc(SCc3ccccc3)ccc2c1I
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(cc1)C(F)(F)F
COc1cc(F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cncc(F)c1
COc1cc(F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)nc1
COc1cc(F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccccn1
COc1cc(c(Cl)cc1-c1nc(cc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1[nH]c(=O)cc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1n(C)c(=O)cc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(9.34,-5.39,;8,-4.62,;6.67,-5.39,;6.67,-6.93,;5.33,-7.7,;4,-6.93,;2.67,-7.7,;4,-5.39,;5.33,-4.62,;5.33,-3.08,;6.67,-2.31,;8,-3.08,;6.67,-.77,;8,,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;;-.77,-1.33,;.77,1.33,;-1.33,.77,;-1.33,2.31,;-.09,3.22,;-.56,4.68,;-2.1,4.68,;-2.58,3.22,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-c1nc(Cl)cc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1c(OC)ncc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-.78,-.1,;.55,-.87,;1.89,-.1,;1.89,1.44,;3.22,2.21,;4.55,1.44,;5.89,2.21,;4.55,-.1,;3.22,-.87,;3.22,-2.41,;4.55,-3.18,;5.89,-2.41,;7.22,-3.18,;4.55,-4.72,;3.22,-5.49,;1.89,-4.72,;.55,-5.49,;-.78,-4.72,;-.78,-3.18,;.55,-2.41,;1.89,-3.18,;-2.12,-5.49,;-2.89,-4.16,;-1.35,-6.83,;-3.45,-6.26,;-4.78,-5.49,;-6.19,-6.12,;-7.22,-4.98,;-6.45,-3.64,;-4.94,-3.96,;3.22,3.75,;4.55,4.52,;4.55,6.06,;3.22,6.83,;1.89,6.06,;.55,6.83,;1.89,4.52,)|
COc1cc(c(Cl)cc1-c1c2ccc(cc2cn(C)c1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-.11,-.1,;1.22,-.87,;2.55,-.1,;2.55,1.44,;3.89,2.21,;5.22,1.44,;6.55,2.21,;5.22,-.1,;3.89,-.87,;3.89,-2.41,;2.55,-3.18,;1.22,-2.41,;-.11,-3.18,;-.11,-4.72,;1.22,-5.49,;2.55,-4.72,;3.89,-5.49,;5.22,-4.72,;6.55,-5.49,;5.22,-3.18,;6.55,-2.41,;-1.45,-5.49,;-2.22,-4.16,;-.68,-6.83,;-2.78,-6.26,;-4.12,-5.49,;-5.52,-6.12,;-6.55,-4.98,;-5.78,-3.64,;-4.28,-3.96,;3.89,3.75,;5.22,4.52,;5.22,6.06,;3.89,6.83,;2.55,6.06,;1.22,6.83,;2.55,4.52,)|
COc1cc(ccc1-c1c2ccc(cc2cn(C)c1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(7.22,-.1,;5.89,-.87,;4.55,-.1,;4.55,1.44,;3.22,2.21,;1.89,1.44,;1.89,-.1,;3.22,-.87,;3.22,-2.41,;1.89,-3.18,;.55,-2.41,;-.78,-3.18,;-.78,-4.72,;.55,-5.49,;1.89,-4.72,;3.22,-5.49,;4.55,-4.72,;5.89,-5.49,;4.55,-3.18,;5.89,-2.41,;-2.12,-5.49,;-2.89,-4.16,;-1.35,-6.83,;-3.45,-6.26,;-4.78,-5.49,;-6.19,-6.12,;-7.22,-4.98,;-6.45,-3.64,;-4.94,-3.96,;3.22,3.75,;4.55,4.52,;4.55,6.06,;3.22,6.83,;1.89,6.06,;.55,6.83,;1.89,4.52,)|
COc1cc(c(Cl)cc1-c1c2ccc(cc2c[nH]c1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-.11,-.1,;1.22,-.87,;2.55,-.1,;2.55,1.44,;3.89,2.21,;5.22,1.44,;6.55,2.21,;5.22,-.1,;3.89,-.87,;3.89,-2.41,;2.55,-3.18,;1.22,-2.41,;-.11,-3.18,;-.11,-4.72,;1.22,-5.49,;2.55,-4.72,;3.89,-5.49,;5.22,-4.72,;5.22,-3.18,;6.55,-2.41,;-1.45,-5.49,;-2.22,-4.16,;-.68,-6.83,;-2.78,-6.26,;-4.12,-5.49,;-5.52,-6.12,;-6.55,-4.98,;-5.78,-3.64,;-4.28,-3.96,;3.89,3.75,;5.22,4.52,;5.22,6.06,;3.89,6.83,;2.55,6.06,;1.22,6.83,;2.55,4.52,)|
COc1cc(c(F)cc1-c1n(C)c(=O)cc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(-.11,-.87,;1.22,-1.64,;2.55,-.87,;2.55,.67,;3.89,1.44,;5.22,.67,;6.55,1.44,;5.22,-.87,;3.89,-1.64,;3.89,-3.18,;5.22,-3.95,;6.55,-3.18,;5.22,-5.49,;6.55,-6.26,;3.89,-6.26,;2.55,-5.49,;1.22,-6.26,;-.11,-5.49,;-.11,-3.95,;1.22,-3.18,;2.55,-3.95,;-1.45,-6.26,;-2.22,-4.93,;-.68,-7.6,;-2.78,-7.03,;-4.12,-6.26,;-5.52,-6.89,;-6.55,-5.75,;-5.78,-4.41,;-4.28,-4.73,;3.89,2.98,;5.22,3.75,;5.22,5.29,;3.89,6.06,;2.55,5.29,;2.55,3.75,;1.22,6.06,;1.22,7.6,;-.11,6.83,;-.11,5.29,)|
COc1cc(c(F)cc1-c1[nH]c(=O)cc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1
COc1cc(c(F)cc1-c1[nH]c(=O)cc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(F)cc1-c1c2ccc(cc2c[nH]c1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-.11,-.87,;1.22,-1.64,;2.55,-.87,;2.55,.67,;3.89,1.44,;5.22,.67,;6.55,1.44,;5.22,-.87,;3.89,-1.64,;3.89,-3.18,;2.55,-3.95,;1.22,-3.18,;-.11,-3.95,;-.11,-5.49,;1.22,-6.26,;2.55,-5.49,;3.89,-6.26,;5.22,-5.49,;5.22,-3.95,;6.55,-3.18,;-1.45,-6.26,;-2.22,-4.93,;-.68,-7.6,;-2.78,-7.03,;-4.12,-6.26,;-5.52,-6.89,;-6.55,-5.75,;-5.78,-4.41,;-4.28,-4.73,;3.89,2.98,;5.22,3.75,;5.22,5.29,;3.89,6.06,;3.89,7.6,;2.55,5.29,;1.22,6.06,;2.55,3.75,)|
COc1cc(c(F)cc1-c1c2ccc(cc2c[nH]c1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(-.11,-.1,;1.22,-.87,;2.55,-.1,;2.55,1.44,;3.89,2.21,;5.22,1.44,;6.55,2.21,;5.22,-.1,;3.89,-.87,;3.89,-2.41,;2.55,-3.18,;1.22,-2.41,;-.11,-3.18,;-.11,-4.72,;1.22,-5.49,;2.55,-4.72,;3.89,-5.49,;5.22,-4.72,;5.22,-3.18,;6.55,-2.41,;-1.45,-5.49,;-2.22,-4.16,;-.68,-6.83,;-2.78,-6.26,;-4.12,-5.49,;-5.52,-6.12,;-6.55,-4.98,;-5.78,-3.64,;-4.28,-3.96,;3.89,3.75,;5.22,4.52,;5.22,6.06,;6.55,6.83,;3.89,6.83,;2.55,6.06,;1.22,6.83,;2.55,4.52,)|
COc1cc(c(F)cc1-c1n(C)c(=O)cc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(9.34,-5.39,;8,-4.62,;6.67,-5.39,;6.67,-6.93,;5.33,-7.7,;4,-6.93,;2.67,-7.7,;4,-5.39,;5.33,-4.62,;5.33,-3.08,;6.67,-2.31,;8,-3.08,;6.67,-.77,;8,,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;;-.77,-1.33,;.77,1.33,;-1.33,.77,;-1.33,2.31,;-.09,3.22,;-.56,4.68,;-2.1,4.68,;-2.58,3.22,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-12.32,;1.33,-13.09,;3.44,-13.65,;1.9,-10.99,)|
COc1cc(c(Cl)cc1-c1[nH]c(=O)cc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(F)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1C
COc1cc(ccc1F)-c1cc(OC)c(cc1C)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(F)cc(c1)-c1cc(OC)c(cc1C)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1ccc(F)c(c1)-c1cc(OC)c(cc1C)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1F
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1F
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)ccc1F
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1c(F)cccc1F |(-.11,-.1,;1.22,-.87,;2.55,-.1,;2.55,1.44,;3.89,2.21,;5.22,1.44,;6.55,2.21,;5.22,-.1,;3.89,-.87,;3.89,-2.41,;5.22,-3.18,;5.22,-4.72,;3.89,-5.49,;2.55,-4.72,;1.22,-5.49,;-.11,-4.72,;-.11,-3.18,;1.22,-2.41,;2.55,-3.18,;-1.45,-5.49,;-2.22,-4.16,;-.68,-6.83,;-2.78,-6.26,;-4.12,-5.49,;-5.52,-6.12,;-6.55,-4.98,;-5.78,-3.64,;-4.28,-3.96,;3.89,3.75,;5.22,4.52,;6.55,3.75,;5.22,6.06,;3.89,6.83,;2.55,6.06,;2.55,4.52,;1.22,3.75,)|
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc2CCCc2c1
COc1cc(c(Cl)cc1-c1cn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1ccc(F)c(Cl)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cc(F)cc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1ccc(C)c(Cl)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cc(F)cc(F)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1cccc(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1ccc(F)c(Cl)c1
COc1cc(c(C)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncccn1)-c1ccc(C)c(Cl)c1
COc1cc(c(Cl)cc1-c1c(Br)cnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-7.45,9.79,;-7.45,11.33,;-6.12,12.1,;-4.79,11.33,;-3.45,12.1,;-3.45,13.64,;-2.12,14.41,;-4.79,14.41,;-6.12,13.64,;-7.45,14.41,;-8.79,13.64,;-8.79,12.1,;-10.12,14.41,;-10.12,15.95,;-8.79,16.72,;-8.79,18.26,;-7.45,19.03,;-6.12,18.26,;-6.12,16.72,;-7.45,15.95,;-7.45,20.57,;-8.79,21.34,;-8.79,19.8,;-6.12,21.34,;-4.79,20.57,;-3.32,21.04,;-2.42,19.8,;-3.32,18.55,;-4.79,19.03,;-2.12,11.33,;-2.12,9.79,;-.79,9.02,;.55,9.79,;.55,11.33,;1.88,12.1,;-.79,12.1,)|
CCc1nnc2cc(ccc2c1-c1cc(Cl)c(cc1OC)-c1cccc(F)c1)S(=O)(=O)Nc1ccon1 |(-3.33,-11.5,;-4.67,-10.73,;-4.67,-9.19,;-6,-8.42,;-6,-6.88,;-4.67,-6.11,;-4.67,-4.57,;-3.33,-3.8,;-2,-4.57,;-2,-6.11,;-3.33,-6.88,;-3.33,-8.42,;-2,-9.19,;-2,-10.73,;-.67,-11.5,;-.67,-13.04,;.67,-10.73,;.67,-9.19,;-.67,-8.42,;-.67,-6.88,;.67,-6.11,;2,-11.5,;2,-13.04,;3.33,-13.81,;4.67,-13.04,;4.67,-11.5,;6,-10.73,;3.33,-10.73,;-3.33,-2.26,;-4.67,-1.49,;-4.67,-3.03,;-2,-1.49,;-.67,-2.26,;.8,-1.79,;1.7,-3.03,;.8,-4.28,;-.67,-3.8,)|
COc1cc(c(Cl)cc1-c1c(C)nnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(.67,-6.11,;-.67,-6.88,;-.67,-8.42,;.67,-9.19,;.67,-10.73,;-.67,-11.5,;-.67,-13.04,;-2,-10.73,;-2,-9.19,;-3.33,-8.42,;-4.67,-9.19,;-4.67,-10.73,;-6,-8.42,;-6,-6.88,;-4.67,-6.11,;-4.67,-4.57,;-3.33,-3.8,;-2,-4.57,;-2,-6.11,;-3.33,-6.88,;-3.33,-2.26,;-4.67,-1.49,;-4.67,-3.03,;-2,-1.49,;-.67,-2.26,;.8,-1.79,;1.7,-3.03,;.8,-4.28,;-.67,-3.8,;2,-11.5,;2,-13.04,;3.33,-13.81,;4.67,-13.04,;4.67,-11.5,;6,-10.73,;3.33,-10.73,)|
COc1cc(c(Cl)cc1-c1c(N)cnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-.11,-.1,;1.22,-.87,;2.55,-.1,;2.55,1.44,;3.89,2.21,;5.22,1.44,;6.55,2.21,;5.22,-.1,;3.89,-.87,;3.89,-2.41,;5.22,-3.18,;6.55,-2.41,;5.22,-4.72,;3.89,-5.49,;2.55,-4.72,;1.22,-5.49,;-.11,-4.72,;-.11,-3.18,;1.22,-2.41,;2.55,-3.18,;-1.45,-5.49,;-2.22,-4.16,;-.68,-6.83,;-2.78,-6.26,;-4.12,-5.49,;-5.52,-6.12,;-6.55,-4.98,;-5.78,-3.64,;-4.28,-3.96,;3.89,3.75,;5.22,4.52,;5.22,6.06,;3.89,6.83,;2.55,6.06,;1.22,6.83,;2.55,4.52,)|
COc1cc(c(Cl)cc1-c1c(OC)nnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-3.33,-5.39,;-3.33,-3.85,;-2,-3.08,;-.67,-3.85,;.67,-3.08,;.67,-1.54,;2,-.77,;-.67,-.77,;-2,-1.54,;-3.33,-.77,;-4.67,-1.54,;-4.67,-3.08,;-6,-3.85,;-6,-.77,;-6,.77,;-4.67,1.54,;-4.67,3.08,;-3.33,3.85,;-2,3.08,;-2,1.54,;-3.33,.77,;-3.33,5.39,;-4.67,6.16,;-4.67,4.62,;-2,6.16,;-.67,5.39,;.8,5.87,;1.7,4.62,;.8,3.37,;-.67,3.85,;2,-3.85,;2,-5.39,;3.33,-6.16,;4.67,-5.39,;4.67,-3.85,;6,-3.08,;3.33,-3.08,)|
COc1cc(c(Cl)cc1-c1c(N)nnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(.67,1.54,;-.67,.77,;-.67,-.77,;.67,-1.54,;.67,-3.08,;-.67,-3.85,;-.67,-5.39,;-2,-3.08,;-2,-1.54,;-3.33,-.77,;-4.67,-1.54,;-4.67,-3.08,;-6,-.77,;-6,.77,;-4.67,1.54,;-4.67,3.08,;-3.33,3.85,;-2,3.08,;-2,1.54,;-3.33,.77,;-3.33,5.39,;-4.67,6.16,;-4.67,4.62,;-2,6.16,;-.67,5.39,;.8,5.87,;1.7,4.62,;.8,3.37,;-.67,3.85,;2,-3.85,;2,-5.39,;3.33,-6.16,;4.67,-5.39,;4.67,-3.85,;6,-3.08,;3.33,-3.08,)|
COc1cc(c(F)cc1-c1c[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1
COc1cc(c(F)cc1-c1c[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1
COc1cc(c(F)cc1-c1c[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1c(O)cnc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(1.33,2.31,;2.67,1.54,;4,2.31,;4,3.85,;5.33,4.62,;6.67,3.85,;8,4.62,;6.67,2.31,;5.33,1.54,;5.33,,;6.67,-.77,;8,,;6.67,-2.31,;5.33,-3.08,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;1.33,-.77,;2.67,,;4,-.77,;,-3.08,;.77,-4.41,;-.77,-1.75,;-1.33,-3.85,;-2.67,-3.08,;-2.83,-1.55,;-4.33,-1.23,;-5.1,-2.56,;-4.07,-3.71,;5.33,6.16,;4,6.93,;4,8.47,;5.33,9.24,;6.67,8.47,;8,9.24,;6.67,6.93,)|
COc1cnc2cc(ccc2c1-c1cc(Cl)c(cc1OC)-c1cccc(F)c1)S(=O)(=O)Nc1ccon1 |(9.34,-.77,;8,,;6.67,-.77,;6.67,-2.31,;5.33,-3.08,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;1.33,-.77,;2.67,,;4,-.77,;5.33,,;5.33,1.54,;6.67,2.31,;6.67,3.85,;8,4.62,;5.33,4.62,;4,3.85,;4,2.31,;2.67,1.54,;1.33,2.31,;5.33,6.16,;4,6.93,;4,8.47,;5.33,9.24,;6.67,8.47,;8,9.24,;6.67,6.93,;,-3.08,;.77,-4.41,;-.77,-1.75,;-1.33,-3.85,;-2.67,-3.08,;-2.83,-1.55,;-4.33,-1.23,;-5.1,-2.56,;-4.07,-3.71,)|
COc1cc(c(F)cc1-c1cn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1
COc1cc(c(F)cc1-c1cn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1
COc1cc(c(F)cc1-c1cn(C)c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccsn1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccc(F)cn1)-c1cccc(F)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C(F)F
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C#N
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C#N
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(Cl)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncon1)-c1cccc(Cl)c1
COc1cc(c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccsn1)-c1cccc(Cl)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1cscn1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1ccc(Cl)c(C)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC2)C1=O
CC(C)(C)OC(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)OC(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)COC(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CS(=O)(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
NC(=O)Cn1ccn(-c2cccc3n(ncc23)-c2ccccc2F)c1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CN1CC(=O)N(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1C(=O)CN(Cc2ccccn2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nc(cs2)C(F)(F)F)C1=O
C[C@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@@H]3C[C@H]2CO3)C1=O |TLB:21:23:28.29:26|
FC1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1C[C@@H](N(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1cc(F)ccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1cccnc1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1ccncc1
CC[C@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(C)C(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CN1CCCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Cc1csc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)n1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@H]3C[C@@H]2CO3)C1=O |TLB:21:23:28.29:26|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cocn2)C1=O
Cc1noc(C)c1CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1ncccn1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nnco2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nnc(s2)C2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2ncco2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@@H]2CCOC2)C1=O
Cc1cnc(nc1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nccs2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cnccn2)C1=O
Fc1ccc(c(F)c1)-n1ncc2c(cccc12)N1CCN(Cc2ncco2)C1=O
Fc1ccc(c(F)c1)-n1ncc2c(cccc12)N1CCN(Cc2cocn2)C1=O
C[C@H]1CN(C(=O)N1Cc1ncco1)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cscn2)C1=O
Cc1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)s1
Cc1cnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
Cc1cncc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)n1
Cc1nccnc1CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Cc1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
CCc1cc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)on1
CC(N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1nc(C)no1
CCOc1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)s1
Cc1nc(CN2CCCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)oc1C
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nnc(o2)C2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nnc(o2)C2CCC2)C1=O
CCS(=O)(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@@H]2CCOC2)C1=O
Cc1cccc(c1)-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC[C@H](F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCNC1=O
NS(=O)(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
COCCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(C)C(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C(=O)C2CC(=O)C2)C1=O
CNS(=O)(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CCN2CCNC2=O)C1=O
CC(C)(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
COC[C@H]1CC[C@H](COC)N1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCN3CCCC3C2)C1=O
CC(C)OC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CN(CC1CCOCC1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
FC1CCN(CC1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC1CN(CC(C)O1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC2CN2CCOCC2)C1=O
CN(CCN1CCOCC1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCOCCNC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NCC2CCOC2)C1=O
CC(C)CCC(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)S(=O)(=O)C1CCCC1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)S(=O)(=O)C1CCCCC1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)S(=O)(=O)c1cccs1
CC(C)CS(=O)(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCCS(=O)(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)S(=O)(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCS(=O)(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(O)[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@H]2CCOC2)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1cccc(OC(F)(F)F)c1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2ccc(cn2)C(F)(F)F)C1=O
C[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC(F)(F)C2)C1=O
CC(C)CNC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCN(CC)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC2)C1=O
CC(C)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)OCC(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cc(ccn2)C(F)(F)F)C1=O
CCOCC1(F)CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCN3CCC[C@H]3C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC3(COC3)C2)C1=O
CC1COCC(C)N1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC3(C2)OCCO3)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC(=O)NC(=O)C2)C1=O
CN1CC2CN(CC2C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCOC3CCCCC23)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC3CCCC3C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@H]3C[C@@H]4C[C@H](C3)C[C@H]2C4)C1=O
CN1C(=O)[C@H]2CN(C[C@H]2C1=O)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
COC1C2CCC1CN(C2)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |THB:10:8:4.5:2|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC3(CC2)OCCO3)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@H]3[C@H]4CC[C@H](C4)[C@H]3C2)C1=O |THB:24:25:27.28:30,32:31:27.28:30|
CN1CCCC2CN(CC12)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
C[C@@H]1COCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CN1[C@H]2CC[C@@H]1CN(CC2)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |TLB:10:7:4.3:1|
CCC1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)C1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CC1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
C[C@@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
COC(=O)[C@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC[C@@H]2C(=O)Nc2ccccc2)C1=O
O[C@@H]1C[C@@H](N(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1cc(F)ccc1F
O[C@H]1C[C@@H](N(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1cc(F)ccc1F
CC(C)CC(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)[C@H]1CCCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)[C@@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)[C@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@@H]1C[C@@H](N(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1cc(F)ccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC[C@@H]2c2ccccc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC2c2ccccc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1ccccn1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C(=O)OC2CCCCC2)C1=O
CC(C)CCCC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CCCC(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)CC2CCCC2)C1=O
OC(CC1CCCC1)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)CC2CCCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CC2CN(CCN2C1=O)C(=O)OC1CCCC1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1cncnc1
OC(CC1CCCCC1)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)CC2CCC2)C1=O
OC(CC1CCC1)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)CC2CC3CCC2C3)C1=O |THB:23:24:27.28:30|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)c2ccccc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)C2CCCC2)C1=O
CC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(O)(CCC=C)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccc(cn1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCC(O)(CC(C)C)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
COc1cccc(c1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1cccc(c1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)c2ccc(cc2)C(F)(F)F)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)c2cccnc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)c2ccc3OCOc3c2)C1=O
Fc1ccncc1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)C[C@@H](O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)C[C@H](O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)CC2CCOC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1cncs1
CC[C@@H](CO)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC[C@@H](O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(C)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)C(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)C2CCC2)C1=O
OC(CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)C1CCC1
OC(N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)C(=O)C1CCC1
CC(C)C[C@@](C)(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)C[C@](C)(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC[C@H]2C(F)(F)F)C1=O
COC[C@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC[C@@H]2C(F)(F)F)C1=O
CC1(C)CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1cccc(CNC(=O)CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)c1
Fc1ccc(F)c(CNC(=O)CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)c1
Cc1ccccc1CNC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
C[C@@H](NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1ccccc1
Fc1cc(F)cc(CNC(=O)CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)c1
C[C@H](NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1ccccc1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nc3ccccc3s2)C1=O
CC(C)C(C)(O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC2CCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC2CCCO2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)C2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CCC2)C1=O
Fc1ccccc1[C@H]1C[C@H](CO1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CC(O)CN1CCCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
C[C@H]1CCCN1C(=O)CN1CCCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CC(=O)CN1CCCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC2CC2(F)F)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1cnn2cccnc12
Cn1cc2cc(ccc2n1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1ccc(o1)C1CC1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CCc2ccccc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC2CC2)C1=O
C[C@]1(C[C@@H](CO1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1cccc(F)c1
Fc1cccc(c1)[C@@H]1C[C@H](CO1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccc(F)c(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)c1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cccnc2)C1=O
Cc1cc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)no1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC2COC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC[C@@H]2C#N)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC3CCC2C3)C1=O |THB:21:23:26.27:29|
C[C@]1(C[C@H](CO1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1cccc(F)c1
OC1CCC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCC1(O)CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
FC1CN(CC1F)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1cncc(c1)N1CCOCC1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1cccnn1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NCC2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2ccncc2)C1=O
Cc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)co1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2[C@H]3CC[C@@H]2CC3)C1=O |r|
CC1(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)COC1
CO[C@H](CC(C)C)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CO[C@@H](CC(C)C)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(=O)N1CC(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)C1
Cc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)cs1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2ncccn2)C1=O
Cc1cnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)nc1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CCc2cccnc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1nccs1
Fc1ccccc1-n1ncc2c(cccc12)N1C(=O)CN(Cc2ccncn2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC2CCO2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@H]2CCOC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCCN(Cc2cocn2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C1=O)c1cnccn1
Cc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)c(C)o1
Cc1cncc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)c1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC2(CC2)OCc2ccccc2)C1=O
COc1cncc(c1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cnco2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CCN(Cc3ccccc3)C2=O)C1=O
CC(C)(C)c1cnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
Cc1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccc(F)cc2F)s1
FC(F)(F)c1ccc(cc1)-n1ncc2c(cccc12)N1CCN(Cc2ncco2)C1=O
Cc1noc(C)c1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)c1cnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
Cc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)oc1C
Cc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)c(C)s1
Cc1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccc(cc2)C(F)(F)F)s1
C[C@@H]1CN(C(=O)N1C(=O)OC(C)(C)C)c1cccc2n(ncc12)-c1ccccc1F
FC(F)(F)c1ccc(cc1)-n1ncc2c(cccc12)N1CCN(Cc2cocn2)C1=O
Cc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccc(F)cc2F)cs1
Cc1cc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)on1
Cc1scnc1CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
C[C@@H]1CN(C(=O)N1)c1cccc2n(ncc12)-c1ccccc1F
C[C@@H]1CN(C(=O)N1Cc1ncco1)c1cccc2n(ncc12)-c1ccccc1F
COc1nccnc1CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)c1cc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)on1
CCc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)cs1
CC(C)c1cc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)no1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cc(on2)C2CC2)C1=O
C[C@@H](N1CCN(C1=O)c1cccc2n(ncc12)-c1ccc(F)cc1F)c1nc(C)no1
COCc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)cs1
Fc1ccccc1-n1ncc2c(cccc12)N1CCCN(Cc2ncco2)C1=O
CC(C)c1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
Cc1cnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)cn1
Cc1noc(C)c1CN1CCCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Cc1cncc(CN2CCCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)n1
Cc1nnc(CN2CCCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
CCc1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
CC(C)(C)c1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)o1
Cc1cnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)s1
Cc1nocc1CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@H]1CC[C@@H](CC1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |r,wU:1.0,wD:4.7,(.53,9.13,;1.44,7.88,;2.97,8.05,;3.88,6.8,;3.25,5.39,;1.72,5.23,;.81,6.48,;4.15,4.15,;5.69,4.15,;6.17,2.68,;4.92,1.78,;3.68,2.68,;2.21,2.21,;4.92,.24,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;2.13,-2.55,;1.22,-1.3,;2.13,-.06,;3.59,-.53,;1.65,-4.01,;2.68,-5.16,;2.2,-6.62,;.7,-6.94,;-.33,-5.8,;.14,-4.33,;-.89,-3.19,)|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CCC(=O)CC2)C1=O
CC(C)(C)OC(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CNC2)C1=O
OC1(CC1)C(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
NC(=O)C(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CS(=O)(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@@H]2CCCC[C@H]2OCc2ccccc2)C1=O
O[C@@H]1CCCC[C@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCCS(=O)(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@H]2CCCC[C@@H]2OCc2ccccc2)C1=O
O[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O=C(CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1)N1CCCC1
O=C(CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccn1)N1CCCC1
CO[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CO[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@H]2CCCCC2=O)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CN(C2)S(=O)(=O)CC2CC2(Cl)Cl)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CN(C2)S(=O)(=O)CC2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CN(C2)S(=O)(=O)CC(F)(F)F)C1=O
CC(C)CS(=O)(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(C)OC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCOC(=O)C=CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |w:6.6|
CCOC(=O)\C=C\N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(C)OC(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
OC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCOCC2)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)C1CCCCC1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC(F)(F)CC2)C1=O
FC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC(CC2)C(F)(F)F)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC(C2)C(F)(F)F)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@@H]3CC[C@H](C2)O3)C1=O |TLB:21:23:27.26:30|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC(=O)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NCC(F)(F)F)C1=O
CC(C)(C)CCn1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC2)C1=O
CC(C)(C)n1ncc2c(cccc12)N1CCN(CC(=O)N2CC[C@H](F)C2)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC[C@@H](C2)C(F)(F)F)C1=O
CC1(F)CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2[C@H]3CC[C@@H]2CC(=O)C3)C1=O |THB:30:29:23:25.26|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC(F)(F)C(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC(=O)CC2)C1=O
F[C@H]1CCN(C1)C(=O)C=CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |w:9.10|
CCNC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
OCC1(CCC1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@@H]1CCCN(C1)C(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCCN(C1)C(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
COC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCOCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2COC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCCC2)C1=O
CC(=O)C1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CO[C@H]1C[C@@H](C1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |r,wU:2.1,wD:4.6,(4.2,14.09,;5.11,12.85,;4.48,11.44,;5.03,10,;3.6,9.45,;3.04,10.89,;2.97,8.05,;3.88,6.8,;5.41,6.96,;3.25,5.39,;4.15,4.15,;5.69,4.15,;6.17,2.68,;4.92,1.78,;3.68,2.68,;2.21,2.21,;4.92,.24,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;2.13,-2.55,;1.22,-1.3,;2.13,-.06,;3.59,-.53,;1.65,-4.01,;2.68,-5.16,;2.2,-6.62,;.7,-6.94,;-.33,-5.8,;.14,-4.33,;-.89,-3.19,)|
CC1(C)CC1NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC(C2)C(F)(F)F)C1=O
FC(F)C1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)O[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@H]1CCC[C@H]1NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC1(CC1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@H]2CCC[C@@H]2OCc2ccccc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@@H]2CCC[C@H]2OCc2ccccc2)C1=O
CC(C)COC1COCC1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CO[C@H]1CCC[C@H]1NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccc(Cl)cc1
CC(C)(C)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@@H]3CCC[C@@H]3C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NCCC(F)(F)F)C1=O
CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
NC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)[C@H](N(C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)C(C)(C)C)C(N)=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCC2(F)F)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1cc(Cl)cc(Cl)c1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CC(=O)C2)C1=O
OC1CC(C1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |(5.11,12.85,;4.48,11.44,;3.04,10.89,;3.6,9.45,;5.03,10,;2.97,8.05,;3.88,6.8,;5.41,6.96,;3.25,5.39,;4.15,4.15,;5.69,4.15,;6.17,2.68,;4.92,1.78,;3.68,2.68,;2.21,2.21,;4.92,.24,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;2.13,-2.55,;1.22,-1.3,;2.13,-.06,;3.59,-.53,;1.65,-4.01,;2.68,-5.16,;2.2,-6.62,;.7,-6.94,;-.33,-5.8,;.14,-4.33,;-.89,-3.19,)|
CN(C1CCC1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2(CCC2)C(F)(F)F)C1=O
[#8]\[#7]=[#6]-1/[#6]-[#6](-[#6]-1)-[#7]-[#6](=O)-[#6]-[#7]-1-[#6]-[#6]-[#7](-[#6]-1=O)-c1cccc2n(ncc12)-c1ccccc1F
[#6]-[#8]\[#7]=[#6]-1/[#6]-[#6](-[#6]-1)-[#7]-[#6](=O)-[#6]-[#7]-1-[#6]-[#6]-[#7](-[#6]-1=O)-c1cccc2n(ncc12)-c1ccccc1F
FC1CCC(CC1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |(1.89,-14.21,;1.26,-12.8,;-.27,-12.64,;-.9,-11.23,;.01,-9.99,;1.54,-10.15,;2.16,-11.55,;-.62,-8.58,;.28,-7.33,;1.82,-7.49,;-.34,-5.93,;.56,-4.68,;2.1,-4.68,;2.58,-3.22,;1.33,-2.31,;.09,-3.22,;-1.38,-2.74,;1.33,-.77,;2.67,,;2.67,1.54,;1.33,2.31,;,1.54,;-1.46,2.02,;-2.37,.77,;-1.46,-.48,;;-1.94,3.48,;-.91,4.63,;-1.39,6.09,;-2.89,6.41,;-3.92,5.27,;-3.45,3.8,;-4.48,2.66,)|
CC(C)(C)CNC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)C[C@@H](N)C(=O)N[C@@H](C)COc1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)C[C@@H](N)C(=O)NC(C)COc1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)CC(N)C(=O)N[C@@H](C)COc1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
CN[C@H](CC(C)C)C(=O)NCCOc1cc(F)cc(c1)C(F)(F)F |r|
CC(C)C[C@@H](N)C(=O)NC(COc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ccccc1 |r|
N[C@H](c1nc2c(cc(cc2[nH]1)C(F)(F)F)C(F)(F)F)c1ccc(Cl)cc1 |r|
N[C@H](Cc1cccc(c1)C(F)(F)F)C(=O)NCc1nc2c(cc(cc2[nH]1)C(F)(F)F)C(F)(F)F |r|
COc1ccccc1-n1ncc(C(=O)Nc2ccc(Cl)cc2)c1N
Cc1ccccc1-n1ncc(C(=O)Nc2ccc(Cl)cc2F)c1N
COCCOc1ccccc1-n1nc(C)c(C(=O)Nc2ccc(cc2F)C(F)(F)F)c1N
Cc1c(F)cccc1-n1ncc(C(=O)Nc2ccc(OC(F)(F)F)cn2)c1N
Cc1c(F)cccc1-n1ncc(C(=O)N2CCc3cc(Cl)ccc23)c1N
COc1ccccc1-n1ncc(C(=O)N2CCc3cc(Cl)ccc23)c1N
Cc1c(F)cccc1-n1nnc(C(=O)Nc2ccc(Cl)cn2)c1N
CCc1nn(c(N)c1C(=O)Nc1ccc(cn1)C(F)(F)F)-c1ccccc1OC
COCCOc1ccccc1-n1nc(C)c(C(=O)Nc2ccc(cc2C)C(F)(F)F)c1N
Cc1nn(c(N)c1C(=O)Nc1ccc(Cl)cn1)-c1cccc(F)c1C
CCc1ccccc1-n1ncc(C(=O)Nc2ccc(OCC(F)(F)F)cn2)c1N
CCc1nn(c(N)c1C(=O)Nc1ccc(cn1)C(F)(F)F)-c1cccc(F)c1C
Cc1nn(c(N)c1C(=O)Nc1ccc(cn1)C(F)(F)F)-c1ccccc1F
Nc1c(cnn1-c1ccccc1-c1cccnc1)C(=O)Nc1ccc(Cl)cn1
COc1cc(ccn1)-c1ccccc1-n1ncc(C(=O)Nc2ccc(Cl)cn2)c1N
Nc1c(cnn1-c1ccccc1O)C(=O)Nc1ccc(cn1)C(F)(F)F
Cc1c(F)cccc1-n1cnc(C(=O)Nc2ccc(cn2)C(F)(F)F)c1N
COc1ccccc1-n1cnc(C(=O)Nc2ccc(Cl)cc2)c1N
Fc1ccc(Oc2ccc(cc2)-n2c(nc3ccccc23)C2CCOCC2)cc1
Cn1cc(Cl)c(n1)-c1nc2ccccc2n1-c1ccc(Oc2ccc(F)cc2)cc1
Fc1ccc(Oc2ccc(cc2)-n2c(nc3ccccc23)-c2c[nH]cn2)cc1
Fc1ccc(Oc2ccc(cc2)-n2c(nc3ccccc23)[C@@H]2CCC(=O)N2)cc1
Cc1nnc(Cc2nc3ccccc3n2-c2ccc(Oc3ccc(F)cc3)cc2)[nH]1
Fc1ccc(Oc2ccc(cc2)-n2c(CCN3CCCCC3)nc3ccccc23)cc1
Fc1ccc(Oc2ccc(cc2)-n2c(Cc3nnn[nH]3)nc3ccccc23)cc1
CCN(CC)C(=O)CN1CCC(CC1)c1nc2ccccc2n1-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)CN1CCC(CC1)c1nc2ccccc2n1-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)CN1CCC[C@H]1c1nc2ccccc2n1-c1ccc(Oc2ccc(F)cc2)cc1
Fc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1ccccc1)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1O[C@@H]1CCCC[C@@H]1c1ccccc1)S(=O)(=O)Nc1ncns1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)N([Na])c1cscn1 |r|
Fc1cc(c(F)cc1O[C@H]1CCC[C@@H]1c1ccccc1)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1O[C@H]1CCCCC[C@@H]1c1ccccc1)S(=O)(=O)Nc1ncns1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Cn1nccc1[C@H]1CCCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)N([Na])c1cscn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)N([Na])c1cscn1 |r|
CCn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
Fc1cc(O[C@H]2CCCC[C@@H]2n2ccnc2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1nccs1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(cc1F)S(=O)(=O)Nc1cc(F)ncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(cc1F)S(=O)(=O)Nc1ccnc(F)n1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(Cl)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(cc1C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1ccn[nH]1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccnc(F)n1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1n1ccnc1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1cn[nH]c1)S(=O)(=O)Nc1ccncn1 |r|
Nc1n[nH]cc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Nc1cc(ccn1)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Nc1cc(ccn1)[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1cccnc1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@H]1CCCC[C@@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@H]1CCCC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCCC[C@@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1ccnnc1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCCC[C@@H]1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCCC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CCc1cc(c(F)cc1O[C@H]1CCC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1C#N)S(=O)(=O)Nc1ccncn1 |r|
Cc1c(O[C@H]2CCC[C@@H]2c2ccnn2C)ccc(c1F)S(=O)(=O)Nc1ccncn1 |r|
Cc1c(O[C@H]2CCCC[C@@H]2c2ccnn2C)ccc(c1F)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CCCC[C@@H]1c1c[nH]nc1N)S(=O)(=O)Nc1ccncn1 |r|
Nc1ncccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cc1ncccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Nc1n[nH]cc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cc1c(F)c(ccc1O[C@H]1CCCC[C@@H]1c1c[nH]nc1N)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1O[C@@H]1CCCC[C@H]1c1ccccc1)S(=O)(=O)Nc1ncns1 |r|
Cn1nccc1[C@@H]1CCC[C@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Nc1nnccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Fc1c(O[C@H]2CCCC[C@@H]2c2cn[nH]c2)ccc(c1F)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@H]1CCC[C@@H]1c1c[nH]nc1N)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1 |r|
Cn1nccc1[C@H]1CC(F)(F)CC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
CCc1cc(ccc1O[C@H]1CCCC[C@@H]1c1c[nH]nc1N)S(=O)(=O)Nc1ccncn1 |r|
Nc1n[nH]cc1[C@H]1CCCC[C@@H]1Oc1ccc(c(F)c1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nncc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
CC(=O)Nc1n[nH]cc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1C)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1C[C@H](C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)OCc1ccccc1 |r|
Cn1nccc1[C@H]1C[C@@H](C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)OCc1ccccc1 |r|
Cn1nccc1[C@@H]1[C@H](CCC1(C)C)Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1[C@@H](CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)OCc1ccccc1 |r|
Cc1cc(c(F)cc1O[C@H]1CCC[C@@H]1c1cn[nH]c1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1O[C@H]1CC(F)(F)CC[C@@H]1c1cn[nH]c1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CC(F)(F)CC[C@@H]2c2cn[nH]c2)cc(F)c1S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC(F)(F)C[C@@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1C[C@@H](F)C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CCCC[C@@H]2c2cn[nH]c2)ccc1S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC(F)(F)C[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccnc(F)n1 |r|
Cn1nccc1[C@H]1C[C@@H](CC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)OCc1ccccc1 |r|
Cn1nccc1[C@H]1CC[C@@H](C[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)OCc1ccccc1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccnc(F)n1 |r|
CCn1nccc1[C@H]1CCC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Nc1n[nH]cc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1cscn1 |r|
Cn1nccc1[C@@H]1[C@H](CCCC1(F)F)Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
CCn1nccc1[C@@H]1CCC[C@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
CO[C@@H]1C[C@H](Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ccncn2)[C@H](C1)c1ccnn1C |r|
CO[C@H]1C[C@H](Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ccncn2)[C@H](C1)c1ccnn1C |r|
Cc1cc(c(F)cc1O[C@H]1CC(F)(F)CC[C@@H]1c1ccnn1C)S(=O)(=O)Nc1nncs1 |r|
Cn1nccc1[C@@H]1CCC[C@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(F)(F)CC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC(F)(F)C[C@@H]1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCC(F)(F)C[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1 |r|
Cn1nccc1[C@H]1CC(F)(F)C[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@@H]1CCCC[C@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@@H]1CC(F)(F)CC[C@H]1c1cn[nH]c1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@H]2CC(F)(F)CC[C@@H]2c2cn[nH]c2)ccc1S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@@H]1CCC[C@H]1c1ccn[nH]1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@@H]2CCC[C@H]2c2ccn[nH]2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccnc(=O)[nH]1 |r|
Fc1cc(O[C@@H]2CCCC[C@H]2c2ccn[nH]2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC[C@@H](O)C[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1C[C@@H](O)CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CC[C@H](O)C[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@@H]1C[C@@H](O)CC[C@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1[C@H]1CCCC[C@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(O[C@@H]2CCCC[C@H]2c2cn[nH]c2)cc(F)c1S(=O)(=O)Nc1ccncn1 |r|
Cc1cc(c(F)cc1O[C@@H]1CCCC[C@H]1c1cn[nH]c1)S(=O)(=O)Nc1ccncn1 |r|
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
C[C@@H]1CNCCN1c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CC(=O)N[C@@H]1CCN(C1)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CCN(CC)C1CCN(C1)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Fc1cc(Nc2ccc(Cl)cc2N2CCC(C2)N2CCCC2)c(Cl)cc1S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(C)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
C[C@H]1CN(CCN1)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CNC1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(F)ccc1Nc1c(F)cc(cc1F)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(F)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(OC(F)(F)F)ccc1Nc1ccc(cc1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(OC(F)(F)F)ccc1Nc1c(F)cc(cc1F)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(OC(F)(F)F)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(OC(F)(F)F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(Cl)cnc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1nc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
CNC1CCN(C1)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CN[C@@H]1CCCN(C1)c1cc(F)ccc1Nc1ccc(cc1)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(F)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCN(C1)c1cc(F)ccc1Nc1c(F)cc(cc1F)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
NC1CCN(C1)c1cc(F)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1
NC1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
NC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1ccccc1Nc1ccc(cc1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1)C(F)(F)F
CNC1CCN(C1)c1cc(ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
CNC1CCN(C1)c1ccccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1ccccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
F[C@@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1)S(=O)(=O)Nc1cscn1 |r|
F[C@@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1 |r|
F[C@@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
F[C@@H]1CCN(C1)c1cc(F)ccc1Nc1c(F)cc(cc1F)S(=O)(=O)Nc1cscn1 |r|
F[C@@H]1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CNC1CCN(C1)c1c(F)cccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1c(F)cccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1c(F)cccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(OC)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(OC)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
CNC1CCN(C1)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CN[C@@H]1CCCN(C1)c1cc(OC)ccc1Nc1ccc(cc1)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(OC)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(OC)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(OC)ccc1Nc1c(F)cc(cc1F)S(=O)(=O)Nc1cscn1 |r|
CN[C@@H]1CCCN(C1)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN1CCN(CC1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
CN1CCN(CC1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CN(C)[C@H]1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN(C)[C@H]1CCN(C1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F |r|
CN1CCN(CC1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
CN1CCN(CC1)c1cc(OC(F)F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CN1CCN(CC1)c1cc(OC(F)(F)F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CN(C)[C@H]1CCN(C1)c1cc(ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F |r|
CN[C@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1 |r|
CN[C@H]1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
COc1ccc(Nc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)N1CC[C@@H](C1)N(C)C |r|
CN(C)[C@H]1CCN(C1)c1cc(OC(F)F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F |r|
CN(C)[C@@H]1CCN(C1)c1cc(OC(F)F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
Fc1ccc(Nc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)N1CCCNCC1
CNC1CCN(C1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C#N
CC(=O)N[C@@H]1CCN(C1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F |r|
CC(=O)N[C@@H]1CCN(C1)c1cc(ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F |r|
CN[C@H]1CCN(C1)c1cc(ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F |r|
CN[C@H]1CCN(C1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F |r|
COC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
COC1CCN(C1)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
CC(=O)N[C@@H]1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
COC1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
COC1CCN(C1)c1cc(ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
CC(=O)N[C@@H]1CCN(C1)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
CN(CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)N(C(=O)OC(C)(C)C)c1cscn1)C(=O)OC(C)(C)C
CN(C)CCN(C)c1cc(F)ccc1Nc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
CN(C)CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
CN(CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)N(C(=O)OC(C)(C)C)c1ncc(F)cn1)C(=O)OC(C)(C)C
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C#N
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)cn1)C#N
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)cn1
CN(CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)N(C(=O)OC(C)(C)C)c1ccc(F)cn1)C(=O)OC(C)(C)C
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccccn1
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1)C#N
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccccn1)C#N
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C#N
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1)C(F)(F)F
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccccn1)C(F)(F)F
CNCCN(C)c1cc(ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccccn1
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
CNCCN(C)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1
CNCCN(C)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
CNCCN(C)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNCCN(C)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)cn1
CNCCN(C)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CNCCN(C)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)cn1
CNCCN(C)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1
CNCCN(C)c1cc(Cl)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(Cl)s1
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(Cl)s1
CNCCN(C)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(Cl)s1
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1
CNCCN(C)c1cc(OC)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1
CN(CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)N(C(=O)OC(C)(C)C)c1cc(C)on1)C(=O)OC(C)(C)C
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cc(C)on1
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cc(C)[nH]n1
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cc(C)[nH]n1
CN(C)CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)N(C(=O)OC(C)(C)C)c1ncc(F)cn1
CN(C)CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
CN(C)CCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(Cl)s1
CN(C)CCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(Cl)s1
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(C)s1
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncco1
CNCCN(C)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cc(on1)C(C)(C)C
CNCCN(C)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cc(on1)C(C)(C)C
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccn(C)n1
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)cn1
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cnccn1
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cc(C)on1
CNC1CCN(C1)c1cc(F)ccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cncnc1
Cn1nccc1-c1cc(ccc1C1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cc(F)ccn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cc(F)ccn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccc(F)cn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccc(F)cn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cnccn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccc1F)C(F)(F)F
Cc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)n1
Cc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)n1
Cc1ccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)nc1
Cc1ccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)nc1
Cc1ccnc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)c1
Cc1ccnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)c1
CC(C)Oc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)n1
CC(C)Oc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2ccnn2C)C(F)(F)F)n1
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnc1F)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1
Cn1nccc1-c1cc(Cl)ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1
CC(C)Oc1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccc(F)n2)c(c1)-c1ccnn1C
CC(C)Oc1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccc(F)n2)c(c1)-c1ccnn1C
Fc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Fc1cnc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-c2ccc(F)nc2)C(F)(F)F)nc1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2ccc(F)nc2)C(F)(F)F)nc1
Fc1ccc(cn1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Fc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Fc1ccc(cn1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
Fc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
Fc1ccc(cc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Fc1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Fc1ccc(cc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Fc1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Fc1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Fc1ccc(cc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
Fc1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)-n1ccnn1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)-n1ccnn1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(c1)-n1ccnn1
Fc1cnc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-n2ccnn2)C(F)(F)F)nc1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-n2ccnn2)C(F)(F)F)nc1
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)-n1ccnn1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)-n1ccnn1
Fc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-n2ccnn2)C(F)(F)F)n1
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-n2ccnn2)C(F)(F)F)n1
Cc1nc(cs1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
Cc1nc(cs1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
Cc1nc(cs1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Cc1nc(cs1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Cc1nc(cs1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Cc1nc(cs1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Cc1nc(cs1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cc1nc(cs1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cc1nc(cs1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
Cc1nc(co1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
CS(=O)(=O)CCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
CS(=O)(=O)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
CS(=O)(=O)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
CS(=O)(=O)CCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CS(=O)(=O)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CS(=O)(=O)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Fc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-n2cccn2)C(F)(F)F)n1
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-n2cccn2)C(F)(F)F)n1
Fc1cnc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2-c2nccs2)C(F)(F)F)nc1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2nccs2)C(F)(F)F)nc1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)-c1nccs1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)-c1nccs1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(c1)-c1nccs1 |r|
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2-c2nccs2)C(F)(F)F)n1 |r|
CC(C)Oc1ccc(cn1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
CC(C)Oc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
CC(C)Oc1ccc(cn1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CC(C)Oc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CCOc1ccc(cn1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CCOc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CCOc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(Cl)c1 |r|
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2Cl)C(F)(F)F)nc1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(Cl)c1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(Cl)c1 |r|
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2Cl)C(F)(F)F)n1 |r|
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)C1CCOCC1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)C1CCOCC1
Fc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2N2CCCC2=O)C(F)(F)F)n1
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCCC2=O)C(F)(F)F)n1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCCC2=O)C(F)(F)F)nc1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCCC1=O |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)N1CCCC1=O |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(c1)N1CCCC1=O |r|
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCOCC1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCOCC1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCOCC2)C(F)(F)F)nc1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)N1CCOCC1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(c1)N1CCOCC1 |r|
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCOCC2)C(F)(F)F)n1 |r|
COCCOc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
COCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
COCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
COCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
COCCCOc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
COCCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
COCCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
COCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
COCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
COCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
COCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
COCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
COCCCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
COCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
COCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
COCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
COCCCCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
COCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
COCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
COCCCCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
COCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
FCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
FCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
FCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
FCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
FCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
FCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
FCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
FCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
FCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
FCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
FCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
FCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
FCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
FCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
FCCCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(OC2CCOCC2)c1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(OC2CCOCC2)c1
Fc1cnc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2OC2CCOCC2)C(F)(F)F)nc1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2OC2CCOCC2)C(F)(F)F)nc1
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(OC2CCOCC2)c1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(OC2CCOCC2)c1
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(OC2CCOCC2)c1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(OC2CCOCC2)c1
Fc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2OC2CCOCC2)C(F)(F)F)n1
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2OC2CCOCC2)C(F)(F)F)n1
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(O[C@H]2CCOC2)c1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(O[C@H]2CCOC2)c1
Fc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2O[C@H]2CCOC2)C(F)(F)F)n1
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2O[C@H]2CCOC2)C(F)(F)F)n1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2O[C@H]2CCOC2)C(F)(F)F)nc1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(O[C@H]2CCOC2)c1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(O[C@H]2CCOC2)c1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(O[C@@H]2CCOC2)c1
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(O[C@@H]2CCOC2)c1
OC(=O)c1ccc(cc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
OC(=O)c1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
OC(=O)c1ccc(cc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
OC(=O)c1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
OC(=O)c1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
OC(=O)c1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
Fc1ccc(nc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Fc1ccc(nc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Fc1ccc(nc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Fc1ccc(nc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Fc1ccc(nc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Fc1ccc(nc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Fc1ccc(nc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
Fc1ccc(nc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
Cc1ccc(cn1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
Cc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
Cc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
Cc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
Cc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
Cc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCOC1=O |r|
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCOC2=O)C(F)(F)F)nc1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(c1)N1CCOC1=O |r|
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCOC2=O)C(F)(F)F)n1 |r|
FC(F)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
FC(F)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
FC(F)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
FC(F)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
FC(F)CCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(OC2COC2)c1
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(OC2COC2)c1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2OC2COC2)C(F)(F)F)nc1 |r|
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2OC2COC2)C(F)(F)F)n1 |r|
FCCCOc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
FCCCOc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Cc1nc(ccc1F)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
Cc1nc(ccc1F)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F |r|
Cc1nc(ccc1F)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
Cc1nc(ccc1F)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
COc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCOCC1=O
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCOCC1=O
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCS(=O)(=O)CC1
Fc1cnc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCS(=O)(=O)CC2)C(F)(F)F)nc1 |r|
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2N2CCS(=O)(=O)CC2)C(F)(F)F)n1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(c1)N1CCS(=O)(=O)CC1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)N1CCS(=O)(=O)CC1 |r|
CCCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
CCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
CCCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
CCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
Fc1cccc(NS(=O)(=O)c2ccc3[C@@H](CCOc3c2)c2ccc(cc2OC2CCOCC2)C(F)(F)F)n1 |r|
Fc1cccc(NS(=O)(=O)c2ccc3[C@H](CCOc3c2)c2ccc(cc2OC2CCOCC2)C(F)(F)F)n1 |r|
CCCc1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
CCCc1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F
FC(F)(F)Oc1ccc(Oc2ccc(cc2)-c2nc(N[C@H]3CCNC3=O)nc(n2)C#N)cc1 |r|
NC(=O)c1nc(N[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1 |r|
FC(F)(F)c1ccc(Oc2ccc(cc2)-c2nc(N[C@H]3CCNC3=O)nc(n2)C#N)nc1 |r|
CCN(C(C)C)c1nc(nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)C(N)=O
CCN(C(C)C)c1nc(nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1)C(N)=O
NC(=O)c1nc(N[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1 |r|
FC(F)(F)Oc1ccc(Oc2ccc(cc2)-c2nc(nc(n2)N2CCOCC2)C#N)cc1
FC(F)(F)c1ccc(Oc2ccc(cc2)-c2nc(nc(n2)N2CCOCC2)C#N)nc1
NC(=O)c1nc(nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)N1CCOCC1
NC(=O)c1nc(nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1)N1CCOCC1
NC(=O)c1nc(N)nc(n1)N1CC(C1)Oc1ccc(cn1)C(F)(F)F
NC(=O)c1nc(NCCO)nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1
NC(=O)c1nc(N)nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1
NC(=O)c1nc(N[C@H]2CCNC2=O)nc(n1)N1CC(C1)Oc1ccc(cn1)C(F)(F)F |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2-c2ccncc2)C#N)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2-c2cccnc2)C#N)cc1
Cn1cccc1-c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C#N
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2-c2ccc(N)cc2)C#N)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2-c2ccsc2)C#N)cc1
COc1ccc(cn1)-c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C#N
Cn1cc(cn1)-c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C#N
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C#N
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2-c2ccc(O)nc2)C#N)cc1
COc1ncccc1-c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C#N
COc1cncc(c1)-c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C#N
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(C#N)c(c2)-c2ccncc2)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(C#N)c(c2)-c2cccnc2)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2-c2ccncc2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2-c2cccnc2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCCC2)C(F)(F)F)cc1
CN(C)CCNCc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CNCCc2ccc(cc2)S(N)(=O)=O)C(F)(F)F)cc1
CN1CCN(Cc2cc(ccc2Oc2ccc(cc2)-c2cccc(n2)C(N)=O)C(F)(F)F)CC1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CNCCN2CCNC2=O)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCNC(=O)C2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CC[C@H](O)C2)C(F)(F)F)cc1 |r|
CN(C)CCN(C)Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CN(C)CCCNCc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CN(C)Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CNCCO)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCC[C@H]2CO)C(F)(F)F)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCC[C@@H]2CO)C(F)(F)F)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCOCC2)C(F)(F)F)cc1
NC(=O)[C@@H]1CCCN1Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCC(F)(F)C2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN[C@H]2CCNC2=O)C(F)(F)F)cc1 |r|
CC(C)(C)OC(=O)NC1CCN(Cc2cc(ccc2Oc2ccc(cc2)-c2cccc(n2)C(N)=O)C(F)(F)F)C1
CC(C)(C)OC(=O)N1CCC(C1)NCc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCCCC2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCC2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCCC(O)C2)C(F)(F)F)cc1
CN(CCO)Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(c(CN3CCC3)c2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(c(CN3CC[C@H](O)C3)c2)C(F)(F)F)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(c(CNCCC(F)(F)F)c2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(c(CN3CCCC3)c2)C(F)(F)F)cc1
CC(N1CCCC1)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2cccc(CN3CCCC3)n2)cc1
NC1CCN(Cc2cc(ccc2Oc2ccc(cc2)-c2cccc(n2)C(N)=O)C(F)(F)F)C1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CNC2CCNC2)C(F)(F)F)cc1
NC1CN(Cc2cc(Oc3ccc(cc3)-c3cccc(n3)C(N)=O)ccc2C(F)(F)F)C1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(O)C[N+]([O-])=O)C(F)(F)F)cc1
NCC(O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NCc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCNC(=O)C2)C(F)(F)F)cc1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CC[C@H](O)C2)C(F)(F)F)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2[C@@H](O)CO)C(F)(F)F)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(O)CN2CCNC(=O)C2)C(F)(F)F)cc1
NC(=O)C(N1CCCC1)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)C(N1CCCCC1)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CCCNC(C(N)=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CN(C)C(C(N)=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CCN(CC)C(C(N)=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1Cl
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(Cl)c1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(c1)C#N
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(c1)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1C(F)(F)F
CN(c1ccccc1)c1cc(ccc1Oc1ccc(F)cc1)-c1cccc(n1)C(N)=O
CN(Cc1cc(ccc1Oc1ccc(F)cc1)-c1cccc(n1)C(N)=O)c1ccc(cc1)C(O)=O
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(COc2ccc(Cl)cc2I)c1
CCN(CC)Cc1cc(ccc1Oc1ccc(F)cc1)-c1cccc(n1)C(N)=O
CCOCc1cc(ccc1Oc1ccc(F)cc1)-c1cccc(n1)C(N)=O
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(CN2CCCC2)c1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(CN2CCOCC2)c1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(c1)-c1ccc(Cl)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(c1)-c1nn[nH]n1
CN(Cc1cc(ccc1Oc1ccc(F)cc1)-c1cccc(n1)C(N)=O)c1ccccc1
COCc1cc(ccc1Oc1ccc(F)cc1)-c1cccc(n1)C(N)=O
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(COc2ccc(F)cc2)c1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)c(COc2ccc(cc2)C#N)c1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(c(CN3CCNC(=O)C3)c2)C(F)(F)F)cc1
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CN2CCCCC2)C(F)(F)F)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CNC2CCCC2)C(F)(F)F)cc1
CCN(CC)S(=O)(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(N2CCCC2)C(=O)N2CCCC2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(N2CCNC(=O)C2)C(=O)N2CCCC2)C(F)(F)F)cc1
CCN(CC)S(=O)(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2CNc2nccs2)C(F)(F)F)cc1
OC[C@H](O)c1ccnc(n1)-c1ccc(Oc2ccc(cc2CN2CCCC2)C(F)(F)F)cc1 |r|
OC[C@@H](O)c1ccnc(n1)-c1ccc(Oc2ccc(cc2CN2CCCC2)C(F)(F)F)cc1 |r|
CCN(C)Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CCN(CC)Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CCN(CCO)Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CCN(CCN(C)C)Cc1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)C1CCCN(Cc2cc(ccc2Oc2ccc(cc2)-c2cccc(n2)C(N)=O)C(F)(F)F)C1
COC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(O)C#N)C(F)(F)F)cc1
NC(C#N)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2\C=C2/SC(=O)NC2=O)C(F)(F)F)cc1
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2C(O)C(F)(F)F)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(=O)C(=O)N2CCCC2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(O)C(=O)N2CCCC2)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(O)=O)C(F)(F)F)cc1
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(=O)N2CCCC2)C(F)(F)F)cc1
CN(CCO)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CN1CCN(CC1)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CNC(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CCN(CC)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(=O)N2CCNC(=O)C2)C(F)(F)F)cc1
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1)-c1nc(cc(n1)C(N)=O)[C@H](O)CO)C(F)(F)F |r|
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)C(N)=O)C(F)(F)F
CCN(CC)Cc1cc(ccc1Oc1ccc(cc1)-c1nc(CCOC(C)=O)cc(n1)C(N)=O)C(F)(F)F
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1)-c1nccc(n1)C(N)=O)C(F)(F)F
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1)-c1nc(N[C@H]2CCNC2=O)cc(n1)C(N)=O)C(F)(F)F |r|
NC(=O)c1cc(CCn2ccnc2)nc(n1)-c1ccc(Oc2ccc(cc2CN2CCOCC2)C(F)(F)F)cc1
CN(C)c1ncc(cn1)-c1cc(ccc1Oc1ccc(cc1)-c1nc(N[C@H]2CCNC2=O)cc(n1)C(N)=O)C(F)(F)F |r|
CN(C)c1cnc(cn1)-c1cc(ccc1Oc1ccc(cc1)-c1nc(N[C@H]2CCNC2=O)cc(n1)C(N)=O)C(F)(F)F |r|
CCN(CC)Cc1cc(ccc1Oc1ccc(cc1)-c1nc(cc(n1)C(N)=O)[C@H](O)CO)C(F)(F)F |r|
CCN(CC)Cc1cc(ccc1Oc1ccc(cc1)-c1nc(cc(n1)C(O)=O)C(N)=O)C(F)(F)F
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2CN2CCOCC2)C(F)(F)F)cc1)C(O)=O
CCN(CC)Cc1cc(ccc1Oc1ccc(cc1)-c1nc(cc(n1)C(N)=O)[C@@H](O)CO)C(F)(F)F |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(cc2-c2cnc(cn2)N(C)C)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1)-c1cc(cc(n1)C(N)=O)[C@H](O)CO)C(F)(F)F |r|
NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(Cl)cc2-c2ccnn2C2CNC2)cc1)[C@H](O)CO |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)-c1ccc(Oc2ccc(Cl)cc2-c2ccnn2C2CNC2)cc1 |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(cc2-c2ccnn2C)C(F)(F)F)cc1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccccc2-c2ccnn2C)cc1)C(N)=O)C(N)=O |r|
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1)-c1nc(N[C@H]2CCNC2=O)cc(n1)C(N)=O |r|
OC[C@H](O)CNC(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
CCN(CC)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
CCN(C)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(=O)N2CC[C@H](O)C2)C(F)(F)F)cc1 |r|
CCN(CCO)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
CCN(CCN(C)C)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
NC(=O)C1CCCN(C1)C(=O)c1cc(ccc1Oc1ccc(cc1)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(=O)Nc2nncs2)C(F)(F)F)cc1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(=O)Nc2nccs2)C(F)(F)F)cc1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc(Oc2ccc(cc2C(=O)NCc2nnn[nH]2)C(F)(F)F)cc1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCCC2)cc1F
Fc1cc(OCC2CCCCC2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(OCC2CCCCC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CC(C)(C)OC(=O)N1CCCC(COc2cc(F)c(cc2F)C(=O)NS(C)(=O)=O)C1
CS(=O)(=O)NC(=O)c1cc(F)c(OCCC2CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(F)c(OCC2CCCNC2)cc1F
CS(=O)(=O)NC(=O)c1cc(F)c(OCC2CCCO2)cc1F
CC(C)(C)OC(=O)N1CCC(CCOc2cc(F)c(cc2F)C(=O)NS(C)(=O)=O)CC1
CC1(C)C2CCC1(C)C(C2)Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O |TLB:10:8:1:5.4|
CS(=O)(=O)NC(=O)c1ccc(CNC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:22:13:20:16.17.18,12:13:16:20.19.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:22:13:20:16.17.18,12:13:16:20.19.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(O)(C4)C2)C3)c(Cl)c1 |TLB:23:13:21:18.17.16,THB:14:13:18:21.15.16,14:15:18:13.23.22,23:17:21:13.14.22,12:13:21:18.17.16|
CC1(C)C(COc2cc(F)c(cc2Cl)C(=O)NS(C)(=O)=O)C1(C)C
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCCC2CCCC2)cc1F
CN(Cc1ccc(cc1Cl)C(=O)NS(C)(=O)=O)C12CC3CC(CC(C3)C1)C2 |TLB:26:17:24:20.21.22,1:17:20:24.23.22,THB:26:21:24:17.25.18,25:17:20:24.23.22,25:23:20:17.26.18|
CN(C(=O)c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)C12CC3CC(CC(C3)C1)C2 |TLB:1:19:22:26.25.24,28:19:26:22.23.24,THB:28:23:26:19.27.20,27:19:22:26.25.24,27:25:22:19.28.20|
COC12CC3CC(CC(COc4cc(F)c(cc4Cl)C(=O)NS(C)(=O)=O)(C3)C1)C2 |TLB:26:8:28:3.4.5,26:4:28:8.7.27,THB:9:8:28:3.4.5,7:8:3:28.6.5,7:6:3:8.26.27|
CCCCCC12CCC(COc3cc(F)c(cc3Cl)C(=O)NS(C)(=O)=O)(CC1)CC2
CS(=O)(=O)NC(=O)c1cc(Cl)c(O[C@H]2C3CC4CC2CC(Cl)(C4)C3)cc1F |r,TLB:12:13:17:22.20.19,13:14:22:17.18.19,23:20:17:14.13.15,THB:13:18:22:14.23.15,23:14:17:22.20.19|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCCCCC2)cc1F
CS(=O)(=O)NC(=O)c1cnc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C1CC1 |TLB:22:13:20:16.17.18,THB:12:13:20:16.17.18,22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(COC2C3CC4CC(C3)CC2C4)cc1F |TLB:15:16:18:20.21.22,THB:16:24:20:18.17.22,16:17:20:24.23.25,23:24:18:20.21.22,23:21:18:24.16.25,(6.49,-1.89,;6.89,-.4,;8.38,-.8,;7.29,1.08,;5.4,-.01,;4.31,-1.09,;4.71,-2.58,;2.83,-.7,;1.74,-1.78,;.25,-1.39,;-.84,-2.48,;-2.33,-2.87,;-1.24,-3.96,;-.15,.1,;-1.64,.5,;-2.04,1.99,;-3.52,2.39,;-4.14,3.79,;-5.67,3.96,;-6.58,2.72,;-8.38,1.68,;-6.87,1.38,;-5.44,3.3,;-6.3,.12,;-4.44,1.15,;-5.96,1.31,;.94,1.19,;2.43,.79,;3.52,1.88,)|
CCc1cc(C(=O)NS(C)(=O)=O)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:27:18:25:21.22.23,THB:17:18:25:21.22.23,27:22:25:18.26.19,26:18:21:25.24.23,26:24:21:18.27.19|
CCc1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:30:21:28:24.25.26,THB:20:21:28:24.25.26,30:25:28:21.29.22,29:21:24:28.27.26,29:27:24:21.30.22|
OC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:29:20:27:23.24.25,THB:19:20:27:23.24.25,29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.29.21|
OCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:27:18:25:21.22.23,THB:17:18:25:21.22.23,27:22:25:18.26.19,26:18:21:25.24.23,26:24:21:18.27.19|
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:28:19:26:22.23.24,THB:18:19:26:22.23.24,28:23:26:19.27.20,27:19:22:26.25.24,27:25:22:19.28.20|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCC3(CC3)CC2)cc1F
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C1CCC1 |TLB:12:13:16:20.19.18,22:13:20:16.17.18,THB:22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)NC(=O)c1cc(Cl)c(COC2C3CC4CC(C3)CC2C4)cc1F |TLB:13:14:16:18.19.20,THB:14:22:18:16.15.20,14:15:18:22.21.23,21:22:16:18.19.20,21:19:16:22.14.23,(6.49,-2.58,;6.89,-1.09,;8.38,-1.49,;7.29,.39,;5.4,-.7,;4.31,-1.78,;4.71,-3.27,;2.83,-1.39,;1.74,-2.48,;.25,-2.08,;-.84,-3.17,;-.15,-.59,;-1.64,-.19,;-2.04,1.3,;-3.52,1.7,;-4.14,3.1,;-5.67,3.27,;-6.58,2.03,;-8.38,.99,;-6.87,.69,;-5.44,2.61,;-6.3,-.57,;-4.44,.45,;-5.96,.62,;.94,.5,;2.43,.1,;3.52,1.19,)|
FC(F)(F)c1cc(ccc1OCC12CC3CC(CC(C3)C1)C2)C(=O)NS(=O)(=O)N1CCC1 |TLB:21:12:19:15.16.17,THB:11:12:19:15.16.17,21:16:19:12.20.13,20:12:15:19.18.17,20:18:15:12.21.13|
CC1(C)[C@H]2C[C@@H]1[C@H](COc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)CC2 |r|
CS(=O)(=O)NC(=O)c1ccc(OCC2C3CC4CC(C3)CC2C4)c(c1)C1CC1 |TLB:12:13:15:17.18.19,THB:13:21:17:15.14.19,13:14:17:21.20.22,20:21:15:17.18.19,20:18:15:21.13.22,(7.75,1.73,;6.42,2.5,;5.65,3.84,;7.19,3.84,;5.08,1.73,;3.75,2.5,;3.75,4.04,;2.41,1.73,;1.08,2.5,;-.25,1.73,;-.25,.19,;-1.59,-.58,;-2.92,.19,;-4.25,-.58,;-5.58,.19,;-6.92,-.58,;-6.92,-2.12,;-7.75,-4.02,;-6.35,-3.37,;-6.34,-.97,;-5.15,-4.04,;-4.25,-2.12,;-5.58,-2.89,;1.08,-.58,;2.41,.19,;1.08,-2.12,;.31,-3.45,;1.85,-3.45,)|
COc1cc(OCC23CC4CC(CC(C4)C2)C3)c(Cl)cc1C(=O)NS(C)(=O)=O |TLB:16:7:14:10.11.12,6:7:10:14.13.12,6:7:14:10.11.12,THB:16:11:14:7.15.8,15:7:10:14.13.12,15:13:10:7.16.8|
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3CCC(C)(C)Cc3c2)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3CC(C)(C)CCc3c2)cc1F
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)c(Br)c1 |TLB:22:13:20:16.17.18,THB:12:13:20:16.17.18,22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C(F)(F)F |TLB:22:13:20:16.17.18,THB:12:13:20:16.17.18,22:17:20:13.21.14,21:13:16:20.19.18,21:19:16:13.22.14|
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3OC(C)(C)CCc3c2)cc1F
CNS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3CCC(C)(C)Oc3c2)cc1F
OCCS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:25:16:23:19.20.21,THB:15:16:23:19.20.21,25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1Cl |TLB:23:14:21:17.18.19,THB:13:14:21:17.18.19,23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15|
Cn1cnc(c1)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:28:19:26:22.23.24,THB:28:23:26:19.27.20,18:19:26:22.23.24,27:19:22:26.25.24,27:25:22:19.28.20|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(Cl)cc1C(=O)NS(=O)(=O)c1c[nH]cn1 |TLB:5:6:9:13.12.11,15:6:13:9.10.11,THB:15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(Cl)cc1C(=O)NS(=O)(=O)N1CCOCC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
Cc1nnn(n1)C12CC3CC(CC(COc4cc(F)c(cc4Cl)C(=O)NS(C)(=O)=O)(C3)C1)C2 |TLB:30:12:32:7.8.9,30:8:32:12.11.31,THB:13:12:32:7.8.9,11:12:7:32.10.9,11:10:7:12.30.31|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3CCC(C)(C)Oc3c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3CC(C)(C)CCc3c2)cc1F
CCCCCC12CCC(COc3cc(F)c(cc3Cl)C(=O)NS(=O)(=O)N(C)C)(CC1)CC2
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(Cl)(C4)C2)C3)cc1F |TLB:26:16:24:21.20.19,THB:15:16:24:21.20.19,17:16:21:24.18.19,17:18:21:16.26.25,26:20:24:16.17.25|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2(F)CCCCC2)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2(CCC2)C(F)(F)F)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3CCC(C)(C)Cc3c2)cc1F
CN(C)S(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C1CC1 |TLB:14:15:18:22.21.20,24:15:22:18.19.20,THB:23:15:18:22.21.20,23:21:18:15.24.16,24:19:22:15.23.16|
CS(=O)(=O)NC(=O)c1cc(Cl)c(COC23CC4CC(CC(C4)C2)C3)cc1F |TLB:13:14:17:21.20.19,23:14:21:17.18.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCC3(CCC3)CC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCC3(CC3)CC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(F)(C4)C2)C3)cc1F |TLB:26:16:24:19.20.21,THB:15:16:24:19.20.21,15:16:19:24.22.21,25:16:19:24.22.21,25:22:19:16.26.17,26:20:24:16.25.17|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC[C@H]2C[C@@H]3CC[C@H](C2)N3CC(F)(F)F)cc1F |r,THB:22:21:14.15.20:17.18|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(C2)C(F)(F)C(C4)C3)cc1F |TLB:15:16:22:19.18.26,THB:17:16:22:19.18.26,17:18:22:16.27.21,27:16:19:22.25.26,27:25:19:16.17.21|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC[C@H]2CC[C@H](CC2)C(F)(F)F)cc1F |r,wU:14.13,17.20,(8.67,3.36,;7.34,2.59,;6.57,3.93,;8.11,1.26,;6,1.82,;4.67,2.59,;4.67,4.13,;3.33,1.82,;3.33,.28,;2,-.49,;2,-2.03,;.67,.28,;-.67,-.49,;-2,.28,;-3.33,-.49,;-3.33,-2.03,;-4.67,-2.8,;-6,-2.03,;-6,-.49,;-4.67,.28,;-7.34,-2.8,;-8.67,-3.57,;-8.11,-1.46,;-6.57,-4.13,;.67,1.82,;2,2.59,;2,4.13,)|
CC1(C)[C@@H]2C[C@H]1[C@@H](COc1cc(F)c(cc1Cl)C(=O)NS(N)(=O)=O)CC2 |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCC3(CCC3)CC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC[C@@H]2CC[C@H]3C[C@@H]2C3(C)C)cc1F |r|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CC3CCC2C3)cc1F |THB:15:16:19.20:22|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCC(F)(F)CC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCCCCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCCCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCCC2)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2(CC2)C(F)(F)F)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(Cl)(C4)C2)C3)cc1F |TLB:24:14:22:17.18.19,THB:13:14:22:17.18.19,24:18:22:14.23.15,23:14:17:22.20.19,23:20:17:14.24.15,21:20:17:14.24.15|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCCC2)cc1F
CC1(C)[C@@H]2C[C@H]1[C@H](COc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)CC2 |r|
COc1ncccc1-c1cc(ccc1OCC12CC3CC(CC(C3)C1)C2)C(=O)NS(C)(=O)=O |TLB:15:16:19:23.22.21,25:16:23:19.20.21,THB:25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2C3CC4CC(C3)CC2C4)cc1F |TLB:13:14:16:18.19.20,THB:14:22:18:16.15.20,14:15:18:22.21.23,21:22:16:18.19.20,21:19:16:22.14.23,(7.75,1.73,;6.42,2.5,;5.65,3.84,;7.19,3.84,;5.08,1.73,;3.75,2.5,;3.75,4.04,;2.41,1.73,;2.41,.19,;1.08,-.58,;1.08,-2.12,;-.25,.19,;-1.59,-.58,;-2.92,.19,;-4.25,-.58,;-5.58,.19,;-6.92,-.58,;-6.92,-2.12,;-7.75,-4.02,;-6.35,-3.37,;-6.34,-.97,;-5.15,-4.04,;-4.25,-2.12,;-5.58,-2.89,;-.25,1.73,;1.08,2.5,;1.08,4.04,)|
CS(=O)(=O)NC(=O)c1cc(Cl)c(COc2ccc3CCCCc3c2)cc1F
CC1(C)C(COc2ccc(cc2Cl)C(=O)NS(C)(=O)=O)C1(C)C
CC1(C)[C@@H]2C[C@H]1C(COc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)=CC2 |r,c:25|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CC3CCC2C3)cc1F |THB:13:14:17.18:20|
CS(=O)(=O)NC(=O)c1cc(Cl)c(O[C@@H]2C[C@@H]3CC[C@H]2C3)cc1F |r|
CC1(C)[C@H]2CC[C@](C)(C2)[C@H]1Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O |r|
CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC2CC3CCC2C3)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC2CC3CC2C2CCCC32)cc1F |THB:12:13:16:22.18,21:22:13.14:16,19:18:13.14:16|
CC(C)[C@H]1CC[C@@H](CC1)Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O |r,wU:6.9,wD:3.2,(-8,.77,;-6.67,1.54,;-6.67,3.08,;-5.33,.77,;-5.33,-.77,;-4,-1.54,;-2.67,-.77,;-2.67,.77,;-4,1.54,;-1.33,-1.54,;,-.77,;,.77,;1.33,1.54,;1.33,3.08,;2.67,.77,;2.67,-.77,;1.33,-1.54,;1.33,-3.08,;4,1.54,;4,3.08,;5.33,.77,;6.67,1.54,;8,2.31,;5.9,2.87,;7.44,.21,)|
CC1(C)CCCC(C1)Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CC1(C)CCC(CC1)Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC2CCCCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(O[C@@H]2C[C@@H]3CC[C@@]2(C)C3(C)C)cc1F |r,TLB:14:15:18.19:22|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCC2CCCCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC2C3CC4CC2CC(Cl)(C4)C3)cc1F |TLB:14:15:17:24.22.25,15:16:24:20.21.19,THB:15:20:24:17.16.25,21:20:17:24.22.25,21:22:17:20.15.19|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCC2CCCC2)cc1F
CC(C)[C@H]1CC[C@@H](CC1)Oc1cc(F)c(cc1Cl)C(=O)NS(=O)(=O)N(C)C |r,wU:6.9,wD:3.2,(-3.16,-5.78,;-4.49,-5,;-5.82,-5.78,;-4.49,-3.47,;-3.16,-2.69,;-3.16,-1.15,;-4.49,-.38,;-5.82,-1.15,;-5.82,-2.69,;-4.49,1.15,;-3.16,1.93,;-3.16,3.46,;-1.82,4.23,;-1.82,5.78,;-.49,3.47,;-.49,1.92,;-1.82,1.15,;-1.82,-.38,;.85,4.23,;.85,5.78,;2.18,3.47,;3.51,4.23,;2.74,5.57,;4.85,5,;4.28,2.9,;3.51,1.57,;5.82,2.9,)|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC2C3CC4CC2CC(Cl)(C4)C3)cc1F |TLB:14:15:17:24.22.25,15:16:24:20.21.19,THB:15:20:24:17.16.25,21:20:17:24.22.25,21:22:17:20.15.19|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC2CCC3(CCCC3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(OC2CCC3(CCCCC3)CC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCC2CCCCCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCCC2CCCCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC2CCC(CC2)C(F)(F)F)cc1F |(5.57,-1.54,;6.34,-.21,;7.88,-.21,;5.57,1.13,;4.8,2.46,;6.9,1.9,;4.23,.36,;2.9,1.13,;2.9,2.67,;1.57,.36,;1.57,-1.18,;.23,-1.95,;.23,-3.49,;-1.1,-1.18,;-2.43,-1.95,;-3.52,-.86,;-3.12,.62,;-4.21,1.71,;-5.7,1.31,;-6.1,-.17,;-5.01,-1.26,;-6.79,2.4,;-7.88,3.49,;-5.7,3.49,;-7.88,1.31,;-1.1,.36,;.23,1.13,;.23,2.67,)|
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCC2CCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OC2CCC3(CCCC3)CC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCCC2CCCC2)cc1F
CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(OCCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:24:23:26:20.19.18,24:19:26:23.25.22,THB:25:23:20:26.17.18,25:17:20:23.24.22|
O[C@H]1CCN(C1)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |r,TLB:28:19:26:22.23.24,THB:18:19:26:22.23.24,28:23:26:19.27.20,27:19:22:26.25.24,27:25:22:19.28.20|
FC1CN(C1)S(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:27:18:25:21.22.23,THB:17:18:25:21.22.23,27:22:25:18.26.19,26:18:21:25.24.23,26:24:21:18.27.19|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(C2)C(F)(F)C(C4)C3)cc1F |TLB:15:16:22:19.18.26,THB:17:16:22:19.18.26,17:18:22:16.27.21,27:16:19:22.25.26,27:25:19:16.17.21|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CCCC1)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CCOCC1)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(F)(C4)C2)C3)cc1F |TLB:15:16:21:24.18.19,26:16:24:21.20.19,THB:17:16:21:24.18.19,17:18:21:16.26.25,26:20:24:16.17.25|
COC12CC3CC(CC(COc4cc(F)c(cc4C4CC4)C(=O)NS(C)(=O)=O)(C3)C1)C2 |TLB:28:8:30:3.4.5,28:4:30:8.7.29,THB:9:8:30:3.4.5,7:8:3:30.6.5,7:6:3:8.28.29|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC3(CC3)CC2)cc1F
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CC(F)(F)C1)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(F)(C4)C2)C3)cc1F |TLB:12:13:18:21.15.16,23:13:21:18.17.16,THB:14:13:18:21.15.16,14:15:18:13.23.22,23:17:21:13.14.22|
Cc1cc(C(=O)NS(C)(=O)=O)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:26:17:24:20.21.22,THB:16:17:24:20.21.22,26:21:24:17.25.18,25:17:20:24.23.22,25:23:20:17.26.18|
Cc1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:29:20:27:23.24.25,THB:19:20:27:23.24.25,29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.29.21|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:26:17:24:20.21.22,THB:16:17:24:20.21.22,26:21:24:17.25.18,25:17:20:24.23.22,25:23:20:17.26.18|
CC(C)(C)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:28:19:26:22.23.24,THB:18:19:26:22.23.24,28:23:26:19.27.20,27:19:22:26.25.24,27:25:22:19.28.20|
CS(=O)(=O)NC(=O)c1ccc(OCC2CCC3(CC3)CC2)cc1F
COCCNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:29:20:27:23.24.25,THB:19:20:27:23.24.25,29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.29.21|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(CC2)C(F)(F)F)cc1F
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OC1(COC1)c1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:23:24:27:31.30.29,33:24:31:27.28.29,THB:33:28:31:24.32.25,32:24:27:31.30.29,32:30:27:24.33.25|
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CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4(F)CC(F)(CC(F)(C4)C2)C3)cc1F |TLB:26:14:24:21.19.18,THB:26:19:24:14.15.25,13:14:24:21.19.18,15:14:21:24.16.18,15:16:21:14.26.25,17:16:21:14.26.25|
CS(=O)(=O)NC(=O)c1cnc(OCC23CC4(F)CC(F)(CC(F)(C4)C2)C3)c(Cl)c1 |TLB:25:13:23:20.18.17,THB:25:18:23:13.14.24,12:13:23:20.18.17,14:13:20:23.15.17,14:15:20:13.25.24,16:15:20:13.25.24|
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCCC2)cc1F
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCCC2)cc1F
COCCS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2(C#N)C3CC4CC(C3)CC2C4)cc1F |TLB:18:17:21:23.24.25,16:17:21:23.24.25,THB:26:27:21:23.24.25,26:24:21:27.28.17,17:27:23:21.20.25,17:20:23:27.26.28|
CNS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2(C#N)C3CC4CC(C3)CC2C4)cc1F |TLB:16:15:19:21.22.23,14:15:19:21.22.23,THB:24:25:19:21.22.23,24:22:19:25.26.15,15:25:21:19.18.23,15:18:21:25.24.26|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2(C#N)C3CC4CC(C3)CC2C4)cc1F |TLB:15:14:18:20.21.22,13:14:18:20.21.22,THB:23:24:18:20.21.22,23:21:18:24.25.14,14:24:20:18.17.22,14:17:20:24.23.25|
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Fc1cc(OCC2C3CC4CC(C3)CC2C4)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:5:6:8:10.11.12,THB:13:14:8:10.11.12,13:11:8:14.15.6,6:14:10:8.7.12,6:7:10:14.13.15,(.14,4.04,;.14,2.5,;-1.2,1.73,;-1.2,.19,;-2.53,-.58,;-3.86,.19,;-5.2,-.58,;-6.52,.19,;-7.86,-.58,;-7.86,-2.12,;-8.69,-4.02,;-7.3,-3.37,;-7.28,-.97,;-6.09,-4.04,;-5.2,-2.12,;-6.52,-2.89,;.14,-.58,;1.47,.19,;1.47,1.73,;2.81,2.5,;2.81,4.04,;4.14,1.73,;5.47,2.5,;4.7,3.84,;6.24,3.84,;6.81,1.73,;7.2,.25,;8.69,.64,;8.29,2.13,;.14,-2.12,;-.63,-3.45,;.91,-3.45,)|
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OCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCCC2)cc1F
CS(=O)(=O)NC(=O)c1ccc(C(O)C2C3CC4CC(C3)CC2C4)c(Cl)c1 |TLB:11:13:15:17.18.19,THB:13:21:17:15.14.19,13:14:17:21.20.22,20:21:15:17.18.19,20:18:15:21.13.22,(7.08,-2.31,;5.75,-1.54,;5.75,-3.08,;7.08,-.77,;4.42,-.77,;3.08,-1.54,;3.08,-3.08,;1.75,-.77,;.41,-1.54,;-.92,-.77,;-.92,.77,;-2.25,1.54,;-2.25,3.08,;-3.59,.77,;-4.92,1.54,;-6.25,.77,;-6.25,-.77,;-7.08,-2.67,;-5.69,-2.03,;-5.67,.37,;-4.48,-2.7,;-3.59,-.77,;-4.92,-1.54,;.41,1.54,;.41,3.08,;1.75,.77,)|
CS(=O)(=O)NC(=O)c1cc(I)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:23:14:21:17.18.19,13:14:17:21.20.19,THB:23:18:21:22.15.14,22:20:17:23.15.14,22:14:17:21.20.19|
CCOCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:19:20:23:27.26.25,19:20:27:23.24.25,29:20:27:23.24.25,THB:29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.21.29|
COCCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:19:20:23:27.26.25,19:20:27:23.24.25,29:20:27:23.24.25,THB:29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.21.29|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4(F)CC(F)(CC(F)(C4)C2)C3)cc1F |TLB:28:16:26:23.21.20,THB:28:21:26:16.17.27,15:16:26:23.21.20,17:16:23:26.18.20,17:18:23:16.28.27,19:18:23:16.28.27|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)C1CCOCC1)C1CC1 |TLB:5:6:9:13.12.11,5:6:13:9.10.11,15:6:13:9.10.11,THB:14:6:9:13.12.11,14:12:9:6.7.15,15:10:13:6.14.7|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)C1CCOC1)C1CC1 |TLB:15:6:13:9.10.11,5:6:9:13.12.11,5:6:13:9.10.11,THB:14:6:9:13.12.11,14:12:9:6.7.15,15:10:13:6.14.7|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2CC[C@H](CC2)C(F)(F)F)cc1F |r,wU:16.16,19.23,(8.67,-3.36,;7.34,-2.59,;6.57,-3.93,;8.11,-1.26,;6,-1.82,;4.67,-2.59,;4.67,-4.13,;3.33,-1.82,;2,-2.59,;.67,-1.82,;-.67,-2.59,;-2.21,-2.59,;-1.44,-3.93,;.67,-.28,;-.67,.49,;-2,-.28,;-3.33,.49,;-4.67,-.28,;-6,.49,;-6,2.03,;-4.67,2.8,;-3.33,2.03,;-7.34,2.8,;-8.67,3.57,;-6.57,4.13,;-8.11,1.46,;2,.49,;3.33,-.28,;4.67,.49,)|
CC(C)OCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:30:21:28:24.25.26,20:21:24:28.27.26,20:21:28:24.25.26,THB:29:21:24:28.27.26,29:27:24:21.22.30,30:25:28:21.29.22|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:23:14:21:17.18.19,THB:23:18:21:14.22.15,13:14:21:17.18.19,22:14:17:21.20.19,22:20:17:14.23.15|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CC(C1)C#N)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(C#N)C3CC4CC(C3)CC2C4)cc1F |TLB:17:16:20:22.23.24,15:16:20:22.23.24,THB:25:26:20:22.23.24,25:23:20:26.27.16,16:26:22:20.19.24,16:19:22:26.25.27|
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FC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCCC2)cc1F
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)C1CCC1)C1CC1 |TLB:5:6:9:13.12.11,5:6:13:9.10.11,15:6:13:9.10.11,THB:14:6:9:13.12.11,14:12:9:6.7.15,15:10:13:6.14.7|
CNS(=O)(=O)NC(=O)c1cc(Cl)c(O[C@@H]2C[C@@H]3C[C@@H]3C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(O[C@@H]2C[C@@H]3C[C@@H]3C2)cc1F |r|
FC1CN(C1)S(=O)(=O)NC(=O)c1cc(Cl)c(O[C@@H]2C[C@@H]3C[C@@H]3C2)cc1F |r|
CC(O)CS(=O)(=O)NC(=O)c1ccc(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:25:16:23:19.20.21,15:16:19:23.22.21,15:16:23:19.20.21,THB:25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17|
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(C#N)C3CC4CC(C3)CC2C4)cc1F |TLB:18:17:21:23.24.25,16:17:21:23.24.25,THB:26:27:21:23.24.25,26:24:21:27.28.17,17:27:23:21.20.25,17:20:23:27.26.28|
Fc1cc(OCC2CCC(F)(F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(COC23CC4CC(CC(C4)C2)C3)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1 |TLB:15:6:13:9.10.11,THB:15:10:13:14.7.6,14:12:9:15.7.6,14:6:9:13.12.11,5:6:13:9.10.11|
Fc1cc(OCC23CC4(F)CC(F)(CC(F)(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:5:6:13:10.8.16,THB:15:14:10:6.7.18,7:6:13:10.8.16,7:8:13:6.17.18,17:6:10:13.14.16,17:14:10:6.7.18|
FC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(CCCCC2)C(F)(F)F)cc1F
Fc1cc(OCC2(CCCCC2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(I)cc1C(=O)NS(=O)(=O)N1CCC1 |TLB:15:6:13:9.10.11,THB:15:10:13:14.7.6,14:12:9:15.7.6,14:6:9:13.12.11,5:6:13:9.10.11|
Fc1cc(OCC2(C#N)C3CC4CC(C3)CC2C4)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1 |TLB:7:6:10:12.13.14,5:6:10:12.13.14,THB:15:16:10:12.13.14,15:13:10:16.17.6,6:16:12:10.9.14,6:9:12:16.15.17|
Fc1cc(OCC2(C#N)C3CC4CC(C3)CC2C4)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:7:6:10:12.13.14,5:6:10:12.13.14,THB:15:16:10:12.13.14,15:13:10:16.17.6,6:16:12:10.9.14,6:9:12:16.15.17|
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC(F)(F)CC2)cc1F
FC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC(F)(F)CC2)cc1F
CC(=O)c1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:31:22:29:25.26.27,THB:31:26:29:30.23.22,30:28:25:31.23.22,30:22:25:29.28.27,21:22:29:25.26.27|
CC(C)(O)c1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:32:23:30:26.27.28,THB:32:27:30:31.24.23,31:29:26:32.24.23,31:23:26:30.29.28,22:23:30:26.27.28|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CCC2(COC2)CC1)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(CCCCC2)C(F)(F)F)cc1F
Fc1cc(OCC2CCCC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
OCC12CC3CC(C1)CC(COc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1)(C3)C2 |TLB:10:9:3:5.6.7,THB:1:2:5:9.8.32,8:9:3:5.6.7,8:6:3:9.33.32,33:9:5:3.2.7,33:2:5:9.8.32|
Fc1cc(OCC23CC4(F)CC(F)(CC(F)(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |TLB:5:6:10:13.14.16,THB:17:6:10:13.14.16,17:14:10:6.7.18,7:6:13:10.8.16,7:8:13:6.17.18,9:8:13:6.17.18|
Fc1cc(OCC2(CCCC2)C(F)(F)F)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CCCCC1
Fc1cc(OCC23CC4CC(C2)CC(C4)(C3)OC(=O)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:5:6:12:14.8.9,11:6:14:12.10.9,THB:7:6:12:14.8.9,7:8:12:6.11.15,11:10:14:6.7.15|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CC2(COC2)C1)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(CCCCC2)C(F)(F)F)cc1F
CC1(C)CCCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)C1
FCC12CC3CC(C1)CC(COc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1)(C3)C2 |TLB:10:9:3:5.6.7,THB:1:2:5:9.8.32,8:9:3:5.6.7,8:6:3:9.33.32,33:9:5:3.2.7,33:2:5:9.8.32|
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC(F)(F)CC2)cc1F
Fc1cc(OCC2CCCC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCC2)cc1F
COC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCC2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCC(F)(F)CC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CCC(F)(F)CC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCC(F)(F)CC1
FC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(C2)C(F)(F)C(C4)C3)cc1F |TLB:19:20:23:26.29.30,THB:31:20:23:26.29.30,31:29:23:20.21.25,21:20:26:23.22.30,21:22:26:20.31.25|
Fc1cc(OCC2(CCCC2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(C2)C(F)(F)C(C4)C3)cc1F |TLB:18:19:22:25.28.29,THB:30:19:22:25.28.29,30:28:22:19.20.24,20:19:25:22.21.29,20:21:25:19.30.24|
CC(C)(F)c1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:32:23:30:26.27.28,22:23:26:30.29.28,22:23:30:26.27.28,THB:32:27:30:23.31.24,31:23:26:30.29.28,31:29:26:23.32.24|
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(C)CCC(F)(F)CC2)cc1F
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(C)CCC(F)(F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CC3CC3C2)cc1F
Fc1cc(OCC2CC3CC3C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2[C@@H]3CCC[C@H]23)cc1F |r|
OC12CC3CC(C1)CC(COc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1)(C3)C2 |TLB:31:8:6:2.3.4,THB:9:8:6:2.3.4,31:3:6:8.7.32,7:8:2:6.5.4,7:5:2:8.31.32|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CC2(CCO2)C1)C1CC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
Fc1cc(OCC23CC4CC(C2)C(F)(F)C(C4)C3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |TLB:5:6:9:12.15.16,THB:17:6:9:12.15.16,17:15:9:6.7.11,7:6:12:9.8.16,7:8:12:6.17.11|
Fc1cc(OCC2CC3CC3C2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(OCC2CC3CC3C2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Fc1cc(OCC23CC2CCCC3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
O=C(NS(=O)(=O)N1CCC1)c1cnc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C1CC1 |TLB:25:16:23:19.20.21,THB:25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17,15:16:23:19.20.21|
COCCS(=O)(=O)NC(=O)c1cnc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C1CC1 |TLB:25:16:23:19.20.21,THB:25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17,15:16:23:19.20.21|
Fc1cc(OCC2(F)CCCCC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(O[C@H]2C3CC4CC2C[C@](Cl)(C4)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r,wU:5.4,wD:12.13,TLB:5:6:14:11.10.9,4:5:11:14.8.9,THB:5:10:14:6.7.15,7:6:11:14.8.9,7:8:11:6.5.15,(2.54,2.48,;1.21,1.71,;-.13,2.48,;-1.46,1.71,;-2.79,2.48,;-4.28,2.09,;-4.28,.55,;-5.18,-1.38,;-6.38,-.71,;-6.36,1.69,;-5.61,2.85,;-6.94,2.09,;-6.94,.55,;-8.43,.15,;-7.78,-1.36,;-5.61,-.23,;-1.46,.17,;-.13,-.6,;1.21,.17,;2.54,-.6,;2.54,-2.14,;3.88,.17,;5.21,-.6,;4.44,-1.93,;5.98,.74,;6.54,-1.37,;6.94,-2.85,;8.43,-2.46,;8.03,-.97,;-2.79,-.6,;-4.33,-.6,;-3.56,-1.93,)|
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC2CCCC3)cc1F
OC1CCN(CC1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:31:22:29:25.26.27,THB:21:22:29:25.26.27,31:26:29:22.30.23,30:22:25:29.28.27,30:28:25:22.31.23|
Fc1cc(OCC2CCC3(CC3)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CS(=O)(=O)NC(=O)c1ccc(OC[C@H]2CC[C@@H](CC2)C(F)(F)F)cc1F |r,wU:16.19,wD:13.12,(8.67,-3.36,;7.34,-2.59,;6.57,-3.93,;8.11,-1.26,;6,-1.82,;4.67,-2.59,;4.67,-4.13,;3.33,-1.82,;2,-2.59,;.67,-1.82,;.67,-.28,;-.67,.49,;-2,-.28,;-3.33,.49,;-3.33,2.03,;-4.67,2.8,;-6,2.03,;-6,.49,;-4.67,-.28,;-7.34,2.8,;-8.67,3.57,;-6.57,4.13,;-8.11,1.46,;2,.49,;3.33,-.28,;4.67,.49,)|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2CC[C@@H](CC2)C(F)(F)F)cc1F |r,wU:19.23,wD:16.16,(8.67,-3.36,;7.34,-2.59,;6.57,-3.93,;8.11,-1.26,;6,-1.82,;4.67,-2.59,;4.67,-4.13,;3.33,-1.82,;2,-2.59,;.67,-1.82,;-.67,-2.59,;-2.21,-2.59,;-1.44,-3.93,;.67,-.28,;-.67,.49,;-2,-.28,;-3.33,.49,;-3.33,2.03,;-4.67,2.8,;-6,2.03,;-6,.49,;-4.67,-.28,;-7.34,2.8,;-8.67,3.57,;-6.57,4.13,;-8.11,1.46,;2,.49,;3.33,-.28,;4.67,.49,)|
Fc1cc(OCC2CCC3(CC3)CC2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CC(F)C2)CCC(F)(F)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC2CCC(CC2)C(F)(F)F)cc1F |(8.72,-.56,;7.18,-.56,;7.18,.98,;7.18,-2.1,;5.64,-.56,;4.87,.77,;5.64,2.1,;3.33,.77,;2.56,-.56,;1.02,-.56,;.25,-1.9,;-1.08,-2.67,;.25,-3.44,;.25,.77,;-1.29,.77,;-2.77,.37,;-3.86,1.46,;-5.35,1.06,;-5.75,-.43,;-4.66,-1.51,;-3.17,-1.12,;-7.24,-.82,;-8.33,.26,;-7.63,-2.31,;-8.72,-1.22,;1.02,2.1,;2.56,2.1,;3.33,3.44,)|
Fc1cc(OC2CCC(Cl)=CC2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1 |c:9|
Fc1cc(OC2CCC(Cl)(Cl)CC2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
CCC1=CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1 |t:2|
Fc1cc(O[C@@H]2C[C@@H]3CC[C@H]2C3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(O[C@@H]2C[C@@H]3CC[C@H]2C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2C[C@@H]3CC[C@H]2C3)cc1F |r|
CO[C@@H]1CCN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |r,TLB:31:22:29:25.26.27,THB:21:22:29:25.26.27,31:26:29:22.30.23,30:22:25:29.28.27,30:28:25:22.31.23|
Fc1cc(OCCC2CCC(F)(F)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(O[C@H]2C[C@@H]3CC[C@H]2C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@H]2C[C@@H]3CC[C@H]2C3)cc1F |r|
CC1(CCC(F)(F)CC1)OCc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(F)c(OCC23CC4CC(CC(C4)C2)C3)c(Cl)c1F |TLB:13:14:17:21.20.19,23:14:21:17.18.19,THB:22:14:17:21.20.19,22:20:17:14.23.15,23:18:21:14.22.15|
Fc1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)c(Cl)c1OCC12CC3CC(CC(C3)C1)C2 |TLB:20:21:24:28.27.26,30:21:28:24.25.26,THB:29:21:24:28.27.26,29:27:24:21.30.22,30:25:28:21.29.22|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@H]2C3CC4CC2C[C@](F)(C4)C3)cc1F |r,wU:15.15,wD:22.24,TLB:15:16:24:21.20.19,14:15:21:24.18.19,THB:15:20:24:16.17.25,17:16:21:24.18.19,17:18:21:16.15.25,(7.33,-1.44,;6,-2.21,;5.23,-3.54,;6.77,-3.54,;4.66,-1.44,;3.33,-2.21,;3.33,-3.75,;2,-1.44,;2,.1,;.66,.87,;.66,2.41,;-.11,3.75,;1.43,3.75,;-.67,.1,;-2,.87,;-3.34,.1,;-3.34,-1.44,;-4.23,-3.36,;-5.44,-2.69,;-5.42,-.29,;-4.67,.87,;-6,.1,;-6,-1.44,;-7.33,-.67,;-6.83,-3.34,;-4.67,-2.21,;-.67,-1.44,;.66,-2.21,;.66,-3.75,)|
CC1(C)CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CCCCC2C3(F)F)cc1F
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CCCCC2C3(F)F)cc1F
Fc1cc(OCC23CCCCC2C3(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC23CCCCC2C3(F)F)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC2CCC3(CCC3)CC2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(OCC2CCC3(CC3)CC2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Fc1cc(OCC2CC3C(C2)C3(F)F)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(OCC2CC3C(C2)C3(F)F)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(C=C)cc1C(=O)NS(=O)(=O)N1CCC1 |TLB:15:6:13:9.10.11,THB:5:6:13:9.10.11,15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7|
CO[C@H]1CCN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |r,TLB:31:22:29:25.26.27,THB:21:22:29:25.26.27,31:26:29:22.30.23,30:22:25:29.28.27,30:28:25:22.31.23|
Fc1cc(COC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:15:6:13:9.10.11,THB:15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7,5:6:13:9.10.11|
Fc1c(F)c(cc(Cl)c1OCC12CC3CC(CC(C3)C1)C2)C(=O)NS(=O)(=O)N1CCC1 |TLB:10:11:14:18.17.16,20:11:18:14.15.16,THB:19:11:14:18.17.16,19:17:14:11.20.12,20:15:18:11.19.12|
Fc1cc(cc(Cl)c1OCC12CC3CC(CC(C3)C1)C2)C(=O)NS(=O)(=O)N1CCC1 |TLB:9:10:13:17.16.15,19:10:17:13.14.15,THB:18:10:13:17.16.15,18:16:13:10.19.11,19:14:17:10.18.11|
CS(=O)(=O)NC(=O)c1cc(F)c(OCC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:13:14:17:21.20.19,23:14:21:17.18.19,THB:22:14:17:21.20.19,22:20:17:14.23.15,23:18:21:14.22.15|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)c(F)c1F |TLB:13:14:17:21.20.19,23:14:21:17.18.19,THB:22:14:17:21.20.19,22:20:17:14.23.15,23:18:21:14.22.15|
Fc1cc(OCC2(CCC2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2(CCC2)C(F)(F)F)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Fc1cc(OCC2(CCC2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC2(CCC2)C(F)(F)F)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
CC1(F)CCC(COc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCC2)CC1 |(-9.05,-2.41,;-7.51,-2.41,;-8.28,-3.75,;-7.51,-.87,;-6.17,-.1,;-4.84,-.87,;-3.51,-.1,;-2.17,-.87,;-.84,-.1,;-.84,1.44,;.49,2.21,;.49,3.75,;1.83,1.44,;1.83,-.1,;.49,-.87,;.49,-2.41,;3.16,2.21,;3.16,3.75,;4.49,1.44,;5.83,2.21,;5.06,3.54,;6.6,3.54,;7.16,1.44,;7.56,-.05,;9.05,.35,;8.65,1.84,;-4.84,-2.41,;-6.17,-3.18,)|
Fc1cc(OC2C3CC4CC(C3)CC2C4)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |TLB:4:5:7:9.10.11,THB:5:13:9:7.6.11,5:6:9:13.12.14,12:13:7:9.10.11,12:10:7:13.5.14,(.51,-3.33,;.11,-1.84,;-1.37,-1.44,;-1.77,.05,;-3.26,.44,;-4.35,-.64,;-5.68,.12,;-7.01,-.64,;-7.01,-2.18,;-7.84,-4.09,;-6.45,-3.44,;-6.43,-1.04,;-5.24,-4.11,;-4.35,-2.18,;-5.68,-2.96,;-.68,1.13,;.8,.74,;1.2,-.75,;2.69,-1.15,;3.09,-2.64,;3.78,-.06,;5.27,-.46,;4.87,-1.95,;6.36,-1.55,;6.36,.63,;6.75,2.12,;7.84,1.03,;-1.08,2.62,;-.68,4.11,;-2.17,3.71,)|
Fc1cc(O[C@H]2C3CC4CC2C[C@](F)(C4)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r,wU:5.4,wD:12.13,TLB:5:6:14:11.10.9,4:5:11:14.8.9,THB:5:10:14:6.7.15,7:6:11:14.8.9,7:8:11:6.5.15,(-.28,-3.75,;-.28,-2.21,;-1.61,-1.44,;-1.61,.1,;-2.95,.87,;-4.28,.1,;-4.28,-1.44,;-5.18,-3.36,;-6.38,-2.69,;-6.36,-.29,;-5.61,.87,;-6.94,.1,;-6.94,-1.44,;-8.28,-.67,;-7.78,-3.34,;-5.61,-2.21,;-.28,.87,;1.05,.1,;1.05,-1.44,;2.39,-2.21,;2.39,-3.75,;3.72,-1.44,;5.06,-2.21,;4.29,-3.54,;5.83,-3.54,;6.39,-1.44,;7.88,-1.84,;8.28,-.35,;6.79,.05,;-.28,2.41,;.49,3.75,;-1.05,3.75,)|
Fc1cc(O[C@H]2C3CC4CC2C[C@](F)(C4)C3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,wU:5.4,wD:12.13,TLB:5:6:14:11.10.9,4:5:11:14.8.9,THB:5:10:14:6.7.15,7:6:11:14.8.9,7:8:11:6.5.15,(-0,-3.75,;-0,-2.21,;-1.34,-1.44,;-1.34,.1,;-2.67,.87,;-4,.1,;-4,-1.44,;-4.9,-3.36,;-6.1,-2.69,;-6.09,-.29,;-5.33,.87,;-6.67,.1,;-6.67,-1.44,;-8.21,-1.44,;-7.5,-3.34,;-5.33,-2.21,;-0,.87,;1.33,.1,;1.33,-1.44,;2.66,-2.21,;2.66,-3.75,;4,-1.44,;5.33,-2.21,;4.56,-3.54,;6.42,-3.3,;6.67,-1.44,;8.21,-1.44,;7.44,-.1,;-0,2.41,;.77,3.75,;-.77,3.75,)|
Fc1cc(OC2C3CC4CC(C3)CC2C4)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |TLB:4:5:7:9.10.11,THB:5:13:9:7.6.11,5:6:9:13.12.14,12:13:7:9.10.11,12:10:7:13.5.14,(.19,-3.33,;-.21,-1.84,;-1.69,-1.44,;-2.09,.05,;-3.58,.44,;-4.67,-.64,;-6,.12,;-7.33,-.64,;-7.33,-2.18,;-8.17,-4.09,;-6.77,-3.44,;-6.75,-1.04,;-5.57,-4.11,;-4.67,-2.18,;-6,-2.96,;-1,1.13,;.48,.74,;.88,-.75,;2.37,-1.15,;2.77,-2.64,;3.46,-.06,;4.95,-.46,;4.18,-1.79,;5.72,-1.79,;6.28,.31,;7.77,-.09,;8.17,1.4,;6.68,1.8,;-1.4,2.62,;-1,4.11,;-2.49,3.71,)|
Fc1cc(OC2CCC(F)(F)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OC2CCC(F)(F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OC2CCC(F)(F)CC2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(OC2CCC(F)(F)CC2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC2CCC3(CC3)CC2)cc1F
Fc1cc(OC2CCC3(CC3)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC3C(C2)C3(F)F)cc1F
Fc1cc(OCC2CCC3C(C2)C3(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCC3C(C2)C3(F)F)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC2CC22CCCCC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC2C3CC4CC(C3)CC2C4)cc1F |TLB:14:15:17:19.20.21,THB:15:23:19:17.16.21,15:16:19:23.22.24,22:23:17:19.20.21,22:20:17:23.15.24,(7.1,.63,;6.01,-.46,;5.24,-1.79,;6.78,-1.79,;4.52,-.06,;3.43,-1.15,;3.83,-2.64,;1.95,-.75,;1.55,.74,;.06,1.13,;-.34,2.62,;.06,4.11,;-1.43,3.71,;-1.03,.05,;-2.52,.44,;-3.6,-.64,;-4.93,.12,;-6.27,-.64,;-6.27,-2.18,;-7.1,-4.09,;-5.7,-3.44,;-5.69,-1.04,;-4.5,-4.11,;-3.6,-2.18,;-4.93,-2.96,;-.63,-1.44,;.86,-1.84,;1.26,-3.33,)|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CC(F)C2)CCCCC1
COC12CC3CC(C1)C(Oc1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O)C(C3)C2 |TLB:9:8:5:3.2.7,THB:8:25:3:5.6.7,8:6:3:25.27.26,27:25:5:3.2.7,27:2:5:25.8.26,1:2:5:25.8.26,(-6.26,-4.15,;-5.17,-3.06,;-5.57,-1.57,;-6.75,-2.55,;-6.44,-.5,;-6.84,.99,;-5.75,2.07,;-6.18,.75,;-4.27,1.68,;-3.18,2.77,;-1.69,2.37,;-.6,3.46,;.89,3.06,;1.98,4.15,;1.29,1.57,;.2,.48,;-1.29,.88,;-2.38,-.21,;2.77,1.17,;3.17,-.32,;3.86,2.26,;5.35,1.86,;6.84,1.46,;5.75,3.35,;4.95,.37,;-3.87,.19,;-4.95,-.9,;-4.23,-1.9,)|
Fc1cc(O[C@H]2C3CC4CC2C[C@@](Cl)(C4)C3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,wU:5.4,12.13,TLB:4:5:9:14.12.11,5:6:14:9.10.11,15:12:9:6.5.7,13:12:9:6.5.7,THB:5:10:14:6.15.7,15:6:9:14.12.11,(2.39,2.41,;1.05,1.64,;-.28,2.41,;-1.61,1.64,;-2.95,2.41,;-4.43,2.01,;-4.43,.47,;-5.76,-.3,;-7.1,.47,;-7.1,2.01,;-5.76,2.78,;-6.52,1.61,;-6.53,-.79,;-6.53,-2.33,;-7.93,-1.43,;-5.33,-1.46,;-1.61,.1,;-.28,-.67,;1.05,.1,;2.39,-.67,;2.39,-2.21,;3.72,.1,;5.06,-.67,;4.29,-2.01,;5.83,.66,;6.39,-1.44,;7.16,-2.78,;7.93,-1.44,;-2.95,-.67,;-4.49,-.67,;-3.72,-2.01,)|
Fc1cc(OC2CCC(Cl)(Cl)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
COCC1CC1c1cc(C(=O)NS(C)(=O)=O)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |w:6.6,3.2,TLB:31:22:29:25.26.27,21:22:25:29.28.27,21:22:29:25.26.27,THB:31:26:29:22.30.23,30:22:25:29.28.27,30:28:25:22.31.23|
Fc1cc(OCC2(CCCCC2)C#N)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC2(CCCCC2)C#N)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(CCCCC2)C#N)cc1F
CC1(C)CCCC(C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1
CC1(C)CCCC(C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC2CCC3(CCCCC3)CC2)cc1F
Fc1cc(OC2CCC3(CCCCC3)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CC1(C)CCCC(C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1
Fc1cc(OC2CCC3(CCCCC3)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CC1(F)CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1 |(-9.05,-2.41,;-7.51,-2.41,;-8.28,-3.75,;-7.51,-.87,;-6.17,-.1,;-4.84,-.87,;-3.51,-.1,;-2.17,-.87,;-.84,-.1,;-.84,1.44,;.49,2.21,;.49,3.75,;1.83,1.44,;1.83,-.1,;.49,-.87,;.49,-2.41,;-.28,-3.75,;1.26,-3.75,;3.16,2.21,;3.16,3.75,;4.49,1.44,;5.83,2.21,;5.06,3.54,;6.6,3.54,;7.16,1.44,;7.56,-.05,;9.05,.35,;8.65,1.84,;-4.84,-2.41,;-6.17,-3.18,)|
Fc1cc(OCC2CCC3(CCC3)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(O[C@H]2C3CC4CC2C[C@@](F)(C4)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r,wU:5.4,12.13,TLB:5:6:14:9.10.11,4:5:9:14.12.11,15:12:9:6.5.7,THB:5:10:14:6.15.7,15:6:9:14.12.11,13:12:9:6.5.7,(-.45,-3.75,;-.45,-2.21,;-1.79,-1.44,;-1.79,.1,;-3.12,.87,;-4.61,.47,;-4.61,-1.07,;-5.94,-1.84,;-7.27,-1.07,;-7.27,.47,;-5.94,1.24,;-6.69,.08,;-6.71,-2.32,;-7.48,-3.66,;-8.1,-2.97,;-5.5,-2.99,;-.45,.87,;.88,.1,;.88,-1.44,;2.22,-2.21,;2.22,-3.75,;3.55,-1.44,;4.88,-2.21,;4.11,-3.54,;5.65,-3.54,;6.22,-1.44,;7.7,-1.84,;8.1,-.35,;6.61,.05,;-.45,2.41,;.32,3.75,;-1.22,3.75,)|
Fc1cc(O[C@H]2C3CC4CC2C[C@@](Cl)(C4)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r,wU:5.4,12.13,TLB:4:5:9:14.12.11,5:6:14:9.10.11,15:12:9:6.5.7,THB:5:10:14:6.15.7,15:6:9:14.12.11,(2.22,2.48,;.88,1.71,;-.45,2.48,;-1.79,1.71,;-3.12,2.48,;-4.61,2.09,;-4.61,.55,;-5.94,-.23,;-7.27,.55,;-7.27,2.09,;-5.94,2.85,;-6.69,1.69,;-6.71,-.71,;-7.1,-2.2,;-8.1,-1.36,;-5.5,-1.38,;-1.79,.17,;-.45,-.6,;.88,.17,;2.22,-.6,;2.22,-2.14,;3.55,.17,;4.88,-.6,;4.11,-1.93,;5.65,.74,;6.22,-1.37,;6.61,-2.85,;8.1,-2.46,;7.7,-.97,;-3.12,-.6,;-4.66,-.6,;-3.89,-1.93,)|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCC=CC2)cc1F |c:17|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCCC(F)(F)C2)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(COC2CCCCC2)cc1F
Fc1cc(COC2CCCCC2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Fc1cc(COC2CCCCC2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
CC1CCCCC1COc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1
CC1CCCCC1COc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1
CO[C@]12CC3CC(C1)[C@H](Oc1cc(F)c(cc1Cl)C(=O)NS(=O)(=O)N1CCC1)C(C3)C2 |r,wU:8.9,2.1,TLB:9:8:29:3.2.30,7:2:29:6.8.5,1:2:29:6.8.5,THB:8:6:3:29.28.30,8:28:3:6.7.5,7:6:29:3.2.30,(-5.37,-2.94,;-6.71,-2.17,;-6.71,-.63,;-8.1,-1.27,;-7.27,.63,;-5.94,-.14,;-4.61,.63,;-5.5,-1.3,;-4.61,2.17,;-3.12,2.57,;-1.79,1.8,;-.45,2.57,;.88,1.8,;2.22,2.57,;.88,.26,;-.45,-.51,;-1.79,.26,;-3.12,-.51,;2.22,-.51,;2.22,-2.05,;3.55,.26,;4.88,-.51,;4.11,-1.85,;5.65,.82,;6.22,-1.28,;6.61,-2.77,;8.1,-2.37,;7.7,-.88,;-5.94,2.94,;-7.27,2.17,;-6.69,1.77,)|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@H]2C3CC4CC2C[C@@](Cl)(C4)C3)cc1F |r,wU:15.15,22.24,TLB:14:15:19:24.22.21,15:16:24:19.20.21,25:22:19:16.15.17,23:22:19:16.15.17,THB:15:20:24:16.25.17,25:16:19:24.22.21,(7.16,-1.67,;5.83,-.9,;5.06,-2.23,;6.6,.44,;4.49,-.13,;3.16,-.9,;3.16,-2.44,;1.82,-.13,;.49,-.9,;-.84,-.13,;-2.18,-.9,;-3.72,-.9,;-2.95,-2.23,;-.84,1.41,;-2.18,2.18,;-3.66,1.78,;-3.66,.24,;-4.99,-.53,;-6.33,.24,;-6.33,1.78,;-4.99,2.55,;-5.75,1.39,;-5.76,-1.01,;-5.76,-2.55,;-7.16,-1.66,;-4.56,-1.68,;.49,2.18,;1.82,1.41,;3.16,2.18,)|
Fc1cc(OCC2CCC(Cl)=CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |c:10|
Fc1cc(OCC2CCC(Cl)(Cl)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1(F)F |TLB:15:6:13:9.10.11,THB:15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7,5:6:13:9.10.11|
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1(F)F |TLB:15:6:13:9.10.11,THB:15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7,5:6:13:9.10.11|
CS(=O)(=O)NC(=O)c1cc(C2CC2(F)F)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:27:18:25:21.22.23,THB:27:22:25:18.26.19,26:18:21:25.24.23,26:24:21:18.27.19,17:18:25:21.22.23|
CCCCOc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1
Fc1cc(OCC2CN(C2)C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC2CN(C2)C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CNS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
FC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@H]2C3CC4CC2C[C@](Cl)(C4)C3)cc1F |r,wU:19.20,wD:26.29,TLB:18:19:25:28.22.23,19:20:28:25.24.23,THB:19:24:28:20.21.29,21:20:25:28.22.23,21:22:25:20.19.29,(9.02,-3.04,;7.69,-2.27,;6.2,-2.67,;5.8,-1.18,;7.29,-.78,;4.47,-.41,;3.7,-1.74,;5.24,.92,;3.13,.36,;1.8,-.41,;1.8,-1.95,;.46,.36,;-.87,-.41,;-2.2,.36,;-3.54,-.41,;-5.08,-.41,;-4.31,-1.74,;-2.2,1.9,;-3.54,2.67,;-5.02,2.27,;-5.02,.73,;-5.92,-1.19,;-7.12,-.53,;-7.11,1.87,;-6.35,3.04,;-7.69,2.27,;-7.69,.73,;-9.02,-.04,;-8.52,-1.17,;-6.35,-.04,;-.87,2.67,;.46,1.9,;1.8,2.67,)|
CC1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1 |(-8.95,-3.18,;-7.61,-2.41,;-7.61,-.87,;-6.28,-.1,;-4.94,-.87,;-3.61,-.1,;-2.28,-.87,;-.94,-.1,;-.94,1.44,;.39,2.21,;.39,3.75,;1.72,1.44,;1.72,-.1,;.39,-.87,;.39,-2.41,;-.38,-3.75,;1.16,-3.75,;3.06,2.21,;3.06,3.75,;4.39,1.44,;5.73,2.21,;4.96,3.54,;6.5,3.54,;7.06,1.44,;7.46,-.05,;8.95,.35,;8.55,1.84,;-4.94,-2.41,;-6.28,-3.18,)|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCC2(CC2)CC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CCC2(CC2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC3CC3C2)cc1F
Fc1cc(OCC2CCC3CC3C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
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FC1CN(C1)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCC3CC3C2)cc1F
CC1CCCC(C)C1COc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1
CC1CCCC(C)C1COc1cc(F)c(cc1Cl)C(=O)NS(=O)(=O)N1CCC1
CC1CCCC(C)C1COc1cc(F)c(cc1Cl)C(=O)NS(=O)(=O)C1CC1
CC1CC1c1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |w:4.4,1.0,TLB:32:23:30:26.27.28,THB:32:27:30:23.31.24,31:23:26:30.29.28,31:29:26:23.32.24,22:23:30:26.27.28|
C\C=C\c1cc(C(=O)NS(=O)(=O)N2CCC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:31:22:29:25.26.27,THB:31:26:29:22.30.23,30:22:25:29.28.27,30:28:25:22.31.23,21:22:29:25.26.27|
CCS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCC3(CC3)CC2)cc1F
Fc1cc(OCC2CCCC(F)(F)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCCC(F)(F)C2)cc1F
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Fc1cc(OCC2CCC(=CC2)C2CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |c:9|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CC3C4CCC(C4)C3C2)cc1F |TLB:17:18:23:20.21,THB:25:24:23:20.21|
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CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCC=CC1 |c:28|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCC2(CC2)CC1
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CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(CCCCC2)C(F)F)cc1F
FC(F)C1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CCCCC1
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CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCC(CC1)C(F)(F)F |(-4.1,-.77,;-4.1,.77,;-2.77,,;-1.44,.77,;-.1,,;1.23,.77,;2.56,,;3.9,.77,;2.56,-1.54,;1.23,-2.31,;-.1,-1.54,;-1.44,-2.31,;-2.98,-2.31,;-2.21,-3.64,;3.9,-2.31,;3.9,-3.85,;5.23,-1.54,;6.57,-2.31,;5.8,-3.64,;7.34,-.98,;7.9,-3.08,;8.67,-4.41,;9.44,-3.08,;-4.1,2.31,;-5.44,3.08,;-6.77,2.31,;-6.77,.77,;-5.44,,;-8.11,3.08,;-9.44,3.85,;-7.34,4.41,;-8.88,1.75,)|
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Fc1cc(OCC2CCC(CC2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |(3.72,.85,;2.39,.08,;1.06,.85,;-.28,.08,;-1.61,.85,;-2.94,.08,;-4.28,.85,;-4.28,2.39,;-5.61,3.16,;-6.94,2.39,;-6.94,.85,;-5.61,.08,;-8.28,3.16,;-9.61,3.93,;-7.51,4.49,;-9.05,1.82,;-.28,-1.46,;1.06,-2.23,;2.39,-1.46,;3.72,-2.23,;3.72,-3.77,;5.06,-1.46,;6.39,-2.23,;5.62,-3.57,;7.16,-.9,;7.73,-3,;8.12,-4.49,;9.61,-4.09,;9.21,-2.6,;-1.61,-2.23,;-3.15,-2.23,;-2.38,-3.57,)|
Fc1cc(OCC2CCC3CC3C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
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CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
Fc1cc(OCC2CCCC(F)(F)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2(CCCCC2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCC(F)(F)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC23CCCCC2C3(F)F)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
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Fc1cc(OCC2CC3CC3C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
O=C(NS(=O)(=O)N1CCC1)c1cnc(OCC23CC4CC(CC(C4)C2)C3)c(c1)C1CC1 |TLB:19:20:17.18.23:24,23:18:25:22.24.21,23:22:25:17.18.19,THB:19:18:24:20.25.21|
Cn1nccc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)-c1ccncc1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Fc1ccc(c(Br)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)Oc1ccc(c(Cl)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Fc1ccc(c(Cl)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Cc1ccc(c(Cl)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)-c1ccncc1
Clc1ccccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)-c1ccccc1
CCOc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCOCC1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCOC(C1)c1ccccc1
CC1(CN(CCO1)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)c1ccccc1
CC1CN(CCO1)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COC(=O)C1CN(CCO1)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
CCC1CN(CCO1)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
CN(C)C(=O)C1CN(CCO1)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
CC(C)(O)C1CN(CCO1)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(c1)-c1cn[nH]c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(c1)[N+]#[C-])-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(Br)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)Oc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Clc1ccc(c(c1)C1=CCNCC1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1 |t:8|
Clc1ccc(c(c1)-c1cn[nH]c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Clc1ccc(c(c1)-c1ccncc1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(Cl)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Nc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
NC(=O)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Clc1ccc(cc1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Fc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Fc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(cc1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Oc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Clc1ccc(c(Cl)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)ONc1nccs1)C(F)(F)F
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccn(CCN(C)C)n1
COc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncco1
COc1cc(Cl)ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)C1=CCNCC1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1 |t:11|
FC(F)(F)c1ccc(c(Cl)c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncco1
FC(F)(F)c1ccc(c(Br)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(Cl)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(c(c1)-c1ccncc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)-c1cn[nH]c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(Cl)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(cc1Cl)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Oc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(OC)c(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1 |(4.67,-5.42,;3.33,-6.19,;2,-5.42,;.67,-6.19,;-.67,-5.42,;-2,-6.19,;-2,-7.73,;-.67,-3.88,;.67,-3.11,;.67,-1.57,;2,-.8,;2,-3.88,;-2,-3.11,;-3.33,-3.88,;-4.67,-3.11,;-4.67,-1.57,;-3.33,-.8,;-3.33,.74,;-2,1.51,;-.67,.74,;-.67,-.8,;-2,-1.57,;-2,3.05,;-3.33,2.28,;-2.77,4.38,;-.67,3.82,;-.67,5.36,;.58,6.27,;.1,7.73,;-1.44,7.73,;-1.91,6.27,)|
Clc1ccc(c(Cl)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Cc1cc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1cc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
Clc1ccc(cc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(c1)-c1ccncc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
FC(F)(F)c1ccc(c(Br)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
CN1CCC(=CC1)c1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |c:4|
FC(F)(F)C(=O)ON(c1ccncn1)S(=O)(=O)c1ccc2c(nccc2c1)-c1ccc(cc1C1=CCNCC1)C(F)(F)F |t:37|
FC(F)(F)c1ccc(c(c1)C1=CCNCC1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1 |t:11|
FC(F)(F)c1ccc(c(c1)-c1ccncc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)-c1ccncc1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
CN1CCC(=CC1)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |c:4|
FC(F)(F)c1ccc(c(c1)C1=CCNCC1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1 |t:11|
CN1CCC(=CC1)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |c:4|
FC(F)(F)c1ccc(c(Cl)c1)-c1cccc2cc(ccc12)S(=O)(=O)Oc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2c(cccc2c1)N1CCCC1c1ccccc1
FC(F)(F)c1ccc(c(c1)-c1ccnn1C1CNC1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1
CN1CC(C1)n1nccc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCCC1c1ccccc1
CN1CCN(CC1)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCCC1c1cccnc1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCC[C@@H]1c1cccnc1 |r|
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCCC1c1ccncc1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCC[C@H]1c1ccncc1
CC1CCCN1c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCC1c1ccccc1
O=C1CCCN1c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1ccccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)C1CCCN1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)C1CCCN1c1ccccn1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)C1CCCN1Cc1ccccc1
O=S(=O)(Nc1ncc[nH]1)c1ccc2c(cccc2c1)C1CCCN1Cc1ccccc1
O=S(=O)(Nc1ncns1)c1ccc2c(NCc3ccccc3)cccc2c1
CN(Cc1ccccc1)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
O=C(N1CCCC1c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1)c1ccccc1
O=S(=O)(Nc1nccs1)c1ccc2c(cccc2c1)C1CCCN1C1CCOCC1
O=S(=O)(Nc1nccs1)c1ccc2c(cccc2c1)[C@@H]1CCCN1C1CCOCC1 |r|
O=S(=O)(Nc1nccs1)c1ccc2c(cccc2c1)[C@H]1CCCN1C1CCOCC1 |r|
Fc1ccc2n(C[N+]#[C-])c(cc2c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
Cn1c(cc2cc(F)ccc12)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
Fc1cnc(NS(=O)(=O)c2ccc3c(cccc3c2)-c2ccc(cc2C2=CCNCC2)C(F)(F)F)s1 |t:28|
CN1CCC(CC1)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
Cn1cncc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
Cn1ccnc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
Fc1cnc(NS(=O)(=O)c2ccc3c(cccc3c2)-c2ccc(cc2-n2ccnc2)C(F)(F)F)s1
Fc1cnc(NS(=O)(=O)c2ccc3c(cccc3c2)-c2ccc(cc2C2CCNCC2)C(F)(F)F)s1
Fc1ccc2[nH]c(cc2c1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccccc1
CN1CCC(CC1)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
CS(=O)(=O)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
FC(F)(F)c1ccc(-c2cccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)C1(F)CNC1
FC(F)(F)c1ccc(c(c1)C1=CCNC1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1 |t:11|
FC(F)(F)c1ccc(c(c1)C1CCNCC1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
FC(F)(F)c1ccc(c(c1)-n1ccnc1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
CN1CCC=C(C1)c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |c:4|
Cn1cncc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cn1ccnc1-c1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C1CC1
Fc1ccc(c(c1)-c1ccncc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3cccnc3)nccc2c1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3ncoc3-c3ccccc3)nccc2c1
C[C@@H](COc1ccc(Cl)cc1)Oc1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1 |r|
Clc1ccc(CCCOc2nccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)cc1
Clc1ccc(Cn2ccnc2COc2nccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)cc1
O=S(=O)(Nc1ccncn1)c1ccc2c(OC[C@H]3CN(Cc4ccccc4)CCO3)nccc2c1 |r|
O=S(=O)(Nc1ccncn1)c1ccc2c(OCC3(CC3)C#N)nccc2c1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3cccc4[nH]ncc34)nccc2c1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3cccc(c3)C#N)nccc2c1
Cc1nn(nc1COc1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccccc1
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
FC(F)(F)c1ccc(cc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(F)c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Cl)ncc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ncccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(c(OC)n1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(OC)c(c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1ccc(OC(F)(F)F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1c(cccc1C(F)(F)F)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(OC(F)(F)F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(F)c(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc2ccccc2cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
FC(F)(F)c1ccc(c(Cl)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1c(F)cccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cccc(F)c1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1 |(3.33,-1.54,;2,-2.31,;2,-3.85,;3.33,-4.62,;3.33,-6.16,;2,-6.93,;.67,-6.16,;-.67,-6.93,;.67,-4.62,;-.67,-3.85,;-2,-4.62,;-3.33,-3.85,;-3.33,-2.31,;-2,-1.54,;-2,,;-.67,.77,;.67,,;.67,-1.54,;-.67,-2.31,;-.67,2.31,;-2.21,2.31,;.87,2.31,;-.67,3.85,;.67,4.62,;.67,6.16,;2,6.93,;3.33,6.16,;3.33,4.62,;2,3.85,)|
Cc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Cl)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
O=S(=O)(Nc1ccncn1)c1ccc2c(nccc2c1)-c1cccc2ccsc12
Fc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cn1ccc2cccc(-c3nccc4cc(ccc34)S(=O)(=O)Nc3ccncn3)c12
Cc1cc2cnn(C)c2cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ncc(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ncc(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cnccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccncc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cccc(OC)c1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1 |(3.33,-.77,;2,-1.54,;2,-3.08,;3.33,-3.85,;3.33,-5.39,;2,-6.16,;.67,-5.39,;-.67,-6.16,;-.67,-7.7,;.67,-3.85,;-.67,-3.08,;-2,-3.85,;-3.33,-3.08,;-3.33,-1.54,;-2,-.77,;-2,.77,;-.67,1.54,;.67,.77,;.67,-.77,;-.67,-1.54,;-.67,3.08,;-2.21,3.08,;.87,3.08,;-.67,4.62,;.67,5.39,;.67,6.93,;2,7.7,;3.33,6.93,;3.33,5.39,;2,4.62,)|
COc1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
CCOc1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
FC(F)(F)COc1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ncc(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(NS(=O)(=O)c2ccc3c(nccc3c2)-c2ccc(cc2OC)C(F)(F)F)ncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccnc(C)n1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncncc1F)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cnccn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cc(C)ncn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
Oc1cc(F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1ccc(Oc2nccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)cc1Cl
COc1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(s1)C#N)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(c1)C#N
COc1cc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)-c1cccc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)-c1cnn(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)-c1cccnc1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
O=S(=O)(Nc1nccs1)c1ccc2c(nccc2c1)-c1ccn(c1)-c1ccccc1
Cc1c(cnn1-c1ccccc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1ccccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(F)ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(Cl)ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(Cl)ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1cc(ccc1-c1nc(Cl)cc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1nc(cc2cc(ccc12)S(=O)(=O)Nc1nccs1)[N+]#[C-])C(F)(F)F
COc1cc2cc(ccc2c(n1)-c1ccc(cc1OC)C(F)(F)F)S(=O)(=O)Nc1nccs1
CNc1cc2cc(ccc2c(n1)-c1ccc(cc1OC)C(F)(F)F)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1nc(cc2cc(ccc12)S(=O)(=O)Nc1nccs1)N(C)C)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)F
COCc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COC(=N)c1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
NC(=O)c1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
Fc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)-n1ccnc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
OCC(O)Cc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cnc(-c2ccc(cc2O)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(c(Br)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ncns1)c1ccc2c(nccc2c1)N1CCCC1c1ccccc1
O=S(=O)(Nc1nccs1)c1ccc2c(nccc2c1)N1CCCC1c1ccccc1
O=S(=O)(Nc1nccs1)c1ccc2c(nccc2c1)N1CCC[C@@H]1c1ccccc1 |r|
O=S(=O)(Nc1nccs1)c1ccc2c(nccc2c1)N1CCC[C@H]1c1ccccc1 |r|
COc1cc(ccc1-c1ncc([N+]#[C-])c2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(Cl)ccc1-c1ncc([N+]#[C-])c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ncc(C#N)c2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
O=S(=O)(Nc1nccs1)c1ccc2c(nccc2c1)N1CCC(C1)c1ccccc1
Cn1cccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2c(nccc2c1)C1CCCN1C1CCOCC1
COCCN1CCCC1c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1ccc(cc1Cl)N1CCN(CC1)c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(Cl)ccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(F)ccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1ccccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(ccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
COc1cc(F)ccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1
COc1ccccc1-c1nncc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncco1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)F
COc1cc(Cl)ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(F)ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(Cl)ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1ccccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(c(Cl)c1)-c1ccnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1c(N)cnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |(2,.77,;.67,,;.67,-1.54,;2,-2.31,;2.05,-3.88,;.67,-4.62,;-.67,-3.85,;-.67,-2.31,;-2,-1.54,;-3.33,-2.31,;-3.33,-3.85,;-4.67,-1.54,;-4.67,,;-3.33,.77,;-3.33,2.31,;-2,3.08,;-.67,2.31,;-.67,.77,;-2,,;-2,4.62,;-2.77,5.95,;-3.54,4.62,;-.67,5.39,;.67,4.62,;1.14,3.16,;2.68,3.16,;3.16,4.62,;1.91,5.53,;3.38,-4.65,;4.72,-5.42,;2.61,-5.98,;4.15,-3.31,)|
COc1cc(ccc1-c1c(cnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N)C(F)(F)F |(2,.77,;.67,,;.67,-1.54,;2,-2.31,;2.05,-3.88,;.67,-4.62,;-.67,-3.85,;-.67,-2.31,;-2,-1.54,;-3.33,-2.31,;-4.67,-1.54,;-4.67,,;-3.33,.77,;-3.33,2.31,;-2,3.08,;-.67,2.31,;-.67,.77,;-2,,;-2,4.62,;-2.77,5.95,;-3.54,4.62,;-.67,5.39,;.67,4.62,;1.14,3.16,;2.68,3.16,;3.16,4.62,;1.91,5.53,;-3.33,-3.85,;-3.33,-5.39,;3.38,-4.65,;4.72,-5.42,;2.61,-5.98,;4.15,-3.31,)|
COc1cc(ccc1-c1cncc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(ccc1-c1cncc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(cnc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(cnc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cn1ncnc1COc1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCCn3ccnn3)nccc2c1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3cc4OCCCn4n3)nccc2c1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3cccnc3N3CCOCC3)nccc2c1
FC(F)(COc1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C1CCOCC1
Cc1cccc(CCCOc2nccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)n1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3ccc(cc3)-n3ccnc3)nccc2c1
FC(F)(F)c1[nH]ncc1CCCOc1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCCn3cccc3)nccc2c1
O=S(=O)(Nc1ccncn1)c1ccc2c(OCc3ccc(cc3)N3CCOCC3)nccc2c1
Cn1cc(CCOc2nccc3cc(ccc23)S(=O)(=O)Nc2ccncn2)cn1
Cn1ncc2cccc(-c3nccc4cc(ccc34)S(=O)(=O)Nc3ccncn3)c12
Cc1c(ccc2n(C)ncc12)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
Cc1cc2n(C)ncc2cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
Cc1ccc2n(C)ncc2c1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1 |(-1.98,-6.93,;-.65,-6.16,;.68,-6.93,;2.02,-6.16,;2.02,-4.62,;3.16,-3.59,;4.65,-3.99,;2.54,-2.18,;1,-2.34,;.68,-3.85,;-.65,-4.62,;-1.98,-3.85,;-3.32,-4.62,;-4.65,-3.85,;-4.65,-2.31,;-3.32,-1.54,;-3.32,,;-1.98,.77,;-.65,,;-.65,-1.54,;-1.98,-2.31,;-1.98,2.31,;-3.52,2.31,;-.44,2.31,;-1.98,3.85,;-.65,4.62,;-.65,6.16,;.68,6.93,;2.02,6.16,;2.02,4.62,;.68,3.85,)|
O=S(=O)(Nc1ccncn1)c1ccc2c(nccc2c1)-c1cccc2cccnc12
Cc1noc(C)c1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1 |(2.9,-2.81,;2.13,-4.14,;3.04,-5.39,;2.13,-6.64,;.67,-6.16,;-.67,-6.93,;.67,-4.62,;-.67,-3.85,;-2,-4.62,;-3.33,-3.85,;-3.33,-2.31,;-2,-1.54,;-2,,;-.67,.77,;.67,,;.67,-1.54,;-.67,-2.31,;-.67,2.31,;-2.21,2.31,;.87,2.31,;-.67,3.85,;.67,4.62,;.67,6.16,;2,6.93,;3.33,6.16,;3.33,4.62,;2,3.85,)|
Cn1nc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccnc(OC)n1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)NC(C)=O)C(F)(F)F
Cn1ccnc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ccncn1)c1ccc2c(nccc2c1)C1CCCN1C1CCOCC1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)C#N
COC(=O)c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCC[C@H]1c1cccnc1
O=S(=O)(Nc1ncns1)c1ccc2c(cccc2c1)N1CCC[C@@H]1c1ccncc1 |r|
Fc1ccc(c(c1)C1=CCOC1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1 |t:8|
Cn1cc(cn1)-c1cc(F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(Cl)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(c(Oc2cccnn2)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(c(Oc2ccccn2)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(c(OCC#N)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ncc(O)c2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(F)ccc1-c1ncc(O)c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccccc1-c1ncc(O)c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)N=C1NC(=O)CS1)C(F)(F)F |w:21.23|
COc1cc(ccc1-c1cnnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1cnnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(C(F)F)c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(F)ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1ccccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1ccnc2cc(cc(C)c12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1cncc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
COc1ccccc1-c1cncc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccccc1-c1cncc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(F)ccc1-c1cncc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1ccnc2cc(ncc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1ccnc2cc(c(F)cc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1ccccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1ccc(cc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
Cc1cc(Cl)ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ncns1
Cc1cc(ccc1-c1ccnc2cc(ccc12)S(=O)(=O)Nc1ncns1)C#N
COc1ccccc1-c1c(cnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N |(-1.33,2.31,;,1.54,;1.33,2.31,;1.33,3.85,;2.67,4.62,;4,3.85,;4,2.31,;2.67,1.54,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;-2.67,-3.08,;-1.9,-4.41,;-3.44,-1.75,;-4,-3.85,;-5.33,-3.08,;-6.74,-3.71,;-7.77,-2.56,;-7,-1.23,;-5.5,-1.55,;5.33,,;6.67,.77,)|
COc1ccccc1-c1c(Br)cnc2cc(ccc12)S(=O)(=O)Nc1nccs1 |(2.82,.1,;1.48,-.67,;1.48,-2.21,;2.82,-2.98,;2.82,-4.52,;1.48,-5.29,;.15,-4.52,;.15,-2.98,;-1.18,-2.21,;-2.52,-2.98,;-2.52,-4.52,;-3.85,-2.21,;-3.85,-.67,;-2.52,.1,;-2.52,1.64,;-1.18,2.41,;.15,1.64,;.15,.1,;-1.18,-.67,;-1.18,3.95,;-2.72,3.95,;-1.95,5.29,;.15,4.72,;1.48,3.95,;1.48,2.41,;2.95,1.94,;3.85,3.18,;2.95,4.43,)|
COc1cc(ccc1-c1ccnc2cc(c(C)cc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1ccnc2cc(c(OC)cc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1ccnc2c(C)c(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C#N
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cnsn1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1
COc1cc(Cl)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C#N
COc1cc(Cl)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2cc(F)cc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2cccc(c2)C(F)(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2cccc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C#N
COc1cc(-c2cccc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)C#N
COc1cc(-c2cccc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1cc(-c2cc(F)cc(F)c2)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C#N
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(c1)C(F)(F)F
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1ccc(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)-c1cccc(F)c1
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(c1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(F)cc1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(c1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(F)nc1
COc1ccc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C1=CCOCC1 |t:32|
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
Cc1cc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
Cc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
Cc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C#N
COc1cc(CC(C)(C)C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(OCC(C)C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(OCC(F)(F)F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1nc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1ccc(F)c(F)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccnc1
COc1cc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncns1)-c1cccc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccnc(C)n1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cc(C)ncn1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nnco1)-c1cc(F)cc(F)c1
FC(F)(F)C(=O)ON(c1nccs1)S(=O)(=O)c1ccc2c(nccc2c1)-c1ccc(Cl)cc1OCC#N
FC(F)(F)c1ccc(c(OCC#N)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)C(=O)ON(c1nccs1)S(=O)(=O)c1ccc2c(nccc2c1)-c1ccccc1OCC#N
FC(F)(F)C(=O)ON(c1ccncn1)S(=O)(=O)c1ccc2c(nccc2c1)-c1ccc(Cl)cc1OCC#N
Cc1cnc(F)c(c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cnc(OC2CCNCC2)c(c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cnc(OCCOc2ccccc2)c(c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
CC(C)(O)c1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(c(c1)[N+]#[C-])-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cnsn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncco1)C(F)(F)F
COc1cc(ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1ccccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(F)ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1ncns1)C#N
COc1ncccc1-c1ncc(F)c2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1cnc(-c2ccccc2C#N)c2ccc(cc12)S(=O)(=O)Nc1nccs1
Fc1cnc(-c2ccccc2OCC#N)c2ccc(cc12)S(=O)(=O)Nc1nccs1
COc1cc(F)ccc1-c1ncc(C#N)c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccccc1-c1ncc([N+]#[C-])c2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1cccc(c1)-c1ccc(cc1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
FC(F)(F)C(=O)ON(c1ncns1)S(=O)(=O)c1ccc2c(nccc2c1)-c1ccc(Cl)cc1OCC#N
COc1cc(F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ncccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1nc(Cl)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ncc(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1ncc(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ncc(C)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1nc(C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)Oc1ccc(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(c(OC2CCOCC2)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
CC(Oc1cc(F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
FC(Oc1cc(F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1)[N+]#[C-]
NC(=O)COc1cc(F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1nc(OCC(C)C)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nc(Cl)cs1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(Cl)s1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nc(cs1)C#N)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cc(Cl)ncn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nc(C)cs1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nnc(Cl)s1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ncc(F)cn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccc(F)cn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nc(cs1)C(F)(F)F)C(F)(F)F
Clc1cccc(c1)-n1cc(cn1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cocn1)C(F)(F)F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccccc1C
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(C)cc1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(F)cc1F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(F)ccc1F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1c(F)cccc1F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(F)c(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(F)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccnc1
COc1cc(c(OC)cc1C(F)F)-c1nccc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(c(OC)cc1C(F)F)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(cc1)C#N
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1nccs1
COc1cc(C(F)F)c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(C(F)F)c(cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C1CC1
COc1cc(Cl)ccc1-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(C)o1
COc1cc(Oc2ccc(F)cc2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2cccc(F)c2)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(Oc2ccccc2F)ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccccc1-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cccc(c1)-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(cc1)-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(C)c(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(C)cc(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(C)c(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(C)cc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccnc1F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccnc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cncc(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccnc1C
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(C)nc1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cncc(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1c(C)ccnc1F
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cnc(F)c(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccnc1OC
COc1ccc(cn1)-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1F)-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(F)c(c1)C#N
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(F)cc(c1)C#N
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(F)c(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc2[nH]ccc2c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(F)c(Cl)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(F)cc(Cl)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(Cl)c(F)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(Cl)c(C)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1ccc(C)c(Cl)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cc(C)cc(Cl)c1
COc1cc(ccc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1cscn1)C(F)(F)F
COc1nc(c(Cl)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1ccc(Cl)cc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(Cl)cc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1ccc(Cl)cc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1ccc(Cl)cc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ncc(F)s1
COc1ccc(CN(c2ncns2)S(=O)(=O)c2ccc3c(n[nH]c(=O)c3c2)-c2ccccc2OC)cc1
COc1ccc(cc1-c1n[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
COc1cc(ccc1-c1nc(C)nc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1nc(-c2ccc(cc2OC)C(F)(F)F)c2ccc(cc2n1)S(=O)(=O)Nc1nccs1
COc1cc(C(F)F)c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(C(F)F)c(F)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1cscn1
COc1cc(C(F)F)c(F)cc1-c1nc(C)nc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1-c1nc(C)nc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)F
COc1cc(ccc1-c1nc(C)nc2cc(ccc12)S(Cl)(=O)=O)C1(F)COC1
COc1cc(ccc1-c1nc(C)nc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(ccc1-c1nc(C)nc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncns1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(c(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1
COc1cc(Cl)ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncns1)-c1cccc(F)c1
COc1cc(Cl)ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccncn1
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ccncn1)-c1cccc(c1)C(F)(F)F
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1ccc(F)c(F)c1
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nncs1)-c1cc(F)cc(F)c1
Cc1cc(Cl)ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1ncns1
Oc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COC[C@H]1CCCN1c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(c(Cl)c1)-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ncc(Cl)cc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(ccc1-c1nc(=O)[nH]c2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1c[nH]c(=O)c2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1cc(Br)c(c(c1)C1=CCNCC1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1 |t:12,(10.61,-23.3,;9.27,-22.53,;10.04,-21.19,;8.5,-23.86,;7.94,-21.76,;7.89,-20.19,;6.56,-19.42,;6.56,-17.88,;5.22,-20.19,;5.22,-21.73,;6.56,-22.5,;3.89,-22.5,;2.56,-21.73,;1.22,-22.5,;1.22,-24.04,;2.56,-24.81,;3.89,-24.04,;3.89,-19.42,;2.56,-20.19,;1.22,-19.42,;1.22,-17.88,;2.56,-17.11,;2.56,-15.57,;3.89,-14.8,;5.22,-15.57,;5.22,-17.11,;3.89,-17.88,;3.89,-13.26,;2.35,-13.26,;5.43,-13.26,;3.89,-11.72,;2.56,-10.95,;1.09,-11.43,;.19,-10.18,;1.09,-8.94,;2.56,-9.41,)|
COc1cc(cc(C2=CCNCC2)c1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |t:7,(7.89,-17.11,;6.56,-17.88,;6.56,-19.42,;7.89,-20.19,;7.94,-21.76,;6.56,-22.5,;5.22,-21.73,;3.89,-22.5,;2.56,-21.73,;1.22,-22.5,;1.22,-24.04,;2.56,-24.81,;3.89,-24.04,;5.22,-20.19,;3.89,-19.42,;2.56,-20.19,;1.22,-19.42,;1.22,-17.88,;2.56,-17.11,;2.56,-15.57,;3.89,-14.8,;5.22,-15.57,;5.22,-17.11,;3.89,-17.88,;3.89,-13.26,;2.35,-13.26,;5.43,-13.26,;3.89,-11.72,;2.56,-10.95,;1.22,-11.72,;-.11,-10.95,;-.11,-9.41,;1.22,-8.64,;2.56,-9.41,;9.27,-22.53,;10.61,-23.3,;10.04,-21.19,;8.5,-23.86,)|
FC(F)(F)c1ccc(c(c1)-c1ccncc1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(c(Br)c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
CC(C)(C)OC(=O)N1CCC(=CC1)c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F |c:10|
FC(F)(F)c1ccc(c(c1)C1=CCNCC1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1 |t:11|
Fc1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(c(Cl)c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
Clc1ccc(cc1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
Fc1cc(Cl)ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
Clc1ccc(c(Cl)c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)N1CCc2c(C1)cccc2-c1cccc2CNCCc12
C[N+]1([O-])CCC(=CC1)c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F |c:5|
CN1CCC(=CC1)c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F |c:4|
Cn1cc(cn1)-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)-c1cn[nH]c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
Nc1cc(ccn1)-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)C1=CCOCC1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1 |t:11|
COc1cncc(c1)-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cc1cncc(c1)-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(-c2cccc3CN(CCc23)S(=O)(=O)Nc2ncns2)c(c1)-c1cccnc1
FC(F)(F)c1ccc(-c2cccc3CN(CCc23)S(=O)(=O)Nc2ncns2)c(c1)-c1cncnc1
O=S(=O)(Nc1ncns1)N1CCc2c(C1)cccc2-c1cccc2ccccc12
O=S(=O)(Nc1ncns1)N1CCc2c(C1)cccc2-c1cncc2ccccc12
COc1ccc(c(OC)c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
COc1ccc(OC)c(c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
COc1cccc(OC)c1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1 |(-.15,-7.55,;-.15,-6.01,;1.18,-5.24,;2.52,-6.01,;3.85,-5.24,;3.85,-3.7,;2.52,-2.93,;2.52,-1.39,;3.85,-.62,;1.18,-3.7,;-.15,-2.93,;-1.48,-3.7,;-2.82,-2.93,;-2.82,-1.39,;-1.48,-.62,;-1.48,.92,;-.15,1.69,;1.18,.92,;1.18,-.62,;-.15,-1.39,;-.15,3.23,;-1.69,3.23,;1.39,3.23,;-.15,4.77,;-1.48,5.54,;-2.95,5.06,;-3.85,6.31,;-2.95,7.55,;-1.48,7.08,)|
COc1ccc(F)cc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
COc1cc(F)ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(c(c1)N1CCOCC1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(-c2cccc3CN(CCc23)S(=O)(=O)Nc2ncns2)c(c1)-n1ccnc1
Fc1cnc(NS(=O)(=O)N2CCc3c(C2)cccc3-c2ccc(cc2C2=CCNCC2)C(F)(F)F)s1 |t:28|
FC(F)(F)c1ccc(c(c1)C1=CCNC1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1 |t:11|
Fc1cnc(NS(=O)(=O)N2CCc3c(C2)cccc3-c2ccc(cc2C2CCNCC2)C(F)(F)F)s1
FC(F)(F)c1ccc(c(c1)C1=CCNCC1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1nccs1 |t:11|
CC(C)(C)OC(=O)N1CCC(=CC1)c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |c:10|
Fc1cnc(NS(=O)(=O)N2CCc3c(C2)cccc3-c2ccc(cc2-n2ccnc2)C(F)(F)F)s1
CN1CCC(=CC1)c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F |c:4|
CN1CCC(=CC1)c1ccc(cc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F |c:4|
CN1CCN(CC1)c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
Cc1cn(cn1)-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
Cc1cncn1-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
COc1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C1CC1
COc1cc(ccc1-c1nccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1cc(ccc1-c1nccc2CN(CCc12)S(=O)(=O)Nc1ncns1)C1CC1
COc1cc(ccc1-c1cccc2CN(CC(C)c12)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cn1nccc1-c1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COc1ncccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)N1CCc2c(C1)cccc2-c1cccc2[nH]ncc12
Clc1ccc2c(ccnc2c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
CN1CCC(=CC1)c1cc(Cl)cc(F)c1-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncc(F)s1 |c:4,(-4.67,-8.6,;-3.33,-7.83,;-2,-8.6,;-.67,-7.83,;-.67,-6.29,;-2,-5.52,;-3.33,-6.29,;.67,-5.52,;2,-6.29,;3.33,-5.52,;4.67,-6.29,;3.33,-3.98,;2,-3.21,;2,-1.67,;.67,-3.98,;-.67,-3.21,;-2,-3.98,;-3.33,-3.21,;-3.33,-1.67,;-2,-.9,;-2,.64,;-.67,1.41,;.67,.64,;.67,-.9,;-.67,-1.67,;-.67,2.95,;-2.21,2.95,;.87,2.95,;-.67,4.49,;-2,5.26,;-3.47,4.78,;-4.37,6.03,;-3.47,7.27,;-4.24,8.6,;-2,6.8,)|
COc1cc(ccc1-c1cccc2CCN(Cc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(c(Br)c1)-c1cccc2CN(CCc12)S(=O)(=O)Nc1ccncn1
CC(C)(C)OC(=O)N1CCC(=CC1)c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1 |c:10|
CC(C)(C)OC(=O)N1CCc2c(C1)cccc2-c1cccc2CN(CCc12)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1ncnc2CN(CCc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1-c1ncnc2CN(CCc12)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
COc1cc(ccc1-c1ncnc2CN(CCc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1cc(ccc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1nncs1)-c1ccc(F)c(F)c1
COc1ccc(cc1-c1cccc2CN(CCc12)S(=O)(=O)Nc1nncs1)-c1ccc(F)c(F)c1
COc1cc(ccc1-c1ncnc2CN(CCc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
OC(=O)CN(c1ccccc1)c1cc(nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O
NC(=O)c1cc(cc(n1)[C@H](O)CO)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NC(=O)CN(c1ccccc1)c1cc(cc(n1)C(N)=O)-c1ccc(Oc2ccc(F)cc2)cc1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=N)\N=N/NCC(N)=O
OC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)N(CCC#N)c1ccccc1
Cn1nccc1-c1cc(Cl)ccc1-c1c[nH]c2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
CC(C)n1cc(-c2ccc(cc2-c2ccnn2C)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
CC(=O)n1cc(-c2ccc(cc2-c2ccnn2C)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1-c1c[nH]c2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COC(=O)n1cc(-c2ccc(cc2-c2ccnn2C)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1-c1cn(c2cc(ccc12)S(=O)(=O)Nc1ncns1)S(C)(=O)=O)C(F)(F)F
Cn1nccc1-c1cc(ccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cn1cc(-c2cccnc2)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cc(F)ccc2F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
Cn1nccc1-c1cc(ccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Cn1nccc1-c1cc(ccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1nncs1)C(F)(F)F
CC#Cc1cncc(c1)-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cc(cc(c2)C(F)(F)F)-c2ccncc2)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(cc2C#N)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cc(Br)cc(c2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(cc2-c2ccncc2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(cc2-c2ccn(n2)C2CNC2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(cc2-c2cn[nH]c2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(cc2C2=CCNCC2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1 |t:11|
Cn1cc(-c2ccc(cc2Cl)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(c(Cl)c2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1-c1c[nH]c2nc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cn1cc(-c2ccc(cc2-c2ccnn2C)C(F)(F)F)c2ccc(nc12)S(=O)(=O)Nc1ncns1
CC(=O)n1cc(-c2ccc(cc2-c2ccnn2C)C(F)(F)F)c2ccc(nc12)S(=O)(=O)Nc1ncns1
COc1cc(F)ccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
COc1cc(OC)cc(c1)-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(F)c(c2)C#N)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(C#N)c(F)c2)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(OC(F)(F)F)cc2)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cccc(OC(F)(F)F)c2)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cccc(c2)C#N)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccccc2)c2ccc(cc12)S(=O)(=O)Nc1ncns1
COc1ccc(-c2cn(C)c3cc(ccc23)S(=O)(=O)Nc2ncns2)c(OC)c1
Cn1cc(-c2cccc3ccccc23)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cccc3ncccc23)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cccc(c2)S(C)(=O)=O)c2ccc(cc12)S(=O)(=O)Nc1ncns1
COc1ccc(-c2cn(C)c3cc(ccc23)S(=O)(=O)Nc2ncns2)c2ccccc12
COc1ccc(-c2cn(C)c3cc(ccc23)S(=O)(=O)Nc2ncns2)c(Cl)c1
Cc1noc(C)c1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1 |(3.21,-3.25,;2.44,-4.59,;2.92,-6.05,;1.67,-6.96,;.42,-6.05,;-.91,-6.82,;.9,-4.59,;-.19,-3.5,;-1.72,-3.66,;-2.35,-2.25,;-3.83,-1.85,;-1.2,-1.22,;-1.2,.32,;.13,1.09,;1.46,.32,;1.46,-1.22,;.13,-1.99,;.13,2.63,;-1.41,2.63,;1.67,2.63,;.13,4.17,;1.46,4.94,;2.93,4.46,;3.83,5.71,;2.93,6.96,;1.46,6.48,)|
Cn1cc(-c2ccc(Br)cc2C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccccc2C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cc1cnc(N)c(c1)-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
Cc1cc(ccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1)C#N
CN(C)c1cccc(c1)-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cccc(c2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
COc1ccc(cc1C(F)(F)F)-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2ccc(cc2-c2ccnn2C)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1nc(Br)ns1
Cn1cc(-c2ccncc2Cl)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cn(C)c2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cccc3CNCCc23)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1cc(-c2cccc3CCNCc23)c2ccc(cc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1-n1cnc2cc(ccc12)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1-n1cnc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cn1cc(-c2ccc(cc2C2=CCNCC2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1nccs1 |t:11|
Cn1cc(-c2ccc(cc2C2=CCNCC2)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1cscn1 |t:11|
Fc1ccc(Oc2ccc(cc2)-c2cccc(n2)C(=O)NCCNS(=O)(=O)c2cccnc2)cc1
CS(=O)(=O)c1cccc(c1)S(=O)(=O)NCCNC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
NCCCC[C@H](NC(=O)c1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O |r|
NC(=O)C[C@H](NC(=O)c1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@@H](O)CO)C(N)=O |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)[N+]#[C-])cc1)[C@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)[N+]#[C-])cc1)[C@@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2C(F)(F)F)[N+]#[C-])cc1)[C@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2C(F)(F)F)[N+]#[C-])cc1)[C@@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2cc(Cl)ccc2F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2cc(Cl)ccc2F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(c(c2)[N+]#[C-])C(F)(F)F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc([N+]#[C-])c(c2)C(F)(F)F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc([N+]#[C-])c(c2)C(F)(F)F)cc1)[C@H](O)CO |r|
COC(=O)[C@H](C)NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO |r|
C[C@H](NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO)C(O)=O |r|
C[C@H](NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)[C@H](O)CO)C(N)=O |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)[C@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cc2)C(F)(F)F)cc1)[C@@H](O)CO |r|
NC(=O)c1cc(nc(n1)-c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1)[C@H](O)CO |r|
C[C@H](Nc1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(O)=O)C(O)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCC2(Cc3ccccc3C2)CC1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCC(CC1)Oc1ccc(cc1)[N+]#[C-])C(N)=O)C(N)=O |r|
CN(C)CCNc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
OCCNc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
NC(=O)[C@H](CO)Nc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1 |r|
Fc1ccc(Oc2ccc(cc2)-c2nc(nc3ccccc23)N2CCNC(=O)C2)cc1
Nc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
COC(=O)[C@@H]1CCCN1c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1 |r|
CN(N)c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
CCN1CCN(CC1)c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
OC1CCN(CC1)c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
OCCN1CCN(CC1)c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
CN1CCN(CC1)c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
NC(=O)[C@@H]1CCCN1c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
COC(=O)[C@@H]1C[C@@H](O)CN1c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1 |r|
Fc1ccc(Oc2ccc(cc2)-c2nc(NCCCn3ccnc3)nc3ccccc23)cc1
CN(C)CCCNc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
CNc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
OC[C@H](O)CNc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1 |r|
OC[C@@H](O)CNc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
NC(=O)C[C@H](Nc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1)C(N)=O
CN1[C@H]2CCC[C@@H]1C[C@@H](C2)Nc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1 |r,THB:10:8:1:3.4.5,0:1:7.9.8:3.4.5|
OCC(CO)Nc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
Fc1ccc(Oc2ccc(cc2)-c2nc(NCCN3CCNC3=O)nc3ccccc23)cc1
NN(CCO)c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
NC(=O)CNc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
NC(=O)c1nc(-c2ccc(Oc3ccccc3)cc2)c2ccccc2n1
CCOC(=O)c1nc(-c2ccc(Oc3ccccc3)cc2)c2ccccc2n1
OC(=O)c1nc(-c2ccc(Oc3ccccc3)cc2)c2ccccc2n1
OC[C@@H](O)c1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1 |r|
CCOc1nc(-c2ccc(Oc3ccc(F)cc3)cc2)c2ccccc2n1
Fc1ccc(Oc2ccc(cc2)-c2nc(Oc3ccccn3)nc3ccccc23)cc1
CCOC(=O)[C@H](O)[C@H](O)c1cn(-c2ccc(Oc3ccc(cn3)C(F)(F)F)cc2)c2ccccc12
CCOC(=O)[C@H](O)[C@H](O)c1cccc(n1)-c1ccc(Oc2ccc(c(c2)C#N)C(F)(F)F)cc1
OC(=O)C(=O)c1cn(-c2ccc(Oc3ccc(c(c3)C#N)C(F)(F)F)cc2)c2ccccc12
OCCc1cn(-c2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)c2cnccc12
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cncc(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-1.33,-10.01,;-1.33,-11.55,;,-9.24,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;6.67,-6.93,;8,-7.7,;8,-9.24,;6.67,-10.01,;5.33,-9.24,;6.67,-11.55,;6.67,-13.09,;5.13,-11.55,;8.21,-11.55,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cnn(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;,-7.7,;-1.41,-7.07,;-2.44,-8.22,;-1.67,-9.55,;-2.29,-10.96,;-.16,-9.23,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)nc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;,-9.24,;-1.33,-10.01,;-2.67,-9.24,;-4,-10.01,;-2.67,-7.7,;-1.33,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;-2.67,-9.24,;-2.67,-7.7,;-1.33,-6.93,;-1.33,-5.39,;,-4.62,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccnn1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;,-7.7,;-1.41,-7.07,;-2.44,-8.22,;-1.67,-9.55,;-.16,-9.23,;.98,-10.26,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cncc(c1)C#N |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-1.33,-10.01,;,-9.24,;-1.33,-11.55,;-1.33,-13.09,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cncc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-1.33,-10.01,;,-9.24,;-1.33,-11.55,;-1.33,-13.09,;.21,-11.55,;-2.87,-11.55,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;6.67,-6.93,;9.34,-6.93,;10.67,-6.16,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cncc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-1.33,-10.01,;-1.33,-11.55,;,-9.24,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccnc1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;,-9.24,;-1.33,-10.01,;-2.67,-9.24,;-2.67,-7.7,;-1.33,-6.93,;-1.33,-5.39,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccnc(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;,-9.24,;-1.33,-10.01,;-2.67,-9.24,;-2.67,-7.7,;-4,-6.93,;-1.33,-6.93,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;6.1,-10.99,;4.56,-13.65,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Br)c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;6.1,-10.99,;4.56,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(cc(F)c1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(-c2cc(F)cc(Cl)c2)c(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;6.67,-8.47,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cc(F)cc(Cl)c1 |(-1.09,-5.71,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
OC[C@H](O)Cc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |wD:2.2,(9.34,-5.39,;8,-4.62,;6.67,-5.39,;6.67,-6.93,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(6.82,-5.02,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nccs1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;2.67,-10.78,;1.13,-9.24,;4.21,-9.24,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nncs1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Br)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(Cl)cc1-n1c2cc(F)c(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
FC(F)(F)c1ccc(c(c1)-c1cn[nH]c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(2.67,-10.78,;2.67,-9.24,;4.21,-9.24,;1.13,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.74,-5.25,;7.77,-4.1,;7,-2.77,;5.5,-3.09,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.53,-2.15,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-2.76,3.22,;-3.23,4.68,;-4.77,4.68,;-5.25,3.22,)|
FC(F)(F)c1ccc(c(c1)-c1cn[nH]c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(2.67,-10.78,;2.67,-9.24,;1.13,-9.24,;4.21,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.74,-5.25,;7.77,-4.1,;7,-2.77,;5.5,-3.09,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.53,-2.15,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-2.76,3.22,;-3.23,4.68,;-4.77,4.68,;-5.25,3.22,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2c(C)cc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;2.67,1.54,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(C)cc1-n1c2ccc(cc2c(C)cc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;2.67,1.54,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(C)cc1-n1c2ccc(cc2c(C)cc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;2.67,1.54,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2c(C)cc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;2.67,1.54,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Br)ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;,-7.7,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1 |(6.42,-5.71,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1nc(N2CC(F)(F)C2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.58,-10.33,;2.67,-11.42,;1.86,-12.73,;3.47,-12.73,;3.76,-10.33,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Fc1cccc(c1)-c1cc(OCC#N)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;-2.67,-4.62,;-4,-3.85,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
CCOc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-2.67,-4.62,;-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
Cc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cc(F)cc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)c(C)c1 |(6.82,-5.02,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccnc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)nc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(-c2cnn(C)c2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.42,-10.15,;1.9,-11.61,;3.44,-11.61,;4.34,-12.86,;3.91,-10.15,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccncc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,)|
COc1cc(N2CC(F)(F)C2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.58,-10.33,;2.67,-11.42,;1.86,-12.73,;3.47,-12.73,;3.76,-10.33,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cnc(C)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(N2CC(C2)C(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.58,-10.33,;2.67,-11.42,;3.76,-10.33,;2.67,-12.96,;2.67,-14.5,;1.13,-12.96,;4.21,-12.96,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)c(F)cc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)cc(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C#N)c(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-15.4,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C#N)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-15.4,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cncc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Cl)ccc1-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2cc(OC)c1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;5.33,,;6.67,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;6.67,-6.93,;9.34,-6.93,;10.67,-6.16,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;6.67,-6.93,;8,-7.7,;9.34,-6.93,;8,-9.24,;6.67,-10.01,;6.67,-11.55,;5.33,-9.24,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;6.67,-6.93,;6.67,-5.39,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;6.67,-6.93,;6.67,-5.39,)|
COc1cc(F)cc(c1)-c1ccc(OC)c(c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(8,-12.32,;6.67,-11.55,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,;5.33,-7.7,;5.33,-9.24,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)ccc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;6.67,-6.93,;6.67,-5.39,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1Cl |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;6.67,-6.93,;6.67,-5.39,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;5.33,-7.7,;6.67,-6.93,;8,-7.7,;8,-9.24,;6.67,-10.01,;5.33,-9.24,;9.34,-10.01,;10.67,-10.78,;10.11,-8.68,;8.57,-11.34,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;6.67,-6.93,;8,-7.7,;8,-9.24,;9.34,-10.01,;6.67,-10.01,;5.33,-9.24,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;6.67,-6.93,;8,-7.7,;8,-9.24,;9.34,-10.01,;6.67,-10.01,;5.33,-9.24,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1cccc(c1)-c1ccc(OC)c(c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(9.34,-5.39,;9.34,-6.93,;8,-7.7,;8,-9.24,;6.67,-10.01,;5.33,-9.24,;5.33,-7.7,;6.67,-6.93,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,;6.67,-5.39,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;6.67,-6.93,;6.67,-5.39,;6.67,-3.85,;8.21,-5.39,;5.13,-5.39,)|
COc1ccc(Br)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1cc(Cl)c(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1cc(Cl)c(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1cc(Cl)cc(c1)-c1ccc(OC)c(c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(8,-12.32,;6.67,-11.55,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,;5.33,-7.7,;5.33,-9.24,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(OC)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;9.34,-6.93,;9.34,-5.39,;6.67,-6.93,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;8,-9.24,;8,-7.7,;6.67,-6.93,;6.67,-5.39,)|
COc1ccc(cc1Cl)-c1ccc(OC)c(c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(10.67,-9.24,;9.34,-10.01,;8,-9.24,;6.67,-10.01,;5.33,-9.24,;5.33,-7.7,;6.67,-6.93,;8,-7.7,;9.34,-6.93,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;9.34,-6.93,;6.67,-6.93,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,;6.67,-5.39,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(OC)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;9.34,-10.01,;8,-7.7,;9.34,-6.93,;9.34,-5.39,;6.67,-6.93,)|
COc1cnc(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(Cl)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1C |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;5.33,-7.7,;5.33,-9.24,;6.67,-10.01,;8,-9.24,;8,-7.7,;9.34,-6.93,;6.67,-6.93,;6.67,-5.39,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(Cl)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(Cl)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(F)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(F)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(F)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(F)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(Cl)c(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(F)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(F)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cnc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-4,-6.93,;-2.67,-9.24,;-1.33,-10.01,;-1.33,-11.55,;,-9.24,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)C1CCOCC1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-1.33,-10.01,;,-9.24,)|
COc1cc(OC)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(OC)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-6.67,.77,;-8,,;-8,-1.54,;-9.34,-2.31,;-6.67,-2.31,;-5.33,-1.54,)|
COc1cc(OC)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(ccc1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(ccc1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,)|
COc1cc(ccc1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cccc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1C)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;2.67,-10.78,;1.13,-9.24,;4.21,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-6.67,.77,;-8,,;-8,-1.54,;-9.34,-2.31,;-6.67,-2.31,;-5.33,-1.54,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;6.1,-10.99,;4.56,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccc(F)cn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-4,6.93,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;6.1,-10.99,;4.56,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncon1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccc(F)cn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-4,6.93,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccsn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnsn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Cl)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Cl)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(Cl)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Cl)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)on1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-5.68,5.93,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cscn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cc(F)cc(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-6.67,.77,;-8,,;-8,-1.54,;-6.67,-2.31,;-5.33,-1.54,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.33,-1.54,;-6.67,-2.31,;-8,-1.54,;-8,,;-6.67,.77,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-6.67,.77,;-8,,;-8,-1.54,;-9.34,-2.31,;-6.67,-2.31,;-5.33,-1.54,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nnc(C)s1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.33,5.93,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnc(C)cn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cncc(C)n1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
FC(F)(F)c1cccc(c1)-c1ccc(cc1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1Cl |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1C |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1ccc(cc1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-8.47,;-.77,-10.57,;.77,-7.91,)|
COc1ccccc1-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(F)cc(c1)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1ccc(cc1C#N)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;6.67,-13.09,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1F)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(C)c1Cl |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(Cl)c1C |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
CCOc1cccc(c1)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-14.63,;5.33,-13.86,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cccc(c1F)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1ccc(F)c(c1)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(ccc1C)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(C)cc(c1)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cccc(c1C)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1C)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cc(C)ccc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
Cc1cc(ccc1Cl)-c1cc(C)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
Cc1cc(ccc1Cl)-c1cc(C)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1 |(5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
Cc1cc(ccc1Cl)-c1cc(C)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
Cc1cc(ccc1Cl)-c1cc(C)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2cc(F)c(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2cc(F)c(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(Cl)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2cc(F)c(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2cc(F)c(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2cc(F)c(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COCc1cc(NS(=O)(=O)c2ccc3n(-c4cc(F)c(Br)cc4OC)c(=O)ccc3c2)ncn1 |(,7.7,;-1.33,6.93,;-1.33,5.39,;-2.67,4.62,;-2.67,3.08,;-4,2.31,;-4,.77,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-7.7,;2.67,-9.24,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-2.31,;5.33,-3.08,;4,-.77,;2.67,,;1.33,-.77,;;-5.33,3.08,;-5.33,4.62,;-4,5.39,)|
COc1cc(NS(=O)(=O)c2ccc3n(-c4cc(F)c(Br)cc4OC)c(=O)ccc3c2)ncn1 |(-1.33,6.93,;-1.33,5.39,;-2.67,4.62,;-2.67,3.08,;-4,2.31,;-4,.77,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-7.7,;2.67,-9.24,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-2.31,;5.33,-3.08,;4,-.77,;2.67,,;1.33,-.77,;;-5.33,3.08,;-5.33,4.62,;-4,5.39,)|
CCc1nccc(NS(=O)(=O)c2ccc3n(-c4cc(F)c(Br)cc4OC)c(=O)ccc3c2)n1 |(-6.67,6.93,;-6.67,5.39,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;-4,2.31,;-4,.77,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-7.7,;2.67,-9.24,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-2.31,;5.33,-3.08,;4,-.77,;2.67,,;1.33,-.77,;;-5.33,3.08,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccc(C)n1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-1.33,5.39,;-2.67,3.08,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nccc(C)n1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-1.33,5.39,;-2.67,3.08,)|
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,)|
CCc1nccc(NS(=O)(=O)c2ccc3n(-c4cc(F)c(cc4OC)-c4cc(F)cc(Cl)c4)c(=O)ccc3c2)n1 |(-6.67,6.93,;-6.67,5.39,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;-4,2.31,;-4,.77,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;4,-2.31,;5.33,-3.08,;4,-.77,;2.67,,;1.33,-.77,;;-5.33,3.08,)|
COc1cc(NS(=O)(=O)c2ccc3n(-c4cc(F)c(cc4OC)-c4cc(F)cc(Cl)c4)c(=O)ccc3c2)ncn1 |(-1.33,6.93,;-1.33,5.39,;-2.67,4.62,;-2.67,3.08,;-4,2.31,;-4,.77,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;4,-2.31,;5.33,-3.08,;4,-.77,;2.67,,;1.33,-.77,;;-5.33,3.08,;-5.33,4.62,;-4,5.39,)|
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,)|
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(ccc1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,)|
COc1cc(ccc1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(ccc1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(cc1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;4.21,-13.86,;1.13,-13.86,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(ccc1F)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(F)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C#N |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(c1)C#N |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C#N |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;,-7.7,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)cc(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)c(F)cc1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1ccc(cc1Cl)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1Cl)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)ccc1Cl |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1ccc(Cl)c(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)ccc1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1ccc(F)c(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1ccc(Cl)cc1-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(C)cc1-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(C)c(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1Cl)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(ccc1Cl)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1Cl)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1Cl)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1Cl)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Fc1cc(F)cc(c1)-c1ccc(c(c1)C1CC1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.1,-3.29,;6.87,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Fc1cc(F)cc(c1)-c1ccc(c(c1)C1CC1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.1,-3.29,;6.87,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
Fc1cc(F)cc(c1)-c1ccc(c(c1)C1CC1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.1,-3.29,;6.87,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
Fc1cc(F)cc(c1)-c1ccc(c(c1)C1CC1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nncs1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.1,-3.29,;6.87,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Fc1cc(F)cc(c1)-c1ccc(c(c1)C1CC1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nncs1 |(,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.1,-3.29,;6.87,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Fc1cc(F)cc(c1)-c1ccc(c(c1)C1CC1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncns1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.1,-3.29,;6.87,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.76,3.22,;-3.23,4.68,;-4.77,4.68,;-5.25,3.22,)|
Fc1cc(F)cc(c1)-c1ccc(c(c1)C1CC1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncns1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-4.62,;6.1,-3.29,;6.87,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-2.76,3.22,;-3.23,4.68,;-4.77,4.68,;-5.25,3.22,)|
COc1cc(Br)ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;6.67,-8.47,;6.1,-10.57,;4.56,-7.91,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(ccc1C)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;,-12.32,;-1.33,-13.09,;.77,-13.65,;-.77,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)ccc1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1Cl |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1Cl |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)cc1Cl |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1ccc(c(Cl)c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;4,-11.55,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cc1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(C)ccc1-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)c(F)cc1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)c(F)cc1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cc(Cl)ccc1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cc(Cl)ccc1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cc(Cl)ccc1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-11.55,;5.33,-13.86,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(Cl)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(ccc1Cl)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1ccc(CC(=O)OC(C)(C)C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;1.33,-10.01,;-1.33,-10.01,;-1.33,-11.55,;-1.33,-13.09,;-2.87,-11.55,;.21,-11.55,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Cc1cc(ccc1Cl)-c1cc(OCC#N)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;-2.67,-4.62,;-4,-3.85,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Oc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1 |(,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
C[C@@H](Oc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)C#N |wU:1.0,(6.67,-6.93,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;8,-4.62,;9.34,-3.85,)|
Fc1cc(c(OCC#N)cc1Br)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;9.34,-3.85,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
Fc1cc(c(O[C@@H]2CCNC2)cc1Br)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wD:6.5,(,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;8.08,-4.76,;9.11,-5.91,;8.34,-7.24,;6.83,-6.92,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
C[C@@H](Oc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(F)c1)C#N |wD:1.0,(-1.33,-6.93,;-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;-2.67,-4.62,;-4,-3.85,)|
Fc1cc(F)cc(c1)-c1cc(OC2CNC2)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;-1.73,-6.88,;-3.22,-6.48,;-2.82,-4.99,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccc(F)cn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-4,6.93,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncon1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnsn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccsn1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nncs1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncns1)-c1ccc(Cl)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.76,3.22,;-3.23,4.68,;-4.77,4.68,;-5.25,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(C2CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;3.91,-10.15,;3.44,-11.61,;1.9,-11.61,;1.42,-10.15,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(CC(C)(C)C)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;5.33,-10.78,;3.23,-11.34,;4.77,-8.68,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(CC2CCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;.94,-11.5,;-.55,-11.1,;-.15,-9.61,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cc(F)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(CC2CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.17,-11.54,;-.33,-11.86,;-1.1,-10.53,;-.07,-9.38,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(CC2C[C@@H]3CC[C@@H]2C3)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |r,wU:8.13,11.12,TLB:5:6:12:9.10,(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.73,-11.5,;.19,-11.5,;-.9,-9.47,;-.4,-7.99,;,-9.24,;-1.18,-12.45,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc([C@@H]2CC[C@H](C)CC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wU:8.8,5.4,(5.45,-2.16,;4.11,-1.39,;2.78,-2.16,;2.78,-3.7,;1.45,-4.47,;1.45,-6.01,;.11,-6.78,;.11,-8.32,;1.45,-9.09,;1.45,-10.63,;2.78,-8.32,;2.78,-6.78,;.11,-3.7,;-1.22,-4.47,;.11,-2.16,;1.45,-1.39,;1.45,.15,;.11,.92,;-1.22,.15,;-2.55,.92,;-2.55,2.46,;-1.22,3.23,;.11,2.46,;1.45,3.23,;2.78,2.46,;2.78,.92,;4.11,.15,;-3.89,3.23,;-4.66,1.9,;-3.12,4.57,;-5.22,4,;-5.22,5.54,;-6.47,6.45,;-5.99,7.91,;-4.45,7.91,;-3.98,6.45,)|
COc1cc(C2CCOCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
CO[C@H]1CC[C@H](CC1)c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |r,wD:5.8,2.1,(4,-14.63,;2.67,-13.86,;2.67,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;1.33,-2.31,;,-3.08,;8,,;7.23,1.33,;8.77,-1.33,;9.34,.77,;10.67,,;10.83,-1.53,;12.34,-1.85,;13.11,-.52,;12.08,.63,)|
COc1cc(CC2C[C@@H]3CC[C@@H]2O3)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |r,wU:8.13,wD:11.12,(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;-.6,-10.61,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;1.33,-2.31,;,-3.08,;8,,;7.23,1.33,;8.77,-1.33,;9.34,.77,;10.67,,;10.83,-1.53,;12.34,-1.85,;13.11,-.52,;12.08,.63,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,)|
COc1cccc(c1)-c1nc(OC)c(cc1Cl)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc([C@@H]2CCOC(C)(C)C2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wD:5.4,(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;.52,-12.86,;-.21,-11.6,;1.33,-10.01,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cc(F)cc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(C2CCC(F)(F)CC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;3.39,-13.68,;1.94,-13.68,;1.33,-11.55,;1.33,-10.01,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
CCOc1cccc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-14.63,;5.33,-13.86,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(F)(F)F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;5.33,-15.4,;6.87,-13.86,;3.79,-13.86,;4,-10.01,)|
COc1cccc(c1Cl)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(C)C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;5.33,-13.86,;6.67,-11.55,)|
COc1cc(ccc1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cccc(c1F)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(F)F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cccc(c1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C1CC1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.87,-12.32,;6.1,-13.65,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc2CCOc12 |(8.92,-7.17,;10.26,-7.94,;11.59,-7.17,;11.59,-5.63,;12.93,-4.86,;14.26,-5.63,;14.26,-7.17,;12.93,-7.94,;12.93,-9.48,;14.26,-10.25,;15.59,-9.48,;16.93,-10.25,;16.93,-11.79,;15.59,-12.56,;14.26,-11.79,;12.93,-12.56,;11.59,-11.79,;11.59,-10.25,;10.26,-9.48,;18.26,-12.56,;19.03,-11.22,;17.49,-13.89,;19.59,-13.33,;19.59,-14.87,;20.84,-15.77,;20.36,-17.24,;18.82,-17.24,;18.35,-15.77,;12.93,-3.32,;14.26,-2.55,;14.26,-1.01,;12.93,-.24,;11.59,-1.01,;10.13,-.53,;9.22,-1.78,;10.13,-3.02,;11.59,-2.55,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C1CC1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.87,-12.32,;6.1,-13.65,)|
CCc1cccc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1OC |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,;6.67,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,;6.67,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(OC)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(n1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(cc1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;1.33,-2.31,;,-3.08,;8,,;8.77,-1.33,;7.23,1.33,;9.34,.77,;10.67,,;10.83,-1.53,;12.34,-1.85,;13.11,-.52,;12.08,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;2.67,-13.86,;1.33,-14.63,;1.33,-16.17,;2.67,-16.94,;2.67,-18.48,;4,-16.17,;4,-14.63,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(cc1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cccc(n1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1ccnc(n1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc2CCOc2c1 |(16.79,-10.01,;18.12,-9.24,;18.12,-7.7,;16.79,-6.93,;16.79,-5.39,;18.12,-4.62,;19.46,-5.39,;19.46,-6.93,;20.79,-7.7,;22.12,-6.93,;22.12,-5.39,;23.46,-4.62,;24.79,-5.39,;24.79,-6.93,;23.46,-7.7,;23.46,-9.24,;22.12,-10.01,;20.79,-9.24,;19.46,-10.01,;26.13,-4.62,;25.36,-3.29,;26.9,-5.95,;27.46,-3.85,;28.79,-4.62,;30.2,-3.99,;31.23,-5.14,;30.46,-6.47,;28.95,-6.15,;15.46,-4.62,;15.46,-3.08,;14.12,-2.31,;12.79,-3.08,;11.32,-2.6,;10.42,-3.85,;11.32,-5.1,;12.79,-4.62,;14.12,-5.39,)|
CCc1cccc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(OC)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;,-7.7,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,;6.67,-10.01,)|
COc1cc(Cl)ccc1-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)[N-][n+]1ccccc1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1nc(OCC2CC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;4.77,-12.88,;3.23,-12.88,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1nc(OC2CCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;.94,-11.5,;-.55,-11.1,;-.15,-9.61,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCC2(C)CC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.78,-11.02,;1.2,-13.08,;-.06,-12.2,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(C)C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1nc(OCC2CCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.25,-12.46,;4.77,-13.92,;3.23,-13.92,;2.76,-12.46,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OC2CCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.17,-11.54,;-.33,-11.86,;-1.1,-10.53,;-.07,-9.38,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-6.67,.77,;-8,,;-8,-1.54,;-9.34,-2.31,;-6.67,-2.31,;-5.33,-1.54,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1nc(C2CC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;3.44,-10.57,;1.9,-10.57,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COCCCOc1nc(OC)c(cc1Cl)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(14.67,-2.31,;13.34,-3.08,;12,-2.31,;10.67,-3.08,;9.34,-2.31,;8,-3.08,;6.67,-2.31,;5.33,-3.08,;4,-2.31,;2.67,-3.08,;2.67,-4.62,;4,-.77,;5.33,,;6.67,-.77,;8,,;2.67,,;1.33,-.77,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;,1.54,;1.33,2.31,;2.67,1.54,;4,2.31,;-2.67,-3.08,;-1.9,-4.41,;-3.44,-1.75,;-4,-3.85,;-5.33,-3.08,;-6.74,-3.71,;-7.77,-2.56,;-7,-1.23,;-5.5,-1.55,)|
COc1nc(OCC(F)(F)C(F)(F)F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;-.21,-11.55,;2.87,-11.55,;1.33,-13.09,;1.33,-14.63,;-.21,-13.09,;2.87,-13.09,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCC(F)(F)F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;1.33,-13.09,;-.21,-11.55,;2.87,-11.55,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccc(F)cn1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-4,6.93,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncon1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cccc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cccc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncon1)-c1cccc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(CC2CCCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cnccn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(C[C@H]2CCCOC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wU:6.5,(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;6.67,-10.01,;6.67,-11.55,;5.33,-12.32,;4,-11.55,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cccc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-6.67,.77,;-8,,;-8,-1.54,;-9.34,-2.31,;-6.67,-2.31,;-5.33,-1.54,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(CC2CCOCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;6.67,-11.55,;6.67,-10.01,;5.33,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC2CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC(C)(C)C)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;2.67,-13.86,;1.13,-12.32,;4.21,-12.32,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C[C@@H]2CCOC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wD:6.5,(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;5.41,-9.38,;6.44,-10.53,;5.67,-11.86,;4.16,-11.54,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(C)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(C#CC(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;2.67,-13.86,;1.13,-12.32,;4.21,-12.32,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(C)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(C)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(C)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(C)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(C)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(C#CC2CC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.44,-13.65,;1.9,-13.65,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cccc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cccc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(C[C@H]2CCCCO2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wU:6.5,(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC2CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(C#CC2CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(C#CC2CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)cnn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-6.67,5.39,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(C#CC2CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccc(C)nn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-4,6.93,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1nc(C#CC2CCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(C#CC(C)(C)OC)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;1.13,-12.32,;4.21,-12.32,;2.67,-13.86,;4,-14.63,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC(C)(C)O)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;2.67,-13.86,;1.13,-12.32,;4.21,-12.32,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(NC2CCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.17,-11.54,;-.33,-11.86,;-1.1,-10.53,;-.07,-9.38,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(c(Cl)c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;4,-11.55,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1Cl)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccccc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,)|
COc1ccc(c(F)c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;4,-11.55,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1ccc(cc1Cl)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1ccc(cc1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(C)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cccc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(F)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1C |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(C)cc1-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)ccc1Cl |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(ccc1C)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;,-12.32,;-1.33,-13.09,)|
COc1ccc(cc1-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)C#N |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-12.32,;-1.33,-13.09,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,)|
COc1cc(ccc1C#N)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-15.4,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cncc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cnc(F)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Cl)cc(c1)-c1cc(OC)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-2.67,-16.94,;-1.33,-16.17,;-1.33,-14.63,;-2.67,-13.86,;-2.67,-12.32,;-4,-11.55,;-1.33,-11.55,;,-12.32,;,-13.86,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;1.33,-2.31,;,-3.08,;8,,;8.77,-1.33,;7.23,1.33,;9.34,.77,;10.67,,;10.83,-1.53,;12.34,-1.85,;13.11,-.52,;12.08,.63,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-11.55,;5.33,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(C)cc(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1ccc(C)c(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)cc1Cl |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1ccc(Cl)c(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
CCOc1cccc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-14.63,;5.33,-13.86,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(F)(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;6.67,-11.55,;8,-10.78,;7.44,-12.88,;5.9,-10.22,;4,-10.01,)|
COc1ccc(cn1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cncc(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cccc(c1Cl)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1ccc(F)c(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cc1F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cccc(c1F)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cccc(c1C)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccnc(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccnc1C |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,)|
COc1cncc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccn1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(F)ccc1-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cc1C |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1C |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,)|
COc1ccc(Cl)cc1-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-10.01,;5.33,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;1.33,-10.01,;2.67,-9.24,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccnc(OC)c1Cl |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;,-13.86,;1.33,-10.01,;,-9.24,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1OC |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;5.33,-9.24,;6.67,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccncc1Cl |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,)|
COc1ccc(cc1C)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(4,-14.63,;2.67,-13.86,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(cc1)C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)cc1C(N)=O |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;4,-10.01,;5.33,-9.24,;5.33,-7.7,;6.67,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(cc1)C1CC1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;3.44,-15.19,;1.9,-15.19,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1C#N |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-9.24,;6.67,-8.47,)|
COc1cc(c(Cl)cn1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;4,-11.55,;2.67,-12.32,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(OC(F)(F)F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;5.33,-15.4,;3.23,-15.96,;4.77,-13.3,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(nc1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;2.67,-13.86,;2.67,-15.4,;1.13,-13.86,;4.21,-13.86,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccnc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-12.32,;-1.33,-13.09,;-.77,-10.99,;.77,-13.65,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(OC(F)F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-14.63,;1.33,-16.17,;,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ncc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(Cl)cc1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cc(Cl)cnc1OC |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;2.67,-12.32,;1.33,-11.55,;1.33,-10.01,;,-9.24,;-1.33,-10.01,)|
COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)C#CC1CCCC1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;-1.33,-8.47,;-2.67,-9.24,;-2.83,-10.77,;-4.33,-11.09,;-5.1,-9.76,;-4.07,-8.61,)|
COc1ccc(CC#N)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;,-10.78,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cnc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(Cl)ccc1F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-4,-6.93,;-2.67,-9.24,;-1.33,-10.01,;,-9.24,;1.33,-10.01,)|
COc1ccccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,)|
COc1cc(OC)cc(c1)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;2.67,-12.32,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;1.33,-10.01,;2.67,-9.24,;4,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cccc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.5,-1.53,;-7,-1.85,;-7.77,-.52,;-6.74,.63,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(F)c(F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-5.33,,;-5.33,-1.54,;-6.67,-2.31,;-8,-1.54,;-8,,;-6.67,.77,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(C#CC2CCCC2)c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(OCC2CC2)ncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-1.33,6.93,;,7.7,;.77,9.03,;1.54,7.7,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(OCC2CCC2)ncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-1.33,6.93,;,7.7,;.4,9.19,;1.89,8.79,;1.49,7.3,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(OCC2CCCC2)ncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-1.33,6.93,;,7.7,;.16,9.23,;1.67,9.55,;2.44,8.22,;1.41,7.07,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
CCCOc1cc(NS(=O)(=O)c2ccc3n(-c4cc(F)c(Br)cc4OC)c(=O)ccc3c2)ncn1 |(,9.24,;,7.7,;-1.33,6.93,;-1.33,5.39,;-2.67,4.62,;-2.67,3.08,;-4,2.31,;-4,.77,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;2.67,-7.7,;2.67,-9.24,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-2.31,;5.33,-3.08,;4,-.77,;2.67,,;1.33,-.77,;;-5.33,3.08,;-5.33,4.62,;-4,5.39,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(OCC(C)C)ncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-1.33,6.93,;,7.7,;,9.24,;1.33,6.93,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(OC2CCC2)ncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-1.33,6.93,;-2.42,8.02,;-1.33,9.11,;-.24,8.02,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Br)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(OCC2(C)CC2)ncn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-1.33,6.93,;,7.7,;-1.18,8.69,;1.4,8.35,;1.26,6.82,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(Cl)cc(c1)-c1ccc(c(OC)c1)-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1 |(,-13.86,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1C)-c1ccc(c(OC)c1)-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1 |(5.33,-13.86,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;4,-6.93,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ncccn1)-c1ccc(Cl)c(C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ncccn1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(ccc1Cl)-c1cc(OC)c(cc1F)-n1c2ccc(cc2ncc1=O)S(=O)(=O)Nc1ncccn1 |(6.67,-11.55,;5.33,-12.32,;4,-11.55,;4,-10.01,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;,-4.62,;-1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;5.33,-7.7,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-5.33,3.08,)|
COc1cc(Oc2ccc(F)cc2)ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-2.67,-12.32,;-1.33,-10.01,;,-9.24,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
Fc1cccc(c1)[C@@H]1CC[C@H](C1)n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1nccc(C)n1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-1.33,5.39,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccc(F)n1)-c1cccc(OC(C)C)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-1.33,5.39,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccc(F)n1)-c1cccc(c1)C(F)(F)F |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-1.33,5.39,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;4.56,-13.65,;6.1,-10.99,)|
COc1cc(C2CC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;3.44,-10.57,;1.9,-10.57,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C2CC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;3.44,-10.57,;1.9,-10.57,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)C1CC1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;3.44,-10.57,;1.9,-10.57,)|
COc1nc(OCC(F)(F)C2CCOCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;-.21,-11.55,;2.87,-11.55,;1.33,-13.09,;,-13.86,;,-15.4,;1.33,-16.17,;2.67,-15.4,;2.67,-13.86,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(O[C@H](C)C(F)(F)C(F)F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wD:6.6,(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;5.33,-9.24,;4,-11.55,;2.46,-11.55,;5.54,-11.55,;4,-13.09,;5.33,-13.86,;2.67,-13.86,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCc2ccc(F)cc2F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-16.17,;5.33,-13.86,;5.33,-12.32,;6.67,-11.55,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCc2ccc(F)cc2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;4,-14.63,;4,-16.17,;2.67,-13.86,;2.67,-12.32,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCc2ccc(F)c(c2)C(F)(F)F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-16.17,;5.33,-13.86,;5.33,-12.32,;6.67,-14.63,;8,-15.4,;5.9,-15.96,;7.44,-13.3,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCc2ccc(F)c(F)c2F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-16.17,;5.33,-13.86,;6.67,-14.63,;5.33,-12.32,;6.67,-11.55,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCc2cc(F)c(F)c(F)c2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-16.17,;2.67,-13.86,;1.33,-14.63,;2.67,-12.32,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OCC2CCCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;4,-14.63,;2.67,-13.86,;2.67,-12.32,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(Oc2ccc(F)cc2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;,-12.32,;-1.33,-11.55,;-2.67,-12.32,;-1.33,-10.01,;,-9.24,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(Oc2ccc(F)cc2F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;-2.67,-12.32,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(Oc2ccc(F)c(F)c2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;-2.67,-12.32,;,-12.32,;,-13.86,;1.33,-11.55,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(OC2C[C@H]3CC[C@@H]2C3)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |r,wU:11.12,wD:8.13,(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;.27,-10.25,;-1.22,-9.86,;-1.61,-8.37,;-.84,-7.03,;.64,-7.43,;-.31,-8.48,;-2.46,-7.22,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(O[C@H]2CCCC[C@H]2C)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wD:11.12,6.5,(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(Oc2cc(F)ccc2F)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;,-9.24,;-1.33,-10.01,;-2.67,-9.24,;-1.33,-11.55,;,-12.32,;1.33,-11.55,;2.67,-12.32,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(Oc2cccc(Cl)c2C)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;,-12.32,;,-13.86,;1.33,-11.55,;2.67,-12.32,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(C2CC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.09,-5.71,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;3.44,-10.57,;1.9,-10.57,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(N(C)C2CCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;1.33,-10.01,;1.17,-11.54,;-.33,-11.86,;-1.1,-10.53,;-.07,-9.38,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(NC[C@H]2CCC(C)(C)O2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wU:7.6,(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.58,-12.46,;2.1,-13.92,;.56,-13.92,;.39,-15.45,;-.84,-14.56,;.09,-12.46,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC2(C)COC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;1.3,-11.62,;2.31,-13.82,;3.81,-14.18,;4.16,-12.68,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC2(O)CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.98,-11.52,;3.31,-13.72,;2.17,-14.76,;.83,-14.01,;1.14,-12.5,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC2(F)CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.98,-11.52,;3.31,-13.72,;2.17,-14.76,;.83,-14.01,;1.14,-12.5,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C[C@H]2CCOC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |wU:6.5,(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;4,-10.01,;5.41,-9.38,;6.44,-10.53,;5.67,-11.86,;4.16,-11.54,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1nc(NCC2(C)CCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.65,-10.75,;1.97,-12.95,;.84,-13.99,;-.5,-13.24,;-.2,-11.73,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,)|
COc1cc(C#CC2(F)CCCC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.98,-11.52,;3.31,-13.72,;2.17,-14.76,;.83,-14.01,;1.14,-12.5,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)C#CC1CCCC1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;2.67,-10.78,;2.67,-12.32,;3.91,-13.23,;3.44,-14.69,;1.9,-14.69,;1.42,-13.23,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccc(F)n1)-c1cccc(c1)C(F)(F)F |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-1.9,1.33,;-3.44,-1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-1.33,5.39,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;4,-11.55,;4,-10.01,;5.33,-12.32,;6.67,-13.09,;6.1,-10.99,;4.56,-13.65,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncc(F)cn1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ncco1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cc(C)ncn1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-1.33,5.39,;-4,5.39,;-5.33,4.62,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccnc(C)n1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-2.67,3.08,;-2.67,4.62,;-4,5.39,;-5.33,4.62,;-6.67,5.39,;-5.33,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccc(F)cn1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-4,6.93,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1cccc(F)n1)-c1cnc(OC)c(Cl)c1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-2.67,4.62,;-1.33,5.39,;-2.67,3.08,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-14.63,;4,-11.55,;5.33,-12.32,;4,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccc(F)cn1)-c1ccc(Cl)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.33,3.08,;-5.33,4.62,;-4,5.39,;-4,6.93,;-2.67,4.62,;-2.67,3.08,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)cc1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;4,-10.01,;4,-11.55,;2.67,-12.32,;2.67,-13.86,;1.33,-11.55,;1.33,-10.01,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(OC(F)F)c1 |(-1.33,-5.39,;,-4.62,;1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;5.33,-7.7,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;-2.67,,;-3.44,-1.33,;-1.9,1.33,;-4,.77,;-4,2.31,;-5.25,3.22,;-4.77,4.68,;-3.23,4.68,;-2.76,3.22,;2.67,-9.24,;1.33,-10.01,;1.33,-11.55,;2.67,-12.32,;2.67,-13.86,;4,-11.55,;5.33,-12.32,;5.33,-13.86,;6.67,-14.63,;4,-14.63,;4,-10.01,)|
COC1(F)C=C(C(F)=CC1n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)c1ccc(F)c(F)c1 |c:4,7|
Oc1ccccc1Cc1cccc(n1)-c1ccc(OCC(F)(F)F)nc1
COc1ncccc1-c1ccccc1Cc1cccc(n1)-c1ccc(OCC(F)(F)F)nc1
Fc1ccc(cn1)-c1ccccc1Cc1cccc(n1)-c1ccc(OCC(F)(F)F)nc1
COc1ncc(cn1)-c1ccccc1Cc1cccc(n1)-c1ccc(OCC(F)(F)F)nc1
CSc1ncc(cn1)-c1ccccc1Cc1cccc(n1)-c1ccc(OCC(F)(F)F)nc1
CN(C)c1ncc(cn1)-c1ccccc1Cc1cccc(n1)-c1ccc(OCC(F)(F)F)nc1
Cc1cc(ccc1OC2CN(C2)c3ccnc(n3)Nc4cccc(c4)C(=O)NC)F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CCC(CC2)c2nc(cs2)-c2ccccc2)ccc1F
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)ccc1F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(cc3)C(F)(F)F)C2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(cc2)C(F)(F)F)ccc1F
CNC(=O)c1cccc(Nc2ccnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)c(C)c2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CCc3cc(OCC(F)(F)F)ccc3C2)ccc1Cl
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)c(F)c2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(Cl)cc2C)c1
CNC(=O)c1cccc(Nc2ncnc(NCCCOc3ccc(OC(F)(F)F)cc3)n2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)ccc1F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)c(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2C)c1
CCc1cccc(OC2CN(C2)c2ncnc(Nc3cccc(c3)C(=O)NC)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cc(Cl)ccc2Cl)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(Cl)c(C)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2C)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc3CCCc3c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(OC(F)(F)F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2nc(cs2)-c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2csc(n2)-c2ccccc2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CCC(CC2)c2nc(cs2)-c2ccccc2)ccc1Cl
COCCNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2Cl)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(OC)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(C)cc2Cl)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(C)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(cc2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)C(=O)c2ccc(Cl)cc2)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)c1
COCCNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)c(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(OCC(F)(F)F)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(cc2)C(C)C)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(c2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(OC)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(=CC2)c2csc(n2)-c2ccccc2)c1 |c:20|
COCCNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2cccc(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(C)c2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)ccc1N(C)C
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2Cl)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(=CC2)c2nc(cs2)-c2ccccc2)c1 |c:20|
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(C)c(C)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2Cl)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(Cl)c(F)c2)c1
CNC(=O)c1cccc(Nc2cccc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)ccc1F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(Cl)c(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(c2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2c(Cl)cccc2Cl)c1
CNC(=O)c1cc(Nc2ncnc(NCCCOc3ccc(OC(F)(F)F)cc3)n2)ccc1F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cc(C)ccc2Cl)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(OC(F)(F)F)cc3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(OC(F)(F)F)c(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(Cl)c2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3)C2)ccc1F
CNC(=O)c1cccc(Nc2ccnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(C2)cccc3C#N)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3C)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(cc2)C(F)(F)F)c1
CNC(=O)c1cc(Nc2ncnc(NCCCOc3ccc(OC(F)(F)F)cc3)n2)ccc1Cl
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(C)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(OCCC(F)(F)F)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(c2)C#C)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)ccc1Cl
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(OC)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(C)c2C)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(SC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(Cl)c(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccccc2Cl)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(OC)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)C(=O)c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccccc2C)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3)C2)ccc1Cl
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)c(F)c3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(ccc3C2)C2CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(COc3ccc(F)c(F)c3)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)OCc2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccccc2F)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(COc3ccc(cc3)C(F)(F)F)C2)ccc1Cl
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)c(Cl)c2)ccc1Cl
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(=CC2)c2ccc(cc2)C#N)c1 |c:20|
CNC(=O)c1cccc(Nc2ncnc(N[C@H](C)CCc3ccccc3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(OCC(F)(F)F)cc2)c1
CCNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CCC(CC2)c2nc(cs2)-c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(Cl)c2Cl)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3F)C2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(F)c(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCCN(CC2)c2ncc(cc2Cl)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(Cl)cn2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CCc3ccccc3)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(OC(F)(F)F)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(OC(F)(F)F)c2)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CC(COc3ccc(cc3)C(F)(F)F)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)OCc2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(C)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccccc2)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(C)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccc(C)c(C)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(cc2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2cccc(OC(F)(F)F)c2)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)c(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2cccc(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(C2)cccc3OC(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)C#Cc2ccccc2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(F)cc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)S(=O)(=O)c2ccc(OC(F)(F)F)cc2)c1
CCn1c2CCN(Cc2c2ccccc12)c1ncnc(Nc2cccc(c2)C(=O)NC)n1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(C#N)c(Cl)c2)c1
CNC(=O)c1ccc(Cl)c(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(Cl)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3Cl)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(=CC2)c2ccc(C)c(C)c2)c1 |c:20|
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(c2)C(C)(C)C)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(=CC2)c2ccc(OC(F)(F)F)cc2)c1 |c:20|
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(C2)cccc3OCC(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(C2)cccc3OC)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)n2cc(cn2)-c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2nc(no2)-c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(Cl)cccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(COc3ccccc3)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(C2)cnn3-c2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(Cl)cc2)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)(C#N)c2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(cc2)C(C)(C)C)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(cc2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(Cc3ccc(F)c(F)c3)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(NCCCOc3ccc(Cl)cc3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2c(F)cc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC[C@@H](C2)Oc2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cc(C)ccc2F)c1
CNC(=O)c1cccc(Nc2ncnc(NCCCOc3ccc(OC(F)(F)F)cc3)n2)c1C
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)c(Cl)c3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(OC)cc2)c1
CNC(=O)c1ccc(C)c(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1c(F)ccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3)C2)c1F
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)ccc1Cl
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(F)cc3)C2)c1
CNC(=O)c1cc(Nc2ncnc(NCCCOc3cccc(c3)C(F)(F)F)n2)ccc1Cl
CNC(=O)c1ccc(F)c(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(Cl)c(OC(F)(F)F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)n2cc(cn2)-c2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2nc(c(C)s2)-c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(NCCCOc3ccc(cc3)C(F)(F)F)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccc(cc2)C#N)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3cccc(OC(F)(F)F)c3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccccc2OC(F)(F)F)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)cc3)C2)c1
Fc1ccc(OC2CN(C2)c2ncnc(Nc3cccc(c3)C(=O)NCC(F)(F)F)n2)cc1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccccn2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(F)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cc(F)ccc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccccc2C(F)(F)F)c1
CNC(=O)c1cccc(Nc2cc(ccn2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(Cc3ccc(OC(F)(F)F)cc3)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2OC(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C)(C2)Oc2ccc(C)cc2)c1
CNC(=O)c1c(F)ccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)c1F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)c2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(C)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)[C@@H](C)Oc2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cc(F)cc(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3cccc(c3)C(F)(F)F)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COCc3ccc(cc3)C(F)(F)F)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)n2cc(cn2)-c2ccccc2Cl)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(Cc3ccccc3OC(F)(F)F)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(F)c(OC(F)(F)F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(cc2Cl)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(cc2)C#N)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(Cc3ccc(F)cc3)CC2)c1
CNC(=O)c1cccc(Nc2ccnc(n2)N2CC(COc3ccc(Cl)cc3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(c2)-c2ccccc2)c1
NC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3cccc(Cl)c3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(OC(F)(F)F)cc2)c1C
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCCN(Cc3ccccc3)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2OC)c1
Fc1ccc(OC2CN(C2)c2ncnc(Nc3cccc(c3)C(=O)NC3CC3)n2)cc1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(CC#N)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)c(c3)C(F)(F)F)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccccc2OC(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(cc2)C#N)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC2COc2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCCC(C2)Oc2ccccc2Cl)c1
CC(C)(C)NC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(OCc3ccccc3)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccc(C#N)c(c2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(ccc3C2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2-c2ccccc2)c1
CNC(=O)c1cccc(Nc2cc(ncn2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)ccc1O
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3ccc(OC)cc3C2)c1
NC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(Br)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(OC)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(OC)cc3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cc(Cl)cc(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(F)cccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)c(F)c2F)c1
Cc1ccc(cc1C)N1CCN(CC1)c1ncnc(Nc2ccc(Cl)c(c2)C(N)=O)n1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(F)c(F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccccc3OC(F)(F)F)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(Cc3ccccc3)CC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2nc(no2)C(C)C)c1
CNC(=O)c1cccc(Nc2ncnc(NCCCc3ccc(Cl)cc3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(OCCOC)ccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc4ccccc4c3)C2)c1
NC(=O)c1cccc(Nc2ncnc(n2)N2CCc3ccccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(NCCOc3ccc(Cl)cc3)n2)c1
NC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccccc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2cccc(c2)C(F)(F)F)c1
CN(C)C(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COCc3ccc(Cl)cc3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3cccc(F)c3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3ccccc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3cccc(OC)c3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)(C#N)c2ccc(F)cc2)c1
CCCc1noc(n1)C1CCN(CC1)c1ncnc(Nc2cccc(c2)C(=O)NC)n1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccccc3Cl)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccc(C#N)c(OC(F)(F)F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Sc2ccc(C)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccccc3F)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(C2)cccc3OCCOC)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3cccc4ccccc34)C2)c1
CNC(=O)c1cccc(Nc2ncnc(NCc3nc(no3)-c3ccccc3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(Cl)c4cccnc34)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2cccc(c2F)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)Nc2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(cc3)C#N)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC3(CC2)OCc2ccccc32)c1
CNC(=O)c1cccc(Nc2ncnc(NCCCOc3cccc(F)c3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(COCC3CC3)CC2)c1
CNC(=O)c1cc(Cl)cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C)(C2)Oc2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(cc2)C2CCCC2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3oc(cc3C2)-c2ccccc2)c1
CNC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)ccc1C
Cc1c(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)cccc1C(N)=O
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3c(C2)cnn3-c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cccc(c3C2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)c1F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2ccc(F)c(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)OCc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C)(COc3ccccc3)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2c(F)cccc2F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(OCC(F)(F)F)ccc3C2)c1C
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccccc3C(F)(F)F)C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2cccc(OC(F)(F)F)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCCC(C2)Oc2cccc(Cl)c2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3ccc(Cl)cc3C2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N(C)Cc2nc(no2)-c2ccccc2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cccc(OC)c3C2)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(NCCCOc3ccc(OC(F)(F)F)cc3)n2)c1
CNC(=O)c1ccc(OC)c(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2)c1
CNC(=O)c1cccc(Nc2nc(C)nc(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncc(F)c(n2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2ncnc(NCc3cn4cc(C)ccc4n3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(NCCc3nnc(o3)-c3ccc(C)s3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(NCCc3nc4cc(Cl)ccc4[nH]3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(NCc3noc(n3)C(=O)NC3CC3)n2)c1
CCN1C(=O)C2(CCN(CC2)c2ncnc(Nc3cccc(c3)C(=O)NC)n2)c2ccccc12
NC(=O)c1cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(F)cc2)ccc1F
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(ccc3C2)C(O)C(F)(F)F)c1
Cc1c(Nc2ncnc(n2)N2CCc3cc(Br)ccc3C2)cccc1C(N)=O
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CCCc3ccccc3)CC2)c1
Cc1ccc(cc1C)N1CCN(CC1)c1ncnc(Nc2ccc(F)c(c2)C(N)=O)n1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCC(C)C)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccccc2C#N)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3ccc(cc3C2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCc3cc(ccc3C2)C#N)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(Cl)cc2Cl)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(C)cc2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(cc2)C(F)(F)F)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(F)c(Cl)c2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(F)c(C)c2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(F)cc2Cl)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(COc3ccc(Cl)cc3)C2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CC(COc3ccc(C)cc3)C2)c1
CCNC(=O)c1cccc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cc(F)cc(Nc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2cc(ccn2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2nc(C)nc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2ccnc(c2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2cccc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cc(Nc2cccc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)ccc1F
CNC(=O)c1cc(Nc2cccc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)ccc1Cl
CNC(=O)c1cccc(Nc2cc(ncn2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2ccnc(c2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2ncnc(N3CC(C3)Oc3ccc(Cl)cc3F)c2F)c1
CNC(=O)c1cccc(Nc2ccnc(NCCCOc3ccc(OC(F)(F)F)cc3)n2)c1
CNC(=O)c1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1C
CNC(=O)c1cccc(Oc2ncnc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2cccc(c2)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2cccc(c2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2nc(ncc2F)N2CC(C2)Oc2ccc(F)cc2)c1
CNC(=O)c1cccc(Nc2nccc(n2)N2CCc3cc(OCC(F)(F)F)ccc3C2)c1
CNC(=O)c1cccc(Nc2ccnc(n2)N2CC(C2)Oc2ccc(Cl)cc2F)c1
CNC(=O)c1cccc(Nc2nc(ncc2F)N2CC(C2)Oc2ccc(Cl)cc2F)c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(Br)c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(Cl)c1
Cn1nccc1-c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(Cl)c1
CC(C)(C)OC(=O)N1CCC(=CC1)c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F |c:10|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)C1=CCNCC1 |t:33|
NCc1nsc(NS(=O)(=O)c2ccc3N(CCOc3c2)c2ccc(cc2Cl)C(F)(F)F)n1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cc(Cl)ncn2)c(Cl)c1
Cc1nsc(NS(=O)(=O)c2ccc3N(CCOc3c2)c2ccc(cc2Cl)C(F)(F)F)n1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cscn2)c(Cl)c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccon2)c(Cl)c1
CN(C)CCn1ccc(NS(=O)(=O)c2ccc3N(CCOc3c2)c2ccc(cc2Cl)C(F)(F)F)n1
Cn1ccc(NS(=O)(=O)c2ccc3N(CCOc3c2)c2ccc(cc2Cl)C(F)(F)F)n1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(Cl)c1
Fc1ccc(NS(=O)(=O)c2ccc3N(CCOc3c2)c2ccc(cc2Cl)C(F)(F)F)nc1
FC(F)(F)c1ccc(N2CCNc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(Cl)c1
CN1CCN(c2ccc(cc2Cl)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
CC(=O)N1CCN(c2ccc(cc2Cl)C(F)(F)F)c2ccc(cc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)-c1cccnc1
CN1CCC(=CC1)c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F |c:4|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)-c1cncnc1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncco2)c(Cl)c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)C1=CCOCC1 |t:33|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)-c1ccncc1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(Cl)c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nncs2)c(Cl)c1
Nc1cc(ccn1)-c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
O=S(=O)(Nc1ncns1)c1ccc2N(CCOc2c1)c1ccccc1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)C#N
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(Cl)c1
O=S(=O)(Nc1ncns1)c1ccc2N(CCOc2c1)c1cccc2ncccc12
FC(F)(F)c1ccc(cc1)N1C(COc2cc(ccc12)S(=O)(=O)Nc1ncns1)c1ccccc1
FC(F)(F)Oc1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)c1ccc2N(CCOc2c1)c1cccc2ccccc12
COc1ccc(cc1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C1=CCNCC1 |t:33|
COCCOc1ccc(cc1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1
Clc1ccc(cc1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(Br)c1
CN1CCC(=CC1)c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |c:4|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)C1=CCNCC1 |t:34|
Clc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(Br)c1
COCCNc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
CN1CCN(CC1)c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
CN1CCC(=CC1)c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |c:4|
Clc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C1=CCNCC1 |t:30|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)-c1ccncc1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)-c1cncnc1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccno2)c(Cl)c1
Clc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
O=S(=O)(Nc1ncns1)c1ccc2N(CCOc2c1)c1ccccc1C#N
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1C#N
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1N1CCNCC1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccccn2)c(Br)c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cscn2)c(Br)c1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccccn2)c(c1)C1=CCNCC1 |t:34|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cscn2)c(c1)C1=CCNCC1 |t:33|
Brc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)N=[N+]=[N-]
[N-]=[N+]=Nc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C1=CCNCC1 |t:32|
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccc2ncccc2c1
Cc1ccc(Cl)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1cccc2ccncc12
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccc2nccnc2c1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccc2scnc2c1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccc2ncsc2c1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1cccc2scnc12
Cc1ccc2cnccc2c1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1ccc(cc1Cl)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccc(cc1)C#N
COc1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1c(F)cccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1ccc(F)cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1ccc(F)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(ccc1F)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1ccc(cc1F)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(F)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(cc1F)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)C1=CCNCC1 |t:34|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cccnn2)c(c1)C1=CCNCC1 |t:34|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cnccn2)c(c1)C1=CCNCC1 |t:34|
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)C#N
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ncco2)c(c1)C#N
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccno2)c(c1)C#N
CC1CN(c2ccc(cc2O1)S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F
C[C@H]1CN(c2ccc(cc2O1)S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F |r|
C[C@@H]1CN(c2ccc(cc2O1)S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F |r|
CC1COc2cc(ccc2N1c1ccc(cc1C#N)C(F)(F)F)S(=O)(=O)Nc1nccs1
C[C@@H]1COc2cc(ccc2N1c1ccc(cc1C#N)C(F)(F)F)S(=O)(=O)Nc1nccs1 |r|
C[C@H]1COc2cc(ccc2N1c1ccc(cc1C#N)C(F)(F)F)S(=O)(=O)Nc1nccs1 |r|
FC(F)(F)c1cnc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(Cl)c1
CCC1CN(c2ccc(cc2O1)S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F
CC[C@H]1CN(c2ccc(cc2O1)S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F |r|
COc1cc(Cl)cnc1N1CC(C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(Cl)ccc1N1C[C@H](C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1 |r|
COc1cc(Cl)ccc1N1C[C@@H](C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1 |r|
COc1cc(ccc1N1CC(C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(ccc1N1C[C@H](C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N |r|
COc1cc(ccc1N1C[C@@H](C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N |r|
COc1ccc(C)nc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(F)cnc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ncc(Cl)cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CC(C)c1ccc(cc1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)COc1ccc(cc1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
Cc1ccc(cc1C#N)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(ccc1C#N)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1cncc(c1)C#N
COc1ccc(cc1C#N)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(cc1OC)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(OC)c1
Clc1cnc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(Cl)c1
FC(F)(F)c1ccc(cn1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)C(F)(F)Oc1ccc(cc1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(cc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
FC(F)(F)c1cc(ccc1Cl)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(cc1Cl)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC1(F)Oc2ccc(cc2O1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)Oc1ccc(C#N)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC1(F)Oc2cccc(N3CCOc4cc(ccc34)S(=O)(=O)Nc3nccs3)c2O1
Clc1cncc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cncc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(C)n1
Cc1cncc(C)c1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(C)cn1
Cc1ccc(C#N)c(n1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1cnc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(F)c1
COc1cc(C)c(cn1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CCOc1ccc(cn1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(OC)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(OC(F)(F)F)ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccc(cc1)-n1cccn1
Clc1cccc(C#N)c1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cnc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(OC)n1
COc1cnc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(OC)c1
COc1ncc(cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
Cc1cc(OC(F)F)cnc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1-c1ccncc1
Cn1nccc1-c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1C1CCOCC1
COc1cc(F)ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(F)cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2cscn2)c(c1)C#N
COc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccc(cc1)-n1ccnc1
Fc1cc(ccc1Cl)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(ccc1Cl)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cnccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1cccc(C#N)c1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=C1CCCc2ccc(cc12)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CN(C)c1c(C)cc(cc1C)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CCOc1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1ccc(cc1Cl)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1cccc2cccnc12
FC(F)(F)Oc1cc(ccc1C#N)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CC(C)c1ccc(C)cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1c(Cl)cccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1cc(Cl)ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1cccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c1Cl
FC(F)Oc1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1cccc(CC#N)c1
Fc1ccc(cc1C#N)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(F)c1
Fc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
Cc1ccc(Cl)cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)Oc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1ccc(Cl)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(nc1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(C#N)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)Oc1cccc(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(Cl)ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Fc1cccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c1C#N
Fc1ccc(C#N)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(C#N)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccncc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
Clc1ccc(C#N)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)Oc1cc(Cl)ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1ccc(C#N)c(c1)N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(Cl)ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
[O-][N+](=O)c1ccc(OC(=O)N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)cc1
Fc1ccccc1-c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
Fc1ccc(cc1)-c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
Fc1cccc(c1)-c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
COc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)-c1cccc(F)c1
CC(C)c1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
CCc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
OCC(O)c1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
OCc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
OCC(O)Cc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
OC[C@@H](O)Cc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
OC[C@H](O)Cc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
OCC(O)Cc1cc(Cl)ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
OCCc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(N2CCOc3cc(c(Cl)cc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
COc1nc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
Fc1cc2N(CCOc2cc1S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F
Fc1c2OCCN(c2ccc1S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F
COc1cc(ccc1N1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1nccs1)C#N
Fc1cc(cc2OCCN(c3ccc(cc3C#N)C(F)(F)F)c12)S(=O)(=O)Nc1nccs1
COc1cc(ccc1CN1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
O=S(=O)(Nc1nccs1)c1ccc2N(Cc3ccccc3)CCOc2c1
Cc1onc(c1CN1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)-c1ccccc1
O=S(=O)(Nc1nccs1)c1ccc2N(Cc3c[nH]c4cccnc34)CCOc2c1
COc1cc(ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
Cc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(ccc1N1CCOc2cc(c(cc12)C#N)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1ccc(cc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COCCOc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CS(=O)(=O)c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1-c1cncnc1
COc1cc(ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
COc1cc(Cl)ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(N2C(=O)COc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C#N
COc1ccccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(cc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(N2C(=O)COc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(Br)c1
Fc1cc(ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(N2C(=O)COc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(Cl)c1
CC(O)c1ccccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1
Clc1ccc(N2CCOc3cc(ccc23)S(=O)(=O)Nc2ccncn2)c(c1)C#N
NC(=O)c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1cc(F)ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1
COc1ccc(F)cc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1
Cc1cc(ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
COc1cc(ccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1ccncn1)C#N
OCC(O)c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CC(=C)c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
Oc1ccc(cn1)-c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
NC(=O)COc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1OCC#N
CC(C)(O)c1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
CCc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc2N(CCOc2c1)c1ccccc1Oc1ccncc1
CC(C)(Oc1ccccc1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C#N
OCc1cc(ccc1N1C(=O)COc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1N1C(=O)C(C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1cc(ccc1N1C(=O)[C@H](C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
COc1cc(ccc1N1C(=O)[C@@H](C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
COc1cc(ccc1N1C(=O)C(C)(C)Oc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
COc1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)cc1
Oc1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)nc1
FC(F)(F)COc1ccc(cn1)C(=O)N1CCCC(C1)c1ccccc1
COc1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)nc1
Fc1ccc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)nc1
CSc1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)nc1
COc1ncccc1-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)nc1
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)nc1
Oc1ccc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)nc1
COc1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1cccnc1N
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=S)Nc1ccc(cc1)C(F)(F)F
COc1ccc(NC(=S)N2CCCC(C2)c2ccccc2-c2cnc(nc2)N(C)C)cc1
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)Nc1ccc(OC(F)(F)F)cc1
COc1ccc(cc1)S(=O)(=O)N1CCCC(C1)c1ccccc1-c1cnc(nc1)N(C)C
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)S(=O)(=O)c1ccc(OC(F)(F)F)cc1
COc1ccc(cc1[C@@H](O)CO)C(=O)N1CCCC(C1)c1ccccc1-c1cnc(nc1)N(C)C |r|
COc1ccc(cc1[C@H](O)CO)C(=O)N1CCCC(C1)c1ccccc1-c1cnc(nc1)N(C)C |r|
COc1ccc(cc1)C(=O)N1CCCC(C1)c1ccccc1-c1cnc(nc1)N(C)C
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1cccc(c1)C(N)=O
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(cc1)C(N)=O
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OC(F)(F)F)cc1
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)C(=O)c1ccc(OCC(F)(F)F)cc1
CN(C)c1ncc(cn1)-c1ccccc1C1CCCN(C1)S(=O)(=O)Nc1ncns1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCC[N+]1(C)CCCCC1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCC[N+]1(C)CCOCC1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)N1CCC(CC1)[N+]1(C)CCCC1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCc1ccc(cc1)[N+](C)(C)C
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCC[N+]1(C)CCCC1
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)NCC[N+](C)(C)C
Cc1cc(cc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(=O)N1CC[N+](C)(C)CC1
CN(C1CC[N+](C)(C)CC1)C(=O)c1cc(C)nc(c1)-c1ccc(Oc2ccc(F)cc2)cc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2C[C@@H]3C[C@H]2CN3)nc1 |r|
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@H]2CCS(=O)(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CCS(=O)(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)N2CCOCC2)nc1
CC(=O)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cc1
NC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CN(CC1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)N2CCOCC2)nc1
C[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)CC2)nc1
CC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cn1
FC(F)(F)C1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCOCC2)nc1
COCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC(F)(F)CC2)nc1
O[C@@H]1CS(=O)(=O)C[C@H]1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)C1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@@H]1CS(=O)(=O)C[C@@H]1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2C[C@@H]3CCCN3C(=O)C2)nc1
OCCN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CS(=O)(=O)C1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(C)(O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)CC2)nc1
CN(C)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@H]1C[C@H](C1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |wU:1.0,3.5,(11.12,-1.96,;9.78,-1.19,;8.3,-1.59,;7.9,-.1,;9.38,.3,;6.56,.67,;5.23,-.1,;5.23,-1.64,;3.9,.67,;3.9,2.21,;2.56,2.98,;1.23,2.21,;-.11,2.98,;-1.44,2.21,;-2.77,2.98,;-4.11,2.21,;-4.11,.67,;-5.44,-.1,;-6.77,.67,;-6.77,2.21,;-5.44,2.98,;-8.11,-.1,;-9.44,-.87,;-7.34,-1.43,;-8.88,1.23,;-1.44,.67,;-.11,-.1,;1.23,.67,;2.56,-.1,)|
FC1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
N[C@H]1[C@@H]2CN(C[C@H]12)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2CCO2)nc1
C[C@@H](O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNC3(CC3)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCNC(=O)C2)nc1
CO[C@@H]1C[C@@H](C1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |wU:2.1,4.6,(12.26,-1.15,;10.93,-1.92,;9.59,-1.15,;9.2,.34,;7.71,-.06,;8.11,-1.55,;6.38,.71,;5.04,-.06,;5.04,-1.6,;3.71,.71,;3.71,2.25,;2.37,3.02,;1.04,2.25,;-.29,3.02,;-1.63,2.25,;-2.96,3.02,;-4.29,2.25,;-4.29,.71,;-5.63,-.06,;-6.96,.71,;-6.96,2.25,;-5.63,3.02,;-8.3,-.06,;-9.63,-.83,;-7.53,-1.39,;-9.07,1.27,;-1.63,.71,;-.29,-.06,;1.04,.71,;2.37,-.06,)|
CN(C)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
C[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCCC2)nc1
CCN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CCN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)C2CCC2)nc1
CC1(COC1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
N[C@H]1[C@@H]2CN(C[C@H]12)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
OC[C@@H]1C[C@H](F)CN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3CC(F)(F)C[C@H]3C2)nc1
Fc1ccc(cc1)N1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
COCCNC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)Oc1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@H]2CNC(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(F)(F)C2)nc1
COCC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CCN(C1CCN(CC)C(=O)C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
COC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
COC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CS(=O)(=O)CCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
NC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CC1CN(CC(C)N1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
C[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
COC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
F[C@@H]1CCN(C1)C1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)[C@@H]1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN1C[C@@H](CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN1C[C@H](CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC(CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1)C(F)(F)F
O=C(N1CCOCC1)c1ccc2cc(Oc3ccccn3)ccc2n1
CN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccccn3)ccc2n1
Cc1noc(n1)C1CCCN(C1)C(=O)c1ccc2cc(Oc3ccccn3)ccc2n1
O=C(NCCN1CCCCC1)c1ccc2cc(Oc3ccccn3)ccc2n1
O=C(Nc1ncns1)c1ccc2cc(Oc3ccccn3)ccc2n1
CN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCCN1CCCCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N1CCOCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(Nc1ccc2cn[nH]c2c1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CN(C)CCCNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCCN1CCOCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCCCN1CCOCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(Nc1nccs1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCc1cccnc1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N[C@H]1CCOC1=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC(C)[C@H](CO)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCc1cccs1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCCc1cccs1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCc1ccco1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC(C)C(CO)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCCN1CCCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCc1ccccn1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NCc1ccncc1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
Cc1ccc(CNC(=O)c2ccc3cc(Oc4ccc(cc4)C#N)ccc3n2)o1
O=C(NCCCN1CCCCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(Nc1ccc(Oc2ccccc2)cc1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
FC(F)(F)Oc1cccc(CNC(=O)c2ccc3cc(Oc4ccc(cc4)C#N)ccc3n2)c1
Cc1ccc(CNC(=O)c2ccc3cc(Oc4ccc(cc4)C#N)ccc3n2)cc1
O=C(NCc1ccc2OCOc2c1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
COc1cccc(CNC(=O)c2ccc3cc(Oc4ccc(cc4)C#N)ccc3n2)c1OC
O=C(N1CCCCCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CCCN(CCOC)C(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CCOCCNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NC1CCN(Cc2ccccc2)C1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
FC(F)(F)C1CCCN(C1)C(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N1CCc2ccccc12)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N1CCNCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N[C@@H]1CCOC1=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NC1CCOC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CS(=O)(=O)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NC1CCCOC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N[C@@H]1CCOC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N[C@H]1CCOC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@H]1CCCC[C@H]1NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@H]1CCCC[C@@H]1NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@H]1CCC[C@@H]1NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC(C)(O)CNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
OCC1(CC1)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC(C)(CO)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@H]1CC[C@@H](CC1)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1 |wU:4.7,wD:1.0,(10.08,-7.2,;8.74,-6.43,;8.74,-4.89,;7.41,-4.12,;6.08,-4.89,;6.08,-6.43,;7.41,-7.2,;4.74,-4.12,;4.74,-2.58,;6.08,-1.81,;3.41,-1.81,;3.41,-.27,;2.08,.5,;.74,-.27,;-.59,.5,;-1.93,-.27,;-3.26,.5,;-3.26,2.04,;-4.59,2.81,;-4.59,4.35,;-3.26,5.12,;-1.93,4.35,;-1.93,2.81,;-3.26,6.66,;-3.26,8.2,;-1.93,-1.81,;-.59,-2.58,;.74,-1.81,;2.08,-2.58,)|
OCC(CO)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC(CO)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC(O)CNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@@H]1CCC[C@@H](C1)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@@H]1CC[C@@H](C1)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@H]1CCC[C@H]1NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@H]1CCC[C@@H](C1)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O[C@H]1CC[C@H](CC1)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1 |wU:1.0,4.7,(10.08,-7.2,;8.74,-6.43,;7.41,-7.2,;6.08,-6.43,;6.08,-4.89,;7.41,-4.12,;8.74,-4.89,;4.74,-4.12,;4.74,-2.58,;6.08,-1.81,;3.41,-1.81,;3.41,-.27,;2.08,.5,;.74,-.27,;-.59,.5,;-1.93,-.27,;-3.26,.5,;-3.26,2.04,;-4.59,2.81,;-4.59,4.35,;-3.26,5.12,;-1.93,4.35,;-1.93,2.81,;-3.26,6.66,;-3.26,8.2,;-1.93,-1.81,;-.59,-2.58,;.74,-1.81,;2.08,-2.58,)|
CC(O)C(C)NC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC(C)C(O)CNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(NC1CCS(=O)(=O)C1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N1CCNC(=O)C1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N1CCC(CC1)N1CCOCC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
Fc1ccc2OCC[C@@H](NC(=O)c3ccc4cc(Oc5ccc(cc5)C#N)ccc4n3)c2c1
CC(C)(C)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CC1(C)C[C@@H](NC(=O)c2ccc3cc(Oc4ccc(cc4)C#N)ccc3n2)c2cc(F)ccc2O1
CC(C)[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CN1CCC(NC(=O)c2ccc3cc(Oc4ccc(cc4)C#N)ccc3n2)C1=O
O=C(NCc1ncco1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
CNC(=O)CNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
NC(=O)CNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
NS(=O)(=O)CCNC(=O)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N1CCS(=O)(=O)CC1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCOC2)nc1
NC(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCc2ccccn2)nc1
FC(F)(F)c1ccnc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)c1
FC(F)(F)c1cccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)n1
FC(F)(F)c1cnc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)c(Cl)c1
FC(F)(F)c1cnc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(COC3)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(CNC3)C2)nc1
O=C(NC1CCS(=O)(=O)C1)c1ccc2cc(Oc3ccc(cn3)C#N)ccc2n1
O=C(N[C@H]1CCS(=O)(=O)C1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
O=C(N[C@@H]1CCS(=O)(=O)C1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
Cc1cnc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)nc1
Cc1cc(C)nc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)n1
Cc1ccnc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2C[C@@H]3CNC[C@@H]3C2)nc1
Clc1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)nn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2C[C@H]3CNC(=O)[C@H]3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2[C@H]3CC[C@@H]2C2CNCC32)nc1 |TLB:19:21:26.30:24.23|
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)nn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3CCNC(=O)C3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCn3cnnc3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3C(C2)C(=O)NCC3=O)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNC(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCn3cncc3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCCCC2)nc1
CS(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(C)S(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)c2ccccc2)nc1
F[C@H]1C[C@@H](N(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1)c1cc(F)ccc1F
F[C@@H]1C[C@@H](N(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1)c1cc(F)ccc1F
FC(F)(F)CN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)c2ccccn2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)c2cccnc2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)N2CCCCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)N2CCOCC2)nc1
COC(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(C)C(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN1C(=O)CN(CC11COC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3CNCCN3C2=O)nc1
OC1CCN(CC1(F)F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@H]1CCN(C[C@H]1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |r|
O[C@@H]1CN(CC[C@@H]1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |r|
OC1CN(CCC1(F)F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC[C@@H]1CN([C@@H]1CO)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@@H]1CCN(C[C@H]1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |r|
O[C@@H]1CN(CC[C@H]1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |r|
C[C@H]1N(CC1(C)C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(O)CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COCC1(C)CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1)Oc1ccccc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)Oc2ccccc2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)n2ccnc2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)Oc2ccc(Cl)cc2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)n2cncn2)nc1
C[C@@H]1N(CC1(C)C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)Oc2ccc(Br)cc2)nc1
CC1(CO)CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNC(=O)C2c2ccccc2)nc1
CC(C)(O)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cc1
NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@H]1C[C@H]2CN(CCC(=O)N2C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC[C@@H]3CN[C@@H]3C2)nc1
CS(=O)(=O)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cc1
FC(F)(F)S(=O)(=O)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CNC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)c2cccnc2)nc1
CC(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC=CC2)nc1 |c:25|
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCSCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCc3ccncc3C2)nc1
O[C@H]1C[C@@H](N(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1)c1cc(F)ccc1F
FC(F)(F)c1ccc(cc1)C1CCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(cc1)S(=O)(=O)N[C@H]1CCN([C@@H]1c1ccccc1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(=O)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCS(=O)(=O)CC2)nc1
CC(C)(C)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
Fc1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CC[C@H]3CN(Cc4ccccc4)C[C@@H]23)nc1
CC(C)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(C2)CCNCC3)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCNC2)nc1
OC[C@@H]1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CNS(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CCNS(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC[C@@H]1CCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCCCC2)nc1
CNC(=O)[C@@H]1CCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC3(CC2)OCCO3)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2C[C@H]3C[C@@H]2CN3)nc1 |r|
O=C(N1CCNCC1)c1ccc2cc(Oc3ncccn3)ccc2n1
OC[C@H]1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
Fc1cnc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1cnc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cn1
FC(F)(F)c1cnnc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)c1
FC(F)(F)c1cnc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
N[C@H]1CC[C@@H]2CN(C[C@H]12)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cc1
Fc1cc(cnc1Oc1ccc2nc(ccc2c1)C(=O)N1CCNCC1)C(F)(F)F
CS(=O)(=O)CCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)C2COC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCc3ccccc3C2)nc1
CS(=O)(=O)C1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(O)CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OCC1C[C@H]2C[C@@H]1CN2C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |r|
OC[C@@H]1C[C@H]2C[C@@H]1CN2C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |r|
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CC[C@@H]3CN(Cc4ccccc4)C[C@H]23)nc1
CN1CCCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)C2CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)c2ccccc2)nc1
CC(C)[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCNCC2)nc1
OCC1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OCC1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC3CCC(C2)N3)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)c2cnccn2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)c2cccnc2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)c2ncccn2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)c2cccnn2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)c2ccc(Cl)cn2)nc1
CC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(C)[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(O)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cc1
CC(C)OC(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2C[C@@H]3CN[C@@H]3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC22CNC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2C[C@@H]3CCN[C@@H]3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NN2CCOCC2)nc1
O[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CCCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CS(=O)(=O)CC1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(CN2CCN(CC2)C(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)COC1
CS(=O)(=O)C1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3C(CCC3=O)C2)nc1
CCOC(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)C(=O)C2CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)C2CCCCC2)nc1
OC1CN(CC1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(C)COC(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CCN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1cnc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)c(Br)c1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCOCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCCC2)nc1
FC(F)CN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)C(=O)N2CCOCC2)nc1
OC[C@@H]1C[C@@H](O)CN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(OC(F)(F)F)cn3)ccc2n1
O[C@H]1C[C@@H](C1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |wU:3.5,wD:1.0,(11.12,-1.96,;9.78,-1.19,;9.38,.3,;7.9,-.1,;8.3,-1.59,;6.56,.67,;5.23,-.1,;5.23,-1.64,;3.9,.67,;3.9,2.21,;2.56,2.98,;1.23,2.21,;-.11,2.98,;-1.44,2.21,;-2.77,2.98,;-4.11,2.21,;-4.11,.67,;-5.44,-.1,;-6.77,.67,;-6.77,2.21,;-5.44,2.98,;-8.11,-.1,;-9.44,-.87,;-7.34,-1.43,;-8.88,1.23,;-1.44,.67,;-.11,-.1,;1.23,.67,;2.56,-.1,)|
OC[C@@H]1[C@@H](O)CCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COC1CN(CC1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1CN(CC1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OCC1CC(CO)CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(Cc3ccccn3)CC2)nc1
CC(C)(C)CC(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
N[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)CCN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCC(F)(F)C2)nc1
O[C@H]1CC[C@@]2(CCCN2C(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)C1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(C2)N2CCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(Cc3cocn3)CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(C2)N2CCOCC2)nc1
NS(=O)(=O)CCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC[C@H](C2)N2CCCCC2)nc1
FC(F)(F)c1nnc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)s1
CC(C)NC(=O)C1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CNC(=O)C1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1[C@H](O)[C@H](O)C(C)N1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COC1CN(CC1OC)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
NC(=O)[C@H]1CCCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCOCC2)nc1
O=C(N1CCNCC1)c1ccc2cc(Oc3ccc(cn3)C#N)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3C(COC3=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(F)(F)CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CCNC2)nc1
FC(F)(F)CCS(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3[C@@H](COC3=O)C2)nc1
CC(C)(O)CCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC[C@H]2CCCN2)nc1
OC1(CNC(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)CCC1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCCC2=O)nc1
NCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OCC1CN(CCO1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FCC1CN(CCO1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CCC11CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCc3nc[nH]c(=O)c3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCNC(=O)C2)nc1
FC(F)(F)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CC2(C1)CCN(C2)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |(2.78,7.1,;4.32,7.1,;5.41,6.01,;6.5,7.1,;5.41,8.19,;7.41,5.85,;8.87,6.33,;8.87,7.87,;7.41,8.35,;10.12,8.78,;9.95,10.31,;11.52,8.15,;11.68,6.62,;13.09,5.99,;14.34,6.9,;15.74,6.27,;16.99,7.18,;18.4,6.55,;19.64,7.45,;19.48,8.99,;20.73,9.89,;22.13,9.26,;22.29,7.73,;21.05,6.83,;23.38,10.17,;24.63,11.08,;22.47,11.42,;24.28,8.92,;16.83,8.71,;15.42,9.33,;14.18,8.43,;12.77,9.05,)|
FCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CS[C@H]1CN(C[C@@H]1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCCS(=O)(=O)C2)nc1
OC1CCN(CC1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CS(=O)(=O)C1CN(CC1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC3(C2)OCCO3)nc1
[#6]-[#8]\[#7]=[#6]-1\[#6]-[#6]-[#7](-[#6]-[#6]-1)-[#6](=O)-c1ccc2cc(-[#8]-c3ccc(cn3)C(F)(F)F)ccc2n1
OC1CC2(C1)CCN(CC2)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)CCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@H]1C[C@@H]2CN(CCN2C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[C@@H]1CN2C[C@@H](F)C[C@@H]2CN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[C@@H]1CN2CC(F)(F)C[C@@H]2CN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@H]1C[C@H]2CN(CCN2C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCc3[nH]cnc3C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2COCCN2Cc2ccccc2)nc1
OC1(CNC(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)CCOCC1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC[C@@H]2CCCN2)nc1
CC1(C)CN(CCNC(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)C1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCSCC2)nc1
CN(CC=C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)C#N)nc1
COCOC1CN(CC1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1(CNC(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)CC1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(=O)C2)nc1
OC1COCC1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O=C(N1CCNCC1)c1ccc2cc(Oc3cnc(cn3)C#N)ccc2n1
CC1(C)OC2CN(CC2O1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(C)CC1CN(CCO1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(=O)CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N(C2CCOCC2)C2CCOCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)N2C[C@@H]3C[C@H]2CO3)nc1 |r|
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)N2C[C@H]3C[C@@H]2CO3)nc1 |r|
COCCN(CCOC)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OCC1(CC1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)C2CCOC2)nc1
COC(=O)CS(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)C2CCOCC2)nc1
COCCn1cc(cn1)S(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)CC2CCOC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)S(=O)(=O)C2CCS(=O)(=O)C2)nc1
Cn1cc(cn1)S(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(=O)Nc1nc(C)c(s1)S(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(=O)Nc1ncc(s1)S(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
Cc1c(cnn1C)S(=O)(=O)N1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@H]2CCOC2)nc1
COCCN(C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CCOC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC[C@H]2CCCO2)nc1
O[C@@H]1C[C@@H](O)CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CO[C@H]1C[C@@H](C1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |wU:4.6,wD:2.1,(12.26,-1.15,;10.93,-1.92,;9.59,-1.15,;9.2,.34,;7.71,-.06,;8.11,-1.55,;6.38,.71,;5.04,-.06,;5.04,-1.6,;3.71,.71,;3.71,2.25,;2.37,3.02,;1.04,2.25,;-.29,3.02,;-1.63,2.25,;-2.96,3.02,;-4.29,2.25,;-4.29,.71,;-5.63,-.06,;-6.96,.71,;-6.96,2.25,;-5.63,3.02,;-8.3,-.06,;-9.63,-.83,;-7.53,-1.39,;-9.07,1.27,;-1.63,.71,;-.29,-.06,;1.04,.71,;2.37,-.06,)|
CN(C1CS(=O)(=O)CC1O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2COC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCSCC2)nc1
O[C@@H]1CCC[C@@H]1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
NC(=O)C1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
NC1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(F)(F)C2)nc1
CC1(C)CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC1CNCCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1CNCCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CS(=O)(=O)NC1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[C@H](O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(C1CCOCC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC1(CNC(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)COC1
CN(C)C(=O)CN(C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)C1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC1CN(CC1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC(=O)NC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC(F)(F)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNC3(CCC3)C2)nc1
CN(C1CCS(=O)(=O)C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCSC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCNC2=O)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCNc2ccccn2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCn2ccnc2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2CCN2)nc1
O[C@H]1CS(=O)(=O)C[C@@H]1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(O)CC(C1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |(11.43,-4.13,;9.89,-4.17,;10.62,-5.52,;9.49,-2.68,;8,-3.08,;8.4,-4.57,;6.67,-2.31,;5.33,-3.08,;5.33,-4.62,;4,-2.31,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-2.67,,;-4,-.77,;-4,-2.31,;-5.33,-3.08,;-6.67,-2.31,;-6.67,-.77,;-5.33,,;-8,-3.08,;-9.34,-3.85,;-7.23,-4.41,;-8.77,-1.75,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,)|
COCCOC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CS(=O)(=O)NC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)N2CCOCC2)nc1
FC(F)C1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)(F)Oc1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(C2)N2CCOCC2)nc1 |(-9.34,-3.85,;-8,-3.08,;-7.23,-4.41,;-8.77,-1.75,;-6.67,-2.31,;-5.33,-3.08,;-4,-2.31,;-4,-.77,;-2.67,,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;4,-.77,;2.67,,;1.33,-.77,;;5.33,-3.08,;5.33,-4.62,;6.67,-2.31,;8,-3.08,;9.49,-2.68,;9.89,-4.17,;8.4,-4.57,;11.22,-4.94,;12.56,-4.17,;13.89,-4.94,;13.89,-6.48,;12.56,-7.25,;11.22,-6.48,;-5.33,,;-6.67,-.77,)|
CC(C)(O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)N2CCOCC2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(F)(F)F)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC(F)(F)CC2)nc1
CC(=O)N[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC[C@H](C2)NC(=O)C2CC2)nc1
OC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
CN(C)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
COCCNC(=O)CN(C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCOCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCOCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCCC2)nc1
CCN(CC)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCCCC2)nc1
CN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCCCC2)nc1
CN1CCN(CC1=O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(C)C(=O)[C@@H]1CCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(CC(=O)NC1CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CCN(CC)C(=O)CCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(C)NC(=O)CN(C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CNC(=O)[C@@H]1CCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCCC2)nc1
COCCNC(=O)CN(C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCOCC2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCOCC2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCCC2)nc1
CCN(CC)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
CN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCCCC2)nc1
CN1CCN(CC1=O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
CN(C)C(=O)[C@@H]1CCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
CN(CC(=O)NC1CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
CCN(CC)C(=O)CCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
CC(C)NC(=O)CN(C)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCNCC2=O)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2CNC2)nc1
CC(C)(O)CNC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CCCC#N)CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CCC#N)CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)C#N)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2COC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(C2)OCCO3)nc1
O[C@@H]1CS(=O)(=O)C[C@H]1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3OCOC3C2)nc1
CS(=O)(=O)C1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
CN(C1COC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2COC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNC(C2)C#N)nc1
O=C(NC1CCNC(=O)C1)c1ccc2cc(Oc3ccc(cc3)C#N)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC(F)(F)C2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC(F)(F)C2)nc1
COCC1(F)CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CCOCC1(F)CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(F)(COc3ccncc3)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(F)(COc3cccnc3)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(F)(COc3ccccc3)C2)nc1
[O-]C(=O)N(CC1CN(CC1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1)Cc1ccccc1
COCCOCC1(F)CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC3(COC3)C2)nc1
OC[C@H]1C[C@H](F)CN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC[C@H]1CC(F)(F)CN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC[C@@H]1CC(F)(F)CN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COc1cccc(c1)N1CCN(CC1=O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CSC2)nc1
Cc1ccccc1NC(=O)CCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(C)C(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COc1ccccc1N1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CS(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CS(=O)(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC22COC2)nc1
CC(=O)C1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(F)(F)C2)nc1
CN(C)C(=O)C1(CC[C@@H](F)C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(Cc3ncco3)CC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC(F)(F)CC2)cn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@H]2CCNC(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCCC2)cn1
COCCNC(=O)CN(C)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCOCC2)cn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCCC2)cn1
CCN(CC)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCCCC2)cn1
CN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC(=O)N2CCCCC2)cn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CCNC(=O)C2)nc1
CN(CC(=O)NC1CC1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CCN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CCN(CC)C(=O)CCNC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CC(C)NC(=O)CN(C)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)N2CCOCC2)cn1
CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
N[C@H]1[C@@H]2CN(C[C@H]12)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CN(C1CCN(C)C(=O)C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CCOC2=O)nc1
Cc1nc(CN2CCN(CC2)C(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)co1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(C2)CCOC3)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(C2)CCCOC3)nc1
CS(=O)(=O)C1CN(C1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)CC2)cn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2COC2)cn1
O[C@@H]1CS(=O)(=O)C[C@@H]1NC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
O[C@@H]1CS(=O)(=O)C[C@H]1NC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC=CC2)cn1 |c:25|
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)N2CC(F)(F)C2)nc1
COC(C)(C)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3CC(F)(F)C[C@H]3C2)nc1
CC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
OC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
OC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
OC1CN(CC1O)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)OCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
C[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
F[C@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
OC(CNC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1)C(F)(F)F
CC1CN(CC(C)N1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)N2CCOCC2)cn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(F)(F)C2)cn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(=O)C2)cn1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)N2CCNCC2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNC3(CC3)C2)nc1
O[C@@H]1CCN(C1)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@H]1CCN(C1)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(O)CCN(C1)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@H]1CN(C[C@@H]1O)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@@H]1CN(C[C@H]1O)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC[C@@H]1C[C@@H](O)CN1C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCC(F)(F)C2)nc1
OC1CN(C1)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(O)CN(C1)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCS(=O)(=O)C2)nc1
COC1CN(C1)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC[C@H]1CCCN1C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCC(=O)C2)nc1
FC1CCN(C1)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(C2)N2CCOCC2)cn1 |(-9.34,-3.85,;-8,-3.08,;-7.23,-4.41,;-8.77,-1.75,;-6.67,-2.31,;-5.33,-3.08,;-4,-2.31,;-4,-.77,;-2.67,,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;4,-.77,;2.67,,;1.33,-.77,;;5.33,-3.08,;5.33,-4.62,;6.67,-2.31,;8,-3.08,;9.49,-2.68,;9.89,-4.17,;8.4,-4.57,;11.22,-4.94,;12.56,-4.17,;13.89,-4.94,;13.89,-6.48,;12.56,-7.25,;11.22,-6.48,;-5.33,,;-6.67,-.77,)|
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC[C@@H](F)C2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC[C@H](F)C2)nc1
CS(=O)(=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC1(O)CC(C1)NC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1 |(11.43,-4.13,;9.89,-4.17,;10.62,-5.52,;9.49,-2.68,;8,-3.08,;8.4,-4.57,;6.67,-2.31,;5.33,-3.08,;5.33,-4.62,;4,-2.31,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-2.67,,;-4,-.77,;-4,-2.31,;-5.33,-3.08,;-6.67,-2.31,;-6.67,-.77,;-5.33,,;-8,-3.08,;-9.34,-3.85,;-7.23,-4.41,;-8.77,-1.75,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,)|
CC(NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1)C(=O)N(C)C
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(F)(F)C2)nc1
O[C@@H]1CCCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
O[C@H]1CCCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
N[C@@H]1CCN(C[C@H]1F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@@H]1CNCC[C@H]1NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
F[C@H]1CCN(C1)C1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN1CCC(NC(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)C1=O
CO[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CO[C@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COC(C)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COC1(CNC(=O)c2ccc3cc(Oc4ccc(cn4)C(F)(F)F)ccc3n2)CCC1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(=O)C2)nc1
COC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)C1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCCC#N)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC2)nc1
FC(F)(F)C1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COCCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2CSC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2CS(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2CS(=O)(=O)C2)nc1
FC(F)[C@H]1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC1CC(C1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1 |(11.22,-4.94,;9.89,-4.17,;9.49,-2.68,;8,-3.08,;8.4,-4.57,;6.67,-2.31,;5.33,-3.08,;5.33,-4.62,;4,-2.31,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-2.67,,;-4,-.77,;-4,-2.31,;-5.33,-3.08,;-6.67,-2.31,;-6.67,-.77,;-5.33,,;-8,-3.08,;-9.34,-3.85,;-7.23,-4.41,;-8.77,-1.75,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;2.67,-3.08,)|
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCN2CCOC2=O)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCc2ccccn2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCCc2ccccn2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCCN2CCCC2=O)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC2CNC(=O)C2)nc1
CC(CNC(C)=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(CCS(C)(=O)=O)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CS(=O)(=O)CCCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CC(=O)NCCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCN3C2CCC3=O)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCCC2CS(=O)(=O)C2)nc1
CN(CC(F)(F)F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(F)C2)nc1 |(-5.33,-4.62,;-5.33,-3.08,;-6.67,-2.31,;-4,-2.31,;-4,-.77,;-2.67,,;-1.33,-.77,;;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;8,-3.08,;9.34,-2.31,;8,-4.62,;9.34,-5.39,;10.8,-4.91,;11.28,-6.38,;12.68,-7.01,;9.81,-6.85,;-1.33,-2.31,;-2.67,-3.08,)|
COCC1(F)CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)COC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[N+]1(C)CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)CNC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(CC(F)F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(C2)CCOCC3)nc1
CS(=O)(=O)Nc1noc2cc(COc3ccc(Cl)c(Cl)c3)c(Cl)cc12
CS(=O)(=O)Nc1noc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cc12)C1CC1 |TLB:16:17:21:15.14.20,20:15:22:19.21.18,20:19:22:15.14.16,THB:16:15:21:22.17.18|
CC(C)COc1ccc(OCc2cc3onc(NS(C)(=O)=O)c3cc2Cl)cc1Cl
COCCS(=O)(=O)Nc1noc2cc(COc3ccc(OCC(C)C)c(Cl)c3)c(Cl)cc12
CC(C)Oc1ncc(OCc2cc3onc(NS(C)(=O)=O)c3cc2Cl)cc1Cl
CC1(C)CCc2ccc(OCc3cc4onc(NS(C)(=O)=O)c4cc3Cl)cc2C1
CS(=O)(=O)Nc1noc2cc(OCc3ccc(Cl)c(Cl)c3)c(Cl)cc12
CC1(C)CCc2cc(OCc3cc4onc(NS(C)(=O)=O)c4cc3Cl)ccc2C1
Clc1ccc(OCc2cc3onc(NS(=O)(=O)C4CC4)c3cc2Cl)cc1Cl
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cccc2nccn12)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnc2nccn12)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cnc2CNCCn12)S(=O)(=O)Nc1ncns1
Fc1cccnc1NS(=O)(=O)c1cc(F)c(Oc2ccc(Cl)cc2-c2cccc3nccn23)cc1F
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1c[nH]c(=O)c2cncn12)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ncc2cnccn12)S(=O)(=O)Nc1ncns1
Nc1nc2cc(ccc2[nH]1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1cnc2c(ncnc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-n1cnc2cncnc12)S(=O)(=O)Nc1ncns1
CN(c1ncns1)S(=O)(=O)c1cc(F)c(Oc2ccc(Cl)cc2-c2ccc3[nH]c(N)nc3c2)cc1F
Nc1cnc2ccc(cn12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Nc1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Nc1n[nH]c2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
NC(=O)c1cnc2ccc(cn12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2[nH]c(=O)[nH]c2c1)S(=O)(=O)Nc1ncns1
Nc1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2ocnc2c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2oc(=O)[nH]c2c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2[nH]c(=O)oc2c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2[nH]c(nc2c1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2CC(=O)Nc2c1)S(=O)(=O)Nc1ncns1
Nc1nc2cc(ccc2o1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Nc1nc2ccc(cc2o1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Nc1noc2ccc(cc12)-c1ccccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2nccnc2c1)S(=O)(=O)Nc1ncns1
Nc1nc2cc(ccc2[nH]1)-c1cc(Cl)ccc1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ncns1
Nc1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncccn1
Nc1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(c(F)c1)S(=O)(=O)Nc1ncns1
Nc1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1ccc(c(F)c1F)S(=O)(=O)Nc1ncns1
CNc1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2[nH]cnc2c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccc2NC(=O)Cc2c1)S(=O)(=O)Nc1ncns1
Fc1cc(ccc1Oc1ccc(Cl)cc1-c1ccc2oc(=O)[nH]c2c1)S(=O)(=O)Nc1ncccn1
Nc1noc2ccc(cc12)-c1cc(F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cc1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(c1)-c1ccc2oc(=O)[nH]c2c1
Nc1noc2ccc(cc12)-c1cccnc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
CN(C)c1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1 |r|
Cn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1 |r|
Cn1cncc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
Cn1nccc1C1CCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1 |r|
N[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CCN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2NCc2ccccc2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CCN(Cc1ccccc1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1CCCC[C@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1CCC[C@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1CCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Br)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2NC2CCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CCN(CC)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CCN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C1CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN[C@H]1CCCC[C@@H]1N(C)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CC(=CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r,c:5|
CN(C)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1CCCC[C@H]1Oc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(Cl)s1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(C)cs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1ccc(cc1[N+]([O-])=O)S(=O)(=O)Nc1nccs1 |r|
CCCN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CN(CC1CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
COCCN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CC(C)N(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CCCN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C)[C@@H]1C[C@@H](CC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(CCF)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(CCO)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C1CNC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(C)s1 |r|
CN(C1CN(C)C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CCN[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CCN[C@@H]1CCCC[C@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CC1CCCN1[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CC(O)CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r|
OC1CN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1CC=C(C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r,c:5|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1 |r|
CN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Br)S(=O)(=O)Nc1nccs1 |r|
CN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
CCN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Br)S(=O)(=O)Nc1nccs1 |r|
CN(C1CNC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1CCCC[C@@H]1N1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1 |r|
CN(C1CNC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(CCO)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
CN(C1CNC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
CNCCN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CC=C(C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cccc(c1)C(F)(F)F |r,c:5|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCCC2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
OC1CCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
OC1CCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C1CN(C)C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CCN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C(F)(F)F)S(=O)(=O)Nc1nccs1 |r|
CN(C1CNC1)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
O[C@H]1CCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
O[C@@H]1CCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCCCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CCN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(CCO)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CCN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C)[C@H]1CC[C@@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C)[C@H]1CC[C@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C)[C@H]1C[C@@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1C(F)(F)F)S(=O)(=O)Nc1nccs1 |r|
CN(CC(N)=O)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CNC(=O)CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1C[C@H](CC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C)[C@@H]1CC[C@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C)[C@@H]1CC[C@@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(Cl)n1 |r|
CC(O)CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C)[C@H]1CC[C@@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1CC[C@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cccc(c1)C(F)(F)F |r|
CN(CCO)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CN(C1CNC1)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CCC1)S(=O)(=O)Nc1nccs1 |r|
Cc1csc(NS(=O)(=O)c2cc(Cl)c(N[C@H]3CCCC[C@@H]3N3CCCC3)cc2F)n1 |r|
CN(C)[C@@H]1CC[C@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cccc(c1)C(F)(F)F |r|
CN(C[C@H](O)C(F)(F)F)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C[C@@H](O)C(F)(F)F)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CCN[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1ccncn1 |r|
CN(C1COC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cccc(NS(=O)(=O)c2cc(Cl)c(N[C@@H]3CCCC[C@H]3N3CCCC3)cc2F)n1 |r|
Fc1cccc(NS(=O)(=O)c2cc(Cl)c(N[C@H]3CCCC[C@@H]3N3CCCC3)cc2F)n1 |r|
CCN[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCOCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CCN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(C)cs1 |r|
CN(C)[C@@H]1CC[C@@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cccc(c1)C(F)(F)F |r|
FC1CCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cccc(NS(=O)(=O)c2cc(Cl)c(N[C@H]3CCCC[C@@H]3N3CC4CC4C3)cc2F)n1 |r|
Fc1cccc(NS(=O)(=O)c2cc(Cl)c(N[C@@H]3CCCC[C@H]3N3CC4CC4C3)cc2F)n1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1cccc(F)n1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCCCC2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
CN(C1CCN(C)CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C1CCNCC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(CCO)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(C)cs1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
FC1CCN(CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C1CCC1)[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(CC(C)(C)O)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cccc(NS(=O)(=O)c2cc(Cl)c(N[C@@H]3CCCC[C@H]3N3CCCCC3)cc2F)n1 |r|
CN(CC(O)CF)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CC[C@@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1CC[C@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(CCCO)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
Fc1cccc(NS(=O)(=O)c2cc(Cl)c(N[C@H]3CCCC[C@@H]3N3CCCCC3)cc2F)n1 |r|
CN(CCC(C)(C)O)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(CCC#N)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(CC(O)C(F)F)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(CCO)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C)[C@H]1CC(CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1CC=C(C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r,c:5|
OC1CCN(CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCC[C@@H]1N1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1nccs1 |r|
OC[C@H]1CCCN1[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
OC[C@@H]1CCCN1[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(CCCF)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(CC1(F)CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cccc(c1)C(F)(F)F |r|
CN(CCO)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
CN(C[C@@H](O)C1CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1cnn(C)c1 |r|
CN(C)[C@H]1CC=CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r,c:5|
CN(C)[C@@H]1CC=CC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r,c:5|
CN(C[C@H](O)C1CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1CCCCC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CC(C)C(=O)N1CC(C1)N(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CC(C)CC(=O)N1CC(C1)N(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C1CN(C1)C(C)=O)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCC(CC2)C#N)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CC1(O)CCN(CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CC3CC3C2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(N[C@@H]2CCCC[C@H]2N2CC3CC3C2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
O[C@H]1CCCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCC3(CC3)CC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CN(C1CN(C1)C(=O)C1CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN([C@@H]1C[C@H](O)C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r,wU:7.7,wD:12.14,2.1,4.4,(-1.68,-2.02,;-3.01,-1.25,;-4.35,-2.02,;-4.75,-3.5,;-6.23,-3.1,;-7.57,-3.87,;-5.84,-1.62,;-3.01,.29,;-4.35,1.06,;-4.35,2.6,;-3.01,3.37,;-1.68,2.6,;-1.68,1.06,;-.35,.29,;.99,1.06,;.99,2.6,;2.32,3.37,;2.32,4.91,;3.65,2.6,;3.65,1.06,;2.32,.29,;2.32,-1.25,;4.99,3.37,;4.22,4.71,;5.76,4.71,;6.32,2.6,;6.32,1.06,;7.57,.16,;7.09,-1.3,;5.55,-1.3,;5.08,.16,)|
CN([C@H]1C[C@H](O)C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r,wU:7.7,4.4,wD:12.14,2.1,(-1.68,-2.02,;-3.01,-1.25,;-4.35,-2.02,;-5.84,-1.62,;-6.23,-3.1,;-7.57,-3.87,;-4.75,-3.5,;-3.01,.29,;-4.35,1.06,;-4.35,2.6,;-3.01,3.37,;-1.68,2.6,;-1.68,1.06,;-.35,.29,;.99,1.06,;.99,2.6,;2.32,3.37,;2.32,4.91,;3.65,2.6,;3.65,1.06,;2.32,.29,;2.32,-1.25,;4.99,3.37,;4.22,4.71,;5.76,4.71,;6.32,2.6,;6.32,1.06,;7.57,.16,;7.09,-1.3,;5.55,-1.3,;5.08,.16,)|
CN(CCO)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
Fc1cc(N[C@@H]2CCCC[C@H]2N2CC3CC3C2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CC3CC3C2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CC[C@H](C2)C#N)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CC[C@@H](C2)C#N)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CN1CCN(CC1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1Cc2ccccc2C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1Cc2ccccc2C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(C)=O |r|
CN(C)CC(=O)N(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
OC[C@H]1CCCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
OC[C@@H]1CCCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C1CNC1)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(C)cs1)C(F)(F)F |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(C)c(Cl)s1 |r|
CN(C)[C@H]1CC[C@@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1ccccc1F |r|
CN(C)[C@H]1CC[C@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1ccccc1F |r|
CN(C1CN(CC(F)(F)F)C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCC[C@H](C2)C#N)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CCC[C@@H](C2)C#N)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(=O)C1CN(C)C1 |r|
CN(C1CCC1)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc2cc(c(cc2Cl)S(=O)(=O)Nc3ccncn3)F)c4cccc(c4)C(F)(F)F
Fc1cc(N[C@@H]2CCCC[C@H]2N2CC3C(C2)C3(F)F)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(N[C@H]2CCCC[C@@H]2N2CC3C(C2)C3(F)F)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
OC[C@H]1[C@@H]2CN(C[C@H]12)[C@@H]1CCCC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
OC[C@H]1[C@@H]2CN(C[C@H]12)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccc(F)n1 |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(Cl)cs1 |r|
CN(C)[C@H]1CC(F)(F)CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1CC(F)(F)CC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CCN(C)[C@H]1CCCC[C@@H]1N1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1nccs1 |r|
CN1CC(C1)N(CC(F)(F)F)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1CCC(F)C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@@H](F)CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@H](F)CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@@H]2[C@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(Cl)Cl |r|
CN(C)[C@@H]1C[C@@H]2[C@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(Cl)Cl |r|
CN(C)[C@H]1C[C@H]2[C@@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(Cl)Cl |r|
CN(C)[C@@H]1C[C@H]2[C@@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(Cl)Cl |r|
CN(C)C(C)(C)C(=O)N(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(=O)[C@H]1CCN(C)C1 |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(=O)[C@@H]1CCN(C)C1 |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(=O)[C@@H]1CCCN1C |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(=O)[C@@H]1CCN1C |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1C1CCC1)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(=O)[C@H]1CCCN1C |r|
CN([C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C(=O)[C@H]1CCN1C |r|
Fc1cc(N[C@H]2CC[C@@H](C[C@@H]2N2CCCCC2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1C[C@H]2[C@@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(F)F |r|
CN(C)[C@@H]1C[C@@H]2[C@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(F)F |r|
CN(C)[C@H]1C[C@@H]2[C@H](C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(F)F |r|
CN(C)[C@@H]1C[C@H]2[C@@H](C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)C2(F)F |r|
CN(C)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(C)c(F)s1 |r|
OC[C@@]1(F)CCCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
OC[C@]1(F)CCCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@H]2C[C@H]2C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1C[C@@H]2C[C@@H]2C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@@H]2C[C@@H]2C[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@H]1C[C@H]2C[C@H]2C[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@H]1C[C@@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C1CC1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
OC[C@@]1(F)CCCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
OC[C@]1(F)CCCN(C1)[C@H]1CCCC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CCCc1cccc(c1)[C@H]1CC[C@H](Nc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ccncn2)[C@H](C1)N(C)C |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccc(cc1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(OC(F)(F)F)c1 |r|
CN[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Br)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccon1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccon1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1C1CC1)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(Cl)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccccc1 |r|
CN(C)[C@H]1CN(CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@@H]1CN(CC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
C[N+](C)([O-])[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1C1CCC1)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(Cl)cc(Cl)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1O)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N[C@H]1CC[C@@H](C[C@@H]1N(C)C)c1cccc(c1)C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(N[C@H]2CC[C@@H](C[C@@H]2N2CCCC2)c2cccc(c2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2ccc(cc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2cccc(F)c2F)c2ccc(cc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(OC(F)(F)F)cc2)c2ccc(cc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccccc2)c2ccc(cc12)C(=O)NS(C)(=O)=O
COc1ncccc1-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2cncc(F)c2)c2ccc(cc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2cccnc2)c2ccc(cc12)C(=O)NS(C)(=O)=O
CCOc1ncc(cn1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cc1ccc(cc1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(cc2Cl)C(F)(F)F)c2ccc(cc12)C(=O)NS(C)(=O)=O
CC(C)Cc1ccc(cc1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2cccc(c2)C(F)(F)F)c2ccc(cc12)C(=O)NS(C)(=O)=O
CCc1ccc(cc1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cc1cccc(c1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)c1cccc(c1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
CCc1cccc(c1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2ccc(cc12)C(=O)NS(=O)(=O)C(F)(F)F
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2ccc(cc12)C(=O)NS(=O)(=O)c1cccs1
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2ccc(cc12)C(=O)NS(=O)(=O)c1ccc(F)c(F)c1
CC(C)COc1ccc(cc1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)COc1ccc(cn1)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)N(C)C
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)N1CCCCC1
CC(C)COc1ncc(cc1Cl)-c1cn(CC(C)C)c2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1cn(CC(C)C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1
CC(C)COc1ncc(cc1Cl)-c1cn(C(C)C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(cc2)C(F)F)c2ccc(cc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(cc2)C(F)F)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
CN(C)S(=O)(=O)NC(=O)c1ccc2c(cn(C)c2c1)-c1ccc(cc1)C(F)F
CN(C)S(=O)(=O)NC(=O)c1ccc2c(cn(C)c2c1)-c1ccc(cc1)C(F)(F)F
Cn1cc(-c2cnc(OCC3CC3)c(Cl)c2)c2ccc(cc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2cnc(OCC3CC3)c(Cl)c2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
CCS(=O)(=O)NC(=O)c1ccc2c(cn(C)c2c1)-c1cnc(OCC(C)C)c(Cl)c1
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C(C)C
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C(C)(C)C
CC(C)COc1ncc(cc1Cl)-c1nn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1n(C)nc2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1n(C)nc2cc(ccc12)C(=O)NS(=O)(=O)C1CC1
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(C(=O)NS(C)(=O)=O)c(F)cc12
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(C(=O)NS(=O)(=O)C3CC3)c(F)cc12
CC(C)COc1ccc(cn1)-c1cn(C)c2cc(C(=O)NS(C)(=O)=O)c(F)cc12
CC(C)COc1ccc(cn1)-c1cn(C)c2cc(C(=O)NS(=O)(=O)C3CC3)c(F)cc12
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2cc(F)c(cc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2cc(F)c(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(-c2ccc(cc2)C(F)F)c2cc(F)c(cc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(cc2)C(F)F)c2cc(F)c(cc12)C(=O)NS(=O)(=O)C1CC1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccnn1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccnn1)c1cc(F)c(cc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(F)cc(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(Cl)cc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(OC)cc(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cccc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(OC)cc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cccc(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cccc(c1)C1CC1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cccc(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(C)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(F)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(C)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(C)cc(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(C)cc(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(F)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(F)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(OC)c(F)c(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(F)c(F)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cc(Cl)c(F)c(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(F)cc(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(Cl)cc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)c(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(Cl)ccc1C
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(OC)cc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cccc(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cccc(c1)C1CC1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cccc(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(cnc1OC)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(Cl)cnc1OC
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(OC)nc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccnc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(F)cc1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(cc1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(c(OC)c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cccc(OC(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cccc(OC(C)C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(F)cc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(C)c(F)c(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(OC)cc(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(F)c(F)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(Cl)cc(c1)C#N
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)c(c1)C#N
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(ccc1F)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(OC(F)(F)F)ccc1OC
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)C1CC1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(C)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(C)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(OC)cc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(OC)c(F)c(OC)c1
CCOc1cc(ccc1F)-c1cc(OC)c(cc1Cl)N(C(=O)NC)c1ccc(cn1)S(=O)(=O)Nc1ccon1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cc(F)c(F)c(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)cc1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1ccc(cc1OC)-c1ccc(F)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1ccc(cc1OC)-c1cc(Cl)cc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1ccc(cc1OC)-c1ccc(Cl)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1ccc(cc1OC)-c1cc(F)cc(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)c(c1)C#N
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)c(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1cc(Cl)cc(c1)C#N
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1cc(OC)cc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(C)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1cc(OC)cc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1cccc(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1cc(F)c(F)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(Cl)c(c1)C(F)(F)F
CONC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(F)c(cc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(F)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(F)c(cc1OC)-c1ccc(F)c(c1)C(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccnn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccnn1)c1cc(Cl)c(cc1OC)-c1cc(F)c(F)c(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccnn1)c1cc(Cl)c(cc1OC)-c1cc(OC)nc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1ccc(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1ccc(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CCCCCCCCCCCCCCc1cc(OC)c(cc1F)N(C(=O)NC)c1ccc(cn1)S(=O)(=O)Nc1ncccn1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1nocc1C)c1cc(F)c(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1nocc1C)c1cc(F)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1nocc1C)c1cc(F)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cnsn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccc(F)n1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncco1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccnc(C)n1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccncn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(OCC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncccn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cnsn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccc(F)n1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncco1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccnc(C)n1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccncn1)c1cc(Cl)c(cc1OC)-c1ccc(F)c(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1cccnn1)c1cc(F)c(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ncco1)c1cc(F)c(cc1OC)-c1ccc(F)c(OC(F)(F)F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(ccc1OC)-c1cc(Cl)cc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(ccc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(ccc1OC)-c1cccc(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(ccc1OC)-c1cc(F)cc(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(ccc1OC)-c1ccc(C)c(Cl)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(c(Cl)cc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(c(Cl)cc1OC)-c1cccc(F)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(c(Cl)cc1OC)-c1cc(Cl)cc(OC)c1
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(c(Cl)cc1OC)-c1ccc(C)c(Cl)c1
COc1cc(c(Cl)cc1N(C(N)=O)c1ccc(cn1)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F
COc1cc(c(Cl)cc1N(C(N)=O)c1ccc(cn1)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(F)c1
COc1cc(c(Cl)cc1N(C(N)=O)c1ccc(cn1)S(=O)(=O)Nc1ccon1)-c1cc(Cl)cc(c1)C#N
COc1cc(cc(c1)C(F)(F)F)-c1cc(OC)c(cc1Cl)N(C(N)=O)c1ccc(cn1)S(=O)(=O)Nc1ccon1
COc1cc(c(Cl)cc1N(C(N)=O)c1ccc(cn1)S(=O)(=O)Nc1ccon1)-c1cccc(OCC(F)(F)F)c1
COC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1cccc(c1)C(F)(F)F
CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)C#CC1CCCC1
COc1ccc(CN(C)C(=O)N(c2ccc(SCc3ccccc3)cn2)c2cc(F)c(CCC(F)(F)F)cc2OC)cc1
COc1cc(ccc1Nc1ccc(cc1)S(=O)(=O)N(Cc1ccc(C=O)cc1)c1ccon1)-c1ccc(Cl)c(C)c1
CNC(=O)N(c1ccc(cc1)S(=O)(=O)N(Cc1ccc(OC)cc1)c1ccon1)c1cc(F)c(Br)cc1OC
COc1cc(C#CC2CCC(F)(F)CC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-.15,-2.31,;1.18,-3.08,;2.52,-2.31,;2.52,-.77,;3.85,,;3.85,1.54,;3.85,3.08,;3.85,4.62,;5.19,5.39,;5.19,6.93,;3.85,7.7,;4.62,9.03,;3.08,9.03,;2.52,6.93,;2.52,5.39,;5.19,-.77,;6.52,,;5.19,-2.31,;3.85,-3.08,;3.85,-4.62,;2.52,-5.39,;1.18,-4.62,;-.15,-5.39,;-.15,-6.93,;1.18,-7.7,;2.52,-6.93,;3.85,-7.7,;5.19,-6.93,;5.19,-5.39,;6.52,-4.62,;-1.48,-7.7,;-2.25,-6.37,;-.71,-9.03,;-2.82,-8.47,;-4.15,-7.7,;-5.61,-8.18,;-6.52,-6.93,;-5.61,-5.68,;-4.15,-6.16,)|
COc1cc(C#CC(C)(C)C(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-.15,-1.26,;1.18,-2.03,;2.52,-1.26,;2.52,.28,;3.85,1.05,;3.85,2.59,;3.85,4.13,;3.85,5.67,;3.08,7.01,;2.31,5.67,;5.19,6.44,;6.52,5.67,;5.19,7.98,;6.52,7.21,;5.19,.28,;6.52,1.05,;5.19,-1.26,;3.85,-2.03,;3.85,-3.57,;2.52,-4.34,;1.18,-3.57,;-.15,-4.34,;-.15,-5.88,;1.18,-6.65,;2.52,-5.88,;3.85,-6.65,;5.19,-5.88,;5.19,-4.34,;6.52,-3.57,;-1.48,-6.65,;-2.25,-5.31,;-.71,-7.98,;-2.82,-7.42,;-4.15,-6.65,;-5.61,-7.12,;-6.52,-5.88,;-5.61,-4.63,;-4.15,-5.11,)|
COc1cc(ccc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)C#CC1CCCC1 |(-.15,-1.29,;1.18,-2.06,;2.52,-1.29,;2.52,.25,;3.85,1.02,;5.19,.25,;5.19,-1.29,;3.85,-2.06,;3.85,-3.6,;2.52,-4.37,;1.18,-3.6,;-.15,-4.37,;-.15,-5.91,;1.18,-6.68,;2.52,-5.91,;3.85,-6.68,;5.19,-5.91,;5.19,-4.37,;6.52,-3.6,;-1.48,-6.68,;-2.25,-5.34,;-.71,-8.01,;-2.82,-7.45,;-4.15,-6.68,;-5.61,-7.15,;-6.52,-5.91,;-5.61,-4.66,;-4.15,-5.14,;3.85,2.56,;3.85,4.1,;3.85,5.64,;5.1,6.55,;4.62,8.01,;3.08,8.01,;2.61,6.55,)|
COc1cc(C#CC2CC2C(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.92,-14.18,;-1.92,-12.64,;-.58,-11.87,;.75,-12.64,;2.09,-11.87,;3.42,-12.64,;4.75,-13.41,;6.09,-14.18,;6.86,-15.51,;5.32,-15.58,;4.01,-16.4,;2.71,-17.21,;3.2,-15.09,;4.83,-17.7,;2.09,-10.33,;3.42,-9.56,;.75,-9.56,;-.58,-10.33,;-1.92,-9.56,;-1.92,-8.02,;-.58,-7.25,;-.58,-5.71,;-1.92,-4.94,;-3.25,-5.71,;-3.25,-7.25,;-4.58,-8.02,;-4.58,-9.56,;-3.25,-10.33,;-3.25,-11.87,;-1.92,-3.4,;-1.92,-1.86,;-3.46,-3.4,;-.38,-3.4,;.39,-2.06,;1.93,-2.06,;2.41,-.6,;1.16,.3,;-.08,-.6,)|
COc1cc(C#C[C@H]2C[C@@H]2C(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |r,wU:9.10,wD:7.6,(-.15,-1.93,;1.18,-2.7,;2.52,-1.93,;2.52,-.39,;3.85,.38,;3.85,1.92,;3.85,3.46,;3.85,5,;4.62,6.34,;3.08,6.34,;1.75,7.11,;.41,6.34,;1.75,8.65,;.41,7.88,;5.19,-.39,;6.52,.38,;5.19,-1.93,;3.85,-2.7,;3.85,-4.24,;2.52,-5.01,;1.18,-4.24,;-.15,-5.01,;-.15,-6.55,;1.18,-7.32,;2.52,-6.55,;3.85,-7.32,;5.19,-6.55,;5.19,-5.01,;6.52,-4.24,;-1.48,-7.32,;-2.25,-5.98,;-.71,-8.65,;-2.82,-8.09,;-4.15,-7.32,;-5.61,-7.79,;-6.52,-6.55,;-5.61,-5.3,;-4.15,-5.78,)|
COc1cc(C#C[C@@H]2C[C@@H]2C(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |r,wU:7.6,9.10,(-.15,-1.93,;1.18,-2.7,;2.52,-1.93,;2.52,-.39,;3.85,.38,;3.85,1.92,;3.85,3.46,;3.85,5,;4.62,6.34,;3.08,6.34,;1.75,7.11,;.41,6.34,;1.75,8.65,;.41,7.88,;5.19,-.39,;6.52,.38,;5.19,-1.93,;3.85,-2.7,;3.85,-4.24,;2.52,-5.01,;1.18,-4.24,;-.15,-5.01,;-.15,-6.55,;1.18,-7.32,;2.52,-6.55,;3.85,-7.32,;5.19,-6.55,;5.19,-5.01,;6.52,-4.24,;-1.48,-7.32,;-2.25,-5.98,;-.71,-8.65,;-2.82,-8.09,;-4.15,-7.32,;-5.61,-7.79,;-6.52,-6.55,;-5.61,-5.3,;-4.15,-5.78,)|
COc1cc(C#CC2(CC2)C(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-.15,-1.26,;1.18,-2.03,;2.52,-1.26,;2.52,.28,;3.85,1.05,;3.85,2.59,;3.85,4.13,;3.85,5.67,;2.31,5.67,;3.08,7.01,;5.19,6.44,;6.52,5.67,;5.19,7.98,;6.52,7.21,;5.19,.28,;6.52,1.05,;5.19,-1.26,;3.85,-2.03,;3.85,-3.57,;2.52,-4.34,;1.18,-3.57,;-.15,-4.34,;-.15,-5.88,;1.18,-6.65,;2.52,-5.88,;3.85,-6.65,;5.19,-5.88,;5.19,-4.34,;6.52,-3.57,;-1.48,-6.65,;-2.25,-5.31,;-.71,-7.98,;-2.82,-7.42,;-4.15,-6.65,;-5.61,-7.12,;-6.52,-5.88,;-5.61,-4.63,;-4.15,-5.11,)|
COc1cc(C#CC2CCCC2)c(Cl)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-.15,-1.29,;1.18,-2.06,;2.52,-1.29,;2.52,.25,;3.85,1.02,;3.85,2.56,;3.85,4.1,;3.85,5.64,;5.1,6.55,;4.62,8.01,;3.08,8.01,;2.61,6.55,;5.19,.25,;6.52,1.02,;5.19,-1.29,;3.85,-2.06,;3.85,-3.6,;2.52,-4.37,;1.18,-3.6,;-.15,-4.37,;-.15,-5.91,;1.18,-6.68,;2.52,-5.91,;3.85,-6.68,;5.19,-5.91,;5.19,-4.37,;6.52,-3.6,;-1.48,-6.68,;-2.25,-5.34,;-.71,-8.01,;-2.82,-7.45,;-4.15,-6.68,;-5.61,-7.15,;-6.52,-5.91,;-5.61,-4.66,;-4.15,-5.14,)|
COc1cc(C#C[C@@H]2CCCC(F)(F)C2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |r,wU:7.6,(-.15,-1.93,;1.18,-2.7,;2.52,-1.93,;2.52,-.39,;3.85,.38,;3.85,1.92,;3.85,3.46,;3.85,5,;5.19,5.77,;5.19,7.31,;3.85,8.08,;2.52,7.31,;.98,7.31,;1.75,8.65,;2.52,5.77,;5.19,-.39,;6.52,.38,;5.19,-1.93,;3.85,-2.7,;3.85,-4.24,;2.52,-5.01,;1.18,-4.24,;-.15,-5.01,;-.15,-6.55,;1.18,-7.32,;2.52,-6.55,;3.85,-7.32,;5.19,-6.55,;5.19,-5.01,;6.52,-4.24,;-1.48,-7.32,;-2.25,-5.98,;-.71,-8.65,;-2.82,-8.09,;-4.15,-7.32,;-5.61,-7.79,;-6.52,-6.55,;-5.61,-5.3,;-4.15,-5.78,)|
COc1cc(C#CC2(CCCC2)OCC(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(-1.48,-1.29,;-.15,-2.06,;1.18,-1.29,;1.18,.25,;2.52,1.02,;2.52,2.56,;2.52,4.1,;2.52,5.64,;2.99,7.11,;1.75,8.01,;.5,7.11,;.98,5.64,;3.85,4.87,;5.19,5.64,;6.52,4.87,;7.85,5.64,;6.52,3.33,;7.85,4.1,;3.85,.25,;5.19,1.02,;3.85,-1.29,;2.52,-2.06,;2.52,-3.6,;1.18,-4.37,;-.15,-3.6,;-1.48,-4.37,;-1.48,-5.91,;-.15,-6.68,;1.18,-5.91,;2.52,-6.68,;3.85,-5.91,;3.85,-4.37,;5.19,-3.6,;-2.82,-6.68,;-3.59,-5.34,;-2.05,-8.01,;-4.15,-7.45,;-5.48,-6.68,;-6.95,-7.15,;-7.85,-5.91,;-6.95,-4.66,;-5.48,-5.14,)|
NC(=O)c1cccc(n1)-c1ccc2[nH]ccc2c1
FC(F)(F)c1ccc(NC(=O)c2cccc(n2)-c2ccc3[nH]ccc3c2)cc1
FC(F)(F)c1ccc(cc1)N(C(=O)c1cccc(n1)-c1ccc2[nH]ccc2c1)c1ccc(cc1)C(F)(F)F
C[C@H](Nc1cc(nc(n1)-c1ccc2[nH]ccc2c1)C(N)=O)C(N)=O |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)-c1ccc2[nH]ccc2c1 |r|
NC(=O)c1cc(O[C@H]2CCNC2=O)nc(n1)-c1ccc2[nH]ccc2c1 |r|
CC(C)Cn1ccc2cc(ccc12)-c1cccc(n1)S(=O)(=O)Nc1ncns1
COc1ccc(-c2nc3cc(ccc3n2-c2ccc(F)cc2)-c2nc(N[C@H]3CCNC3=O)cc(n2)C(N)=O)c(OC)c1 |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)-c1ccc2ncn(-c3ccc(cc3)C(F)(F)F)c2c1 |r|
NC(=O)c1cc(N[C@H]2CCNC2=O)nc(n1)-c1ccc2n(cnc2c1)-c1ccc(cc1)C(F)(F)F |r|
CC(C)Cn1ccc2cc(ccc12)-c1nc(N[C@@H](C)C(N)=O)cc(n1)C(N)=O |r|
OC[C@H](O)c1ccnc(n1)-c1ccc2ncn(-c3ccc(cc3)C(F)(F)F)c2c1 |r|
OC[C@@H](O)c1ccnc(n1)-c1ccc2ncn(-c3ccc(cc3)C(F)(F)F)c2c1 |r|
NC(=O)c1cccc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1
NC(=O)c1cccc(n1)-c1ccc2n(ccc2c1)S(=O)(=O)c1ccc(cc1)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc2n(CC3CCCCC3)ccc2c1
NC(=O)c1cccc(n1)-c1ccc2n(ccc2c1)S(=O)(=O)C1CCCCC1
NC(=O)c1cccc(n1)-c1ccc2n(Cc3ccc(F)cc3)ccc2c1
Cc1ccc(Cn2ccc3cc(ccc23)-c2cccc(n2)C(N)=O)cc1
NC(=O)c1cccc(n1)-c1ccc2n(CCC3CCCCC3)ccc2c1
NC(=O)c1cccc(n1)-c1ccc2n(Cc3ccncc3)ccc2c1
NC(=O)c1cccc(n1)-c1ccc2n(CCN3CCOCC3)ccc2c1
Cc1noc(C)c1Cn1ccc2cc(ccc12)-c1cccc(n1)C(N)=O
CC(C)Cn1ccc2cc(ccc12)-c1cccc(n1)C(N)=O
Cc1nc(Cn2ccc3cc(ccc23)-c2cccc(n2)C(N)=O)cs1
Cn1ccc2cc(ccc12)-c1cccc(n1)C(=O)Nc1ccc(cc1)C(F)(F)F
O=C(NC1CCCCC1)c1cccc(n1)-c1ccc2[nH]ccc2c1
FC(F)(F)c1ccc(NC(=O)c2cccc(n2)-c2ccc3[nH]ncc3c2)cc1
FC(F)(F)c1ccc(NC(=O)c2cc(N[C@H]3CCNC3=O)nc(n2)-c2ccc3[nH]ccc3c2)cc1 |r|
C[C@H](Nc1cc(nc(n1)-c1ccc2occc2c1)C(=O)Nc1ccc(cc1)C(F)(F)F)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc2[nH]ccc2c1)C(=O)Nc1ccc(cc1)C(F)(F)F)C(N)=O |r|
FC(F)(F)c1ccc(NC(=O)c2cccc(n2)-c2ccc3occc3c2)cc1
O=C(NCC1CCCCC1)c1cccc(n1)-c1ccc2[nH]ccc2c1
O=C(N1CCCC1)c1cccc(n1)-c1ccc2[nH]ccc2c1
O=C(NC1CCCC1)c1cccc(n1)-c1ccc2[nH]ccc2c1
CC1CN(CC(C)O1)C(=O)c1cccc(n1)-c1ccc2[nH]ccc2c1
O=C(Nc1nnn[nH]1)c1cccc(n1)-c1ccc2[nH]ccc2c1
FC(F)(F)c1ccc(NC(=O)c2cc(N[C@H]3CCNC3=O)cc(n2)-c2ccc3[nH]ccc3c2)cc1 |r|
NC(=O)c1cccc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ncc2c1
OC[C@@H](O)c1cccc(n1)-c1cnc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ncc2c1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2nn(Cc3ccc(cc3)C(F)(F)F)cc2c1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)cnc2c1 |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2n(ccc2c1)S(=O)(=O)N1CCCCC1 |r|
C[C@H](Nc1cc(nc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)-c1ccc2n(CC3CCCCC3)ccc2c1)C(N)=O)C(N)=O |r|
OC[C@H](O)c1cc(nc(c1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1)C#N |r|
NC(=O)c1cc(cc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1)[C@@H](O)CO |r|
NC(=O)c1cc(cc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1)[C@H](O)CO |r|
NC(=O)c1cc(cc(n1)[C@@H](O)CO)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1 |r|
NC(=O)c1cc(cc(n1)[C@H](O)CO)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1 |r|
CC(C)Cn1ccc2cc(ccc12)-c1cc(cc(n1)C(N)=O)[C@H](O)CO |r|
CC(C)Cn1ccc2cc(ccc12)-c1cc(cc(n1)C(N)=O)[C@@H](O)CO |r|
CC(C)Cn1ccc2cc(ccc12)-c1cc(nc(c1)C(N)=O)[C@H](O)CO |r|
Cn1cc(-c2cccc(c2)C(F)(F)F)c2cc(ccc12)-c1cccc(n1)C(N)=O
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2cc(ccc12)-c1cccc(n1)C(N)=O
CCN(CC)CCn1cc(-c2ccc(F)cc2)c2ccc(cc12)-c1cccc(n1)C(N)=O
Nc1cc(nc(n1)-c1ccc2occc2c1)C(=O)Nc1ccc(cc1)C(F)(F)F
OC(=O)c1c[nH]c2ccc(cc12)-c1cccc(n1)C(=O)Nc1ccc(cc1)C(F)(F)F
NC(=O)c1c[nH]c2ccc(cc12)-c1cccc(n1)C(=O)Nc1ccc(cc1)C(F)(F)F
NC(=O)CC[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1cccc(n1)C(=O)Nc1ccc(cc1)C(F)(F)F)C(N)=O |r|
NC(=O)c1cn(Cc2ccc(cc2)C(F)(F)F)c2ccc(cc12)-c1cccc(n1)C(N)=O
C[C@H](NC(=O)c1cn(Cc2ccc(cc2)C(F)(F)F)c2ccc(cc12)-c1cccc(n1)C(N)=O)C(N)=O |r|
NC(=O)c1cccc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)cc(CN[C@H]3CCNC3=O)c2c1 |r|
NC(=O)c1cccc(n1)-c1ccc2n(CC3CCCCC3)cc(CN[C@H]3CCNC3=O)c2c1 |r|
CC(C)Cn1ccc2cc(ccc12)-c1cccc(n1)[C@H](O)[C@@H](O)C(N)=O |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc2n(CC3CCCCC3)ccc2c1 |r|
NC(=O)[C@H](O)[C@@H](O)c1cccc(n1)-c1ccc2n(CC3CC3)ccc2c1 |r|
CC(C)Cn1ncc2cc(ccc12)-c1cccc(n1)[C@H](O)[C@@H](O)C(N)=O |r|
NC(=O)c1csc(n1)-c1ccc2n(Cc3ccc(cc3)C(F)(F)F)ccc2c1
C[C@H](Nc1cc(nc(n1)N1CCc2c(C1)cccc2-c1ccc(cc1)C(F)(F)F)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCc2c(C1)cccc2-c1ccc(cn1)C(F)(F)F)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCc2c(C1)cccc2-c1ccccc1C(F)(F)F)C(N)=O)C(N)=O |r|
NC(=O)c1cccc(n1)N1CCc2c(C1)cccc2-c1ccc(cc1)C(F)(F)F
NC(=O)[C@@H](O)[C@H](O)c1cccc(n1)N1CCc2c(C1)cccc2-c1ccc(cc1)C(F)(F)F |r|
C[C@H](Nc1cc(nc(n1)N1CCc2c(C1)cccc2-c1cccc(c1)C(F)(F)F)C(N)=O)C(N)=O |r|
C[C@H](Nc1cc(nc(n1)N1CCc2c(C1)cccc2C1=CCCCC1)C(N)=O)C(N)=O |r,t:22|
FC(F)(F)c1ccc(cc1)-c1cccc2CN(CCc12)c1cccc(n1)S(=O)(=O)Nc1ncns1
C[C@H](Nc1cc(nc(n1)N1CCc2c(C1)cccc2C1CCCCC1)C(N)=O)C(N)=O |r|
NC(=O)c1cc(cc(n1)[C@H](O)CO)N1CCc2c(C1)cccc2-c1ccc(cc1)C(F)(F)F |r|
NC(=O)c1cc(cc(n1)[C@@H](O)CO)N1CCc2c(C1)cccc2-c1ccc(cc1)C(F)(F)F |r|
NC(=O)c1cc(C2CC2)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:21:12:19:15.16.17,THB:21:16:19:20.13.12,20:18:15:21.13.12,20:12:15:19.18.17,11:12:15:19.18.17,11:12:19:15.16.17|
NC(=O)c1cc(C2CC2)c(COc2ccc(Cl)cc2C#N)cc1F
NC(=O)c1cc(C2CC2)c(COc2cc(Cl)cc(Cl)c2)cc1F
NC(=O)c1cc(Cl)c(OCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:19:10:17:13.14.15,THB:19:14:17:18.11.10,18:16:13:19.11.10,18:10:13:17.16.15,9:10:13:17.16.15,9:10:17:13.14.15|
Cc1ccc(OCc2cc(F)c(cc2C2CC2)C(N)=O)cc1C
Fc1cc(C(=O)NS(=N)(=O)C2CC2)c(F)cc1Oc1ccc(OC(F)(F)F)c(Cl)c1
FC(F)C(F)(F)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=N)(=O)C2CC2)cc1Cl
Fc1cc(COc2cc(Cl)cc(OC(F)(F)F)c2)c(cc1C(=O)NS(=N)(=O)C1CC1)C1CC1
Fc1cc(OCc2cc(F)c(cc2C2CC2)C(=O)NS(=N)(=O)C2CC2)cc(c1)C(F)(F)F
FC(F)C(F)(F)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=N)(=O)N2CCC2)cc1Cl
Fc1cc(OCC23CC4CC(CC(C4)C2)C3)c(cc1C(=O)NS(=N)(=O)N1CCC1)C1CC1 |TLB:15:6:13:9.10.11,THB:15:10:13:6.14.7,14:6:9:13.12.11,14:12:9:6.15.7,5:6:13:9.10.11|
Fc1cc(Oc2cnc(OCC(F)(F)F)c(Cl)c2)c(Cl)cc1C(=O)NS(=N)(=O)C1CC1
COc1ncccc1-c1cc(C(=O)NS(=N)(=O)C2CC2)c(F)cc1Oc1cnc(OC(C)C)c(Cl)c1
CC(C)Oc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=N)(=O)C2CC2)cc1Cl
Fc1cc(O[C@@H]2CCCN(Cc3c(Cl)cccc3Cl)C2)c(cc1C(=O)NS(=N)(=O)C1CC1)C1CC1 |r|
COc1cc(C(=O)NS(=N)(=O)C2CC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:29:20:27:23.24.25,19:20:23:27.26.25,THB:29:24:27:20.28.21,28:20:23:27.26.25,28:26:23:20.29.21|
Fc1cc(OCC2(F)CCN(Cc3cc(cc(Cl)c3F)C(F)(F)F)CC2)c(cc1C(=O)NS(=N)(=O)C1CC1)C1CC1
C[C@H](N1CCC(COc2ccc(cc2C2CC2)C(=O)NS(=N)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=N)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
Fc1cc(NCCC2CCNCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CCCNC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CCCCN2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Fc1cc(NCCC2CCCCN2)c(Cl)cc1S(=O)(=O)Nc1nccs1
CN1CCC(CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1
Fc1cc(NCC2CNCCO2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2COCCO2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2(CN3CCOCC3)CC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2CCCOC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2CCCCO2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2CCOCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2(CN3CCCC3)CC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CCNC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
COCCN1CCCC1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
Fc1cc(NCC2CNC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CNC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
N[C@H]1CC[C@@H](CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |r,wU:4.4,1.0,(2.3,-59.56,;2.29,-58.02,;.96,-57.25,;.96,-55.71,;2.3,-54.94,;2.3,-53.39,;3.62,-52.63,;3.61,-51.07,;4.95,-50.28,;4.95,-48.74,;6.28,-47.97,;6.28,-46.43,;7.61,-48.73,;7.61,-50.28,;6.27,-51.05,;6.28,-52.59,;8.95,-47.95,;8.18,-46.61,;9.72,-46.61,;10.3,-48.72,;11.63,-47.94,;11.62,-46.41,;13.08,-45.93,;13.99,-47.17,;13.09,-48.42,;3.62,-55.7,;3.62,-57.25,)|
N[C@H]1CC[C@H](CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |r,wU:1.0,wD:4.4,(12.18,-61.35,;12.18,-59.81,;10.84,-59.04,;10.84,-57.5,;12.18,-56.73,;12.18,-55.19,;13.5,-54.42,;13.49,-52.86,;14.83,-52.07,;14.83,-50.53,;16.16,-49.76,;16.16,-48.22,;17.49,-50.53,;17.49,-52.07,;16.16,-52.84,;16.16,-54.38,;18.83,-49.74,;18.06,-48.41,;19.6,-48.4,;20.18,-50.51,;21.51,-49.73,;21.5,-48.2,;22.96,-47.73,;23.87,-48.96,;22.97,-50.21,;13.51,-57.5,;13.5,-59.05,)|
N[C@H]1CC[C@@H](CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)CC1 |r,wU:4.4,1.0,(19.01,-58.71,;20.34,-57.93,;20.34,-56.39,;21.68,-55.62,;23.01,-56.39,;24.33,-55.62,;24.31,-54.07,;25.66,-53.28,;25.66,-51.74,;26.98,-50.96,;26.98,-49.43,;28.32,-51.73,;28.32,-53.28,;26.99,-54.05,;26.98,-55.58,;29.66,-50.95,;28.88,-49.61,;30.43,-49.61,;31.01,-51.72,;32.33,-50.94,;32.32,-49.41,;33.78,-48.94,;34.69,-50.16,;33.79,-51.42,;23.01,-57.93,;21.68,-58.7,)|
N[C@H]1CC[C@@H](CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |r,wU:4.4,1.0,(32.42,-58.42,;33.76,-57.64,;33.76,-56.1,;35.1,-55.33,;36.43,-56.1,;37.75,-55.33,;37.73,-53.78,;39.08,-52.99,;39.08,-51.45,;40.4,-50.67,;40.4,-49.14,;41.74,-51.44,;41.74,-52.99,;40.41,-53.75,;40.4,-55.29,;43.08,-50.66,;42.3,-49.32,;43.85,-49.32,;44.43,-51.43,;45.75,-50.65,;45.74,-49.12,;47.2,-48.65,;48.11,-49.87,;47.21,-51.13,;36.43,-57.64,;35.1,-58.41,)|
N[C@H]1CC[C@H](CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |r,wU:1.0,wD:4.4,(46.21,-58.36,;47.55,-57.58,;47.55,-56.04,;48.89,-55.27,;50.21,-56.04,;51.54,-55.27,;51.52,-53.72,;52.86,-52.92,;52.86,-51.39,;54.19,-50.61,;54.19,-49.08,;55.53,-51.38,;55.53,-52.93,;54.19,-53.69,;54.19,-55.23,;56.86,-50.6,;56.09,-49.26,;57.63,-49.26,;58.21,-51.37,;59.53,-50.59,;59.53,-49.05,;60.99,-48.58,;61.89,-49.81,;61,-51.06,;50.21,-57.58,;48.88,-58.35,)|
Fc1cc(NCC2CCC(CC2)NC2CC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |(.5,5.9,;.5,4.36,;-.83,3.59,;-.83,2.05,;-2.17,1.28,;-2.17,-.26,;-3.5,-1.03,;-4.83,-.26,;-6.17,-1.03,;-6.17,-2.57,;-4.83,-3.34,;-3.5,-2.57,;-7.5,-3.34,;-7.5,-4.88,;-8.27,-6.21,;-6.73,-6.21,;.5,1.28,;.5,-.26,;1.83,2.05,;1.83,3.59,;3.17,4.36,;1.83,5.13,;4.5,5.13,;4.5,3.59,;5.83,4.36,;7.24,3.73,;8.27,4.88,;7.5,6.21,;6,5.89,)|
CNC1CCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |(-7.89,-5.55,;-7.89,-4.01,;-6.55,-3.24,;-6.55,-1.7,;-5.22,-.93,;-3.89,-1.7,;-2.55,-.93,;-2.55,.61,;-1.22,1.38,;-1.22,2.92,;.11,3.69,;.11,5.23,;1.45,2.92,;1.45,1.38,;.11,.61,;.11,-.93,;2.78,3.69,;1.45,4.46,;4.12,4.46,;4.12,2.92,;5.45,3.69,;6.86,3.07,;7.89,4.21,;7.12,5.55,;5.61,5.23,;-3.89,-3.24,;-5.22,-4.01,)|
CN(C)C1CCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |(-7.99,-2.58,;-7.59,-4.06,;-8.18,-5.49,;-6.26,-3.29,;-6.26,-1.75,;-4.93,-.98,;-3.59,-1.75,;-2.26,-.98,;-2.26,.56,;-.92,1.33,;-.92,2.87,;.41,3.64,;.41,5.18,;1.74,2.87,;1.74,1.33,;.41,.56,;.41,-.98,;3.08,3.64,;1.74,4.41,;4.41,4.41,;4.41,2.87,;5.74,3.64,;7.15,3.01,;8.18,4.15,;7.41,5.49,;5.91,5.17,;-3.59,-3.29,;-4.93,-4.06,)|
Fc1cc(NCC2CCC(CC2)N2CCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |(1.2,5.01,;1.2,3.47,;-.14,2.7,;-.14,1.16,;-1.47,.39,;-1.47,-1.15,;-2.81,-1.92,;-4.14,-1.15,;-5.47,-1.92,;-5.47,-3.46,;-4.14,-4.23,;-2.81,-3.46,;-6.81,-4.23,;-7.88,-3.14,;-8.97,-4.23,;-7.88,-5.32,;1.2,.39,;1.2,-1.15,;2.53,1.16,;2.53,2.7,;3.86,3.47,;2.53,4.24,;5.2,4.24,;5.2,2.7,;6.53,3.47,;7.94,2.84,;8.97,3.99,;8.2,5.32,;6.69,5,)|
Fc1cc(NCC2CCC(CC2)N2CCOCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |(1.45,5.62,;1.45,4.08,;.11,3.31,;.11,1.77,;-1.22,1,;-1.22,-.54,;-2.55,-1.31,;-3.89,-.54,;-5.22,-1.31,;-5.22,-2.85,;-3.89,-3.62,;-2.55,-2.85,;-6.55,-3.62,;-7.89,-2.85,;-9.22,-3.62,;-9.22,-5.16,;-7.89,-5.93,;-6.55,-5.16,;1.45,1,;1.45,-.54,;2.78,1.77,;2.78,3.31,;4.12,4.08,;2.78,4.85,;5.45,4.85,;5.45,3.31,;6.78,4.08,;8.19,3.45,;9.22,4.6,;8.45,5.93,;6.94,5.61,)|
CN1CCN(CC1)C1CCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |(-9.89,-5.93,;-8.55,-5.16,;-8.55,-3.62,;-7.22,-2.85,;-5.89,-3.62,;-5.89,-5.16,;-7.22,-5.93,;-4.55,-2.85,;-4.55,-1.31,;-3.22,-.54,;-1.89,-1.31,;-.55,-.54,;-.55,1,;.78,1.77,;.78,3.31,;2.12,4.08,;2.12,5.62,;3.45,3.31,;3.45,1.77,;2.12,1,;2.12,-.54,;4.78,4.08,;3.45,4.85,;6.12,4.85,;6.12,3.31,;7.45,4.08,;8.86,3.45,;9.89,4.6,;9.12,5.93,;7.61,5.61,;-1.89,-2.85,;-3.22,-3.62,)|
NC1CCCC(C1)Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
NC1(CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CCCCC1
CC1CC(C)(C)C(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1N
NC1CCCC1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
NCC1CCCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1
OC1CCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CC1 |(-8.55,-3.62,;-7.22,-2.85,;-7.22,-1.31,;-5.89,-.54,;-4.55,-1.31,;-3.22,-.54,;-1.89,-1.31,;-.55,-.54,;-.55,1,;.78,1.77,;.78,3.31,;2.12,1,;2.12,-.54,;.78,-1.31,;.78,-2.85,;3.45,1.77,;2.36,2.86,;4.54,2.86,;4.78,1,;6.12,1.77,;7.52,1.14,;8.55,2.29,;7.78,3.62,;6.28,3.3,;-4.55,-2.85,;-5.89,-3.62,)|
OC1(CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CCCC1
Fc1cc(N[C@@H]2CC[C@H](Cl)CC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r,wU:5.4,8.8,(.11,2.92,;.11,1.38,;-1.22,.61,;-1.22,-.93,;-2.55,-1.7,;-3.89,-.93,;-3.89,.61,;-5.22,1.38,;-6.55,.61,;-7.89,1.38,;-6.55,-.93,;-5.22,-1.7,;.11,-1.7,;.11,-3.24,;1.45,-.93,;1.45,.61,;2.78,1.38,;1.69,2.47,;3.87,2.47,;4.12,.61,;5.45,1.38,;6.86,.76,;7.89,1.9,;7.12,3.24,;5.61,2.92,)|
Fc1cc(NCCCC2CCOC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2CCOC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CCCO2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2CCCO2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC23CCOC2OCC3)c(Cl)cc1S(=O)(=O)Nc1nccs1
CC1(O)CC(CC(C)(O)N1O)Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
Fc1cc(NC[C@@H]2CCCNC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
Fc1cc(c(F)cc1OCCC1(CCNCC1)c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1
Fc1cc(OCCC2(CCNCC2)c2ccc(Cl)cc2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Fc1cc(ccc1Cl)C1(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)CCNCC1
Fc1cc(ccc1Cl)C1(CCOc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)CCNCC1
OC1CCC(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1
NC1CCC(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1
NC1CCC(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1
NC1CCC(CCOc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1
CNC1CCC(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1
Fc1cc(c(F)cc1OCCC1(CCC(CC1)NC1CC1)c1ccccc1)S(=O)(=O)Nc1ncns1
NC1CCC(CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)(CC1)c1ccccc1
NC1CCC(CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)(CC1)c1ccccc1
CC1(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)CCC(N)CC1
CC1(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)CCC(N)CC1
NC1CCC(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccc(Cl)cc1
NC1CCC(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccc(Cl)cc1
NC1CCC(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)CC1 |(-5.22,-6.7,;-5.22,-5.16,;-6.55,-4.39,;-6.55,-2.85,;-5.22,-2.08,;-5.22,-.54,;-3.89,.23,;-3.89,1.77,;-2.55,2.54,;-2.55,4.08,;-1.22,4.85,;-1.22,6.39,;.11,4.08,;.11,2.54,;-1.22,1.77,;-1.22,.23,;1.45,4.85,;.11,5.62,;2.78,5.62,;2.78,4.08,;4.12,4.85,;5.52,4.22,;6.55,5.37,;5.78,6.7,;4.28,6.38,;-3.89,-2.85,;-3.89,-4.39,)|
NC1CCC(COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(Cc2ccc(Cl)c(F)c2)CC1
NC1CCC(COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(Cc2ccc(Cl)c(F)c2)CC1
CNC1CCC(COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(Cc2ccc(Cl)c(F)c2)CC1
OC1CCC(COc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(Cc2ccc(Cl)c(F)c2)CC1
Fc1cc(NC2CCC3CNCC23)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(N2CCCC(C2)C2CCNCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(N2CCC3CCNCC3C2)c(Cl)cc1S(=O)(=O)Nc1nccs1
COCC1CCN(C1)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
OCC1CCN(C1)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CCOCC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CCCOC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC2CCS(=O)(=O)CC2)c(Cl)cc1S(=O)(=O)Nc1nccs1
OC1CCCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1
ON1CCCCC1CCNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cc(ccc1F)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cc(ccc1F)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |r|
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1F)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1F)C(F)(F)F |r|
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(Cl)c1 |r|
COc1cc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)F |r|
COc1cc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)F |r|
COc1cc(ccc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(ccc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(cc(F)c1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(cc(F)c1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1nc(c(F)cc1N1[C@@H]2CCN(C[C@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1nc(c(F)cc1N1[C@H]2CCN(C[C@@H]2OCC1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
Fc1cc(N2[C@@H]3CCN(C[C@H]3OCC2=O)S(=O)(=O)Nc2ccon2)c(cc1-c1cccc(c1)C(F)(F)F)C#N |r|
Fc1cc(N2[C@H]3CCN(C[C@@H]3OCC2=O)S(=O)(=O)Nc2ccon2)c(cc1-c1cccc(c1)C(F)(F)F)C#N |r|
COc1cc(c(F)cc1N1CCO[C@@H]2CN(CC[C@@H]12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1CCO[C@H]2CN(CC[C@H]12)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1CCO[C@@H]2CN(CC[C@@H]12)S(=O)(=O)Nc1ccncn1)-c1cccc(c1)C(F)(F)F |r|
COc1cc(c(F)cc1N1CCO[C@H]2CN(CC[C@H]12)S(=O)(=O)Nc1ccncn1)-c1cccc(c1)C(F)(F)F |r|
[H][C@@]12CN(CC[C@@]1([H])N(C(=O)CO2)c1cc(F)c(cc1OC)-c1cccc(OC(F)(F)F)c1)S(=O)(=O)Nc1ccon1 |r|
[H][C@]12CN(CC[C@]1([H])N(C(=O)CO2)c1cc(F)c(cc1OC)-c1cccc(OC(F)(F)F)c1)S(=O)(=O)Nc1ccon1 |r|
[H][C@@]12CN(CC[C@@]1([H])N(CCO2)c1cc(F)c(cc1OC)-c1cccc(OC(F)(F)F)c1)S(=O)(=O)Nc1ccon1 |r|
[H][C@]12CN(CC[C@]1([H])N(CCO2)c1cc(F)c(cc1OC)-c1cccc(OC(F)(F)F)c1)S(=O)(=O)Nc1ccon1 |r|
[H][C@]12COC(=O)N(c3cc(F)c(cc3OC)-c3cccc(c3)C(F)(F)F)[C@]1([H])CCN(C2)S(=O)(=O)Nc1ccon1 |r|
[H][C@@]12COC(=O)N(c3cc(F)c(cc3OC)-c3cccc(c3)C(F)(F)F)[C@@]1([H])CCN(C2)S(=O)(=O)Nc1ccon1 |r|
[H][C@]12CCC(=O)N(c3cc(F)c(cc3OC)-c3cccc(c3)C(F)(F)F)[C@]1([H])CCN(C2)S(=O)(=O)Nc1ccon1 |r|
[H][C@@]12CCC(=O)N(c3cc(F)c(cc3OC)-c3cccc(c3)C(F)(F)F)[C@]1([H])CCN(C2)S(=O)(=O)Nc1ccon1 |r|
[H][C@@]12CCC(=O)N(c3cc(F)c(cc3OC)-c3cccc(c3)C(F)(F)F)[C@@]1([H])CCN(C2)S(=O)(=O)Nc1ccon1 |r|
[H][C@]12CCC(=O)N(c3cc(F)c(cc3OC)-c3cccc(c3)C(F)(F)F)[C@@]1([H])CCN(C2)S(=O)(=O)Nc1ccon1 |r|
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCOCC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1
FC(F)(F)S(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1
O=C(NS(=O)(=O)C1CC1)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC(F)(F)C3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCC(F)(F)CC3)nc2)cc1
Cc1cc(OCC2CC2)ncc1-c1cccc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCCC3)nc2)cc1
Cc1cc(cnc1OCC1CC1)-c1cccc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
CC(C)(C)OC(=O)N1CCC(COc2ccc(cn2)-c2cccc(OCc3ccc(cc3)C(=O)NS(C)(=O)=O)c2)CC1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(ccc2Cl)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(Cl)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCC3)nc2)cc1
CS(=O)(=O)NC(=O)c1cc(Cl)c(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1F
Fc1cc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
O=C(NS(=O)(=O)c1cccs1)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1
O=C(NS(=O)(=O)c1nccs1)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1
Fc1cc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(Cl)cc1C(=O)NS(=O)(=O)c1cccs1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(Cl)cc(c2)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2ccc(Cl)c(c2)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1F
CS(=O)(=O)NC(=O)c1cc(F)c(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1F
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCOCC3)nc2)c(F)c1
CS(=O)(=O)NC(=O)c1cc(OC(F)F)c(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1F
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)cc1F
CS(=O)(=O)NC(=O)c1cc(F)c(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(F)c1
O=C(NS(=O)(=O)C1CC1)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCOCC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1cc(F)c(COc2cc(F)cc(c2)-c2ccc(OCC3CC3)nc2)cc1F
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccc(OCC3CC3)nc2)c(F)c1
Fc1cc(OCc2ccc(cc2F)C(=O)NS(=O)(=O)C2CC2)cc(c1)-c1ccc(OCC2CC2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(cc(c2)-c2ccc(OCC3CC3)nc2)C2CC2)cc1
Cc1cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)cc(c1)-c1ccc(OCC2CC2)nc1
Cc1cc(OCc2ccc(cc2F)C(=O)NS(=O)(=O)C2CC2)cc(c1)-c1ccc(OCC2CC2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(cc(c2)C(F)(F)F)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2F)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(c1)C#N
O=C(NS(=O)(=O)C1CC1)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(c1)C#N
CS(=O)(=O)NC(=O)c1ccc(COc2ccc(F)c(c2)-c2ccc(OCC3CC3)nc2)cc1
Fc1ccc(OCc2ccc(cc2)C(=O)NS(=O)(=O)C2CC2)cc1-c1ccc(OCC2CC2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(ccc2F)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(Br)cc(c2)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2ccc(F)c(c2)-c2ccc(OCC3CC3)nc2)c(F)c1
Fc1ccc(OCc2ccc(cc2F)C(=O)NS(=O)(=O)C2CC2)cc1-c1ccc(OCC2CC2)nc1
Cc1ccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)cc1-c1ccc(OCC2CC2)nc1
Cc1ccc(OCc2ccc(cc2F)C(=O)NS(=O)(=O)C2CC2)cc1-c1ccc(OCC2CC2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2ccc(Cl)c(c2)-c2ccc(OCC3CC3)nc2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCC3)nc2)c(F)c1
CCS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(F)c1
CC(C)S(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)c(F)c1
Fc1cc(ccc1COc1cccc(c1)-c1ccc(OCC2CC2)nc1)C(=O)NS(=O)(=O)C1CC1
Fc1cc(ccc1COc1cccc(c1)-c1ccc(OCC2CC2)nc1)C(=O)NS(=O)(=O)CC1CC1
Fc1cc(ccc1COc1cccc(c1)-c1ccc(OCC2CC2)nc1)C(=O)NS(=O)(=O)c1cccs1
Fc1cc(ccc1COc1cccc(c1)-c1ccc(OCC2CC2)nc1)C(=O)NS(=O)(=O)c1nccs1
COc1cc(ccc1COc1cccc(c1)-c1ccc(OCC2CC2)nc1)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cccnc2OCC2CC2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cncc(OCC3CC3)c2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)nc2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccc(OCC3CC3)nc2)nc1
O=C(NS(=O)(=O)C1CC1)c1ccc(COc2cc(ccn2)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(n2)-c2ccc(OCC3CC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cccc(OCC3CC3)n2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ncc(OCC3CC3)cc2Cl)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ncc(OCC3CC3)cc2F)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccnc(OCC3CC3)c2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CC3)cn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CC3)cn2)c(F)c1
O=C(NS(=O)(=O)C1CC1)c1ccc(COc2cccc(c2)-c2cnc(OCC3CC3)cn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cncc(OCC3CC3)n2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ncc(OCC3CC3)cn2)c(F)c1
O=C(NS(=O)(=O)C1CC1)c1ccc(COc2cccc(c2)-c2ncc(OCC3CC3)cn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)cc2)cc1
CNC(=O)c1cc(ccc1OCC1CC1)-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CN(C)C(=O)c1cc(ccc1OCC1CC1)-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccn(CC3CC3)n2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cc(CC3CC3)on2)c(F)c1
Cc1nc(OCC2CC2)ccc1-c1cccc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1nc(OCC2CC2)ccc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCOC3)nc2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccc(OCC3CCOC3)nc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(cc(c2)-c2ccc(OCC3CC3)nc2)C#N)cc1
Cc1nc(OCC2CCC2)ccc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1cc(cnc1OCC1CC1)-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1cc(cnc1OCC1CC1)-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1nc(OCC2CC2)ccc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1cc(OCC2CC2)ncc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1cc(OCC2CC2)ncc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CC3)c(Cl)c2)c(F)c1
CC(C)(C)OC(=O)N1CC(COc2ccc(cn2)-c2cccc(OCc3ccc(cc3F)C(=O)NS(C)(=O)=O)c2)C1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cnc(OCC3CC3)c(Cl)c2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2ccc(F)c(c2)-c2cnc(OCC3CC3)c(Cl)c2)c(F)c1
Cc1nc(OCC2CC2)ccc1-c1cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)ccc1F
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CCC3)c(CO)c2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cnc(OCC3CCC3)c(CO)c2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CCC3)c(CO)c2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cnc(OCC3CCC3)c(CO)c2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCC3)nc2CO)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCC3)nc2CO)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(cc(c2)-c2ccc(OCC3CC3)nc2)-c2ccccc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(cc(c2)-c2cncnc2)-c2ccc(OCC3CC3)nc2)cc1
Cn1cc(cn1)-c1cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)cc(c1)-c1ccc(OCC2CC2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(cc(c2)-c2ccc(OCC3CC3)nc2)-c2cccnc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cncc(OCC3CC3)c2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cncc(OCC3CC3)c2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCC3)nc2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cccc(OCC3CC3)n2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cccc(OCC3CC3)n2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2ccc(F)c(c2)-c2cccc(OCC3CC3)n2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ncc(OCC3CC3)cc2F)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ncc(OCC3CC3)cc2F)cc1
Cc1cc(OCC2CC2)cnc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1cc(OCC2CC2)cnc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1cc(OCC2CCC2)cnc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1cc(OCC2CCC2)cnc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1cc(OCC2CCC2)cnc1-c1cccc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccc(OCC3CC3)cn2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccc(OCC3CC3)cn2)cc1
Cc1c(OCC2CC2)ccnc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1c(OCC2CC2)ccnc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cc(OCC3CC3)ccn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cc(OCC3CC3)ccn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cc(OCC3CC3)ccn2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2ccnc(OCC3CC3)c2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccnc(OCC3CC3)c2)cc1
Cc1c(OCC2CC2)nccc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1c(OCC2CC2)nccc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1c(OCC2CC2)nccc1-c1cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)ccc1F
CN(CC1CC1)c1cc(ccn1)-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CCC3)cn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cnc(OCC3CC3)cn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2ccc(F)c(c2)-c2cnc(OCC3CC3)cn2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CCC3)cn2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cncc(OCC3CC3)n2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cncc(OCC3CC3)n2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ncc(OCC3CC3)cn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ncc(OCC3CCC3)cn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cc(OCC3CC3)ncn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cc(OCC3CC3)ncn2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cc(OCC3CC3)ncn2)c(F)c1
Cc1c(OCC2CC2)ncnc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1c(OCC2CC2)ncnc1-c1cc(F)cc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
Cc1c(OCC2CC2)ncnc1-c1cccc(OCc2ccc(cc2)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cnc(OCC3CC3)nc2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cnc(OCC3CC3)nc2)cc1
Cc1nc(OCC2CC2)ncc1-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CN(CC1CC1)c1ncc(cn1)-c1cccc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cc(OCC3CC3)cc(OCC(N)=O)c2)c(F)c1
COCCOc1cc(OCC2CC2)cc(c1)-c1cc(F)cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cc(OCCO)cc(OCC3CC3)c2)c(F)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2cc(OCC3CC3)cc(c2)C(=O)N2CCOCC2)c(F)c1
CN(C)C(=O)c1cc(OCC2CC2)cc(c1)-c1cc(F)cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CN(C)C(=O)COc1cc(OCC2CC2)cc(c1)-c1cc(F)cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
COC1CN(C1)C(=O)c1cc(OCC2CC2)cc(c1)-c1cc(F)cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CN(CCO)Cc1cc(OCC2CC2)cc(c1)-c1cc(F)cc(OCc2ccc(cc2F)C(=O)NS(C)(=O)=O)c1
CCOC(=O)N1CCC(COc2ccc(cn2)-c2cccc(OCc3ccc(cc3)C(=O)NS(C)(=O)=O)c2)CC1
CCS(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccc(OCC3CC3)nc2)cc1
CC(C)S(=O)(=O)NC(=O)c1ccc(COc2cc(F)cc(c2)-c2ccc(OCC3CC3)nc2)cc1
Fc1cc(OCc2ccc(cc2)C(=O)NS(=O)(=O)C2CC2)cc(c1)-c1ccc(OCC2CC2)nc1
Fc1cc(OCc2ccc(cc2)C(=O)NS(=O)(=O)CC2CC2)cc(c1)-c1ccc(OCC2CC2)nc1
Fc1cc(OCc2ccc(cc2)C(=O)NS(=O)(=O)c2cccs2)cc(c1)-c1ccc(OCC2CC2)nc1
Fc1cc(OCc2ccc(cc2)C(=O)NS(=O)(=O)C(F)(F)F)cc(c1)-c1ccc(OCC2CC2)nc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)C2CCNCC2)cc1
Cc1c(OCc2cc(F)c(cc2F)C(=O)NS(C)(=O)=O)cccc1-n1cccn1
CN1CCC(CC1)c1cccc(OCc2cc(F)c(cc2F)C(=O)NS(C)(=O)=O)c1
Cc1nc(no1)-c1cccc(OCc2cc(F)c(cc2F)C(=O)NS(C)(=O)=O)c1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cccnc2)cc1
CS(=O)(=O)NC(=O)c1ccc(COc2cccc(c2)-c2cccnc2)c(F)c1
CS(=O)(=O)NC(=O)c1cc(F)c(COc2cccc(c2)-c2cccnc2)cc1F
CN(C)[C@H]1C[C@H](CC[C@@H]1N1C(=O)COc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1N1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1n1c2cc(F)c(cc2oc1=O)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccc(Cl)c(Cl)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1OC(F)F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccc(F)c(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccc(Cl)c(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@@H](Cc2cccc(c2)C(F)(F)F)CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1n1ccc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(C)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(OC(F)F)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(F)cc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1F)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(ccc1F)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C1(CC1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(OC(F)(F)F)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)-n1cccn1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)-c1ccnn1C |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)-c1cnn(C)c1 |r|
Fc1cc(c(F)cc1N[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cccc(c1)C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(Cl)cc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(F)cc(Cl)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(F)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(CC(F)(F)F)c1 |r|
CN(C)CC(=O)N[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)CC(=O)N(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CC(C)[C@H](N)C(=O)N[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CC(C)[C@H](N)C(=O)N(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(C)(F)F |r|
CN([C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F)C(=O)[C@H]1CCN(C)C1 |r|
CN([C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F)C(=O)[C@@H]1CCN(C)C1 |r|
CN(C)[C@H]1C[C@](O)(CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@@](O)(CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@@H]1C[C@@](O)(CC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN([C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F)C(=O)C1CN(C)C1 |r|
CN(C1CCC1)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(CCO)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C1CNC1)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(OC2CC2)c1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C1COC1 |r|
CN(C1CN(C)C1)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
Oc1cc(c(F)cc1N[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cccc(c1)C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc2N(CCOc2cc1S(=O)(=O)Nc1ccncn1)[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
Fc1cc2N([C@H]3CC[C@@H](C[C@@H]3N3CCCC3)c3cccc(c3)C(F)(F)F)C(=O)COc2cc1S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1N[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cc(ccc1F)C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1N(C)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@]2([C@@H](C[C@@H]1N(C)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)C2(Cl)Cl)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@@H]1C[C@@]2(C(C[C@H]1N(C)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)C2(Cl)Cl)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1N1CCCc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1N1C(=O)CCc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Br)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
Fc1cc(c(F)cc1O[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cccc(c1)C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(OC(F)(F)F)c1 |r|
Fc1cc(O[C@H]2CC[C@@H](C[C@@H]2N2CCCC2)c2cccc(c2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1N[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cccc(OC(F)(F)F)c1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(c(F)cc1N[C@H]1CC[C@@H](C[C@@H]1N1CCCCC1)c1cccc(c1)C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
CN[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
Fc1cc(O[C@H]2CC[C@@H](C[C@@H]2N2CCCC2)c2cccc(OC(F)(F)F)c2)c(Cl)cc1S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(Cl)ccc1Cl |r|
CN(CCO)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccc(Cl)c(Cl)c1 |r|
CCN[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CNCCN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
Fc1cc(c(F)cc1O[C@H]1CC[C@@H](C[C@@H]1N1CCCC1)c1cccc(c1F)C(F)(F)F)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@H]1CN(CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(ccn1)C(F)(F)F |r|
CN(C)[C@H]1CN(CC[C@@H]1Nc1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1)c1cc(ccn1)C(F)(F)F |r|
CN(C)[C@H]1CN(CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(ccc1F)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(Cl)c1Cl |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccnc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccccc1C(F)(F)F |r|
CN(C)[C@@H]1C[C@@H](CC[C@H]1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1ccccc1C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1ccc(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C1CN(C)C1)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C1CCOCC1 |r|
Fc1ccc(cc1C(F)(F)F)[C@H]1CC[C@H](Nc2cc(F)c(cc2F)S(=O)(=O)Nc2ccncn2)[C@H](C1)N1CCCC1 |r|
Fc1cc(cc(c1)C(F)(F)F)[C@H]1CC[C@H](Nc2cc(F)c(cc2F)S(=O)(=O)Nc2ccncn2)[C@H](C1)N1CCCC1 |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cc(ccc1Cl)C(F)(F)F |r|
CN1CC(C1)N[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1c(F)cc(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1ccc(cc1F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
OC1CCN(C1)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(C)(F)F |r|
CN(C)[C@H]1C[C@H](CC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1)c1cccc(c1Cl)C(F)(F)F |r|
CC(C)C(=O)Nc1cc(ccn1)C(=O)NCCOc1ncc(cc1Cl)C(F)(F)F
CC(C)C(=O)Nc1cc(cc(C)n1)C(=O)NCCOc1ncc(cc1Cl)C(F)(F)F
FC(F)(F)c1cnc(OCCNC(=O)c2cccnc2C(F)(F)F)c(Cl)c1
FC(F)(F)c1cnc(OCCNC(=O)c2ncccc2Cl)c(Cl)c1
Fc1ccc(Oc2ccc(cc2)N2CCC3(CC2)NC(=O)NC3=O)cc1
Fc1cccc(Oc2ccc(cc2)N2CCC3(CC2)NC(=O)NC3=O)c1
FC(F)(F)c1cccc(Oc2ccc(cc2)N2CCC3(CC2)NC(=O)NC3=O)c1
FC(F)(F)Oc1ccc(cc1)-c1ccnc(c1)N1CCC2(CC1)NC(=O)NC2=O
Fc1ccc(Oc2ccc(nc2)N2CCC3(CC2)NC(=O)NC3=O)cc1
FC(F)(F)c1ccc(Oc2ccc(nc2)N2CCC3(CC2)NC(=O)NC3=O)cc1
FC(F)(F)c1cccc(Oc2ccc(nc2)N2CCC3(CC2)NC(=O)NC3=O)c1
FC(F)(F)c1ccc(Oc2ccc(cc2)N2CCC3(CC2)NC(=O)NC3=O)cc1
Fc1ccc(Oc2cccnc2N2CCC3(CC2)NC(=O)NC3=O)cc1
FC(F)(F)Oc1cccc(c1)-c1ccnc(c1)N1CCC2(CC1)NC(=O)NC2=O
CN(C)[C@]1(CCc2ccc(Cl)c(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1
CN(C)[C@]1(CCc2ccc(cc2Cl)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccon1 |r|
CN([C@@H]1CCOC1)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN([C@H]1CCOC1)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCC2CCCCC2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1
CN(C)[C@]1(CCC2CCCCC2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1)C1C[C@@H](C1)c1cccc(c1)C(F)(F)F |r,wD:3.29,29.34,(-7.16,-1.57,;-5.62,-1.57,;-4.85,-2.91,;-4.85,-.24,;-6.18,.53,;-6.18,2.07,;-4.85,2.84,;-3.51,2.07,;-3.51,.53,;-2.18,2.84,;-2.18,4.38,;-.85,5.15,;-.85,6.69,;.49,4.38,;.49,2.84,;1.82,2.07,;-.85,2.07,;1.82,5.15,;1.05,6.49,;2.59,3.82,;3.16,5.92,;4.49,5.15,;4.49,3.61,;5.82,2.84,;7.16,3.61,;7.16,5.15,;5.82,5.92,;-4.08,-1.57,;-2.54,-1.49,;-2.46,-3.03,;-3.99,-3.11,;-1.37,-4.12,;-1.76,-5.6,;-.68,-6.69,;.81,-6.29,;1.21,-4.81,;.12,-3.72,;2.7,-4.41,;3.79,-5.5,;3.1,-2.92,;4.19,-4.01,)|
CN(C)C1(CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1)C1CC(C1)c1cccc(c1)C(F)(F)F |(-7.16,-1.57,;-5.62,-1.57,;-4.85,-2.91,;-4.85,-.24,;-6.18,.53,;-6.18,2.07,;-4.85,2.84,;-3.51,2.07,;-3.51,.53,;-2.18,2.84,;-2.18,4.38,;-.85,5.15,;-.85,6.69,;.49,4.38,;.49,2.84,;1.82,2.07,;-.85,2.07,;1.82,5.15,;1.05,6.49,;2.59,3.82,;3.16,5.92,;4.49,5.15,;4.49,3.61,;5.82,2.84,;7.16,3.61,;7.16,5.15,;5.82,5.92,;-4.08,-1.57,;-3.99,-3.11,;-2.46,-3.03,;-2.54,-1.49,;-1.37,-4.12,;-1.76,-5.6,;-.68,-6.69,;.81,-6.29,;1.21,-4.81,;.12,-3.72,;2.7,-4.41,;3.79,-5.5,;3.1,-2.92,;4.19,-4.01,)|
CN(C)[C@@]1(CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1)C1C[C@@H](C1)c1cccc(c1)C(F)(F)F |r,wU:3.29,wD:29.34,(-7.16,-1.57,;-5.62,-1.57,;-4.85,-2.91,;-4.85,-.24,;-6.18,.53,;-6.18,2.07,;-4.85,2.84,;-3.51,2.07,;-3.51,.53,;-2.18,2.84,;-2.18,4.38,;-.85,5.15,;-.85,6.69,;.49,4.38,;.49,2.84,;1.82,2.07,;-.85,2.07,;1.82,5.15,;1.05,6.49,;2.59,3.82,;3.16,5.92,;4.49,5.15,;4.49,3.61,;5.82,2.84,;7.16,3.61,;7.16,5.15,;5.82,5.92,;-4.08,-1.57,;-2.54,-1.49,;-2.46,-3.03,;-3.99,-3.11,;-1.37,-4.12,;-1.76,-5.6,;-.68,-6.69,;.81,-6.29,;1.21,-4.81,;.12,-3.72,;2.7,-4.41,;3.79,-5.5,;3.1,-2.92,;4.19,-4.01,)|
CN(C)[C@@]1(CCc2cccc(n2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1
CN(C)[C@]1(CCc2cccc(n2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CC2CCCC2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CC2CCCC2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2ccccc2)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2ccccc2)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2ccc(cc2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2ccc(cc2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(C)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(C)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1nccs1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2ccc(Cl)c(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2ccc(Cl)c(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Fc1cc(ccc1S(=O)(=O)Nc1ccncn1)N1CCC[C@@](CCc2cccc(c2)C(F)(F)F)(C1)N1CCC1 |r|
Fc1cc(ccc1S(=O)(=O)Nc1ccncn1)N1CCC[C@](CCc2cccc(c2)C(F)(F)F)(C1)N1CCC1 |r|
Fc1cc(ccc1S(=O)(=O)Nc1ccncn1)N1CCC[C@@](CCc2cccc(c2)C(F)(F)F)(C1)N1CCCCC1 |r|
Fc1cc(ccc1S(=O)(=O)Nc1ccncn1)N1CCC[C@](CCc2cccc(c2)C(F)(F)F)(C1)N1CCCCC1 |r|
CN(C)CCN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)CCN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(CC1CN(C)C1)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(CC1CN(C)C1)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(CC1CCN(C)C1)C1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1
CN(C)[C@@]1(CCc2cc(ccc2Cl)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1
CN(C)[C@]1(CCc2cc(ccc2Cl)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C1CN(C)C1)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C1CN(C)C1)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C1CCN(C)CC1)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C1CCN(C)CC1)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(cc1F)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2Cl)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cc(Cl)cc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cc(Cl)cc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN([C@@H]1CCN(C)C1)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN([C@H]1CCN(C)C1)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(C[C@@H]2CCc3ccc(cc23)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(C[C@H]2CCc3ccc(cc23)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(C[C@H]2CCc3ccc(cc23)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(C[C@@H]2CCc3ccc(cc23)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2ccc(c(Cl)c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2ccc(c(Cl)c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ncccn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ncccn1 |r|
CN(C)[C@@]1(CCc2ccc(Cl)c(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2ccc(cc2Cl)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccon1 |r|
CN(CCO)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(CCO)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(C)c(c(C)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(C)c(c(C)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(Cl)c(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(Cl)c(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(C)c(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(C)c(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2c(Cl)cccc2Cl)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2c(Cl)cccc2Cl)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(Cl)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(C)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1ccc(c(C)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CN(CC[C@H]1O)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CN(CC[C@@H]1O)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CN(CC[C@@H]1O)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CN(CC[C@H]1O)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CCN(C)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CCN(C)[C@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN([C@H]1CCOC1)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN([C@@H]1CCOC1)[C@@]1(CCc2cccc(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2ccc(C)c(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2ccc(C)c(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2ccc(C3CC3)c(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2ccc(C3CC3)c(c2)C(F)(F)F)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(c2)C2CC2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(c2)C2CC2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@@]1(CCc2cccc(Cl)c2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
CN(C)[C@]1(CCc2cccc(Cl)c2)CCCN(C1)c1cc(F)c(c(F)c1)S(=O)(=O)Nc1ccncn1 |r|
Clc1ccc(cc1)-c1ccc(o1)C(=O)N\N=C\c1cccs1
COc1cc(OC)cc(\C=N\NC(=O)c2ccc(o2)-c2ccc(Cl)cc2)c1
CCOc1ccc(cc1)-c1ccc(o1)C(=O)N\N=C\c1cccs1
CC(C)Oc1ccc(cc1)-c1ccc(o1)C(=O)N\N=C\c1cccs1
COc1cc(OC)cc(\C=N\NC(=O)c2cccc(n2)-c2ccc(Cl)cc2)c1
Clc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1cccs1
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1cccs1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(c2)-c2ccc(Cl)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(c2)-c2ccc(OC(F)(F)F)cc2)c1
CCOc1ccc(cc1)-c1cncc(c1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(c2)-c2ccc(OC(C)C)cc2)c1
CCOc1ccc(cc1)-c1cc(ccn1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2ccnc(c2)-c2ccc(OC(C)C)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cccc(n2)-c2ccc(OC(C)C)cc2)c1
COc1ccc(cc1)-c1cncc(c1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCOc1ccc(cc1)-c1cncc(c1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCCOc1ccc(cc1)-c1cncc(c1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(c2)-c2ccc(OC3CCCC3)cc2)c1
COc1ccc(cc1)-c1cc(ccn1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCOc1ccc(cc1)-c1cc(ccn1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1ccccc1F
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1ccccc1Cl
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1c(Cl)cccc1Cl
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1c(F)cccc1Cl
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1ccccc1OC
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1cccnc1N1CCOCC1
COc1cc(OC)cc(\C=N\NC(=O)c2cc(ccn2)-c2ccc(Cl)cc2)c1
Clc1ccc(cc1)-c1ccnc(c1)C(=O)N\N=C\c1cccs1
CCOc1ccc(cc1)-c1ccnc(c1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1ccnc(c1)C(=O)N\N=C\c1cccs1
COc1cc(OC)cc(\C=N\NC(=O)c2cc(ccn2)-c2ccc(OC(C)C)cc2)c1
CC(C)Oc1ccc(cc1)-c1ccnc(c1)C(=O)N\N=C\c1cccs1
COc1cc(OC)cc(\C=N\NC(=O)c2cc(ccn2)-c2ccc(OC3CCCC3)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cc(ccn2)-c2ccc(OC(F)(F)F)cc2)c1
O=C(N\N=C\c1cccs1)c1cc(ccn1)-c1ccc(OC2CCCC2)cc1
FC(F)(F)Oc1ccc(cc1)-c1ccnc(c1)C(=O)N\N=C\c1cccs1
COc1cc(OC)cc(\C=N\NC(=O)c2ccnc(n2)-c2ccc(Cl)cc2)c1
CCOc1ccc(cc1)-c1nccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2ccnc(n2)-c2ccc(OC3CCCC3)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2ccnc(n2)-c2ccc(OC(F)(F)F)cc2)c1
COc1ccc(cc1)-c1nccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCOc1ccc(cc1)-c1nccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCCOc1ccc(cc1)-c1nccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCCOc1ccc(cc1)-c1ccnc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\N(C)C(=O)c2ccc(o2)-c2ccc(Cl)cc2)c1
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N(C)\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCCOc1ccc(cc1)-c1cc(ccn1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2ccnc(c2)-c2ccc(OC3CCCC3)cc2)c1
CCCCOc1ccc(cc1)-c1cccc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cccc(n2)-c2ccc(OC(F)(F)F)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2ccnc(n2)-c2ccc(OC(C)C)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccc(n2)-c2ccc(Cl)cc2)c1
CCOc1ccc(cc1)-c1ccnc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccc(n2)-c2ccc(OC(C)C)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccc(n2)-c2ccc(OC3CCCC3)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccc(n2)-c2ccc(OC(F)(F)F)cc2)c1
COc1ccc(cc1)-c1ccnc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCOc1ccc(cc1)-c1ccnc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cc(F)cc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cc(cc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1)C(F)(F)F
COc1ccc(cc1)-c1ccc(o1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1ccc(s1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1ncc(o1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1nc(co1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1noc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1nc(cs1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OCCN(C)C)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc2ncoc12
CCOc4ccc(c3cncc(C(=O)N/N=C/c1cc(OC)cc2ncsc12)n3)cc4
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cncc(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)ccn1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)n1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(OC)cc1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccncc1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccn1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(OC)c(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C(/C)c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(Cl)cc2)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)ccc1OC
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc2ocnc12
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccnc(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(C)cc(C)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1OC
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1OCC
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(F)cc(OC)c1
CCCOc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OCC)cc2)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)c(F)c(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)ccc1Cl
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1Cl
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)ccc1F
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1F
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1OC
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1OC
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC(C)C)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC3CCCC3)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC(F)(F)F)cc2)c1
CCCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc[nH]c(=O)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(F)c(c1)C(N)=O
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccnc(c1)C(N)=O
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(CN(C)C)c1
CCOc1cccc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC)cc2)c1
CCCOc1cccc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC)cc2)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC(C)C)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1OC
CCOc1ccccc1\C=N\NC(=O)c1cncc(n1)-c1ccc(OC)cc1
CCCOc1ccccc1\C=N\NC(=O)c1cncc(n1)-c1ccc(OC)cc1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1OC(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1F
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1Cl
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1Br
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1C(F)(F)F
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1N(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1C(C)(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(F)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(Cl)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(Br)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(c1)C(F)(F)F
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(c1)N(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(C)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(c1)C(C)(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(F)cc1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(Cl)cc1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(Br)cc1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(cc1)C(F)(F)F
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(cc1)N(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(C)cc1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(cc1)C(C)(C)C
CCOc1cc(OCC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC)cc2)c1
CCCOc1cc(OCCC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC)cc2)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC(C)C)cc(OC(C)C)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(F)cc(F)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(Cl)cc(Cl)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(Br)cc(Br)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(cc(c1)C(F)(F)F)C(F)(F)F
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(cc(c1)N(C)C)N(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(C)cc(C)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(cc(c1)C(C)(C)C)C(C)(C)C
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccnc1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(OC)cc1OC
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1c(OC)cccc1OC
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1OC
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)c(OC)c(OC)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(OC)c(OC)c1OC
CCCCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(C)cc(C)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OCC(C)C)cc2)c1
CC(C)COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(C)cc(C)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC(C)(C)C)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC3CC3)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC3CCCCC3)cc2)c1
COc1ccc(cc1)-c1nccnc1C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1cnc(cn1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(F)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2cccc(Cl)c2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2cccc(F)c2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccc2Cl)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(C)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccc2F)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccc2C)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2cccc(C)c2)c1
COc1cccc(c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccc2OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccncc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2cccnc2)c1
CCOc1ccc(c(OC)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(F)cc(OC)c1
CCCOc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OCC)cc2OC)c1
CCOc1ccc(c(OC)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)c(F)c(OC)c1
CCOc1ccc(c(OC)c1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
COc1ccc(c(C)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(c(Cl)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(c(Cl)c1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
COc1ccc(c(OC(F)(F)F)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCCc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccc2N2CCOCC2)c1
CCCCOc1ccccc1-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(CC(C)C)cc2)c1
CCOc1ccc(cc1Cl)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCSc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(c(F)c1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
CCOc1ccc(-c2cncc(n2)C(=O)N\N=C\c2cccc(OC)c2)c(c1)C(F)(F)F
COc1ccc(c(F)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(c(Cl)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(-c2cncc(n2)C(=O)N\N=C\c2cc(OC)cc(OC)c2)c(c1)C(F)(F)F
COc1ccc(c(OC)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccn2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)N2CCOCC2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)N2CCCCC2)c1
CCCN1CCN(CC1)c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(Oc2nccnc2C(=O)N\N=C\c2cc(OC)cc(OC)c2)cc1
COc1ccc(Oc2cnc(cn2)C(=O)N\N=C\c2cc(OC)cc(OC)c2)cc1
CCOc1ccc(Oc2cncc(n2)C(=O)N\N=C\c2cc(OC)cc(OC)c2)cc1
CCc1nccnc1C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCc1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)C(C)C)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccnc2C(C)C)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cnc(cn2)C(C)C)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(C)n2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cnc(C)cn2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccnc2C)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(OC)n2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccnc2OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cnc(OC)cn2)c1
CCOc1ccc(cc1)-c1cnc(C)c(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cnc(CC)c(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cnc(OC)c(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cnc(Oc2ccccc2)c(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1cnc(-c2ccccc2)c(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC3CCC3)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OCSC)cc2)c1
Cc1cc(C)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC3CCCC3)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OCCN(C)C)cc2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OCC3CC3)cc2)c1
CCOc1ccc(c(OCC)c1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
CCOc1ccc(c(OC(C)C)c1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
CCOc1cc(OC)ccc1-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(c(OC(C)C)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC3CCCC3)cc2Cl)c1
CCCCOc1ccc(c(Cl)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OCC(C)C)cc2Cl)c1
COc1ccc(c(OCCN(C)C)c1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccccc2OC2CCCC2)c1
CCNc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(Cl)n2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cnc(Cl)cn2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2nccnc2Cl)c1
CCc1cnc(cn1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N(C)\N=C\c1cc(OC)cc(OC)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)N2CCC(F)(F)C(C)C2)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCCCC1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCC(F)(F)CC1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCCCC1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCC(F)(F)CC1
CC(C)Oc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCCCC1
CC(C)Oc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCC(F)(F)CC1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(cc2)C(F)F)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)N2CCCC(F)(F)CC2)c1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)N2CCC(F)(F)CC2)c1
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCCCCC1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCCCCC1
CC(C)Oc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1CCCCCC1
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(OC)nc2)c1
COc1ccc(nc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(-c2cncc(n2)C(=O)N\N=C\c2cc(OC)cc(OC)c2)c(c1)C(F)(F)F
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccc(cc1)C(=O)NS(C)(=O)=O
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cccc(c1)C(=O)NS(C)(=O)=O
COc1cc(OC)cc(\C=N\NC(=O)c2cncc(n2)-c2ccc(cc2)C(=O)NS(C)(=O)=O)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1CS(C)(=O)=O
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1S(C)(=O)=O
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1ccccc1NS(C)(=O)=O
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1=C(C)CCCC1 |c:21|
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1=C(C)CCCC1 |c:22|
CC(C)Oc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1=C(C)CCCC1 |c:23|
COc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1=C(C)CCCCC1 |c:21|
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1=C(C)CCCCC1 |c:22|
CC(C)Oc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\C1=C(C)CCCCC1 |c:23|
CCOc1ccc(cc1)-c1nc(cnc1N)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1nc(cnc1C)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1nc(cnc1CC)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1nc(cnc1Cl)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1nc(cnc1C(F)(F)F)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1nc(cnc1OC)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1ccc(cc1)-c1nc(cnc1OCC)C(=O)N\N=C\c1cc(OC)cc(OC)c1
CCOc1cc(C)c(c(C)c1)-c1cncc(n1)C(=O)N\N=C\c1cccc(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(CCO)cc(OC)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)N\N=C\c1cc(OC)cc(c1)C(C)O
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)cn1
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Nc1ccc(S(=O)(=O)Nc2ccncn2)cn1
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1Cl
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Nc1ncc(S(=O)(=O)Nc2ccncn2)cc1Cl
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Nc1ccc(S(=O)(=O)Nc2ccncn2)nc1
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1C#N
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1C1CC1
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Nc1ccc(S(=O)(=O)Nc2ccncn2)cn1
O=S(=O)(Nc1ccncn1)c1ccc(N[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCCC2)nc1
O=S(=O)(Nc1ccncn1)c1ccc(O[C@H]2CC[C@H](c3cccc(OC(F)(F)F)c3)C[C@@H]2N2CCCC2)nc1
CN(C)[C@H]1C[C@@H](c2ccc(Cl)c(C(F)(F)F)c2)CC[C@@H]1Nc1ccc(S(=O)(=O)Nc2ccncn2)cn1
CN(C)[C@H]1C[C@@H](c2ccc(Cl)c(C(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)cn1
CN(C)[C@H]1C[C@@H](c2cccc(OC(F)(F)F)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1Cl
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1C(F)(F)F
Cc1cc(S(=O)(=O)Nc2ccncn2)cnc1O[C@H]1CC[C@H](c2cccc(C(F)(F)F)c2)C[C@@H]1N(C)C
O=S(=O)(Nc1ccncn1)c1ccc(N[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCCC2)nc1
O=S(=O)(Nc1ccncn1)c1ccc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCCC2)nc1
O=S(=O)(Nc1ccncn1)c1cnc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCCC2)c(Cl)c1
O=S(=O)(Nc1ccncn1)c1cnc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCCCC2)c(Cl)c1
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1Br
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1F
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)c(Cl)n1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
CCc1cc(S(=O)(=O)Nc2ccncn2)cnc1O[C@H]1CC[C@H](c2cccc(C(F)(F)F)c2)C[C@@H]1N(C)C
CN(C)[C@H]1C[C@@H](c2cccc(OC(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)cn1
O=S(=O)(Nc1ccncn1)c1ccc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCCCC2)nc1
CN(C)[C@H]1C[C@@H](c2cccc(Cl)c2)CC[C@@H]1Oc1ncc(S(=O)(=O)Nc2ccncn2)cc1Cl
Cc1nc(O[C@H]2CC[C@H](c3cccc(OC(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCCC2)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cccc(OC(F)(F)F)c3)C[C@@H]2N2CCCC2)ccc1S(=O)(=O)Nc1ccncn1
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1cc(Cl)c(S(=O)(=O)Nc2ccncn2)cn1
Cc1cc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N(C)C)ncc1S(=O)(=O)Nc1ccncn1
CCc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
CN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)c(C2CC2)n1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N(C)C2CCC2)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3ccc(Cl)c(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3ccc(Cl)c(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cc(C(F)(F)F)ccc3Cl)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cc(Cl)ccc3Cl)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
O=S(=O)(Nc1ccncn1)c1cnc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)n3)C[C@@H]2N2CCCC2)c(Cl)c1
Cc1nc(O[C@H]2CC[C@H](c3cc(C(C)(F)F)ccc3Cl)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cc(F)cc(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cc(C(F)(F)F)ccc3F)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
CN(C)[C@H]1C[C@@H](c2cc(C(F)(F)F)ccc2F)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)c(Cl)n1
Cc1nc(O[C@H]2CC[C@H](c3ccc(F)c(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3F)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
CCN(CC)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)c(C)n1
CCN(C)[C@H]1C[C@@H](c2cccc(C(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)c(C)n1
Cc1nc(O[C@H]2CC[C@H](c3cc(Cl)cc(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cc(Cl)cc(C(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)n3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cccc(OC(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N(C)C)c(F)cc1S(=O)(=O)Nc1ccncn1
Cc1ccc(C(F)(F)F)cc1[C@H]1CC[C@H](Oc2ccc(S(=O)(=O)Nc3ccncn3)c(C)n2)[C@@H](N(C)C)C1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3)C[C@@H]2N2CCOCC2)ccc1S(=O)(=O)Nc1ccncn1
Cc1ccc([C@H]2CC[C@H](Oc3ccc(S(=O)(=O)Nc4ccncn4)c(C)n3)[C@@H](N(C)C)C2)cc1C(F)(F)F
Cc1nc(O[C@H]2CC[C@H](c3cccc(Cl)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1cc([C@H]2CC[C@H](Oc3ccc(S(=O)(=O)Nc4ccncn4)c(C)n3)[C@@H](N(C)C)C2)cc(C(F)(F)F)c1
Cc1nc(O[C@H]2CC[C@H](c3cccc(CC(F)(F)F)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1nc(O[C@H]2CC[C@H](c3cccc(C(F)(F)F)c3C)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
COc1cc(S(=O)(=O)Nc2ccncn2)cnc1O[C@H]1CC[C@H](c2cccc(C(F)(F)F)c2)C[C@@H]1N(C)C
Cc1nc(O[C@H]2CC[C@H](c3ccc(Cl)c(C(F)(F)F)n3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
CN(C)[C@H]1C[C@@H](c2cccc(SC(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)cn1
COc1cc([C@H]2C[C@@H](C(C)(C)C)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc2cc([C@H]1C[C@@H](C(C)(C)C)C1)c(F)cc2n5c(=O)ccc4cc(S(=O)(=O)Nc3ccon3)ccc45
COc1cc(C2CC(F)(F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc(C2CC(F)(C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@@H](C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@](F)(C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@@](F)(C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@](F)(C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@@](F)(C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@@H](C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc(C2CCC2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc([C@H]2C[C@@H](C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc(C2CCC2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3cccnn3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(C)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc(C2CCC2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc(C2CCC2)c(C)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc(C2CCC2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3cccnn3)ccc21
COc1cc(C2CCC2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncco3)ccc21
COc1cc(C2CCC2)ccc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc(C2CCC2)ccc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc(C2CCC2)c(C)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc(C2CCC2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc(C2CCC2)ccc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncco3)ccc21
COc1cc(C2CCC2)c(C)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3cccnn3)ccc21
COc1cc(C2CCC2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncco3)ccc21
COc1cc(C2CCC2)c(C)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncco3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)ccc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)ccc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(C)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)ccc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3cccnn3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3cccnn3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)c(F)cc21
COc1cc(C2CC(F)(F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)c(F)cc21
COc1cc(C23CC(C(F)(F)F)(C2)C3)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncco3)ccc21
COc1cc([C@H]2C[C@H](OC(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@@H](OC(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(F)cc1-n1c(=O)ccc2c(F)c(S(=O)(=O)Nc3ccon3)ccc21
COc1cc(C23CC(C(F)(F)F)(C2)C3)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
COc1cc(C2CC(F)(F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
COc1cc([C@H]2C[C@H](C(F)(F)F)C2)c(Cl)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncco3)ccc21
Cn6cc(c5cc(c3ccc(N2CCN(C(=O)C#Cc1ccccc1)CC2)nc3)c4c(C#N)cnn4c5)cn6
CN(C)[C@H]1C[C@@H](c2cccc(OC(F)(F)F)c2)CC[C@@H]1Nc1ccc(S(=O)(=O)Nc2ccncn2)cn1
O=S(=O)(Nc1ccncn1)c1ccc(N[C@H]2CC[C@H](c3cccc(OC(F)(F)F)c3)C[C@@H]2N2CCCC2)nc1
Cc1nc(O[C@H]2CC[C@H](c3ccc(Cl)c(Cl)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
CN(C)[C@H]1C[C@@H](c2ccc(F)c(C(F)(F)F)c2)CC[C@@H]1Oc1ccc(S(=O)(=O)Nc2ccncn2)c(Cl)n1
Cc1nc(O[C@H]2CC[C@H](c3cc(Cl)cc(Cl)c3)C[C@@H]2N(C)C)ccc1S(=O)(=O)Nc1ccncn1
Cc1ccc([C@H]2CC[C@H](Oc3ccc(S(=O)(=O)Nc4ccncn4)c(C)n3)[C@@H](N(C)C)C2)cc1C(F)(F)F
Fc1ccc(C2=CCCNC2CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)c(Cl)c1 |t:5|
Fc1cc(NC[C@H]2NCCC=C2c2ccc(Cl)cc2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r,c:10|
Fc1cnc(NS(=O)(=O)c2cc(Cl)c(NC[C@H]3NCCC=C3c3ccc(F)cc3)cc2F)s1 |r,c:20|
Fc1ccc(cc1)C1=CCCN[C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r,t:8|
Fc1cc(OCC2NCCC=C2c2ccccc2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |c:10|
Fc1cc(OCC2NCCC=C2c2ccc(Cl)cc2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |c:10|
Cc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |t:8|
COc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |t:9|
COc1cccc(c1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |t:9|
Fc1cc(OCC2NCCC=C2c2cccc(Cl)c2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |c:10|
Fc1ccc(cc1F)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |t:9|
Fc1ccc(C2=CCCNC2COc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(Cl)c1 |t:5|
Fc1cc(OCC2NCCC=C2c2ccc(Cl)s2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |c:10|
Fc1cc(OCC2NCCC=C2c2ccco2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |c:10|
Cn1cc(cn1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |t:7|
Fc1cc(OCC2NCCC=C2C2=CCOCC2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |c:10,t:13|
Fc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1 |t:8|
Fc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |t:8|
Fc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1 |t:8|
Fc1ccc(cc1)C1=CCCN[C@@H]1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r,t:8|
Fc1ccc(cc1)C1=CCCN[C@@H]1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |r,t:8|
Fc1ccc(cc1)C1=CCCN[C@@H]1CNc1ccc(cc1Cl)S(=O)(=O)Nc1nccs1 |r,t:8|
N[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1 |r,c:4|
Fc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |t:8|
Fc1ccc(cc1)C1=CCCN[C@@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |r,t:8|
Fc1cccc(c1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1 |t:8|
Fc1ccc(C2=CCCNC2COc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(F)c1 |t:5|
Fc1cc(OCC2NCCC=C2c2ccncc2)c(Cl)cc1S(=O)(=O)Nc1cscn1 |c:10|
Fc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1 |t:8|
Fc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)cn1 |t:8|
Fc1ccc(cc1)C1=CCCN[C@@H]1CNc1cc(F)c(cc1F)S(=O)(=O)Nc1nccs1 |r,t:8|
Fc1ccc(cc1)C1=CCCN[C@@H]1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nc(Cl)cs1 |r,t:8|
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Fc1cc(NCC23CCCN2CCC3)c(Cl)cc1S(=O)(=O)Nc1nccs1
CC1(C)CN2CCC[C@]2(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1 |r|
CC1(C)CN2CCC[C@@]2(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1 |r|
F[C@@H]1CN2CCC[C@]2(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1 |r|
F[C@H]1CN2CCC[C@@]2(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1 |r|
Fc1cc(NCC23CCCN2CC(F)(F)C3)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC23CCCCN2CCCC3)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCCC23CCCN2CCC3)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC23CCCN2CCC3)c(Cl)cc1S(=O)(=O)Nc1ccncn1
Fc1cccc(NS(=O)(=O)c2cc(Cl)c(NCC34CCCN3CCC4)cc2F)n1
Fc1cc(NCC23CCCN2CCC3)c(Cl)cc1S(=O)(=O)Nc1cscn1
Cc1nc(NS(=O)(=O)c2cc(Cl)c(NCC34CCCN3CCC4)cc2F)sc1F
Cc1csc(NS(=O)(=O)c2cc(Cl)c(NCC34CCCN3CCC4)cc2F)n1
Cc1cnc(NS(=O)(=O)c2cc(Cl)c(NCC34CCCN3CCC4)cc2F)s1
Fc1cc(NCC23CCCN2CCC3)c(Cl)cc1S(=O)(=O)Nc1ncc(Cl)s1
Fc1cnc(NS(=O)(=O)c2cc(Cl)c(NCC34CCCN3CCC4)cc2F)s1
Fc1cc(NCC23CCCN2CCC3)c(Cl)cc1S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1NCC12CCCN1CCC2)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ncns1)c1ccc2n(Cc3ccccc3)ncc2c1
O=C1COc2cc(ccc2N1Cc1ccccc1)S(=O)(=O)Nc1ncns1
O=c1oc2cc(ccc2n1Cc1ccccc1)S(=O)(=O)Nc1ncns1
C[C@H](c1cccc2CCNCc12)n1c2cc(F)c(cc2oc1=O)S(=O)(=O)Nc1cc(Cl)ccn1 |r|
C[C@H](c1cccc2CCNCc12)n1c2cc(F)c(cc2oc1=O)S(=O)(=O)Nc1ccc(F)cn1 |r|
C[C@H](c1cccc2CCNCc12)n1c2cc(F)c(cc2oc1=O)S(=O)(=O)Nc1cccc(F)n1 |r|
O=c1oc2cc(ccc2n1Cc1cccc2CCNCc12)S(=O)(=O)Nc1ncns1
C[C@H](c1ccccc1)n1c2ccc(cc2oc1=O)S(=O)(=O)Nc1ncns1 |r|
C[C@H](c1cccc2CCNCc12)n1c2ccc(cc2oc1=O)S(=O)(=O)Nc1ncns1 |r|
C[C@H](c1ccccc1CN)n1c2cc(F)c(cc2oc1=O)S(=O)(=O)Nc1cccc(F)n1 |r|
O=c1sc2cc(ccc2n1Cc1ccccc1)S(=O)(=O)Nc1ncns1
Fc1ccc(Nc2n[nH]c3cc(OC(F)(F)F)cnc23)cc1F
FC(F)(F)Oc1ccc2c(n[nH]c2c1)-c1ccc(cc1)C#N
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(cc2-c2ccnnc2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1nncs1
CCN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
c1cc(c(cc1S(=O)(=O)Nc2nccs2)C#N)Oc3ccc(cc3c4c[nH]nc4)Cl
Nc1n[nH]cc1-c1cc(ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1)C(F)(F)F
Nc1n[nH]cc1-c1cc(ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
CN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1
CCN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nncs1
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Cc1[nH]ncc1-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccncn1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccnn1
Fc1cc(Oc2ccc(cc2-c2ccnnc2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1cscn1
CN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(NC[C@H]2CCCOC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
FC(F)(F)c1cccc(NC(=O)c2cccc(c2)-c2ccccn2)c1-c1cccnc1
FC(F)(F)c1cccc(NC(=O)c2cccc(c2)-c2ncccc2Cl)c1-c1cccnc1
FC(F)(F)c1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1cccnc1)C(F)(F)F
Nc1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1cccnc1)C(F)(F)F
FC(F)c1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1cccnc1)C(F)(F)F
FC(F)Oc1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1cccnc1)C(F)(F)F
FC(F)(F)c1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1ccncc1)C(F)(F)F
FC(F)(F)c1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1ccccn1)C(F)(F)F
FC(F)c1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1ccccn1)C(F)(F)F
FC(F)Oc1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1ccccn1)C(F)(F)F
FC(F)(F)c1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1ncccc1Cl)C(F)(F)F |(49.28,-2.81,;50.05,-4.15,;50.82,-2.81,;51.39,-4.92,;48.72,-4.93,;47.39,-4.17,;46.06,-4.95,;46.07,-6.5,;47.41,-7.25,;48.73,-6.47,;50.07,-7.23,;51.4,-6.45,;52.74,-7.22,;52.74,-8.75,;51.41,-9.52,;50.08,-8.77,;51.41,-11.06,;52.75,-11.82,;50.08,-11.83,;50.09,-13.37,;51.42,-14.14,;51.43,-15.69,;50.09,-16.46,;48.76,-15.69,;48.76,-14.14,;47.43,-13.37,;46.1,-14.14,;44.77,-13.38,;44.77,-11.83,;46.1,-11.06,;47.43,-11.83,;48.77,-11.06,;47.42,-16.45,;48.51,-17.54,;47.02,-17.94,;46.09,-15.68,)|
Fc1cccnc1-c1c(NC(=O)c2cccc(c2)-c2ncccc2C(F)(F)F)cccc1C(F)(F)F |(59.44,-10.99,;58.1,-11.76,;56.77,-10.99,;55.44,-11.76,;55.44,-13.3,;56.77,-14.07,;58.1,-13.3,;59.43,-14.07,;60.76,-13.3,;60.75,-11.76,;62.08,-10.98,;63.42,-11.75,;62.08,-9.44,;63.41,-8.68,;63.41,-7.14,;62.07,-6.37,;60.74,-7.15,;60.75,-8.69,;59.4,-6.39,;58.08,-7.17,;56.74,-6.42,;56.73,-4.87,;58.06,-4.09,;59.39,-4.85,;60.72,-4.07,;59.95,-2.74,;61.49,-2.73,;62.06,-4.84,;62.09,-14.06,;62.1,-15.61,;60.76,-16.38,;59.43,-15.61,;58.09,-16.38,;59.18,-17.47,;57.69,-17.86,;56.76,-15.61,)|
C[C@H]1CN(C[C@@H](C)O1)c1c(NC(=O)c2cccc(c2)-c2ccccn2)cccc1C(F)(F)F |r|
O=C(COc1cccc2cccnc12)Nc1ccccc1N1CCOCC1
CN(C(=O)COc1cccc2cccnc12)c1ccccc1N1CCOCC1
CC(Oc1cccc2cccnc12)C(=O)Nc1ccccc1N1CCOCC1
Cc1cccc(N2CCOCC2)c1NC(=O)COc1cccc2cccnc12
O=C(Nc1ccccc1N1CCOCC1)\C=C\c1cccc2cccnc12
O=C(Nc1ccccc1N1CCOCC1)c1cccc(c1)-c1ccccn1
O=C(Nc1ccccc1N1CCOCC1)c1cccc(c1)-c1ccccc1
FC(F)(F)c1cccc(NC(=O)c2cccc(c2)-c2ccccn2)c1N1CCOCC1
FC(F)(F)c1cccc(NC(=O)c2cccc(c2)-c2ccccn2)c1N1CCNCC1
CN1CCN(CC1)c1c(NC(=O)c2cccc(c2)-c2ccccn2)cccc1C(F)(F)F
Cc1ncccc1-c1c(NC(=O)c2cccc(c2)-c2ncccc2C(F)(F)F)cccc1C(F)(F)F |(5.46,-28.34,;4.12,-29.11,;2.79,-28.34,;1.45,-29.11,;1.46,-30.66,;2.79,-31.42,;4.12,-30.65,;5.45,-31.42,;6.78,-30.65,;6.77,-29.11,;8.1,-28.34,;9.44,-29.1,;8.1,-26.8,;9.44,-26.03,;9.43,-24.49,;8.09,-23.73,;6.76,-24.51,;6.77,-26.04,;5.42,-23.75,;4.1,-24.53,;2.76,-23.77,;2.75,-22.22,;4.08,-21.44,;5.41,-22.21,;6.74,-21.43,;5.97,-20.09,;7.51,-20.08,;8.08,-22.19,;8.11,-31.41,;8.12,-32.97,;6.78,-33.74,;5.45,-32.97,;4.11,-33.73,;5.2,-34.82,;3.71,-35.22,;2.78,-32.96,)|
COc1ncccc1-c1c(NC(=O)c2cccc(c2)-c2ccccn2)cccc1C(F)(F)F |(16.5,-26.79,;16.5,-28.33,;15.17,-29.09,;13.83,-28.33,;12.5,-29.1,;12.5,-30.64,;13.84,-31.41,;15.16,-30.64,;16.49,-31.41,;17.82,-30.64,;17.83,-29.1,;19.15,-28.32,;20.49,-29.09,;19.14,-26.78,;20.48,-26.02,;20.48,-24.48,;19.14,-23.71,;17.8,-24.49,;17.81,-26.03,;16.47,-23.73,;16.46,-22.19,;15.12,-21.43,;13.79,-22.21,;13.81,-23.76,;15.14,-24.51,;19.16,-31.4,;19.16,-32.95,;17.83,-33.72,;16.49,-32.95,;15.15,-33.72,;16.24,-34.8,;14.75,-35.2,;13.82,-32.95,)|
FC(F)(F)c1cccnc1-c1cccc(c1)C(=O)Nc1cccc(c1-c1cccnn1)C(F)(F)F
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1F)-c1nnc([nH]1)S(=O)(=O)C1CCC1
CC(C)COc1ncc(cc1Cl)-c1cc(F)c(cc1F)-c1nnc([nH]1)S(=O)(=O)NC1CC1
Cc1ccc(Cl)c(Oc2ncc(cc2Cl)-c2cc(F)c(cc2F)-c2nnc([nH]2)S(=O)(=O)CC2CC2)c1
CS(=O)(=O)c1nnc([nH]1)-c1cc(F)c(COc2ccc(Cl)c(Cl)c2)cc1F
Clc1cc(Cl)cc(Oc2ncc(cc2Cl)-c2nnc([nH]2)S(=O)(=O)CC2CC2)c1
Clc1ccc(Oc2cccc(c2)-c2nnc([nH]2)S(=O)(=O)C2CCC2)cc1Cl
CC(C)COc1ncc(cc1Cl)-c1cc(F)c(cc1F)-c1nnc([nH]1)S(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1cc(F)c(cc1F)-c1nnc([nH]1)S(=O)(=O)C1CCC1
COc1cc(ccc1-c1cnc(OCC(C)C)c(Cl)c1)-c1nnc([nH]1)S(=O)(=O)C1CCC1
COc1cc(-c2nnc([nH]2)S(=O)(=O)C2CCC2)c(F)cc1-c1cnc(OCC(C)C)c(Cl)c1
COc1cc(ccc1-c1cnc(OCC(C)C)c(Cl)c1)-c1nnc([nH]1)S(=O)(=O)N1CCC1
CC(C)COc1ncc(cc1Cl)-c1cc(F)c(cc1F)-c1nnc([nH]1)S(=O)(=O)CC1CC1
Fc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2F)-c2nnc([nH]2)S(=O)(=O)CC2CC2)c(Cl)c1
Fc1ccc(Oc2ncc(cc2Cl)-c2cc(F)c(cc2F)-c2nnc([nH]2)S(=O)(=O)CC2CC2)c(F)c1
Fc1cc(c(F)cc1-c1nnc([nH]1)S(=O)(=O)CC1CC1)-c1cnc(Oc2ccccc2C(F)(F)F)c(Cl)c1
CS(=O)(=O)NC(=O)c1cc(F)c(COc2ccc(Cl)c(Cl)c2)cc1F
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](CC#C)NC(=O)[C@@H](N)CCC(O)=O |r|
CCCC[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@@H]3NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CCCC)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CO)NC(=O)[C@H](CC(O)=O)NC3=O)C(=O)N[C@@H](CCC(O)=O)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N2)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C)[C@@H](C)O |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](CC#C)NC(=O)[C@@H](N)CCC(O)=O |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](CC#C)NC(=O)[C@@H](N)CCC(O)=O |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5cc(C)ccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CCc4ccccc4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4cccc5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4ccc5ccccc5c4)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
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CCCC[C@@H]1NC(=O)[C@H](CCc2ccccc2)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
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CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5c(Br)cccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
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CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Cl)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4ccc5ccccc5c4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCc4ccccc4)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4ccccc4)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CC(=O)N1CCC(CCNCc2cc(ccn2)-c2cc(ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)-c2cccc(c2)C(F)(F)F)CC1
Fc1cc(Oc2ccc(Cl)cc2-c2ccnc(CN3CCC3)c2)c(Cl)cc1S(=O)(=O)Nc1cscn1
Fc1cc(Oc2ccc(Cl)cc2-c2cccc(CN3CCC3)c2)c(Cl)cc1S(=O)(=O)Nc1nncs1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccc(CN2CCC2)c1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccc(CNCCC2CCNCC2)c1
NCc1cccc(c1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1cc(C)n2c1C=C1C=CC(CCCCC(=O)NCCOCCOCCC(=O)N3CCC(CCNCc4cc(ccn4)-c4cc(ccc4Oc4ccc(cc4C#N)S(=O)(=O)Nc4ncns4)-c4cccc(c4)C(F)(F)F)CC3)=[N+]1[B-]2(F)F |c:10,85,t:8|
FC(F)(F)c1cccc(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(CNCCC2CCN(CC2)C(=O)CCc2ccc(cc2)C(=O)c2ccc(OCCC#C)cc2)c1
FC(F)(F)c1cccc(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(CNCCC2CCNCC2)c1
NCc1cc(ccn1)-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)-c1cccc(c1)C(F)(F)F
COCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCC(=O)N1CCC(CCNCc2cc(ccn2)-c2cc(ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)-c2cccc(c2)C(F)(F)F)CC1
NCc1cc(ccn1)-c1cc(ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1)-c1cccc(c1)C(F)(F)F
Fc1cc(Oc2ccc(Cl)cc2-c2ccnc(CN3CCC3)c2)c(Cl)cc1S(=O)(=O)Nc1nncs1
CN[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
CC(C)N[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
CC(=O)N[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1 |r,c:7|
N[C@@H]1CCC=C([C@H]1CSc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
N[C@@H]1CCC=C([C@H]1CSc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1ccc(F)cc1
CCN[C@@H]1CCC=C([C@H]1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1ccc(F)cc1
CCN[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
CN(C)[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
CCN(CC)[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
Fc1ccc(cc1)C1=CCC[C@H]([C@@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)N1CCC1
Fc1ccc(cc1)C1=CCC[C@H]([C@@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)n1ccnc1
Fc1ccc(cc1)C1=CCC[C@H]([C@@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)n1cnnc1
N[C@@H]1CCC=C([C@H]1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
N[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1ccc(F)cc1
N[C@@H]1CCC=C([C@H]1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1ccc(F)cc1
CCN[C@@H]1CCC=C([C@H]1CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
CCN[C@@H]1CCC=C([C@H]1CSc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)c1ccc(F)cc1
CCN[C@@H]1CCC=C([C@H]1COc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)c1ccc(F)cc1
CCCCNc1ccc(cc1)C(=O)OCCN(C)C
CC(C)[C@H]1c2ccc(cc2CC[C@@]1(CCN(C)CCCc3[nH]c4ccccc4n3)OC(=O)COC)F
Fc1cc(c(F)cc1OC1OCCNC1c1ccc(Cl)nc1)S(=O)(=O)Nc1ncns1
CC(C)C[C@@H]1COC(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C(N1)c1cc(Cl)cc(Cl)c1 |r|
Fc1cc(c(F)cc1OC1OCCNC1c1ccc2cnccc2c1)S(=O)(=O)Nc1ncns1
COc1cccc(c1)C1NCCOC1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1cccc2nccnc12)S(=O)(=O)Nc1ncns1
CC1(C)CNC(C(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)O1)c1cc(Cl)cc(Cl)c1
CN(C)c1noc2ccc(cc12)C1NCCOC1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1ccc2ncccc2c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1cccc(c1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC[C@H]1NCCO[C@@H]1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
CC(C)[C@H]1COC(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C(N1)c1cc(Cl)cc(Cl)c1 |r|
CC(C)C[C@H]1COC(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C(N1)c1cc(Cl)cc(Cl)c1 |r|
Cn1nc(cc1C1NCCOC1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cn1nccc1C1NCCOC1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1ccc2OCOc2c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1cc(Cl)cc(Cl)c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1ccc(Cl)c(Cl)c1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1ccc(Cl)cc1Cl)S(=O)(=O)Nc1ncns1
COc1ccc(cc1)C1NCCOC1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1cccc(c1)C#N)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1ccc(cc1)C#N)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1OC1OCCNC1c1ccc(cc1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Fc1ccc(cc1)C1NCCOC1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
CC1(C)COC(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C(N1)c1ccc(Cl)cc1
CC1(C)CN[C@@H]([C@@H](Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)O1)c1cc(Cl)cc(Cl)c1 |r|
Fc1ccc(cc1)[C@H]1NCCO[C@@H]1OCc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
COc1ccccc1C1NCCOC1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
CC(C)[C@@H]1COC(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)C(N1)c1cc(Cl)cc(Cl)c1 |r|
CC1(C)CN[C@H]([C@H](Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)O1)c1cc(Cl)cc(Cl)c1 |r|
Fc1cc(c(F)cc1OC[C@H]1OCCN[C@@H]1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
[H][C@]12CSSC[C@]3([H])NC(=O)[C@@]([H])(NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@]([H])(NC(=O)[C@]([H])(CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC1=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c4ccccc14)C(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CC(O)=O)NC3=O)C(=O)N[C@@H](CCC(O)=O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](C(C)C)C(=O)N2)NC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CSSC[C@@H]2NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@@H]3CCCN3C(=O)[C@H](CC(N)=O)NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)CN)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](Cc4ccccc4)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C)C(=O)N3)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1)C(N)=O |r|
COc1c(O)cccc1C(=O)N1CCC2(CC1)Oc1ccccc1-n1c(ccc21)C#N
CS(=O)(=O)Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(Cl)cn12 |TLB:12:13:16.15.20:18,THB:14:15:18:22.13.21,14:13:16.15.20:18,21:13:16:20.19.18,21:19:16:22.14.13|
CC(C)c1cn2c(NS(C)(=O)=O)nnc2cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:18:19:22.21.26:24,THB:20:21:24:28.19.27,20:19:22.21.26:24,27:19:22:26.25.24,27:25:22:28.20.19|
CS(=O)(=O)Nc1noc2cc(COc3ccc(Cl)c(Cl)c3)c(cc12)C1CC1
CNS(=O)(=O)Nc1nnc2cc(OCC3CCCCC3)c(cn12)C1CC1
CNS(=O)(=O)Nc1nnc2cc(OCC34CCC(F)(CC3)CC4)c(cn12)C1CC1
[H][C@]12C[C@@]([H])(CC(COc3cc4nnc(NS(=O)(=O)NC)n4cc3C3CC3)C1)C2(C)C |r|
CNS(=O)(=O)Nc1nnc2cc(OCCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1 |TLB:18:19:17.16.22:23,THB:18:17:19.24.20:23,20:19:16:22.21.23,20:21:18.19.24:16|
CS(=O)(=O)Nc1nnc2cc(OCC3C4CC5CC(C4)CC3C5)c(cn12)C1CC1 |TLB:19:18:22:15.14.13,19:14:17.18.20:22,THB:12:13:17.18.20:22,13:14:17:20.21.22,13:21:17:15.19.14,(61.13,-36.21,;59.78,-35.45,;59.24,-34.01,;60.77,-34.26,;58.46,-36.25,;58.48,-37.79,;59.35,-39.06,;58.41,-40.29,;56.95,-39.77,;55.59,-40.51,;54.28,-39.7,;52.92,-40.44,;52.88,-41.98,;51.53,-42.71,;51.54,-44.12,;50.26,-44.45,;49.03,-44.02,;47.95,-45.21,;49.32,-44.8,;50.62,-45.31,;49.3,-43.35,;50.23,-42.2,;49,-42.66,;54.32,-38.16,;55.68,-37.42,;57,-38.23,;53.01,-37.36,;52.27,-36,;51.46,-37.31,)|
CS(=O)(=O)Nc1noc2cc(OCC34CC5CC(CC(C5)C3)C4)c(Cl)cc12 |TLB:12:13:16.15.20:18,THB:14:15:18:22.13.21,14:13:16.15.20:18,21:13:16:20.19.18,21:19:16:22.14.13|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc(c3)C(F)(F)F)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@]12O[C@@]3(O)O[C@]([H])([C@]4([H])[C@@H](O)N=C(N)N[C@]4([C@H]1O)[C@@H]3O)[C@@]2(O)CO |r,t:12,TLB:23:21:2:16.17.19,23:21:2.3.5:16.17.8,22:21:2:16.17.19,22:21:2.3.5:16.17.8,18:17:2:5.6.21,10:8:17:2.3.19,15:16:2:5.6.21,THB:23:21:17:2.3.19,22:21:17:2.3.19,4:3:17:6.8.21,20:19:17:6.8.21,20:19:2:5.6.21,5:3:17:6.8.21,5:6:17:2.3.19,8:16:2:5.6.21,8:6:2:16.17.19|
CC(C)COc1ncc(cc1Cl)-n1nc(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
OC(=O)[C@@H]1C[C@@H](F)CN1C(=O)c1cc(C2CC2)c(OCC2CCN(Cc3c(Cl)cccc3Cl)CC2)cc1F |r|
NC(=O)OC[C@@H]1NC(=N)N2CCC(O)(O)[C@@]22NC(=N)N[C@@H]12 |r|
Fc1ccc(cc1)[C@H]1C[C@H](CCN1[C@H]1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)Cc1cccc(Cl)c1 |r|
CCCCCN1C(=O)C2(COc3cc(OC)ccc23)c2ccccc12
COc1cc2c(OCC22C(=O)N(C[C@H]3CCCO3)c3ccccc23)cn1 |r|
COc1ccc2OCC3(C(=O)N(Cc4ccccn4)c4ccccc34)c2n1
CCCCCN1C(=O)C2(COc3cc(F)c(F)cc23)c2ccccc12
COc1cc2c(OCC22C(=O)N(Cc3ccc(o3)C(F)(F)F)c3ccccc23)cn1
COc1cc2c(OCC22C(=O)N(CC3CCCCO3)c3ccccc23)cn1
Cc1cc2OCC3(C(=O)N(Cc4ccccn4)c4ccccc34)c2cc1C
COc1ccc2OCC3(C(=O)N(Cc4ccc5OCCOc5c4)c4ccccc34)c2n1
COc1ccc2OCC3(C(=O)N(Cc4csc(n4)C(C)C)c4ccccc34)c2n1
COc1ccc2OCC3(C(=O)N(Cc4ccc(o4)C(F)(F)F)c4ccccc34)c2n1
COc1ccc2OCC3(C(=O)Nc4ccccc34)c2n1
COc1cc2c(OCC22C(=O)N(C[C@@H]3CCCO3)c3ccccc23)cn1 |r|
COc1cc2OCC3(C(=O)N(Cc4ccc(Cl)s4)c4ccccc34)c2cc1OC
COc1ccc2c(OCC22C(=O)N(C[C@H]3CCCO3)c3ccccc23)c1 |r|
COc1ccc2c(OCC22C(=O)N(CC3CCCCO3)c3ccccc23)c1
COc1cc2OCC3(C(=O)N(Cc4ccccn4)c4ccccc34)c2cc1C
COc1cc2OCC3(C(=O)N(Cc4ccccn4)c4ccccc34)c2cc1F
COc1ccc2c(OCC22C(=O)N(Cc3ccccn3)c3ccccc23)c1
CCCCCN1C(=O)C2(COc3cc4OCOc4cc23)c2ccccc12
COc1ccc2OCC3(C(=O)N(Cc4ncccc4C(F)(F)F)c4ccccc34)c2n1
COc1ccc2OCC3(C(=O)N(Cc4ccc(Cl)o4)c4ccccc34)c2n1
COc1cc2OCC3(C(=O)N(Cc4ccc(o4)C(F)(F)F)c4ccccc34)c2cc1F
Fc1cc2OCC3(C(=O)N(Cc4ccccn4)c4ccccc34)c2cc1F
COc1cc2c(OCC22C(=O)Nc3ccccc23)cn1
COCCOc1ccc2c(OCC22C(=O)N(Cc3ccccn3)c3ccccc23)c1
Fc1cc2OCC3(C(=O)N(Cc4ncccc4C(F)(F)F)c4ccccc34)c2cc1C#N
COc1cc2c(OCC22C(=O)N(Cc3ccccn3)c3ccccc23)cc1F
CCOc1nnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(c2)C#N)s1
COc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)ccc1-n1ccnc1C
FC(F)(F)c1cccc(c1)-n1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cn1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3Oc3ccccc3)c(c2)C#N)s1
O=S(=O)(Nc1ccon1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1nn(C)c(C)c1Cc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)cc1
COc1cc(ccc1Oc1ccn(Cc2ccc(Cl)cc2)n1)S(=O)(=O)Nc1ncns1
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1C1CC1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccnc1
Cn1nccc1-c1cc(I)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ccccc1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Fc1cc(c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1Cl)-c1ccnnc1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1C1CCNCC1)S(=O)(=O)Nc1ncns1
Cc1cc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(c2)C#N)no1
Fc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(cc1OC(F)(F)F)-c1ccnnc1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccc(CN2CCC2)c1
Fc1cc(c(F)cc1Oc1ccc(cc1C1=CCNCC1)C(F)(F)F)S(=O)(=O)Nc1ncns1 |t:17|
Fc1ccc(-c2ccn[nH]2)c(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)c1
Cn1nccc1-c1cc(OC(F)(F)F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1ccc(I)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cc1cn(C)nc1-c1cc(C)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC(F)n1cc(cn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
O=S(=O)(Nc1cscn1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1coc(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)cc1)C(F)(F)F
CN(C)c1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
OCC1(CO)CN(Cc2cccc(c2)-c2cc(Cl)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)C1
Fc1cc(Oc2ccc(OC(F)(F)F)cc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1ncns1
CN(C)c1ncc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccc(F)cc1
O=S(=O)(Nc1ncns1)c1ccc(Oc2ccccc2-c2ccc(cc2)C#N)c(c1)C#N
Cc1cc(C)n(n1)-c1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)cc1
Cc1n[nH]cc1-c1ccccc1Oc1ccc(cc1C(N)=O)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccc(Oc3ccccc3)nc2)c(c1)C#N
Fc1ccc(cc1F)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Clc1cc(ccc1Oc1ccc(CC2CC2)cc1)S(=O)(=O)Nc1ncns1
Fc1ccc(cc1F)-n1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F
Cn1nccc1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
CC(C)Oc1ccc(c(C)c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(cc2F)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1ccnnc1
Fc1cc(Oc2cnn(Cc3ccc(Cl)cc3)c2)ccc1S(=O)(=O)Nc1nccs1
Fc1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)-c1ccn[nH]1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)c(F)c1)C(F)(F)F
NC(=O)c1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1nccs1
Cn1nc(Cc2ccc(Cl)cc2)cc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Fc1cn[nH]c1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
COCc1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
Cn1nccc1-c1ccc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)C(F)(F)F
CN(C)c1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
OCCCc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)c(c1)-c1cn[nH]c1
Fc1cc(ccc1Oc1ccc(cc1-c1ccnnc1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Fc1ccc(NS(=O)(=O)c2cc(F)c(Oc3ccc(Cl)cc3-c3ccnnc3)cc2F)nc1
Cn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncc(Cl)s1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccon1
Fc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1nccs1
CC(C)Oc1ccc(cc1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cc1nc(cs1)-c1ccccc1Oc1ccc(c(F)c1)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)cn1
Cc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1nccs1
O=C1CCCN1c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
CC(C)Oc1cc(-c2cc(F)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)n(C)n1
FC(F)(F)c1ccn(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cn1nccc1-c1cc(ncc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1)C(F)(F)F
Cn1nccc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cn1
COc1ccc(cn1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cc1n[nH]cc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncccn1
Nc1ccc(nc1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1C
Fc1ccc(F)c(c1)-n1nc(cc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1)C(F)(F)F
Cn1nc(cc1-c1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)c(c1)C#N)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
Fc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)c(Cn4cccn4)c3)c(c2)C#N)s1
COc1cc(-c2cc(Cl)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)n(C)n1
Fc1ccccc1-n1nc(cc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncns1)C(F)(F)F
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cnn[nH]1
O=S(=O)(Nc1nccs1)c1ccc(Oc2cccc(c2)-c2ccccc2)c(c1)C#N
Cc1cnn(C)c1-c1cc(C)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1 |(14.53,-24.61,;15.44,-23.36,;14.96,-21.9,;16.2,-20.99,;17.46,-21.9,;18.92,-21.42,;16.98,-23.36,;17.88,-24.61,;19.41,-24.44,;20.32,-25.7,;21.85,-25.55,;19.68,-27.11,;18.15,-27.27,;17.25,-26.02,;15.71,-26.18,;15.08,-27.58,;15.99,-28.83,;15.36,-30.23,;13.82,-30.4,;12.91,-29.14,;13.54,-27.74,;12.64,-26.49,;11.75,-25.24,;13.2,-31.8,;11.87,-31.02,;12.11,-32.88,;13.95,-33.15,;15.48,-33.17,;16.36,-34.44,;17.84,-33.99,;17.87,-32.45,;16.41,-31.94,)|
Cc1cn[nH]c1-c1cc(C)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ncns1)c1ccc(Oc2ccccc2Oc2ccccc2)c(c1)C#N
Fc1cc(ccc1Oc1cnn(Cc2ccc(Cl)cc2)c1)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ccncn1
CCn1cc(nc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
CN(C)C(=O)c1cccc(-c2ccccc2)c1Oc1ccc(cc1C#N)S(=O)(=O)c1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccc(cn1)C#N
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3cn[nH]c3)c(c2)C#N)nc1
Cc1cnsc1-c1ccccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)-c1cn[nH]c1
Fc1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c1-c1ccn[nH]1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cocn1
Cc1cc(Oc2ccccc2-c2ccccc2)ccc1S(=O)(=O)Nc1ncns1
Cc1cc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)n(n1)-c1ccccc1
CCOC(=O)Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(CCO)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)s1
CC(C)(C)n1nc(cc1-c1ccc(Oc2ccc(c(F)c2)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
Fc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1CC(F)(F)F
OCc1ccc(cc1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
OCc1cc(nn1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccc(F)cn1
OC1CCN(Cc2cc(Cl)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)C1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1ccc(Cl)nn1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Fc1ccc(c(F)c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC1(F)CCN(Cc2cc(Cl)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)CC1
Fc1ccc(Oc2ccccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ccncn1
CCc1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-n1ccc(n1)C(F)(F)F
FC(F)(F)Oc1ccc(cc1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC(F)(F)c1cc([nH]n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Fc1cc(Oc2ccc(cc2)-c2ccccc2)ccc1S(=O)(=O)Nc1nccs1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(CN2CCOCC2)c1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-n1ccnn1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccccc2-c2ccccc2)cc1
Fc1cc(ccc1Oc1ccc(OC(F)(F)F)cc1-c1cn[nH]c1)S(=O)(=O)Nc1cscn1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2cccnn2)c(c1)-c1ccnnc1
Fc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)s1
Fc1cc(ccc1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1cscn1
Cc1nccn1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Ic1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cn[nH]c1
Fc1cc(Oc2ccc(Cl)cc2C2CCNCC2)c(Cl)cc1S(=O)(=O)Nc1ccncn1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ncccn1
Cn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(OC(F)(F)F)cc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1nncs1
FCCCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(F)c1)C(F)(F)F
CC(C)(C)n1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncc(F)s1
OCc1cccc(c1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ncns1)c1ccc(Oc2ccccc2-c2cn[nH]c2)c(c1)C#N
CC(C)Cc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1C
Fc1cc(Oc2ccc(Cl)cc2-c2cccc(CN3CCC3)n2)c(Cl)cc1S(=O)(=O)Nc1nncs1
OCCc1cccc(c1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cccnc1
CN1CCC(CC1)c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)c(c1)-c1cn[nH]c1
Fc1cc(c(Oc2ccc(cc2F)S(=O)(=O)Nc2ncns2)cc1Cl)-c1ccnnc1
Nc1cc([nH]n1)-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Fc1cc(Oc2cc(ccc2-c2ccnnc2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1nncs1
Fc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
CC(C)(C)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ncns1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)C#N)C(F)(F)F
Clc1ccc(-c2ccn[nH]2)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Cn1nccc1-c1cc(Br)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1cc(c(F)cc1Oc1ccc(cc1-c1ccnnc1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Cc1[nH]ncc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccc(c1)C(=O)NC1CC1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cccc(c1)C(=O)N1CCC1)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(OC2CCC2)c1
CN1CC(C1)n1nccc1-c1cc(ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1)C(F)(F)F
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccncc1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1C1CNC1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnc(c1)N1CCNCC1)S(=O)(=O)Nc1cscn1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(cc2-c2cn[nH]c2)C#N)c(Cl)cc1S(=O)(=O)Nc1ncns1
FC(F)(F)Oc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
FC(F)Oc1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)C1CCNCC1
FC(F)(F)c1ccc(Oc2ccc(cc2C(F)(F)F)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
Fc1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Fc1cc(Oc2ccc(Cl)cc2C2CCNCC2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1ccn[nH]1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnc(c1)N1CCNCC1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnc(CN2CCC2)c1)S(=O)(=O)Nc1ncns1
Nc1cc(ccn1)-c1cc(OC(F)(F)F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
CCN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1ncns1
Brc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cn[nH]c1
Fc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1cn[nH]c1
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ncns1
Ic1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccc(CN2CCC2)c1
Fc1ccc(Oc2ccccc2)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c1
Cc1cc(Oc2ccc(cc2)S(=O)(=O)Nc2nccs2)n(n1)-c1ccccc1
Cc1nn(C)cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
COCc1cc(nn1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)F
CC(C)(C)n1nc(cc1-c1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
COc1ccccc1-c1ccccc1Oc1ccc(c(F)c1)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(Br)ccc1Oc1ccc(cc1C(N)=O)S(=O)(=O)Nc1ncns1
FC(F)(F)c1cccc(n1)-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Clc1ccc(Cn2cc(Oc3ccc(cc3C#N)S(=O)(=O)Nc3nccs3)cn2)cc1
COc1ccc(cc1)-n1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)c(n1)C(C)C
CC(C)(C)n1nc(Cc2ccc(Cl)cc2)cc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Cc1cc(-c2ccc(Oc3ccc(cc3C#N)S(=O)(=O)Nc3nccs3)cc2)n(CCO)n1
CN(C)C(=O)Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1c(F)cccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1 |(15.56,-41.61,;16.8,-40.7,;18.27,-41.16,;19.17,-39.91,;18.25,-38.68,;16.79,-39.16,;15.53,-38.27,;14.21,-39.04,;14.21,-40.58,;12.87,-38.27,;12.87,-36.73,;14.21,-35.96,;15.53,-36.73,;16.87,-35.96,;16.87,-34.42,;15.53,-33.65,;15.53,-32.11,;16.87,-31.34,;18.21,-32.11,;18.21,-33.65,;19.54,-34.42,;20.87,-35.19,;16.86,-29.8,;15.32,-29.8,;16.09,-28.46,;18.21,-29.03,;18.24,-27.49,;17.02,-26.56,;17.52,-25.11,;19.06,-25.14,;19.51,-26.61,)|
Cc1nc(cs1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CCOC(=O)Cn1nc(Cc2ccc(Cl)cc2)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)cn2)cc1)C(F)(F)F
COc1ccc(cc1)-c1cccc(C)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
CN(C)CCn1nc(C)cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
CC(=O)N1CC(C1)c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cc1scnc1NS(=O)(=O)c1cc(Cl)c(Oc2ccc(F)cc2-c2ccnn2C)cc1F
Nc1nccc(n1)-c1cc(F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncc(Cl)s1
OC(=O)c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)ccc1-n1cc(Cl)cn1
O=C1NCCN1c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
FC(F)(F)c1ccnc(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
COc1cccc(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1cnn(CC(F)(F)F)c1
Cn1cc(cn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
CC(C)(C)NC(=O)c1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cn1ncnc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncc(F)s1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncccn2)cc1)C(F)(F)F
Cn1nc(cc1-c1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nncs2)c(c1)C#N)C(F)(F)F
Fc1cc(Oc2cc(ccc2-c2cncnc2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1cscn1
CC(C)C1CN(C(=O)N1)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
CC1CN(C(=O)N1)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
FCCCn1nc(cc1C(F)(F)F)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(F)c1
Cc1cc(ccc1Oc1ccccc1-c1ccnn1C)S(=O)(=O)Nc1cscn1
Cc1cc(C)n(n1)-c1ccc(Oc2ccc(c(F)c2)S(=O)(=O)Nc2nccs2)cc1
FC(F)(F)n1ccc(n1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
CCn1nc(cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)c1)C(F)(F)F
Cn1nccc1-c1cc(ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncc(Cl)s1)C#N
CC(=O)N1CC(C1)n1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Cn1cnnc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
FC(F)(F)Oc1cccc(c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1ccc(n1)-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cnccn1
Fc1ccc(Oc2c(F)cc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
CC(C)Oc1ccc(cc1)-c1cccc(C)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1cscn1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2ncc(F)s2)cc1)C(F)(F)F
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccc(cc2)-c2ccccc2)c(c1)C#N
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccc(cc2)-n2ccc(n2)C2CC2)c(c1)C#N
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cccnn1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cncc(c1)C#N
NC(=O)Cn1nc(Cc2ccc(Cl)cc2)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncsc1F
Clc1cc(Oc2ccccc2-c2ccccc2)ccc1S(=O)(=O)Nc1ncns1
Cn1ccc(n1)-c1c(F)cccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3C3CC3)c(c2)C#N)s1
Fc1cc(Oc2ccc(Cl)cc2-c2cnn[nH]2)c(Cl)cc1S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccccn1
Cc1nsc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
COC(=O)N1CC(C1)c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cc1nc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)sc1F
FC(F)(F)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
CCc1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-n1cccn1
Fc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1cscn1
Cc1c(Cl)ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1-c1nnco1
CCOCn1nncc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CCn1nc(C)c(c1C)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1 |(60.69,-2.04,;60.45,-3.56,;61.64,-4.53,;63.13,-4.13,;63.97,-5.42,;65.51,-5.5,;63,-6.62,;61.56,-6.07,;60.27,-6.9,;63.4,-8.1,;62.31,-9.2,;62.71,-10.68,;64.19,-11.09,;65.29,-9.99,;64.89,-8.5,;65.98,-7.42,;67.46,-7.82,;67.86,-9.3,;69.35,-9.71,;70.44,-8.61,;70.04,-7.12,;68.56,-6.72,;68.16,-5.24,;67.76,-3.75,;71.93,-9.01,;71.53,-10.5,;73.01,-10.1,;73.04,-7.94,;72.66,-6.44,;73.66,-5.27,;72.84,-3.96,;71.34,-4.32,;71.23,-5.86,)|
COC(=O)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1C
Cc1nn(cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1)C(C)(C)C
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1nncs1
Fc1cc(Oc2ccc(cc2-c2cncc(c2)C#N)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1ncns1
CN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncccn1
Cn1nc(cc1-c1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncccn1
CC(C)Oc1ccc(cc1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC(F)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1cn[nH]c1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1cccnn1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1cn[nH]c1
CCn1nc(cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)c1)C(F)(F)F
Fc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c(c1)-c1ccn[nH]1
CCOC(=O)Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ncc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1)C(F)(F)F
CC(C)c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-n1cc(Cl)cn1
Cn1nccc1-c1cc(CCCO)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)s1
OCCn1nccc1-c1cc(F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Fc1ccc(c(F)c1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccn(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1Cl
Fc1cc(ccc1Oc1ccc(Cl)cc1C1CCOCC1)S(=O)(=O)Nc1ncns1
CC(C)c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-n1ccc(n1)C(F)(F)F
Nc1cccc(n1)-c1cc(F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(Cl)cc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncns1
Fc1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncc(Cl)s2)c(c1)-c1cn[nH]c1
Cc1cnncc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ccncn2)c(c1)C1CCNCC1
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1)C#N
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)cc1F)C(F)(F)F
CCc1cc(c(F)cc1Oc1ccc(F)cc1-c1ccnn1C)S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(F)c(F)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Fc1cc(ccc1Oc1ccc(Cl)cc1-c1ccnn1Cc1ccccc1)S(=O)(=O)Nc1nccs1
Fc1cc(ccc1Oc1cc(Cl)ccc1-c1ccn[nH]1)S(=O)(=O)Nc1nccs1
Cn1nc(cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1F)C(F)(F)F
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cnccn1
COCCn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
Cn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1
OC(=O)Cc1cccc(c1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ccc(F)cn1
Nc1[nH]ncc1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Fc1cc(ccc1Oc1cc(nn1-c1ccccc1)C(F)(F)F)S(=O)(=O)Nc1nccs1
Nc1ccnc(c1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)(F)F
CC(C)c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-n1nc(cc1C)C(F)(F)F
ON1CC=CC(=C1)c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F |c:3,5|
Clc1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1-c1ccn[nH]1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1-c1ccccc1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1nncs1
Cc1n[nH]cc1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
OCCn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1ccccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1cscn1
CCn1nc(cc1-c1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
Nc1cc(ccn1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)C1CCOCC1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ccncn2)c(c1)-c1ccn[nH]1
Fc1cc(Oc2ccc(cc2-c2cn[nH]c2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1cscn1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
CCn1nccc1-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1)C(F)(F)F
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(F)c1)C(F)(F)F
Fc1cc(ccc1Oc1ccc(OC(F)(F)F)cc1-c1cn[nH]c1)S(=O)(=O)Nc1nccs1
FC(F)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
FC1(F)CN(Cc2cccc(n2)-c2cc(Cl)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)C1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1F)C(F)(F)F
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cc(ncn1)N1CCOCC1
Fc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c(c1)-c1cn[nH]c1
FC(F)(F)c1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncns1
COc1ccc(cc1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccc(F)c(F)c1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)F
Nc1cc([nH]n1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1ncnc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)s1
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1cn[nH]c1
OCc1cc(nn1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)F
O=S(=O)(Nc1cccs1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
OC(=O)c1ccc(cc1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)s1
FC(F)(F)c1nccc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
O=S(=O)(Nc1nccs1)c1ccc(Oc2cccc(c2)-c2ccccn2)c(c1)C#N
O=S(=O)(Nc1ncns1)c1ccc(Oc2ccccc2-c2ccccc2)cc1C#N
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(cc3)-c3cocn3)c(c2)C#N)nc1
Cc1nc(no1)-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)c1
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(cc3)-n3ccnc3)c(c2)C#N)nc1
CCc1nnc(C)n1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)cc1
FC(F)(F)c1ccccc1NS(=O)(=O)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cn1ncnc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Fc1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)-c1c[nH]nn1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccc(nc2)-c2ccccc2)c(c1)C#N
FC(F)(F)Cn1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-c1ccc(Cl)cc1
O=S(=O)(Nc1ncns1)c1ccc(Oc2ccc(CC3CC3)cc2)c(c1)C#N
Cc1cn(nc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)F
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3OCc3ccccc3)c(c2)C#N)s1
Cc1cn(Cc2ccccc2)nc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Cn2cccn2)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CCn1nc(cc1C1CC1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cc1nnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(F)c2)s1
Cn1ccc(n1)-c1ccc(F)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccon2)cc1)C(F)(F)F
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nc(C)ns2)cc1)C(F)(F)F
NC(=O)c1cc(ccc1Oc1cnn(Cc2ccc(Cl)cc2)c1)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ncns1)c1ccc(Oc2ccccc2Oc2ccncc2)c(c1)C#N
Cc1cccnc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)cc1Cn1ccnc1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1Cn1cncn1
Cc1cc(ccc1Oc1ccn(Cc2ccc(Cl)cc2)n1)S(=O)(=O)Nc1ncns1
OCCn1nc(Cc2ccc(Cl)cc2)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(ccc1Oc1ccc(cc1)-c1ccccc1)S(=O)(=O)Nc1cscn1
Cn1ncnc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc(Oc2cc(nn2C2CCCCC2)C2CC2)c(c1)C#N
NC(=O)c1ccccc1Oc1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ncns1)c1ccc(Oc2nnccc2-c2ccccc2)c(c1)C#N
O=S(=O)(Nc1ncns1)c1ccc(Oc2nccnc2-c2ccccc2)c(c1)C#N
Nc1c(cnn1CC(F)(F)F)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
O=S(=O)(Nc1cnoc1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1nonc1NS(=O)(=O)c1ccc(Oc2ccc(Cl)cc2-c2ccnn2C)c(c1)C#N
Cn1nccc1NS(=O)(=O)c1ccc(Oc2ccc(Cl)cc2-c2ccnn2C)c(c1)C#N
O=S(=O)(Nc1nccs1)c1ccc(Oc2cccc(c2)-c2ccn[nH]2)c(c1)C#N
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccc(cc2)-n2cc(cn2)C#N)c(c1)C#N
Fc1ccccc1-c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)n(CC(F)(F)F)n1
CC(C)(C)n1ccc(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(F)c1
CC(C)(C)n1ccc(Cc2cccc(Oc3ccc(cc3C#N)S(=O)(=O)Nc3cscn3)c2)n1
NC(=O)c1cc(ccc1Oc1ccc(cc1)-c1cc(n[nH]1)C(F)(F)F)S(=O)(=O)Nc1nccs1
CN1CCC(CC1)c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)c1
Nc1cccc(n1)-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Cc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c(c1)-c1ccn(C)n1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cnccn1
Cc1cccc(-c2ccc(F)c(F)c2)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1cnsn1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
COc1cc(-c2cc(F)ccc2Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)n(C)n1
Cc1noc(C)c1Cc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)cc1
CC(C)c1nn(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)-c1ccccc1Cl
O=S(=O)(Nc1ccncn1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cc(ncn1)N1CCOCC1)S(=O)(=O)Nc1nncs1
COCc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)ccc1-n1cc(Cl)cn1
CSc1nc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(c2)C#N)ns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cnsn2)cc1)C(F)(F)F
Fc1cc(F)cc(c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
CC(C)c1nn(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1)-c1ccccc1Cl
CC(C)Oc1cccc(c1)-c1cccc(C)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
COc1cc(C)ccc1Oc1cccc(F)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(ccc1Oc1ncncc1-c1ccccc1)S(=O)(=O)Nc1nccs1
Cn1ccnc1NS(=O)(=O)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
O=S(=O)(Nc1ncc(s1)C#N)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
COc1ccc(cc1)-n1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)C(C)C
Fc1cc(ccc1Oc1ccccc1-c1ccccn1)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1cccc(n1)C#N)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncsc1Cl
O=S(=O)(Nc1cscn1)c1ccc(Oc2cccc(Cc3cc[nH]n3)c2)c(c1)C#N
Cc1nn(C)c(C)c1Cc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)cc1
Cn1ncc(c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1)-c1ccccc1
Cn1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)-c1ccccc1
FC(F)(F)Cn1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)C1CC1
Clc1ncc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)cn1
CCc1ccc(cc1)-c1ncccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(cn2)C(F)(F)F)cc1)C(F)(F)F
Fc1cc(ccc1Oc1ccc(cc1)-c1cocn1)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccc(cn1)C(F)(F)F
Fc1cc(CN2CCC2)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1ccc(cn1)C#N)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
O=S(=O)(Nc1cnsc1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
O=S(=O)(Nc1ncn[nH]1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1ccnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
Cc1cc(sn1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccc(F)cn1
Cc1cncnc1NS(=O)(=O)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Fc1cc(ccc1Oc1cc(nn1-c1ccccc1)C(F)(F)F)S(=O)(=O)Nc1cscn1
O=S(=O)(Nc1nccs1)c1ccc(Oc2cc(nn2-c2ccccn2)C2CC2)c(c1)C#N
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccccc2-c2nncn2-c2ccccc2)c(c1)C#N
Fc1cc(ccc1Oc1ccc(Oc2ccccc2)cc1)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)nc1
Cn1nccc1-c1cc(F)cc(F)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)ccc1CN1CCC1
Cc1cccc(c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)-c1ccccc1F
Fc1cc(ccc1Oc1cccc(OCc2ccccc2)c1)S(=O)(=O)Nc1nccs1
CCc1nnc(C)n1-c1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)cc1
FC(F)(F)c1cc(Oc2ccccc2-c2ccccc2)ccc1S(=O)(=O)Nc1ncns1
CC(C)(C)n1ccc(n1)-c1cc(F)ccc1Oc1ccc(c(F)c1)S(=O)(=O)Nc1nccs1
Cc1scnc1NS(=O)(=O)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1nsc(NS(=O)(=O)c2cc(Cl)c(Oc3ccc(Cl)cc3-c3ccnn3C)cc2F)n1
Nc1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccnn1
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)s1)C(F)(F)F
Cn1nccc1-c1ccc(I)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)s1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccc(c1)C#N
FC(F)(F)c1ccc(c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c1)-c1ccnnc1
Fc1cc(Oc2cc(OC(F)(F)F)ccc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1nncs1
Fc1cc(Oc2cc(ccc2-c2ccnnc2)C#N)c(Cl)cc1S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)C1CCOCC1
FC(F)(F)c1cc(-c2ccc(Oc3ccc(cc3C#N)S(=O)(=O)Nc3nccs3)cc2)n(n1)C1CNC1
FC(F)(F)Oc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnnc1
Fc1cc(ccc1Oc1ccc(OC(F)(F)F)cc1-c1ccn[nH]1)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(I)s2)c(c1)-c1cn[nH]c1
CN1CC(C1)n1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Fc1cc(-c2cn[nH]c2)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1Cl
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1
NCc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
CC(=O)c1cccc(c1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1C1CNC1
Fc1cc(Oc2ccc(cc2-c2cn[nH]c2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1nncs1
Fc1cc(Oc2ccccc2-c2ccccc2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Fc1cc(ccc1Oc1ccc(Cl)cc1-c1ccnn1-c1ccccc1)S(=O)(=O)Nc1nccs1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccccc1
Cn1nccc1-c1cc(ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1)C(F)(F)F
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cccnn1
Cc1cnccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Nc1n[nH]cc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1)C1CC1
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
Nc1cc(ccn1)-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1
Fc1cc(c(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nncs2)cc1OC(F)(F)F)-c1ccnnc1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnc(c1)N1CCC1
Nc1cccc(n1)-c1cc(OC(F)(F)F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1ccc(Cl)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Nc1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncccn1
CCN1CC(C1)n1nccc1-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1)C(F)(F)F
Fc1cc(Oc2ccc(Cl)cc2-c2cccc(c2)C(=O)N2CCC2)c(Cl)cc1S(=O)(=O)Nc1cscn1
Cc1ncccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1OC(F)(F)F)-c1ccnnc1
Brc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccn[nH]1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Nc1cccc(n1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Br)S(=O)(=O)Nc1cscn1
CC(C)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1C
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnc(c1)N1CCOCC1
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ccncn2)c(c1)-c1cccc(c1)C(=O)N1CCC1
CN1CC(C1)n1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1cscn1
CC(C)N1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
Fc1cc(-c2ccn[nH]2)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1Cl
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
Fc1cc(c(F)cc1Oc1ccc(OC(F)(F)F)cc1-c1cn[nH]c1)S(=O)(=O)Nc1nccs1
Fc1cc(Oc2ccc(Cl)cc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Cc1[nH]ncc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
Nc1cc(ccn1)-c1cc(F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1ccc(I)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Ic1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Fc1cc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nncs2)c(cc1C(F)(F)F)-c1ccnnc1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1ccnn1C1CNC1)C(F)(F)F)S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1ccnn1C1CNC1
Fc1cc(Oc2ccc(Cl)cc2-c2cn[nH]c2)c(Cl)cc1S(=O)(=O)Nc1nncs1
Clc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1ccnnc1
Fc1cc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1ccnnc1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cccc(c1)C(=O)N1CCC1
Cc1[nH]ncc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1ccnnc1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(Cl)cc2-c2ccnn2C2CNC2)c(Cl)cc1S(=O)(=O)Nc1cscn1
Fc1cc(c(F)cc1Oc1ccc(OC(F)(F)F)cc1-c1ccnnc1)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(n1)N1CCNCC1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)cc2F)cc1)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(cn1)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cncnc1
Cc1cccc(-c2cccc(F)c2)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
COc1nsc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
Cc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)nc1
CCN1CC(C1)n1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
FC(F)(F)c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)n(Cc2ccccc2)n1
Cn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1csnn1
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
Cn1ncc(F)c1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1 |(30.58,-40,;29.12,-40.48,;27.86,-39.57,;26.62,-40.48,;27.1,-41.94,;26.19,-43.19,;28.63,-41.94,;29.53,-43.19,;31.07,-43.02,;31.97,-44.28,;33.5,-44.13,;31.34,-45.69,;29.81,-45.85,;28.9,-44.6,;27.37,-44.75,;26.74,-46.16,;27.64,-47.41,;27.02,-48.81,;25.48,-48.98,;24.56,-47.72,;25.2,-46.32,;24.3,-45.07,;24.86,-50.38,;23.36,-49.97,;24.08,-51.7,;25.61,-51.72,;27.15,-51.74,;28.08,-50.5,;29.53,-50.99,;29.51,-52.53,;28.05,-53,)|
FC(F)(F)Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3Oc3ccncc3)c(c2)C#N)s1
Cn1nc(cc1-c1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)C#N)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cnsn1
Cn1cc(nc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
OCc1coc(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1
FC(F)(F)c1cn(cn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
Cn1cnnc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Cn1nc(cc1-c1cc(F)c(F)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)(F)F
COc1ccc(cc1F)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)c(Cn4ccnn4)c3)c(c2)C#N)s1
Cc1cccc(-c2cccc(OC(F)(F)F)c2)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1nn(Cc2ccccc2)cc1-c1ccccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cc(ccn2)C#N)cc1)C(F)(F)F
O=S(=O)(Nc1ncco1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cc[nH]n1
Cc1cc(CN2CCCC2)cc(C)c1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Cn1ccc(n1)-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1ccn(n1)C1CCNCC1
CCn1nc(cc1C(F)(F)F)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)c(F)c1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccc(cc2)-n2cccn2)c(c1)C#N
CNc1ncc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccc(F)cc1
Fc1cc(ccc1Oc1ccccc1C1CCCCO1)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1ncc(cn1)C#N)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
FC(F)(F)c1cc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)ncn1
Fc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(I)cc3-c3ccn[nH]3)c(c2)C#N)s1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
O[C@@H]1CCN(Cc2cccc(c2)-c2cc(ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)C(F)(F)F)C1 |r|
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnnc1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)C#N)C(F)(F)F
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1ccnn1C1CNC1
FC(F)(F)c1cc(ccc1Oc1ccn(Cc2ccc(Cl)cc2)n1)S(=O)(=O)Nc1ncns1
COc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)ccc1-n1cccn1
Fc1cc(ccc1Oc1ccc(cc1)-c1ccccc1)S(=O)(=O)Nc1nccs1
Cn1cc(c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)n1)-c1ccc(Cl)cc1
Fc1cc(Oc2nc(Cc3ccc(Cl)cc3)cs2)ccc1S(=O)(=O)Nc1nccs1
OC(=O)Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccccc2-c2nnco2)c(c1)C#N
Fc1c(Oc2ccccc2-c2ccccc2)ccc(c1F)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(C)(C)C#N
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cnccn1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1ccnnc1)C(F)(F)F)S(=O)(=O)Nc1cscn1
Cn1nc(cc1-c1ccc(F)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)(F)F
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Fc1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ccncn2)c(c1)-c1ccnnc1
CC(C)(C)n1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)cc1)C(F)(F)F
Nc1n[nH]cc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ccncn1
Cc1[nH]ncc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cnco1)S(=O)(=O)Nc1ncns1
Fc1ccc(Oc2c(F)cc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Fc1ccc(F)c(c1)-n1nc(cc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncns1)C(F)(F)F
CCOc1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)c(c1)-c1ccn[nH]1
Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)c(c1)-c1cn[nH]c1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)C1CNC1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)C1CCNCC1
Fc1cc(Oc2ccc(Cl)cc2C2CNC2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Cn1nccc1-c1ccc(cc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncc(Cl)s1)C#N
Clc1cccnc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cn1nc(cc1C(F)(F)F)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
FC(F)(F)c1ccn(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)C(F)(F)F
Cn1nccc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
CCn1nc(cc1-c1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ccc(F)cn2)cc1)C(F)(F)F
Fc1ccc(c(F)c1)-n1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccon3)c(c2)C#N)s1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(Cl)c1
Nc1ncccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
Cn1cc(c(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)n1)-c1ccccc1
OCc1cncc(c1)-c1cc(ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1nncs1
O=S(=O)(Nc1nccs1)c1ccc(Oc2cccc(c2)-n2cccn2)c(c1)C#N
Cc1cc(nn1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)(F)F
Cc1ccc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)nc1
Cc1cnn(c1-c1cc(C)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1)C(C)(C)C |(29.61,-21.15,;31.06,-20.66,;32.32,-21.54,;33.55,-20.62,;33.05,-19.16,;31.52,-19.18,;30.6,-17.95,;31.37,-16.62,;30.6,-15.29,;31.37,-13.96,;29.06,-15.29,;28.29,-16.62,;29.06,-17.95,;28.29,-19.29,;26.75,-19.29,;25.98,-17.95,;24.45,-17.95,;23.67,-19.29,;24.45,-20.62,;25.98,-20.62,;26.75,-21.95,;22.14,-19.29,;20.82,-18.48,;22.17,-17.74,;21.34,-20.6,;19.8,-20.56,;18.93,-19.28,;17.45,-19.71,;17.4,-21.25,;18.85,-21.78,;33.94,-17.9,;35.47,-18.04,;33.29,-16.51,;34.7,-16.56,)|
Nc1cc(ccn1)-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1C1CCC1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccn[nH]1
Cc1cc(ccn1)-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F
Fc1cc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1cn[nH]c1
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Fc1cc(c(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)cc1Cl)-c1ccnnc1
Fc1cc(Oc2ccc(Cl)cc2-c2cccc(c2)C(=O)N2CCC2)c(Cl)cc1S(=O)(=O)Nc1nncs1
Fc1cc(c(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nncs2)cc1C(F)(F)F)-c1ccnnc1
Cn1nccc1-c1cc(Br)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CCNC(=O)c1ccc(cc1)-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)c1
NC1=NCN=C1c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |c:4,t:1|
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)nc1
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(F)cc3C3CC3)c(c2)C#N)nc1
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cn[nH]c1
Fc1ccc(Oc2ccc(Oc3ccc(cc3F)S(=O)(=O)Nc3nccs3)cc2)cc1
Ic1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(NC2CCC2)c1
Cc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnnc1)S(=O)(=O)Nc1nncs1
CC(C)Oc1cccc(c1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F
Fc1cc(Oc2ccc(Cl)cc2C2CCNCC2)c(Cl)cc1S(=O)(=O)Nc1cscn1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-n1nccn1
COc1ccc(c(C)c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC(F)Oc1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Fc1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Cc1ccnn1-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cc1cccc(-c2ccc(OC(F)(F)F)cc2)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1n[nH]c(C)c1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1 |(49.34,-42.98,;50.83,-42.58,;51.38,-41.14,;52.92,-41.22,;53.32,-42.71,;54.76,-43.26,;52.03,-43.55,;51.95,-45.09,;50.58,-45.79,;50.5,-47.33,;51.79,-48.16,;53.16,-47.46,;53.24,-45.93,;54.61,-45.22,;55.95,-45.99,;55.95,-47.53,;57.28,-48.3,;58.62,-47.53,;58.62,-45.99,;57.28,-45.22,;57.28,-43.68,;57.28,-42.14,;59.95,-48.29,;60.71,-49.62,;59.18,-49.61,;61.27,-47.49,;61.23,-45.95,;62.45,-45.01,;61.94,-43.56,;60.4,-43.6,;59.96,-45.08,)|
Cc1cn(C)nc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cc1cccc(c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)-c1ccc(F)cc1F
Cc1cnsc1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccc(F)cn1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccccc2-c2ccno2)c(c1)C#N
Fc1cc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)ccc1OCc1ccccc1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(cn1)C#N
O=S(=O)(Nc1nccc(n1)C#N)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Nc1cccc(n1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Fc1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1C1CNC1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(c1)N1CCNCC1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1cn[nH]c1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1nc(ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
Cn1nccc1-c1ccccc1Oc1ccc(cc1I)S(=O)(=O)Nc1cscn1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)cc1F)C(F)(F)F
COc1cc(ccc1C#N)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
COc1cc(ccc1C#N)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
COc1ccc(-c2ccnn2C)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
COc1cccc(c1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1cnccn1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Cc1c(Cl)ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c1-c1nnco1
Cc1csc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cnn(CC(F)(F)F)c1
CC(C)(C)n1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Cc1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)s1)-c1ccnn1C
Fc1cc(Oc2ccc(Cl)cc2-c2cn[nH]c2)ccc1S(=O)(=O)Nc1cscn1
Nc1nn(CC(F)(F)F)cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Fc1cc(Oc2ccc(Cl)cc2-c2ccn[nH]2)c(Cl)cc1S(=O)(=O)Nc1nncs1
Cn1ccc(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(Cl)c1
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccccc3C3CCCCO3)c(c2)C#N)nc1
O=S(=O)(Nc1cncs1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
CC(C)(C)n1nccc1-c1c(Cl)cccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1 |(13.14,-17.62,;14.55,-18.25,;14.71,-19.79,;13.2,-19.01,;15.8,-17.34,;17.27,-17.81,;18.18,-16.56,;17.27,-15.32,;15.81,-15.79,;14.2,-14.62,;12.86,-15.39,;12.86,-16.92,;11.52,-14.62,;11.52,-13.08,;12.86,-12.31,;14.2,-13.08,;15.52,-12.31,;15.52,-10.78,;14.2,-10,;14.2,-8.47,;15.52,-7.69,;16.85,-8.47,;16.85,-10,;18.19,-10.78,;19.52,-11.54,;15.52,-6.16,;13.98,-6.16,;14.76,-4.82,;16.86,-5.4,;16.84,-3.87,;15.58,-2.97,;16.04,-1.5,;17.58,-1.48,;18.08,-2.94,)|
OCCn1nccc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccncn1
FC(F)(F)c1n[nH]cc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Fc1ccc(NS(=O)(=O)c2cc(F)c(Oc3ccc(Cl)cc3C3CCNCC3)cc2F)nc1
Clc1ccc(c(Cl)c1)-n1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cn1
Fc1ccc(Oc2ccc(SNc3ncns3)cc2C#N)c(c1)C1CC1
FC(F)(F)c1ccn(n1)-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Cc1nccnc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(OC(F)(F)F)cc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1ncccn1
CC(C)Oc1cccc(c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1-c1ccn[nH]1
Cn1nccc1-c1cc(Br)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)c(F)c1)C(F)(F)F
Fc1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(c1)-c1ccn[nH]1
Fc1cc(ccc1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
Cc1cc(c(F)cc1Oc1ccc(OC(F)(F)F)cc1-c1ccnnc1)S(=O)(=O)Nc1nncs1
OCCn1nc(cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)(F)F
Fc1cc(Oc2ccc(Cl)cc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1cscn1
CC(C)c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-c1cc(nn1C)C(F)(F)F
Fc1cc(Oc2ccc(Cl)cc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1ncccn1
FC(F)(F)c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)n(n1)-c1ccccc1
Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ccncn1
NC(=O)c1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
COCc1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1C
Clc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(cc1-c1cn[nH]c1)C#N)S(=O)(=O)Nc1ncc(Cl)s1
Fc1ccc(Oc2ccc(c(F)c2)S(=O)(=O)Nc2nccs2)c(c1)-c1ccn[nH]1
Cn1ccc(n1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2nncs2)c(c1)-c1ccn[nH]1
Fc1cc(c(F)cc1Oc1ccc(OC(F)(F)F)cc1-c1cn[nH]c1)S(=O)(=O)Nc1cscn1
Cn1nc(cc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1)C(F)(F)F
Fc1cc(c(F)cc1Oc1ccc(cc1-c1cccnn1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Fc1ccc(cc1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
OCc1cccc(c1)-c1ccc(cc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1)C(F)(F)F
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1nccs1
FC(F)(F)c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)n(Cc2ccccc2)n1
Fc1ccc(NS(=O)(=O)c2cc(F)c(Oc3ccc(cc3C3CCNCC3)C(F)(F)F)cc2F)nc1
Fc1cc(Oc2cc(ccc2-c2cn[nH]c2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1cscn1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(F)c1)C(F)(F)F
Fc1cc(c(F)cc1Oc1ccc(cc1-c1ccnnc1)C(F)(F)F)S(=O)(=O)Nc1nncs1
Fc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)c(Cn4ccnc4)c3)c(c2)C#N)s1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnnc1
Cc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncns1
Nc1ccc(cn1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
Fc1cc(cc(C#N)c1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccsn1
OCCn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3C3CNC3)c(c2)C#N)s1
OCc1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)cc1)C(F)(F)F
Cn1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1
Fc1cc(Oc2ccc(Cl)c(F)c2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1nncs1
Cc1cc(c(F)cc1Oc1ccc(F)cc1-c1ccnn1C)S(=O)(=O)Nc1cscn1
Nc1nccc(n1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(Cl)cc2-c2ccnn2-c2ccccc2)ccc1S(=O)(=O)Nc1nccs1
Nc1cccc(n1)-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Cn1ncc(F)c1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1 |(17.32,-22.36,;17.65,-23.86,;16.61,-25.01,;17.38,-26.34,;18.89,-26.02,;20.03,-27.04,;19.05,-24.49,;20.38,-23.72,;21.72,-24.49,;23.05,-23.72,;24.38,-24.49,;23.05,-22.18,;21.72,-21.41,;20.38,-22.18,;19.05,-21.41,;19.05,-19.87,;20.38,-19.1,;20.38,-17.56,;19.05,-16.8,;17.72,-17.56,;17.72,-19.1,;16.38,-19.87,;15.05,-20.64,;19.05,-15.26,;17.51,-15.26,;18.65,-13.77,;20.38,-14.49,;20.38,-12.95,;21.63,-12.05,;21.15,-10.58,;19.62,-10.58,;19.14,-12.04,)|
Nc1ccc(cn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cnco1
CC(C)(C)OC(=O)n1cc(cn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncc(F)s1
Cc1nsc(NS(=O)(=O)c2cc(Cl)c(Oc3ccc(cc3-c3ccnnc3)C(F)(F)F)cc2F)n1
CN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
CN1CCC(CC1)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1ccnnc1
COCCn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccn[nH]1)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cn[nH]c1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnn1C1CCS(=O)(=O)C1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnc(CN2CCC2)c1)S(=O)(=O)Nc1cscn1
Cc1nsc(NS(=O)(=O)c2cc(Cl)c(Oc3ccc(Cl)cc3-c3c[nH]nc3N)cc2F)n1
Fc1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(c1)-c1cn[nH]c1
Fc1cc(c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1C(F)(F)F)-c1ccnnc1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1cccnn1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)C1CCOCC1
Cc1nocc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(Cl)cc2-c2cccc(c2)C(=O)N2CCC2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnnc1)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnc(c1)N1CCNCC1)S(=O)(=O)Nc1nncs1
Cn1nc(cc1-c1cc(F)cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)(F)F
Fc1ccc(F)c(c1)-n1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)C1CC1
Fc1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cn1ccnc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CC(C)(C)n1ccc(n1)-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Cn1cc(c(N)n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
O=S(=O)(Nc1cc(ccn1)C#N)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
CN(C)Cc1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
CCn1nc(cc1C(F)(F)F)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(F)c1
COC(=O)c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)ccc1-n1cc(Cl)cn1
OCc1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1
Fc1cc(ccc1Oc1ccc(Cl)cc1-c1ccn[nH]1)S(=O)(=O)Nc1nccs1
Clc1cc(ccc1Oc1ccc(cc1)-c1ccccc1)S(=O)(=O)Nc1ncns1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)s1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1C1CNC1)S(=O)(=O)Nc1cscn1
FC(F)(F)Oc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
Nc1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
OC1CN(C1)C(=O)c1cccc(c1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncns1
Cc1ncsc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1ccnn1C1CCNCC1
Cn1cc(cn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CCn1nc(cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nc(C)ns2)c1)C(F)(F)F
Cc1nsc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(F)c2)n1
Fc1cc(ccc1Oc1ccn(Cc2ccc(Cl)cc2)n1)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1Cl
Cn1nccc1-c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)ccc1Cl
Fc1ccc(F)c(c1)-n1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C1CC1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccon1
Fc1cc(Oc2cccc(c2)-c2ccccc2)ccc1S(=O)(=O)Nc1nccs1
CC(C)(C#N)c1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnnc1
FC(F)(F)c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)n(n1)-c1ccccc1
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(cc3-c3cn[nH]c3)C(F)(F)F)c(c2)C#N)nc1
Cn1nccc1-c1cc(CO)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(OC(F)(F)F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(Cl)cc2-c2cccc(n2)C(=O)N2CCC2)c(Cl)cc1S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1ccnc(c1)N1CCNCC1
FC(F)(F)c1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnnc1
Cc1[nH]ncc1-c1cc(Cl)c(F)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Ic1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccn[nH]1
Nc1cc(ccn1)-c1cc(OC(F)(F)F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc(-c2cn[nH]c2)c(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)cc1Cl
Cn1nccc1-c1cc(Cl)cc(Cl)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)nc1
Fc1cc(ccc1Oc1cccc(Oc2ccccc2)c1)S(=O)(=O)Nc1nccs1
COc1ccc(cc1F)-c1cccc(C)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccnn1C1CNC1)S(=O)(=O)Nc1ncns1
CCn1nc(c(Cl)c1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
FC1(F)CCN(Cc2cc(Cl)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)C1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nncs1
Cc1nnc(NS(=O)(=O)c2cc(Cl)c(Oc3ccc(Cl)cc3-c3ccnn3C)cc2F)s1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
Fc1cc(cc(F)c1Oc1ccn(Cc2ccc(Cl)cc2)n1)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccc(cn1)C#N
Cc1snnc1NS(=O)(=O)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1nc(cs1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ccc(F)cn1
Cc1ccc(cc1)-c1ncccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cccnc1NS(=O)(=O)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
O=S(=O)(Nc1ncc[nH]1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1cccc(c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)-c1cc(F)ccc1F
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncccc2Cl)cc1)C(F)(F)F
COCc1cccc(c1)-c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)ccc1Cl
FC(F)(F)c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)n(n1)-c1ccccc1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C1CC1
Fc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)ccc1-n1ccc(n1)C(F)(F)F
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cc(ncn1)N1CCC1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1CC(F)(F)F
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1ccnnc1
Brc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(CN2CCCC2)c1
Clc1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1Cl
Cn1cc(c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)n1)-c1ccc(Cl)cc1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)cc1)C(F)(F)F
CCOC(=O)c1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
CCn1nc(C)cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Cn1nc(cc1-c1ccc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncc(F)s2)cc1)C(F)(F)F
Fc1cccc(c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1ccc(Oc2ccc(cc2)C#N)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c1
CC(C)n1cc(cn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1ccc(-c2ccn[nH]2)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)c1
Fc1ccc(cc1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
FC(F)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)cc1)C(F)(F)F
COCc1cccc(c1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CC(C)(C)OC(=O)n1cc(cn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1nccs1
Fc1ccc(NS(=O)(=O)c2cc(Cl)c(Oc3ccc(cc3C3CCNCC3)C(F)(F)F)cc2F)nc1
Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Fc1ccc(NS(=O)(=O)c2cc(Cl)c(Oc3ccc(Cl)cc3C3CCNCC3)cc2F)nc1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)c(c1)-c1cn[nH]c1
O=S(=O)(Nc1ncns1)c1ccc(Oc2cccnc2-c2ccccc2)c(c1)C#N
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncc(F)cc1F
Cc1nnc(o1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)cc1
CC(C)Oc1cc(-c2cc(F)ccc2Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)n(C)n1
Cn1cc(cn1)-c1cc(OC(F)(F)F)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1
Cn1nncc1-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Clc1ccc(Oc2ccc(cc2)S(=O)(=O)Nc2cscn2)c(c1)-c1cn[nH]c1
CC(C)(C)n1nccc1-c1c(F)cccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1 |(2.75,-17.94,;4.16,-18.57,;4.32,-20.11,;2.82,-19.33,;5.42,-17.66,;6.88,-18.14,;7.79,-16.89,;6.88,-15.64,;5.42,-16.12,;3.81,-14.94,;2.47,-15.72,;2.47,-17.25,;1.13,-14.94,;1.13,-13.41,;2.47,-12.64,;3.81,-13.41,;5.13,-12.64,;5.13,-11.1,;3.81,-10.33,;3.81,-8.8,;5.13,-8.02,;6.46,-8.8,;6.46,-10.33,;7.8,-11.1,;9.13,-11.87,;5.13,-6.49,;3.59,-6.48,;4.37,-5.15,;6.47,-5.73,;6.45,-4.19,;5.19,-3.3,;5.65,-1.83,;7.19,-1.81,;7.69,-3.27,)|
Fc1cc(cc(F)c1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncns1
O=S(=O)(Nc1nccs1)c1ccc(Oc2ccccc2-c2cncnc2)c(c1)C#N
Cn1nccc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(Cl)c1
FC(F)(F)c1ccn(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cn1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnn1C1CCOC1
CN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
Fc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1ccn[nH]1
Fc1cc(ccc1Oc1cc(nn1-c1ccccc1F)C(F)(F)F)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(OC(F)(F)F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
CN1C(CCC1=O)c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncccc2F)cc1)C(F)(F)F
Cn1nccc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-n1cnnn1
FC(F)(F)c1cc(ccc1Oc1ccc(Cl)cc1-c1ccnnc1)S(=O)(=O)Nc1nncs1
Fc1cc(c(F)cc1Oc1ccc(Cl)cc1-c1ccn[nH]1)S(=O)(=O)Nc1nncs1
Cn1nccc1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ccc(F)cn1
FC(F)(F)C(=O)OCc1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)cc1
Fc1cnc(NS(=O)(=O)c2cc(F)c(Oc3ccc(Cl)cc3-c3cn[nH]c3)cc2F)s1
CC(C)(C)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Nc1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ccncn1
CC(C)c1nsc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cccnc1
Cc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(c2)C#N)cn1
FC(F)(F)Cn1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-c1ccccc1
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3nnco3)c(c2)C#N)nc1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)cn1
Cc1cn(Cc2ccccc2)nc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
CN(C)c1ncc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccccc1F
Fc1cc(ccc1Oc1cc(Cc2ccc(Cl)cc2)n[nH]1)S(=O)(=O)Nc1nccs1
Fc1cc(ccc1Oc1ccc(cc1)-c1cc(n[nH]1)C(F)(F)F)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccc(nc1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3cn[nH]c3)c(c2)C#N)s1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)C1CNC1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1ccnnc1
CC(C)(C)n1nccc1-c1cc(F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
FC(F)(F)c1ccnc(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
OCCc1ccc(cc1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2ncns2)c(c1)C1CCNCC1
Fc1cc(Oc2ccc(cc2-c2ccn[nH]2)C#N)c(Cl)cc1S(=O)(=O)Nc1ncns1
Nc1cc(ccn1)-c1cc(ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1)C(F)(F)F
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
COc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(F)cn2)ccc1-n1cnc(C)c1
CN1CC(C1)n1nccc1-c1cc(OC(F)(F)F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
CC(C)(C)OC(=O)N1CCC(CC1)c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1CC(F)(F)F
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(Cl)c1)C(F)(F)F
Fc1cc(Oc2ccc(Cl)cc2C2CCNCC2)c(Cl)cc1S(=O)(=O)Nc1nncs1
Cn1nccc1-c1cc(F)ccc1Oc1c(F)cc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1coc(n1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
COc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncns1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2F)S(=O)(=O)Nc2ncc(F)s2)cc1)C(F)(F)F
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1cn[nH]c1
Cc1nnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(c2)C#N)s1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1cc(ncn1)N1CCNCC1
Fc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3cn[nH]c3)c(F)c2)s1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ccc(cn2)C#N)cc1)C(F)(F)F
Fc1ccc(NS(=O)(=O)c2ccc(Oc3ccc(CN4CCC4)c(F)c3)c(c2)C#N)nc1
Cc1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
Cc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccccc1
CC(C)(C)n1nccc1-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)c(Cl)c1)C(F)(F)F
CCc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccnn1C
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(c(F)c1)S(=O)(=O)Nc1cscn1
OC(=O)Cc1ccc(cc1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1ccc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)-c1ccnn1C1CNC1
COCCn1ccc(n1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nncs1
FC(F)(F)c1cccnc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Fc1cnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)nc1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1cscn1
OC(=O)c1cccc(c1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
COc1cccc(c1)-c1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)ccc1Cl
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ccncn1
Cc1nc(cs1)-c1ccccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
CN(C)c1ncc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccc(C)cc1
CCc1nsc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
Cn1ccc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(c2)C#N)n1
O=S(=O)(Nc1ncsn1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Cc1ccnc(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
Fc1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-c1cc[nH]n1
FC(F)(F)c1ccnc(NS(=O)(=O)c2ccc(Oc3ccccc3-c3ccccc3)c(c2)C#N)n1
Fc1cc(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)c(cc1Cl)-c1ccn[nH]1
CCN1CC(C1)n1nccc1-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C3CNC3)c(c2)C#N)s1
Fc1ccccc1-n1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1)C(F)(F)F
Fc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccc(F)nc1
CN(C)CCn1nc(cc1-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1)C(F)(F)F
Clc1ccc(Oc2ccc(cc2Cl)S(=O)(=O)Nc2cscn2)c(c1)-c1ccn[nH]1
Fc1cc(ccc1Oc1ccc(Cl)cc1-c1cn[nH]c1)S(=O)(=O)Nc1nccs1
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3C3CCNCC3)c(c2)C#N)s1
Cc1ccccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Nc1cccc(n1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
Fc1cc(-c2ccn[nH]2)c(Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)cc1Cl
CSc1nnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3-c3ccnn3C)c(c2)C#N)s1
CN1CCN(C1=O)c1ccc(Oc2ccc(SNc3nccs3)cc2C#N)cc1
COCc1ccc(cc1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CC(C)(C)n1nccc1-c1cc(F)ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(cc1C(F)(F)F)-c1ccnnc1
COc1cc(-c2ccc(Oc3ccc(cc3)S(=O)(=O)Nc3nccs3)c(F)c2)n(C)n1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(Oc2ccccc2)c1
CC(C)(C)n1cc(Cc2cccc(Oc3ccc(cc3C#N)S(=O)(=O)Nc3cscn3)c2)cn1
Cc1cc(sn1)-c1ccccc1Oc1ccc(cc1F)S(=O)(=O)Nc1nccs1
Cn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cn1)C(F)(F)F
Fc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1nncs1
O=S(=O)(Nc1nncs1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
Nc1cccc(n1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
CC(C)Oc1ccc(cc1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
Cn1cc(ccc1=O)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
CCc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccccc1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1ccccn1
Fc1cc(Oc2ccc(Cl)cc2-c2cn[nH]c2)c(Cl)cc1S(=O)(=O)Nc1cscn1
Cn1nccc1-c1ccc(F)cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
OCCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1)C(F)(F)F
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1F)C(F)(F)F
CC(C)(C)n1ccc(n1)-c1c(F)cccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Cc1cc(C)n(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
FC(F)(F)c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)-n1cccn1
Clc1ccc(cc1)-n1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cn1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nncs2)c(c1)-c1cc(ncn1)N1CCOCC1
Fc1ccccc1-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Nc1cc(ccn1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(Cl)s1
Nc1cc(ccn1)-c1cc(F)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncccn1
Cn1nccc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(F)s2)c(c1)C#N
Cc1cccc(-c2ccc(F)cc2)c1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
FC(F)(F)c1ccnc(c1)-c1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Fc1cc(ccc1Oc1ccccc1-c1ccccc1)S(=O)(=O)Nc1ncc(Cl)s1
Fc1ccc(F)c(c1)-c1ccccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Nc1cc(ccn1)-c1cc(ccc1Oc1ccc(cc1Cl)S(=O)(=O)Nc1ccncn1)C(F)(F)F
Fc1cc(c(F)cc1Oc1ccc(cc1C1CCOCC1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Cn1nccc1-c1cc(ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)C1CC1
COC(=O)c1cccc(c1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nncs2)c(cc1OC(F)(F)F)-c1ccnnc1
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncc(Cl)s1
Brc1cccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c1-c1cn[nH]c1
Fc1cc(ccc1Oc1cc(nn1-c1ccccc1)C(F)(F)F)S(=O)(=O)Nc1ncns1
Clc1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c(c1)-c1cncnc1
Fc1ccccc1-n1nc(cc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1)C1CC1
Fc1cc(Oc2ccc(Cl)cc2C2CNC2)c(Cl)cc1S(=O)(=O)Nc1ncc(Cl)s1
COc1nccnc1NS(=O)(=O)c1ccc(Oc2ccc(Cl)cc2-c2ccnn2C)c(c1)C#N
Clc1cnc(NS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3C3COC3)c(c2)C#N)s1
Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncc(F)s1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1cnn(c1)C1CNC1
Cc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncc(Cl)s2)n(n1)C1CCCCC1
Nc1cccc(n1)-c1cc(ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1)C(F)(F)F
Fc1cc(Oc2ccc(Cl)cc2-c2ccnnc2)c(Cl)cc1S(=O)(=O)Nc1nncs1
CCn1nc(cc1-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)cc1)C(F)(F)F
Fc1ccc(F)c(c1)-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Nc1ncc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccc(Cl)cc1
Brc1cnc(NS(=O)(=O)c2ccc(Oc3c(Br)cc(Br)cc3-c3ccccc3)c(c2)C#N)s1
FC(F)(F)c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2cscn2)c(c1)-c1ccnn1C1CNC1
Nc1cc(ccn1)-c1cc(ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1)C(F)(F)F
Nc1ncc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(n1)-c1ccccc1
FC(F)(F)c1cccc(n1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
FC(F)(F)Oc1ccc(c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c1)-c1ccnnc1
Fc1cc(Oc2ccc(cc2-c2ccnnc2)C#N)c(Cl)cc1S(=O)(=O)Nc1nncs1
Cc1ccc(-c2ccnn2C)c(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)c1
Clc1cc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)ccc1-c1cc(n[nH]1)C1CC1
Cn1nccc1-c1cc(F)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncc(F)s1
Cn1cnc(n1)-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1nccs1
CN(C)c1n[nH]cc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
O=S(=O)(Nc1ncns1)c1ccc(Oc2ccccc2-c2ccccc2)c(c1)C#N
CN(C)C(=O)c1cnn(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2nccs2)cc1
CC1CC1N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O |r|
Fc1ccccc1C[C@@H](NC(=O)C1CC1C(F)(F)F)C(=O)N[C@@H]1CCc2c(F)c(F)cc(F)c2N(C2CC2)C1=O |r|
Fc1ccc(C(=O)N[C@H](Cc2ccccc2F)C(=O)N[C@@H]2CCc3c(F)c(F)cc(F)c3N(C3CC3)C2=O)c(c1)C(F)(F)F |r|
CC(C)N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccccn2)C1=O |r|
CC(C)N1c2ccc(cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O)C(F)(F)F |r|
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2c(F)cc(F)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O |r|
CC(C)N1c2cc(ccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O)C(F)(F)F |r|
CC(C)N1c2ccc(F)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O |r|
CC(C)N1c2cc(F)ccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O |r|
CC(C)N1c2c(F)cccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O |r|
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O |r|
CC(C)N1c2c(F)cc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O |r|
CC(C)N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccccc2C(F)(F)F)C1=O |r|
CC(C)N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)C2CC2C(F)(F)F)C1=O |r|
CC(C)N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O |r|
CC(C)N1c2ccc(F)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O |r|
CC(C)N1c2ccc(cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O)C(F)(F)F |r|
CC(C)N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)C2CC2C)C1=O |r|
CC(C)N1c2c(F)cc(F)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O |r|
CC1CC1N1c2c(F)cc(F)c(F)c2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)C2CC2C(F)(F)F)C1=O |r|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O
Nc1nc2CCC(CNC(=O)c3ccc[nH]3)Cc2s1
Nc1nc2CC[C@@H](Cc2s1)NC(=O)c1cc(Br)c(Br)[nH]1 |r|
Nc1nc2CC[C@@H](Cc2s1)NC(=O)c1ccco1 |r|
Nc1nc2CC[C@@H](Cc2s1)NC(=O)[C@@H]1CCCN1
CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)N[C@H]1CCc2nc(N)sc2C1 |r|
CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCC1CCc2nc(N)sc2C1 |r|
Nc1nc2CCC(CNC(=O)c3cc4ccccc4[nH]3)Cc2s1
Nc1nc2CC[C@@H](Cc2s1)NC(=O)c1ccc[nH]1 |r|
Nc1nc2CCC(CNC(=O)c3cc(Br)c(Br)[nH]3)Cc2s1
Nc1nc2CCC(CNC(=O)[C@@H]3CCCN3)Cc2s1
Cn1cccc1C(=O)N[C@H]1CCc2nc(N)sc2C1 |r|
Nc1nc2CC[C@@H](Cc2s1)NC(=O)c1cc2ccccc2[nH]1 |r|
Nc1nc2CCC(CNC(=O)c3cc(Br)c[nH]3)Cc2s1
Nc1nc2CC[C@@H](Cc2s1)NC(=O)c1cc(Br)c[nH]1 |r|
Nc1nc2CC[C@@H](Cc2s1)NCc1ccc[nH]1 |r|
Nc1nc(c[nH]1)-c1ccc(NC(=O)c2ccc[nH]2)cc1
CC(C)(C)OC(=O)n1cc(nc1N)-c1ccc(NC(=O)[C@H]2CCCN2)cc1 |r|
Nc1nc(c[nH]1)-c1cccc(NC(=O)c2ccc[nH]2)c1
Nc1nc(c[nH]1)-c1ccc(NC(=O)c2cc3ccccc3[nH]2)cc1
Nc1nc(c[nH]1)-c1ccc(NC(=O)[C@@H]2CCCN2)cc1
CNc1nc(cn1C(=O)OC(C)(C)C)-c1cccc(NC(=O)c2cc3ccccc3[nH]2)c1
Nc1nc(c[nH]1)-c1ccc(NC(=O)[C@H]2CCCN2)cc1
CC(C)(C)OC(=O)n1cc(nc1N)-c1cccc(NC(=O)[C@H]2CCCN2)c1 |r|
Nc1nc(c[nH]1)-c1cccc(NC(=O)c2c[nH]c3ccccc23)c1
CC(C)(C)OC(=O)n1cc(nc1N)-c1ccc(NC(=O)c2cc3ccccc3[nH]2)cc1
CC(C)(C)OC(=O)n1cc(nc1N)-c1cccc(NC(=O)c2cc3ccccc3[nH]2)c1
CC(C)(C)OC(=O)n1cc(nc1N)-c1ccc(NC(=O)c2ccc[nH]2)cc1
CC(C)(C)OC(=O)n1cc(nc1N)-c1cccc(NC(=O)c2ccc[nH]2)c1
CCN(CC)CC(=O)Nc1c(cccc1C)C
CNc1nc(c[nH]1)-c1cccc(NC(=O)c2cc3ccccc3[nH]2)c1
CC(C)(C)OC(=O)n1cc(nc1N)-c1cccc(NC(=O)c2cc[nH]c2)c1
CC(C)(C)OC(=O)n1cc(nc1N)-c1ccc(NC(=O)c2ccco2)cc1
Nc1nc(c[nH]1)-c1cccc(NC(=O)c2cc3ccccc3[nH]2)c1
CC(C)(C)OC(=O)n1cc(nc1N)-c1cccc(NC(=O)c2c[nH]c3ccccc23)c1
CNc1nc(cn1C(=O)OC(C)(C)C)-c1cccc(NC(=O)c2ccco2)c1
CC(C)(C)OC(=O)n1cc(nc1N)-c1ccc(NC(=O)[C@@H]2CCCN2)cc1 |r|
Nc1nc(cn1C(=O)c1ccc[nH]1)-c1cccc(NC(=O)c2ccc[nH]2)c1
CCCCCN1C(COCC1=O)c1cncc(c1)-c1ccc(OC(F)(F)F)cc1
CN1CC[C@@]2(CC[C@@H](N2)c2nc(C)cc(n2)-c2ccc(cc2)C(F)(F)F)C1=O |r|
CN(C)c1ccc(C(=O)NC2CC22CCN(CC2)c2ccccc2)c2ccccc12
CC(C)Oc1ncc(OCc2cc(F)c(cc2F)C(=O)NS(=O)(=O)N(C)C)cc1Cl
CC1(COc2ccc(cn2)-n2nc(C3CC3)c3cc(ccc23)C(=O)NS(C)(=O)=O)CC1
Fc1cc(c(F)cc1OC[C@@H]1CNCC[C@H]1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1 |r|
C[C@H](c1ccccc1C1(F)CNC1)n1c2cc(F)c(cc2oc1=O)S(=O)(=O)Nc1nccs1 |r|
NC(=O)c1cnc(nc1[C@@H](O)CO)-c1ccc(Oc2cc(F)cc(Cl)c2)cc1 |r|
CS(=O)(=O)N[C@@H](Cc1cnc[nH]1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Cc1oc2nc(nn2c1CNCCc1ccccc1Cl)-c1ccccc1Cl
CC(C)COc1ccc(C)cc1-c1cccc(c1)[C@H]1CC[C@]2(CCN(C)C2=O)N1 |r|
COc1cc(ccc1OC(C)C)C(=O)N1CCC2(CC1)N(C)CCn1c(ccc21)C(F)(F)F
CCOC1CC(OC2(CCN(CC2)C(=O)c2ccc(OC(C)C)c(C)c2)C1)c1scnc1C
CCOc1ncccc1-c1cc(ccc1Oc1ccc(Cl)c(c1)C(F)(F)F)C(=O)NS(C)(=O)=O
CN1CC[C@@]2(CC[C@@H](N2)c2cc(ccn2)-c2cccc(OC(F)(F)F)c2)C1=O |r|
FC(F)(F)c1cc(Oc2ccc(cc2)C(=O)NCC2CCCCN2)cc(c1)C(F)(F)F
COc1cc(ccc1OC(C)C)C(=O)N1CCC2(CC1)CN(CC(F)F)CC(O2)c1ccccn1
Fc1ccc2n(nc(OCCN3CCOC3=O)c2c1)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CN1CCN(CC1=O)c1cccc2n(ncc12)-c1ccccc1F |r|
Fc1ccc(c(F)c1)-n1nc(OCCN2CCNC2=O)c2cc(F)ccc12
Fc1ccc2n(nc(OCCN3CCNC3=O)c2c1)-c1ccccc1F
CC(Oc1nn(-c2ccccc2F)c2ccc(F)cc12)C(=O)N1CCOCC1
Fc1ccc2n(nc(OCC(=O)N3CCOCC3)c2c1)-c1ccccc1F
Fc1ccc2n(nc(OCCn3cc[nH]c3=O)c2c1)-c1ccccc1F
CN1CCN(CCOc2nn(-c3ccccc3F)c3ccc(F)cc23)C1=O
CC(C)(C)OC(=O)NCCOc1cccc2n(ncc12)-c1ccccc1F
[H][C@@]12CN(C[C@]1([H])C(=O)N(C2)c1cccc2n(ncc12)-c1ccccc1F)C(=O)CC(C)(C)O |r|
[H][C@@]12CCN(C(=O)CC(C)(C)O)[C@]1([H])C(=O)N(C2)c1cccc2n(ncc12)-c1ccccc1F |r|
Fc1ccc(cc1)-n1nc(OCCN2CCNC2=O)c2cc(F)ccc12
Fc1ccc2n(nc(OCCn3ccnc3)c2c1)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CC2CN(Cc3ccccc3)CC2C1=O
CSCC[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@@H]3NC(=O)[C@H](CC(O)=O)NC(=O)CNC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc4ccc(O)cc4)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4ccc(O)cc4)NC(=O)[C@H](CCCCN)NC1=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]c4ccccc14)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H]([C@@H](C)O)C(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC3=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2)NC(=O)[C@@H](N)CC(O)=O |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(ccc3Cl)C(F)(F)F)CC2)cc1F
C[C@@H](N1CC[C@H](C1)n1nc(C)c2cc(C(=O)NS(=O)(=O)C3CC3)c(F)cc12)c1cc(Cl)cc(Cl)c1 |r|
C[C@H]([C@H](N)c1nc2ccc(cc2[nH]1)C(C)(C)C)C(N)=O
Cn1cc(C2=CCOCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1 |t:4|
Cn1cc(C2C3CC4CC2CN(C4)C3)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1 |TLB:13:11:8:6.5.4,3:4:12.11.10:8,4:5:12:10.9.8,THB:13:5:12.11.10:8,4:9:12:6.13.5,(6.89,-14.98,;7.37,-16.45,;6.46,-17.69,;7.36,-18.94,;6.89,-20.4,;8.03,-21.42,;7.37,-22.7,;6.13,-23.37,;5,-22.4,;5.53,-21.07,;5.77,-22.67,;6.97,-23.71,;6.3,-25.11,;8.33,-23.02,;8.83,-18.47,;10.16,-19.24,;11.5,-18.47,;11.5,-16.91,;10.16,-16.15,;8.83,-16.93,;12.83,-16.14,;12.82,-14.6,;14.17,-16.9,;15.5,-16.13,;14.72,-14.79,;16.27,-14.78,;16.84,-16.89,;17.62,-18.22,;18.38,-16.89,)|
COc1ncc(cc1C#N)-c1c(C2CCCCC2)c2ccc(cc2n1C)C(=O)NS(=O)(=O)C1CC1
Cc1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1
Cc1nn(-c2cnc(OCC3(C)CC3)c(Cl)c2)c2ccc(cc12)C(=O)NS(C)(=O)=O
Cn1c(c(C2CCCCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1)-c1ccc(nc1)N1CCCC1
COc1ncc(cn1)-c1c(C2CCCCC2)c2ccc(cc2n1C)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2CCN(CC2)C(=O)OC(C)(C)C)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1c(-c2ccoc2)c(C2CCCCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1c(c(C2CCCCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1)-c1ccc(nc1)C#N
Cn1ccc2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1)C(C)(C)C
CCC(c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1)C(C)(C)C
C[C@H]1CC[C@H](C1)c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1 |r|
Cn1cc(C2CCCC(C)(C)C2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1)C1(C)CCCCO1
Cn1cc(C2=CCNCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1 |t:4|
Cn1cc(C2=CCN(CC2)C(=O)OC(C)(C)C)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1 |t:4|
Cn1cc(C2CCCNC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2C3CC4CC(C3)CC2C4)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1 |TLB:10:9:13:6.5.4,10:5:8.9.11:13,THB:3:4:8.9.11:13,4:5:8:11.12.13,4:12:8:6.10.5,(8.01,-1.2,;8.49,-2.66,;7.58,-3.91,;8.48,-5.16,;8.01,-6.61,;9.15,-7.63,;8.49,-8.91,;7.25,-9.58,;7.42,-11.33,;8.09,-9.92,;9.45,-9.24,;6.89,-8.88,;6.65,-7.28,;6.13,-8.61,;9.95,-4.68,;11.28,-5.45,;12.62,-4.68,;12.62,-3.13,;11.28,-2.37,;9.95,-3.14,;13.95,-2.35,;13.94,-.81,;15.29,-3.12,;16.62,-2.34,;15.84,-1,;17.39,-1,;17.96,-3.11,;18.73,-4.44,;19.5,-3.1,)|
Cc1cn(C2CCCC=C2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1 |c:8|
O=C(NS(=O)(=O)C1CC1)c1ccc2c(C3CCCCC3)c3C(=O)CCCCn3c2c1
C[C@@H]1CC[C@H](C1)c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1 |r|
Cn1cc(C2CCNCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2CCCCC2)c2cc(F)c(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2CCCCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2CCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2CCC(CC2)C(C)(C)C)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1 |(26.71,-11.56,;27.18,-13.03,;26.27,-14.27,;27.18,-15.52,;26.7,-16.98,;25.19,-17.29,;24.71,-18.75,;25.74,-19.9,;27.25,-19.58,;27.73,-18.12,;25.25,-21.36,;23.74,-21.67,;26.28,-22.51,;24.7,-22.85,;28.64,-15.05,;29.97,-15.82,;31.31,-15.05,;31.31,-13.49,;29.97,-12.73,;28.64,-13.51,;32.64,-12.72,;32.63,-11.18,;33.97,-13.48,;35.3,-12.71,;34.52,-11.37,;36.07,-11.37,;36.64,-13.47,;37.42,-14.8,;38.18,-13.47,)|
CN1CCC(CC1)c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2CCCN(C2)C(=O)OC(C)(C)C)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
OC1CCCCn2c1c(C1CCCCC1)c1ccc(cc21)C(=O)NS(=O)(=O)C1CC1
Cn1cc(C2CCCCCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cc1cn(C2CCCCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1
Cn1c(c(C2CCCCC2)c2ccc(cc12)C(=O)NS(=O)(=O)C1CC1)-c1cnc(nc1)N1CCOCC1
CC(C)COc1ccc(cn1)-c1nn(C)c2cc(C(=O)NS(=O)(=O)C3CC3)c(F)cc12
CC(C)COc1ncc(cc1C#N)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
COc1cc(cnc1OCC(C)C)-c1cn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2cnc(OCC(C)(C)O)c(Cl)c2)c2ccc(cc12)C(=O)NS(C)(=O)=O
COc1cc(cnc1OCC(C)C)-c1cn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1
Cn1nc(-c2ccc(cc2)C(F)(F)F)c2cc(F)c(cc12)C(=O)NS(C)(=O)=O
Cn1nc(-c2ccc(cc2)C(F)(F)F)c2cc(F)c(cc12)C(=O)NS(=O)(=O)C1CC1
CC(C)COc1ccc(cn1)-c1nn(C)c2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)COc1ccc(cn1)-c1nn(C)c2cc(C(=O)NS(C)(=O)=O)c(F)cc12
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2ccc(nc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2ccc(nc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(-c2ccc(cc2)C(F)(F)F)c2cnc(cc12)C(=O)NS(C)(=O)=O
Cn1nc(-c2ccc(cc2)C(F)(F)F)c2ccc(cc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(cnc12)C(=O)NS(C)(=O)=O
Cn1cc(-c2cnc(OCC(F)F)c(Cl)c2)c2ccc(cc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1nn(C)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1
CC(C)COc1ncc(cc1Cl)-c1n[nH]c2cc(ccc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2cc(cnc12)C(=O)NS(=O)(=O)C1CC1
Cn1cc(-c2cnc(OCC(F)(F)F)c(Cl)c2)c2ccc(cc12)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1cn(C)c2nc(ccc12)C(=O)NS(C)(=O)=O
FC(F)(F)[C@H]1CCN([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)[C@H](C1)c1ccccc1 |r|
Cn1nccc1[C@H]1C[C@H](CCN1[C@H]1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
Fc1cc(c(F)cc1CN1CC[C@@H](C[C@@H]1c1ccccc1)C(F)(F)F)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1CN1CCCC[C@H]1c1ccccc1)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)[C@H]1C[C@H](CCN1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F |r|
Fc1ccc(cc1)[C@H]1C[C@H](CCN1[C@H]1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1ccc(F)cn1)C(F)(F)F |r|
Fc1ccc(cc1)[C@H]1C[C@H](CCN1[C@H]1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1cccnn1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1cc[nH]n1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1cnco1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1ccncc1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1cccnc1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1ccncn1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1cnccn1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1ccccn1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1cn[nH]c1)C(F)(F)F |r|
Fc1cc(c(F)cc1CN1CCCC[C@@H]1c1ccccc1)S(=O)(=O)Nc1ncns1 |r|
Fc1cc(c(F)cc1CN1CC[C@H](C[C@H]1c1ccccc1)C(F)(F)F)S(=O)(=O)Nc1ncns1 |r|
Fc1ccc(cc1)[C@H]1C[C@H](CCN1[C@H]1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1ccon1)C(F)(F)F |r|
Cn1ccc(n1)[C@H]1C[C@H](CCN1[C@H]1CCOc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)C(F)(F)F |r|
Fc1cc2[C@H](CCOc2cc1S(=O)(=O)Nc1ccncn1)N1CC[C@@H](C[C@@H]1c1ccnnc1)C(F)(F)F |r|
CC(C)(C)c1ccccc1-n1nnnc1Oc1ccc(cc1)[C@H]1CC[C@H](N1)C(N)=O |r|
NC(=O)[C@@H]1CC[C@@H](N1)c1ccc(Oc2nnnn2-c2ccccc2OC(F)(F)F)cc1 |r|
CN(C)C(=O)[C@@H]1CC[C@@H](N1)c1ccc(Oc2nnnn2-c2ccccc2OC(F)(F)F)cc1 |r|
COc1ccc(C)c(c1)-n1nnnc1Oc1ccc(cc1)[C@H]1CC[C@H](N1)C(N)=O |r|
Cc1cccc(C)c1-n1nnnc1Oc1ccc(cc1)[C@H]1CC[C@H](N1)C(N)=O |r,wU:20.22,23.28,(59.86,-27.72,;58.37,-28.12,;57.97,-29.6,;56.47,-30,;55.39,-28.9,;55.8,-27.42,;54.72,-26.32,;57.29,-27.03,;57.7,-25.55,;56.67,-24.41,;57.44,-23.07,;58.94,-23.39,;59.1,-24.92,;60.44,-25.69,;61.77,-24.92,;61.77,-23.38,;63.1,-22.61,;64.44,-23.37,;64.44,-24.92,;63.11,-25.69,;65.77,-22.59,;65.92,-21.06,;67.43,-20.73,;68.2,-22.07,;67.18,-23.21,;69.74,-22.22,;70.64,-20.97,;70.37,-23.63,)|
Cc1ccc(Cl)cc1-n1nnnc1Oc1ccc(cc1)[C@H]1CC[C@H](N1)C(N)=O |r|
CN1[C@@H](CC[C@@H]1c1ccc(Oc2nnnn2-c2ccccc2C(F)(F)F)cc1)C(N)=O |r|
NC(=O)[C@@H]1CC[C@@H](N1)c1ccc(Oc2nnnn2-c2cc(F)ccc2OC(F)(F)F)cc1 |r|
NC(=O)[C@@H]1CC[C@@H](N1)c1ccc(Oc2nnnn2-c2cc(Cl)ccc2OC(F)(F)F)cc1 |r|
Cc1cc(ccc1-n1nnnc1Oc1ccc(cc1)[C@H]1CC[C@H](N1)C(N)=O)C(F)(F)F |r|
CS(=O)(=O)NC(=O)c1ccc(cc1)-c1ccc(Cl)c(Cl)c1
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1Cl)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cnc2OC)c(Cl)c1)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(F)c(Oc2ccc(Cl)c(Cl)c2)cc1F
CC(C)COc1ncc(cc1Cl)-c1ccc(C(=O)NS(C)(=O)=O)c(C)c1
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1OC(F)(F)F)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1ccc2c(Oc3ccc(Cl)c(c3)C(F)(F)F)nccc2c1
CS(=O)(=O)NC(=O)c1cc(F)c(cc1F)-c1ccc(Cl)c(Cl)c1
CC(C)COc1ncc(cc1Cl)-c1cc(F)c(cc1F)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1ccc(C(=O)NS(C)(=O)=O)c(F)c1
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1ccc(C(=O)NS(C)(=O)=O)c(Cl)c1
CC(C)COc1ncc(cc1Cl)-c1ncc(cc1F)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1C1=CCOC1)C(=O)NS(C)(=O)=O |t:20|
COc1cc(ccc1-c1cnc(OCC(C)C)c(Cl)c1)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1C(=O)N(C)C)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(OC2CCC2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Sc2cccc(C)c2)c(Cl)c1)C(=O)NS(C)(=O)=O
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(OCC2(C)CC2)c(Cl)c1
CS(=O)(=O)NC(=O)c1ccc2c(nccc2c1)-c1ccc(c(Cl)c1)C(F)(F)F
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1C(F)(F)F)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(Oc2cc(Cl)cc(Cl)c2)c(c1)C(F)(F)F)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(Oc2nccc3cc(ccc23)C(=O)NS(C)(=O)=O)cc1Cl
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1F)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1c(F)cc(cc1F)C(=O)NS(C)(=O)=O
CC(C)COc1ncc(cc1Cl)-c1ccc(cc1C#N)C(=O)NS(C)(=O)=O
COc1cc(ccc1-c1cnc(OCC2(C)CC2)c(Cl)c1)C(=O)NS(C)(=O)=O
COC(=O)[C@@H]1Cc2c([nH]c3ccccc23)[C@H](N1Cc1ccccc1)c1ccccc1 |r|
Fc1ccc(CNC(=O)[C@@H]2Cc3c(CN2)[nH]c2ccccc32)cc1 |r|
Cn1nccc1-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Cn1nccc1-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)-c1nccs1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)-c1nccs1 |r|
Cc1nc(co1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Cc1nc(co1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)-n1ccnn1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)-n1ccnn1 |r|
Fc1ccc(cn1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Fc1ccc(cn1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Fc1ccc(nc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Fc1ccc(cc1)-c1cc(ccc1[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Fc1ccc(cc1)-c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)N1CCOCC1=O |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)N1CCOC1=O |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)N1CCS(=O)(=O)CC1 |r|
FC(F)(F)c1ccc([C@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)N1CCNCC1 |r|
CN1CCN(CC1)c1cc(ccc1[C@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Cn1nccc1-c1cc(ccc1[C@H]1CCc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
Fc1ccc(cn1)-c1cc(ccc1[C@H]1CCc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
Cc1ccc(cn1)-c1cc(ccc1[C@H]1CCc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F |r|
FC(F)(F)c1ccc([C@H]2CCc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCOCC1 |r|
CC1(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)CCCN1
Fc1cc(NCC2CCCN2)c(Cl)cc1S(=O)(=O)Nc1nccs1
Fc1cc(NCC2(Cc3ccccc3)CCCN2)c(Cl)cc1S(=O)(=O)Nc1nccs1
CNC(C)(CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)Cc1ccccc1
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)Cc1ccccc1 |r|
N[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)Cc1ccccc1 |r|
CN(C)[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1)Cc1ccccc1 |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1)Cc1ccccc1 |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncns1)Cc1ccccc1 |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1)CC1CCC1 |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1)CC1CC1 |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1)CC1(C)CC1 |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1)CC(C)(C)C
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1)C[Si](C)(C)C |r|
CN[C@H](CNc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ncc(F)s1)CC12CC(C1)C2 |r|
FC(F)(F)Oc1ccc(cc1)-c1ccc2OCCN(Cc3ncccn3)C(=O)c2c1
Fc1cccc(NS(=O)(=O)c2cc(F)c(O[C@H]3CCN(CC(F)(F)F)C[C@@H]3c3ccc(F)c(F)c3)c(F)c2)n1 |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)CNC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](C)NC1=O)[C@@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N3)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC2=O)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N1C[C@@H](O)C[C@H]1C(=O)N1C[C@@H](O)C[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O)NC(=O)CN |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)CNC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](C)NC1=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N3)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC2=O)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N1C[C@@H](O)C[C@H]1C(=O)N1C[C@@H](O)C[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O)NC(=O)CN |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)CNC(=O)[C@H](CSSC[C@H](NC(=O)CNC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC1=O)[C@@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N3)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC2=O)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N1C[C@@H](O)C[C@H]1C(=O)N1C[C@@H](O)C[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O)NC(=O)CN |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)CNC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CO)NC1=O)[C@@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N3)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC2=O)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N1C[C@@H](O)C[C@H]1C(=O)N1C[C@@H](O)C[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O)NC(=O)CN |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4cnc[nH]4)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)CNC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](C)NC1=O)[C@@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N3)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC2=O)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N1C[C@@H](O)C[C@H]1C(=O)N1C[C@@H](O)C[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O)NC(=O)CN |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4cnc[nH]4)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)CNC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC1=O)[C@@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N3)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC2=O)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N1C[C@@H](O)C[C@H]1C(=O)N1C[C@@H](O)C[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O)NC(=O)CN |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4cnc[nH]4)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)CNC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](NC(=O)[C@@H]4CCCN4C1=O)C(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N3)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC2=O)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@H](CCCCN)C(=O)N1C[C@@H](O)C[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O)NC(=O)CN |r|
[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O)NC(C)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O)NC(C)=O |r|
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[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(F)(F)F)NC(=O)[C@H](Cc1c[nH]c3ccc(Br)cc13)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O)NC(C)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(F)(F)F)NC(=O)[C@H](Cc1cccc(Cl)c1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O)NC(C)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(F)(F)F)NC(=O)[C@H](CC1CCCCC1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC4CCCCC4)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O)NC(C)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(F)(F)F)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O)NC(C)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(F)(F)F)NC(=O)[C@H](Cc1ccc(Cl)cc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(O)=O)NC(C)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(F)(F)F)NC(=O)[C@H](CC1CCCCC1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O)NC(C)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(F)(F)F)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]1NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC2=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC1=O)C1CCCCC1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(N)=O)NC(C)=O |r|
COc1cc(c(Cl)cc1-n1c2ncc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(-3.32,-7.39,;-3.32,-5.85,;-1.99,-5.08,;-.65,-5.84,;.67,-5.07,;.67,-3.53,;2.01,-2.76,;-.66,-2.76,;-1.99,-3.53,;-3.32,-2.76,;-3.33,-1.23,;-2.01,-.46,;-2.01,1.08,;-3.33,1.85,;-4.67,1.08,;-4.67,-.47,;-6,-1.25,;-5.98,-2.79,;-4.65,-3.54,;-4.65,-5.08,;-3.33,3.39,;-4.11,4.72,;-4.88,3.39,;-2,4.16,;-2,5.7,;-3.33,6.47,;-2.99,8,;-1.49,8.15,;-.87,6.73,;2.01,-5.84,;2.01,-7.39,;3.34,-8.15,;4.67,-7.38,;4.67,-5.84,;6,-5.07,;3.34,-5.07,)|
COc1cc(c(F)cc1-n1c2ccc(cc2cnc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1 |(50.95,-11.98,;49.62,-12.76,;49.63,-14.3,;50.96,-15.06,;50.97,-16.61,;49.64,-17.39,;49.65,-18.93,;48.3,-16.62,;48.3,-15.08,;46.96,-14.32,;46.95,-12.77,;48.28,-12,;48.28,-10.47,;46.94,-9.7,;45.62,-10.48,;45.62,-12,;44.29,-12.77,;44.29,-14.32,;45.63,-15.09,;45.62,-16.63,;46.93,-8.16,;45.43,-7.75,;46.53,-6.66,;48.26,-7.39,;48.25,-5.84,;47,-4.95,;47.47,-3.48,;49.01,-3.47,;49.49,-4.94,;52.31,-17.38,;52.32,-18.92,;53.65,-19.68,;54.99,-18.9,;54.97,-17.36,;56.3,-16.57,;53.63,-16.6,)|
COc1cc(ccc1N(C(=O)N(C)C)c1ccc(cn1)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
COc1cc(ccc1N(C(C)=O)c1ccc(cn1)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(C)c1
CNC(=O)N(c1ccc(cc1)S(=O)(=O)Nc1ccon1)c1ccc(cc1OC)-c1ccc(Cl)c(C)c1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)c2ccccc2C(=O)NCc2ccc(s2)-c2cccs2)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
CS(=O)(=O)c1ccccc1CCCN[C@H]1CCC[C@@H]1C(=O)NCc1ccc(s1)-c1cccs1
Brc1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
Cc1ccccc1-c1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
CC(C)(CC(=O)NCc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)NCc1ccc(s1)-c1cccs1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)CCCC(=O)NCc2ccc(s2)-c2cccs2)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)CCC(=O)NCc2ccc(s2)-c2cccs2)cc1
CN(Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)[C@H]1CCC[C@@H]1C(=O)NCc1cccc(OC(F)(F)F)c1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)c2cccc(c2)C(=O)NCc2ccc(s2)-c2cccs2)cc1
CN(Cc1ccc(s1)-c1cccs1)C(=O)[C@H]1CCC[C@@H]1C(=O)NCc1ccc(cc1)-c1ccccc1S(N)(=O)=O
CN(Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)[C@H]1CCC[C@@H]1C(=O)NCc1ccc(cc1)C(F)(F)F
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)\C=C/C(=O)NCc2ccc(s2)-c2cccs2)cc1
O=C(NCc1ccc(s1)-c1cccs1)[C@H]1CCC[C@@H]1NCc1ccc(cc1)-c1ccccc1
CC(NC(=O)[C@H]1CCC[C@@H]1C(=O)NCc1ccc(s1)-c1cccs1)c1ccc(cc1)-c1ccccc1S(N)(=O)=O
FC(F)(F)c1ccc(cc1)-c1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(cc2)-c2ccccc2C(F)(F)F)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)CC(=O)NCc2ccc(s2)-c2cccs2)cc1
CS(=O)(=O)c1ccccc1C#CCN[C@H]1CCC[C@@H]1C(=O)NCc1ccc(s1)-c1cccs1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2cccc(OC(F)(F)F)c2)cc1
CN(Cc1ccc(s1)-c1cccs1)C(=O)[C@H]1CCC[C@@H]1C(=O)N(C)Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccccc2)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(cc2)-c2ccccc2)cc1
COc1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
CS(=O)(=O)c1ccccc1-c1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
COc1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(cc2)-c2ccccc2S(N)(=O)=O)cc1
CN(Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)[C@H]1CCC[C@@H]1C(=O)NCc1ccc(OC(F)(F)F)cc1
COc1ccccc1-c1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(cc2)[N+]([O-])=O)cc1
Cc1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(cc2)-c2ccccc2S(N)(=O)=O)cc1
CC(NC(=O)[C@H]1CCC[C@@H]1C(=O)N(C)Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)c1ccc(s1)-c1cccs1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@@H]2[C@@H](C(=O)NCc3ccc(s3)-c3cccs3)C2=C)cc1
FC(F)(F)c1cccc(c1)-c1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
CC(NC(=O)[C@H]1CCC[C@@H]1C(=O)NCc1ccc(cc1)-c1ccccc1S(N)(=O)=O)c1ccc(s1)-c1cccs1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
FC(F)(F)c1ccccc1-c1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
COc1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)N(C)Cc2ccc(cc2)-c2ccccc2S(N)(=O)=O)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
COc1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(cc2)-c2ccccc2S(N)(=O)=O)cc1
NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@H]2CCC[C@@H]2C(=O)NCc2ccc(OC(F)(F)F)cc2)cc1
CN(Cc1ccc(cc1)-c1ccccc1C(F)(F)F)[C@H]1CCC[C@@H]1C(=O)N(C)Cc1ccc(s1)-c1cccs1
CN(Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)[C@H]1CCC[C@@H]1C(=O)NCc1ccc(s1)-c1cccs1
CS(=O)(=O)c1ccccc1\C=C\CN[C@H]1CCC[C@@H]1C(=O)NCc1ccc(s1)-c1cccs1
FC(F)(F)c1cccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)c1
Fc1ccc(CN[C@H]2CCC[C@@H]2C(=O)NCc2ccc(s2)-c2cccs2)cc1
CN(Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)[C@H]1CCC[C@@H]1C(=O)NCc1ccccc1
CC(C(C)C(=O)NCc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)NCc1ccc(s1)-c1cccs1
COc1cccc(C(=O)N2CCCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
COc1cccc(C(=O)N2CCCC2)c1OC(C)c1ccccc1
Clc1ccc(cc1)-c1nc(COc2ccccc2C(=O)N2CCCCCC2)cs1
COc1cccc(C(=O)N2CCCC2)c1OCc1ccc(cc1)C(C)(C)C
COc1cccc(C(=O)N2CCCC2)c1OCc1nc(no1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1nc(COc2ccccc2CN2CCCCCCC2)cs1
COc1cccc(C(=O)N2CCCC2)c1OCc1ccc(s1)-c1cccs1
CCOc1cccc(C(=O)N2CCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
COc1cccc(C(=O)N2CCCC2)c1OCCc1ccccc1
COc1cccc(CN2CCCCCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
COc1cccc(C(=O)N2CCCCCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
Cc1cccc(C(=O)N2CCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
CC(C)(C)Oc1cccc(C(=O)N2CCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1nc(COc2c(Cl)cccc2C(=O)N2CCCC2)cs1
CC(C)Oc1cccc(C(=O)N2CCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
COc1cccc(C(=O)N2CCCC2)c1OC(C)c1csc(n1)-c1ccc(Cl)cc1
COc1cccc(C(=O)N2CCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1nc(COc2ccccc2C(=O)N2CCCC2)cs1
COc1cccc(C(=O)N2CCCCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1nc(COc2ccccc2C(=O)N2CCCCC2)cs1
Clc1ccc(cc1)-c1nc(COc2ccccc2C(=O)N2CCCCCCC2)cs1
Oc1cccc(C(=O)N2CCCC2)c1OCc1csc(n1)-c1ccc(Cl)cc1
COc1cccc(CN2CCCCCCC2)c1OCc1csc(n1)-c1ccccc1
COc1cccc(C(=O)N2CCCC2)c1OCc1ccc(cc1)-c1ccccc1
COc1cccc(C(=O)N2CCCC2)c1OCCCc1ccccc1
[H][C@@]12NC(=N)N[C@]11N(CCC1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](OC(=O)c3ccc(F)cc3Cl)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](OC(=O)c3ccccc3C(F)(F)F)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3ccccc3C(F)(F)F)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)C3(CCC3)C(F)(F)F)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3ccc(cc3C(F)(F)F)C(F)(F)F)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cc(ccc3C(F)(F)F)C(F)(F)F)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc4CCCc34)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc4c3OCC4(C)C)C1(O)O)C(=N)N[C@H]2CO |r|
[H][C@@]12NC(=N)N[C@]11N(CCC1(O)O)C(=N)N[C@H]2COC(C)=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](OC(=O)c3ccccc3)C1(O)O)C(=N)N[C@H]2C(O)=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](OC(=O)c3cc(ccc3C(F)(F)F)C(F)(F)F)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc(c3)C(F)(F)F)C1(O)O)C(=N)N[C@H]2C(O)=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cc(ccc3C(F)(F)F)C(F)(F)F)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3ccccc3C(F)(F)F)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3ccc(cc3)C(F)(F)F)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc4CCCc34)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc4CCCCc34)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc4c3OCCC4(C)C)C1(O)O)C(=N)N[C@H]2CN1C(=O)CCC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc4c3OCCC4(C)C)C1(O)O)C(=N)N[C@H]2CN1C(=O)CNC1=O |r|
[H][C@@]12NC(=N)N[C@]11N(C[C@H](NC(=O)c3cccc4c3OCCC4(C)C)C1(O)O)C(=N)N[C@H]2CN1C(=O)CN(C)C1=O |r|
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1CNC(=O)c1ccc(OC(F)(F)F)cc1
OC(CCc1ccccc1OC(F)(F)F)[C@@H]1CCC[C@H]1C(=O)NCc1cc(Cl)cc(Cl)c1
OC(CCc1cccc(OC(F)(F)F)c1)[C@@H]1CCC[C@H]1C(=O)NCc1cc(Cl)cc(Cl)c1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1OCCc1cc(Cl)cc(Cl)c1
OC(CCc1cccc(OC(F)(F)F)c1)[C@@H]1CCC[C@H]1C(=O)NCc1ccccc1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1CNC(=O)c1cc(Cl)cc(Cl)c1
OC(CCc1ccc(OC(F)(F)F)cc1)[C@@H]1CCC[C@H]1C(=O)NCc1cc(Cl)cc(Cl)c1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1COCc1cc(Cl)cc(Cl)c1
OC(CCc1cccc(OC(F)(F)F)c1)[C@@H]1CCC[C@H]1C(=O)NCc1ccccc1C(F)(F)F
CN(Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)[C@@H]1CCC[C@H]1C(=O)NCc1ccc(OC(F)(F)F)cc1
CN(Cc1ccccc1)C(=O)[C@@H]1CCC[C@H]1C(=O)NCc1ccc(OC(F)(F)F)cc1
COc1ccc(CCC(O)[C@@H]2CCC[C@H]2C(=O)NCc2cc(Cl)cc(Cl)c2)cc1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1C(=O)NCc1ccccc1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1COCc1ccc(OC(F)(F)F)cc1
CS(=O)(=O)c1ccc(CCC(O)[C@@H]2CCC[C@H]2C(=O)NCc2ccc(OC(F)(F)F)cc2)cc1
OC(CCc1ccccc1OC(F)(F)F)[C@@H]1CCC[C@H]1C(=O)NCc1ccccc1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1CNS(=O)(=O)c1cc(Cl)cc(Cl)c1
OC(CCc1ccc(OC(F)(F)F)cc1)[C@@H]1CCC[C@H]1C(=O)NCc1ccccc1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1OCCc1ccc(OC(F)(F)F)cc1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1C(=O)NCc1cc(Cl)cc(Cl)c1
OC(CCc1ccccc1)[C@@H]1CCC[C@H]1CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1
Cc1cccc(c1OC[C@@H](C)N)C
c1ccc2c(c1)C=Cc3ccccc3N2C(=O)N
c1ccc(c(c1)COc2ccc(cc2)[C@H]3CC[C@H](N3)C(=O)N)F
CC(=O)N[C@H](COC)C(=O)NCc1ccccc1
CS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(C3CC3)c(Cl)c2)cc1F
Fc1cc(COc2cnc(C3CC3)c(Cl)c2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
CC(C)(C)NC(=O)OC(Cc1ccccc1)C(=O)Nc1cnc2ccccc2c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1C
Fc1cc(NCCCCNC[C@H]2CCCN2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
Fc1cc(C(=O)NS(=O)(=O)C2CC2)c(F)cc1OCCC1CCC2(C1)CCN(Cc1ccccc1)CC2
Fc1cc(OCCC2CCC3(C2)CCN(Cc2ccccc2)CC3)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Cc1cc(C(=O)NS(=O)(=O)C2CC2)c(F)cc1OCCC1CCC2(C1)CCN(Cc1ccccc1)CC2
Fc1cc(OCCC2CCC3(C2)CCN(Cc2ccco2)CC3)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Fc1cc(OCCC2CCC3(C2)CCN(Cc2ccsc2)CC3)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
C[C@H](NCc1ccc(OCc2ccccc2F)cc1)C(N)=O
Fc1cc(OCCC2(F)CCN(Cc3cc(Cl)cc(Cl)c3)CC2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCOCC2)cc1F
CC(C)c1cc(C(=O)NS(C)(=O)=O)c(F)cc1OCC12CC3CC(CC(C3)C1)C2 |TLB:26:21:28:25.24.27,26:25:28:22.21.20,THB:24:23:26.25.27:20,24:25:28.23.22:20|
CCC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCC(F)(F)CC1
c1cc2c(cc1OC(F)(F)F)sc(n2)N
FC(F)(F)Oc1ccc2nc(sc2c1)N1CCNCC1
C1CN(CCN1)c1nc2ccc(Oc3ccccc3)cc2s1
COc1cc(NC(=O)c2ccc(o2)-c2ccc(Cl)cc2)cc(OC)c1
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2cccc(F)c2C(F)(F)F)NC(=O)OC(C)(C)C)C1=O
C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1N=C(c2ccccc2)c2ccccc2N(C)C1=O |t:14|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)C23CC4CC(CC(C4)C2)C3)C1=O)c1ccccc1 |c:9,TLB:23:25:28:32.30.31,THB:30:29:26:32.31.33,30:31:28.29.34:26,33:31:28:34.25.26,33:25:28:32.30.31|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](CCc2ccccc2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1=O)c1ccccc1 |c:9|
CN1C[C@@H](CCc2ccccc12)NC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2c(F)cccc2C(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2CC[C@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccc(F)cc2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CC(C)(C)OC(=O)N[C@@H](CN[C@@H]1CCc2ccccc2N(CC(F)(F)F)C1=O)Cc1ccccc1
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NCCC(C)(C)C)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1=O)c1ccccc1 |c:9|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1=O
COC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H]1N=C(c2ccccc2)c2ccccc2N(C)C1=O |t:18|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@H](N)Cc2ccccc2)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)C(C)(C)C)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)C2CC2)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)CCc2ccccc2)C1=O)c1ccccc1 |c:9|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2cccc(c2)C(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccc(cc2)C(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2cnc[nH]2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NS(C)(=O)=O)C1=O)c1ccccc1 |c:9|
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCc2ccccc2N(CC2CC2)C1=O
CC(C)S(=O)(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H]1N=C(c2ccccc2)c2ccccc2N(C)C1=O |t:20|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2cccc(F)c2)NC(=O)OC(C)(C)C)C1=O
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NS(=O)(=O)c2ccccc2)C1=O)c1ccccc1 |c:9|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccc(F)cc2)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2c(F)cccc2F)NC(=O)OC(C)(C)C)C1=O
CN([C@H](Cc1ccccc1)C(=O)N[C@@H]1N=C(c2ccccc2)c2ccccc2N(C)C1=O)C(=O)OC(C)(C)C |t:15|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2cc(F)ccc2F)NC(=O)OC(C)(C)C)C1=O
CN1CCCC[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1=O
CN1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCc2ccccc2N(CC(F)(F)F)C1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCc2ccccc2N(CC(F)(F)F)C1=O
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2cccnc2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2cscn2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1 |c:9|
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccc(cc2)C(F)(F)F)C1=O
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccc(F)cc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2cccc(F)c2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2c(Cl)cccc2Cl)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)C(F)(F)F)C1=O
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2c(F)cccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(C)=O)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2cncnc2)C1=O
CC(C)N1c2ncccc2CCC(NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccc(F)cc2)C1=O
CC(C)N1c2ccc(Cl)cc2CC[C@@H](NC(=O)[C@@H](Cc2cc(F)ccc2F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ncccn2)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccccc2)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccncc2)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccccn2)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccc(F)cc2C(F)(F)F)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)C(C)(C(F)(F)F)C(F)(F)F)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)C(C)(C)C)C1=O
CC(C)N1c2ccccc2CC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)c2ccccc2C(F)(F)F)C1=O
CC(C)N1c2ccccc2OC[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CCN(CC)CCOC(=O)Oc1c(C(C)C)cccc1C(C)C
CC(C)(C)c1cc(C(=O)Nc2cccc(S(N)(=O)=O)c2)n(Cc2ccccc2)n1
COc1ccccc1NC(=O)c1nc2ccccc2nc1N1CCCCC1
O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1cccn1Cc1ccc(Cl)cc1
O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1cc(Br)c(Br)n1-c1ccccc1
O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1cc(Br)c(Br)n1Cc1ccccc1
O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)C1CC1c1ccc(F)c(F)c1
O=C(Nc1nccs1)c1ccc(NC(=O)[C@@H]2C[C@H]2c2ccccc2)cc1
[#6]-[#7](-[#6])-[#6]-[#6]\[#6]=[#6]-1/c2ccccc2-[#6]-[#6]-c2ccccc-12
CC(C)N1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2c(F)cccc2F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2OC(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1F)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CC(C)N1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1=O
CN1C[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C(=O)N(C)c2ccccc12
CC(C)(C)OC(=O)N[C@H](Cc1ccc(F)cc1)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CN1c2ccccc2NC[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2cccc(F)c2)NC(=O)OC(C)(C)C)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1cc(ccc1C(F)(F)F)C(F)(F)F)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CN1c2ccccc2N(CC2CCCCC2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
CN1c2ccccc2N(CC2CCC2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1OC(F)(F)F)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CN1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
CC(C)N1c2ccccc2N(CC2CC2)C[C@@H](NC(=O)[C@@H](Cc2ccc(F)cc2)NC(=O)OC(C)(C)C)C1=O
CC(C)(C)OC(=O)N[C@H](Cc1ccc(F)cc1F)C(=O)N[C@@H]1CN(CC2CC2)c2ccccc2N(CC(F)(F)F)C1=O
CN1c2ccccc2N(CC(F)(F)F)C[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
CN1c2ccccc2N(Cc2ccccc2)C[C@@H](NC(=O)[C@@H](Cc2ccccc2F)NC(=O)OC(C)(C)C)C1=O
NCCCC[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc6cnc[nH]6)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N3)C(=O)N[C@H](CC(N)=O)C(=O)N2)C(N)=O |r|
CC(C)Oc1ccc(CNC(=O)[C@@H]2CCC[C@H]2C2=NOC(C)(C2)c2ccccc2)cc1 |r,t:18|
FC(F)(F)Oc1ccc(CNC(=O)[C@@H]2CCC[C@H]2C2=NC(CO2)c2ccc(Cl)cc2)cc1 |r,t:19|
FC(F)(F)Oc1ccc(CNC(=O)[C@@H]2CCC[C@H]2C2=NOC(C2)c2ccccc2)cc1 |r,t:19|
CC1(CC(=NO1)[C@@H]1CCC[C@H]1C(=O)NCc1ccc(cc1)C(F)(F)F)c1ccccc1 |r,c:3|
CC1(CC(=NO1)[C@@H]1CCC[C@H]1C(=O)NCc1ccc(OC(F)(F)F)cc1)c1ccccc1 |r,c:3|
COC(=O)c1ccc(cc1)C1CC(=NO1)[C@@H]1CCC[C@H]1C(=O)NCc1ccc(OC(F)(F)F)cc1 |r,c:13|
FC(F)(F)Oc1ccc(CNC(=O)[C@@H]2CCC[C@H]2C2=NOC(C2)c2ccc(OC(F)(F)F)cc2)cc1 |r,t:19|
FC(F)(F)Oc1ccc(CNC(=O)[C@@H]2CCC[C@H]2C2=NOC(C2)c2ccc(Cl)cc2)cc1 |r,t:19|
FC(F)(F)Oc1ccc(CNC(=O)[C@@H]2CCC[C@H]2C2=NOC(C2)c2cccc(Cl)c2)cc1 |r,t:19|
COC(=O)c1cccc(c1)C1CC(=NO1)[C@@H]1CCC[C@H]1C(=O)NCc1ccc(OC(F)(F)F)cc1 |r,c:13|
FC(F)(F)Oc1ccc(CNC(=O)[C@@H]2CCC[C@H]2C2=NCC(O2)c2ccccc2)cc1 |r,t:19|
CC(C)(NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1)c1ccccc1 |r|
FC1CC(C1)(NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1)c1ccccc1 |r,wU:12.14,wD:8.8,(20.43,-12.76,;20.54,-11.08,;19.46,-9.99,;20.56,-8.9,;21.65,-10,;21.34,-7.57,;22.88,-7.57,;23.57,-8.94,;23.79,-6.33,;23.32,-4.86,;24.56,-3.94,;25.81,-4.86,;25.33,-6.33,;26.24,-7.57,;27.78,-7.57,;28.26,-9.04,;27,-9.95,;25.75,-9.04,;29.79,-9.08,;30.52,-10.44,;32.06,-10.48,;32.86,-9.17,;32.13,-7.82,;30.59,-7.78,;19.03,-8.9,;18.26,-7.57,;16.72,-7.57,;15.95,-8.9,;16.73,-10.24,;18.26,-10.23,)|
Clc1ccccc1-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
Oc1c(cccc1C(F)(F)F)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
CC(NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1)c1ccccc1 |r|
O=C(NC1(CCCCC1)c1ccccc1)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
FC(F)(F)c1cccc(c1)C1(CCC1)NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
COc1cccc(n1)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
COc1ccc(cc1)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
O=C(NC1(CCCC1)c1ccccc1)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
FC(F)(F)Oc1cccc(c1)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
OC1CC(C1)(NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1)c1ccccc1 |r,wU:12.14,wD:8.8,(19.04,-1.41,;19.04,-.09,;17.96,1.01,;19.06,2.09,;20.14,1,;19.83,3.43,;21.38,3.43,;22.07,2.05,;22.29,4.67,;21.82,6.14,;23.06,7.05,;24.31,6.14,;23.83,4.67,;24.74,3.42,;26.28,3.43,;26.76,1.96,;25.51,1.04,;24.26,1.96,;28.3,1.91,;29.02,.56,;30.56,.51,;31.37,1.82,;30.63,3.18,;29.1,3.22,;17.53,2.09,;16.76,3.42,;15.22,3.43,;14.45,2.09,;15.22,.76,;16.76,.76,)|
Oc1ccc(cc1)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
Oc1cc(ccc1-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1)C(F)(F)F |r|
O=C(NC1(CC1)c1ccccc1)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
Oc1cccc(c1)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
Oc1c(OC(F)(F)F)cccc1-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
Fc1ccc(cc1)C1(CCC1)NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
COC1CC(C1)(NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1)c1ccccc1 |r,wU:13.15,wD:9.9,(-3.39,-12.23,;-4.65,-11.14,;-4.71,-9.81,;-5.79,-8.72,;-4.7,-7.63,;-3.61,-8.73,;-3.92,-6.3,;-2.38,-6.3,;-1.69,-7.67,;-1.47,-5.06,;-1.94,-3.59,;-.7,-2.67,;.56,-3.59,;.08,-5.06,;.98,-6.3,;2.52,-6.3,;3,-7.77,;1.75,-8.68,;.5,-7.77,;4.54,-7.81,;5.27,-9.17,;6.8,-9.21,;7.61,-7.9,;6.87,-6.55,;5.34,-6.51,;-6.23,-7.63,;-7,-6.3,;-8.54,-6.3,;-9.31,-7.63,;-8.53,-8.97,;-7,-8.96,)|
FC(F)(F)c1cccc(n1)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
O=C(NC1(CCC1)c1ccccc1)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
Fc1ccccc1C1(CCC1)NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
COc1ccccc1-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
COc1cccc(c1)-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
Fc1cccc(c1)C1(CCC1)NC(=O)[C@@H]1CCC[C@H]1c1cc(on1)-c1ccccc1 |r|
FC(F)(F)c1ccccc1-c1cc(no1)[C@@H]1CCC[C@H]1C(=O)NC1(CCC1)c1ccccc1 |r|
[H][C@@](C)(NCc1ccc(OCc2cccc(F)c2)cc1)C(N)=O |r|
Cc1cc(nn1-c1cccc(c1)-c1cccc(F)c1C(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1cc(ccc1C(F)(F)F)C(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1ccc(Cl)cc1C(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1ccccc1OCC(F)(F)F)C(N)=O
NC(=O)n1ccc(n1)-c1ccc(cc1)-c1ccccc1Cl
NC(=O)c1cc(N)n(n1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
Cc1cc(nn1-c1cccc(c1)-c1ccccc1Cl)C(N)=O
NC(=O)n1ccc(n1)-c1cccc(c1)-c1ccccc1Cl
Cc1cc(nn1-c1cccc(c1)-c1ccccc1OC(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1ccccc1C(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1ccc(cc1C(F)(F)F)C(F)(F)F)C(N)=O
NC(=O)c1cc(n[nH]1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
Cc1cc(nn1-c1ccc(F)c(c1)-c1ccccc1OC(F)(F)F)C(N)=O
NC(=O)c1ccn(n1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
CC(C)(C)c1cc(nn1-c1cccc(c1)-c1ccccc1OC(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1c(cccc1C(F)(F)F)C(F)(F)F)C(N)=O
NC(=O)c1nc(cs1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
Cc1cc(nn1-c1cccc(c1)-c1ccccc1Oc1ccccc1)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1ccccc1OCC(F)(F)C(F)(F)F)C(N)=O
NC(=O)n1ccc(n1)-c1ccc(Oc2ccc(Cl)cc2F)cc1
Cc1cc(nn1-c1cc(ccc1F)-c1ccccc1OC(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1cc(F)ccc1C(F)(F)F)C(N)=O
Cc1cc(nn1-c1ccc(OC(F)(F)F)c(c1)-c1ccccc1OC(F)(F)F)C(N)=O
Cc1cc(nn1-c1cccc(c1)-c1c(F)cccc1C(F)(F)F)C(N)=O
Cn1cc(nc1C(N)=O)-c1cccc(c1)-c1ccccc1C(F)(F)F
NC(=O)c1csc(n1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
FC(F)(F)Oc1ccccc1-c1cccc(c1)-c1cscn1
Cc1nc(cs1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
FC(F)(F)c1ccccc1-c1cccc(c1)-c1c[nH]cn1
Cn1cc(nc1C(N)=O)-c1ccc(F)c(c1)-c1ccccc1OC(F)(F)F
NC(=O)c1nc(co1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
FC(F)(F)Oc1ccccc1-c1cccc(c1)-c1csc(n1)-c1ncc[nH]1
FC(F)(F)c1ccccc1-c1cccc(c1)-c1cocn1
FC(F)(F)Oc1ccccc1-c1cccc(c1)-c1cocn1
Cc1nc(co1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
NC(=O)NN=Cc1ccc(Oc2ccc(F)cc2)cc1 |w:5.5|
OCc1nc(cs1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
CN(C)C(=O)c1nc(cs1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
Cc1sc(nc1-c1cccc(c1)-c1ccccc1OC(F)(F)F)C(N)=O
NC(=O)Cc1nc(cs1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
NC(=O)c1nc(c(Cl)[nH]1)-c1cccc(c1)-c1ccccc1C(F)(F)F
OC1=NC(=O)C(S1)=Cc1cccc(c1)-c1ccccc1OC(F)(F)F |w:7.8,t:1|
FC(F)(F)Oc1ccccc1-c1cccc(c1)-c1csc(n1)-c1cnccn1
NC(=O)c1nc(c[nH]1)-c1cccc(c1)-c1ccccc1C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cc(ccc1C(F)(F)F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1c(cccc1C(F)(F)F)C(F)(F)F
NC(=O)c1cn(nc1C(N)=O)-c1cccc(c1)-c1ccccc1OC(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cccc(OC(F)(F)F)c1F
Cc1c(C(N)=O)c(nn1-c1cccc(c1)-c1ccccc1OC(F)(F)F)C(N)=O
NC(=O)c1nn(c(C(N)=O)c1C(N)=O)-c1cccc(c1)-c1ccccc1OC(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1c(F)cccc1OC(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cc(ccc1OC(F)(F)F)C(F)(F)F
CCOC(=O)c1cc(nn1-c1cccc(c1)-c1ccccc1OC(F)(F)F)C(N)=O
NC(=O)c1cc(C(N)=O)n(n1)-c1ccc(F)c(c1)-c1ccccc1OC(F)(F)F
CCNC(=O)c1cc(nn1-c1cccc(c1)-c1ccccc1OC(F)(F)F)C(N)=O
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1ccc(F)cc1OCC(F)(F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cc(F)ccc1OCC(F)(F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cccc(Cl)c1Cl
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cccc(OC(F)(F)F)c1OCC(F)(F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1ccccc1C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cccc(c1OCC(F)(F)C(F)(F)F)C(F)(F)F
C([C@@]1([C@H]2[C@@H]3[C@H](N=C(N[C@@]34[C@@H]([C@@H]1O[C@]([C@H]4O)(O2)O)O)N)O)O)O
OC1(C(=O)N(Cc2ccc(F)c(F)c2)c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(CC2CCC2)c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(CC2CCCCC2)c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(F)cc2)c2ccccc12)c1ccc2OCOc2c1
CCCCCCN1C(=O)C(O)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(CC2CC2)c2ccccc12)c1ccc2OCOc2c1
CC(C)(C(=O)c1cccs1)C1(O)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
OC1(CC(=O)c2cccs2)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
OC1(CC(=O)c2ccco2)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
CCCCCN1C(=O)C2(OCc3cc4OCOc4cc23)c2ccccc12
CC(C)CCN1C(=O)C(O)(c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C2(CCCc3cc4OCOc4cc23)c2ccccc12
OC1(C(=O)N(CCCC(F)(F)F)c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C2(CCc3cc4OCOc4cc23)c2ccccc12
OC1(C(=O)N(Cc2ccc3OCOc3c2)c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)s2)c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C2(CCC(=O)c3cc4OCOc4cc23)c2ccccc12
OC1(C(=O)N(Cc2ccccc2)c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C2(CC(=O)c3cc4OCOc4cc23)c2ccccc12
COc1ccc(CN2C(=O)C(O)(c3ccccc23)c2ccc3OCOc3c2)cc1
CCCCCN1C(=O)C(CC(=O)N(C)C)(c2ccccc12)c1ccc2OCOc2c1
CCC(C)CCN1C(=O)C(O)(c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C(CC(=O)NC)(c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C(O)(c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C(CC(N)=O)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(CCC2CC2)c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C(CCC(O)=O)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12)c1ccc2ccoc2c1
CCCCCN1C(=O)C(CC(O)=O)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12)c1ccc2OC(F)(F)Oc2c1
CCCCCN1C(=O)C(CCC(=O)OC)(c2ccccc12)c1ccc2OCOc2c1
COc1ccc(cc1)C1(O)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
CCCCCN1C(=O)C(CC(=O)OC)(c2ccccc12)c1ccc2OCOc2c1
CCCCCN1C(=O)C(N)(c2ccccc12)c1ccc2OCOc2c1
COc1ccc(cc1OC)C1(O)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
COc1ccccc1C1(O)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
CCCCCN1C(=O)C(C(=O)NCc2ccccc2)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12)c1ccoc1
CCCCCN1C(=O)C(C(=O)NC)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12)c1ccc2OCCCOc2c1
CCCCCN1C(=O)C(C(=O)OC)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12)c1ccccc1
CCCCCN1C(=O)C(C)(c2ccccc12)c1ccc2OCOc2c1
COc1cccc(c1)C1(O)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
CCCCCN1C(=O)C(OC)(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12)c1ccc2OCCOc2c1
CCCCCN1C(=O)C(CO)(c2ccccc12)c1ccc2OCOc2c1
COc1ccc(cn1)C1(O)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
CCCCCN1C(=O)C(c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)Nc2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)c2cccs2)C(=O)N(Cc2ccc(Cl)cc2)c2ccccc12
OC1(C(=O)N(Cc2cccc3ccccc23)c2ccccc12)c1ccc2OCOc2c1
OC1(C(=O)N(Cc2ccc(cc2)C(F)(F)F)c2ccccc12)c1ccc2OCOc2c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCCCC2)c1
CC1CCN(CC1)c1ncnc(Nc2cccc(NC(C)=O)c2)n1
COC1CCN(CC1)c1ncnc(Nc2cccc(NC(C)=O)c2)n1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)C(N)=O)c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccccc2)c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(Cc3ccccc3)CC2)c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(O)(CC2)c2ccccc2)c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCN(CC2)C(=O)c2ccccc2)c1
CC(=O)Nc1cccc(Oc2ncnc(n2)N2CCc3ccccc3C2)c1
CC(=O)Nc1cccc(Nc2ncnc(N)n2)c1
CN(C(C)=O)c1cccc(Nc2ncnc(n2)N2CCc3ccccc3C2)c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCc3ccccc3C2)c1
CC(=O)Nc1cccc(Nc2ccnc(n2)N2CCc3ccccc3C2)c1
CC(=O)Nc1cccc(Nc2nccc(n2)N2CCc3ccccc3C2)c1
CC(=O)Nc1cccc(Nc2cc(ncn2)N2CCc3ccccc3C2)c1
CN(c1cccc(NC(C)=O)c1)c1ncnc(n1)N1CCc2ccccc2C1
CC(=O)Nc1cccc(Nc2cc(ncn2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(cc2)C(C)(C)C)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(cc2)C(N)=O)c1C
COc1ccc(COC2CCN(CC2)c2ncnc(Nc3cccc(NC(C)=O)c3C)n2)cc1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(cc2)C(F)(F)F)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccc(OC(F)(F)F)cc2)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2cccc(c2)C(F)(F)F)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(cc2)C(F)(F)F)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(C)cc2)c1C
CC(C)c1ccc(COC2CCN(CC2)c2ncnc(Nc3cccc(NC(C)=O)c3C)n2)cc1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)c2ccccc2)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccccc2)c1C
CC(OC1CCN(CC1)c1ncnc(Nc2cccc(NC(C)=O)c2C)n1)c1ccccc1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccccc2F)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2cccc(F)c2)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(F)cc2)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccccc2C(F)(F)F)c1C
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)Oc2ccccc2)c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccccc2)c1
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccccc2)c1C
CC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H]1CC(=O)NCCCC[C@H](NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCN=C(N)N)NC1=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O |r,wU:4.3,27.28,36.72,wD:13.12,58.61,40.42,72.75,50.53,(15.7,-6.02,;15.75,-7.56,;17.12,-8.27,;14.45,-8.38,;14.51,-9.92,;15.89,-10.62,;15.96,-12.17,;17.32,-12.87,;17.39,-14.42,;18.76,-15.12,;13.22,-10.75,;11.85,-10.03,;13.29,-12.27,;11.99,-13.1,;10.62,-12.4,;9.32,-13.23,;9.23,-14.77,;7.75,-15.15,;6.91,-13.85,;5.39,-13.6,;4.86,-12.15,;5.83,-10.96,;7.34,-11.22,;7.89,-12.66,;12.06,-14.65,;13.42,-15.36,;10.76,-15.48,;10.82,-17.01,;12.2,-17.73,;12.26,-19.26,;10.96,-20.09,;13.84,-20.4,;15.19,-19.66,;16.51,-20.46,;16.47,-22,;15.12,-22.74,;15.08,-24.28,;13.73,-25.02,;12.41,-24.22,;12.46,-22.68,;11.07,-24.96,;11.02,-26.49,;12.34,-27.3,;13.77,-26.71,;14.76,-27.88,;13.96,-29.19,;12.47,-28.83,;9.75,-24.15,;8.39,-24.9,;8.36,-26.43,;7.07,-24.09,;5.74,-24.86,;4.4,-24.08,;4.4,-22.54,;3.06,-24.85,;7.04,-22.54,;8.36,-21.74,;9.72,-22.47,;8.3,-20.21,;6.93,-19.49,;5.63,-20.33,;4.26,-19.61,;2.97,-20.44,;1.6,-19.73,;1.53,-18.19,;.3,-20.56,;9.59,-19.38,;9.53,-17.85,;8.16,-17.13,;16.39,-25.08,;16.36,-26.62,;17.75,-24.34,;19.07,-25.15,;19.03,-26.68,;20.34,-27.49,;20.31,-29.03,;21.62,-29.83,;21.59,-31.37,;20.24,-32.11,;22.9,-32.17,;20.41,-24.4,;21.73,-25.21,;20.45,-22.87,)|
CC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H]1CCCCNC(=O)C[C@H](NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCN=C(N)N)NC1=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O |r,wU:4.3,27.28,36.72,wD:13.12,58.61,40.42,72.75,50.53,(13.52,-4.74,;13.58,-6.28,;14.94,-6.99,;12.27,-7.1,;12.33,-8.63,;13.71,-9.34,;13.78,-10.89,;15.14,-11.59,;15.21,-13.14,;16.58,-13.84,;11.04,-9.46,;9.68,-8.74,;11.11,-10.99,;9.82,-11.82,;8.44,-11.12,;7.14,-11.94,;7.05,-13.48,;5.57,-13.87,;4.73,-12.56,;3.22,-12.31,;2.68,-10.87,;3.65,-9.68,;5.16,-9.94,;5.71,-11.38,;9.89,-13.37,;11.25,-14.08,;8.58,-14.2,;8.64,-15.73,;10.02,-16.44,;10.08,-17.98,;11.44,-18.69,;12.74,-17.86,;14.11,-18.58,;14.28,-20.72,;15.6,-21.52,;12.94,-21.46,;12.91,-23,;11.55,-23.74,;10.23,-22.94,;10.28,-21.4,;8.89,-23.67,;8.84,-25.21,;10.16,-26.01,;11.59,-25.43,;12.59,-26.6,;11.78,-27.91,;10.29,-27.55,;7.57,-22.87,;6.22,-23.62,;6.18,-25.15,;4.89,-22.81,;3.56,-23.57,;2.23,-22.8,;2.22,-21.26,;.89,-23.57,;4.86,-21.26,;6.18,-20.46,;7.54,-21.19,;6.12,-18.93,;4.75,-18.21,;3.45,-19.04,;2.08,-18.33,;.79,-19.16,;-.58,-18.45,;-.64,-16.91,;-1.88,-19.28,;7.41,-18.09,;7.35,-16.56,;5.99,-15.85,;14.21,-23.8,;14.19,-25.34,;15.57,-23.06,;16.89,-23.86,;16.85,-25.4,;18.17,-26.2,;18.13,-27.75,;19.45,-28.54,;19.41,-30.09,;18.06,-30.82,;20.73,-30.88,;18.24,-23.12,;19.55,-23.92,;18.28,-21.59,)|
Cn1c(SCc2ccc(cc2)C(C)(C)C)nc(N)cc1=O
CCCCCCCSc1nc(N)cc(=O)[nH]1
CCCCCCSc1nc(N)cc(=O)[nH]1
CC(=O)Nc1cc(=O)[nH]c(SCc2ccc(cc2)C(C)(C)C)n1
CC(C)(C)c1ccc(CSc2nc(O)cc(=O)[nH]2)cc1
CC(C)(C)c1ccc(CSc2nccc(=O)[nH]2)cc1
CS(=O)(=O)c1ccc(CSc2nc(N)cc(=O)[nH]2)cc1
Nc1cc(=O)[nH]c(SCc2ccc(cc2)-c2ccccc2)n1
Nc1cc(=O)[nH]c(SCc2ccc(OC(F)(F)F)cc2)n1
Nc1cc(=O)[nH]c(SCc2ccc(cc2)C(F)(F)F)n1
Nc1cc(=O)[nH]c(SCc2ccc(cc2)C#N)n1
Nc1cc(=O)[nH]c(SCc2ccc(F)cc2)n1
Cc1ccc(CSc2nc(N)cc(=O)[nH]2)cc1
Nc1cc(=O)[nH]c(SCc2ccccc2)n1
CC(C)CSc1nc(N)cc(=O)[nH]1
Nc1cc(=O)[nH]c(SCc2ccc(Cl)cc2)n1
CC(C)(C)c1ccc(CSc2nc(N)cc(=O)[nH]2)cc1
Cn1c(N)cc(=O)nc1SCc1ccc(cc1)C(C)(C)C
COc1cc(N)nc(SCc2ccc(cc2)C(C)(C)C)n1
CC(C)(C)c1ccc(CSc2nc3nc[nH]c3c(=O)[nH]2)cc1
CC(C)(C)c1ccc(CSc2nc(N)c(N)c(=O)[nH]2)cc1
CC(C)(C)c1ccc(CSc2nc(N)c(Cl)c(=O)[nH]2)cc1
CC(C)(C)c1ccc(CSc2nc(NS(C)(=O)=O)cc(=O)[nH]2)cc1
CC(C)(C)OC(=O)Nc1cc(=O)[nH]c(SCc2ccc(cc2)C(C)(C)C)n1
CC(C)(C)c1ccc(CSc2nc(NC(=O)C3CC3)cc(=O)[nH]2)cc1
CCCCCCCC(O)(C(N)=O)c1cccc(Cl)c1
CCCCCCC[C@](O)(C(N)=O)c1cccc(Cl)c1 |r|
CCCCCCC[C@@](O)(C(N)=O)c1cccc(Cl)c1 |r|
O=C1NC(=O)C(N1)(c1ccccc1)c1ccccc1
CC(C1CC1)n1c(CNC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)nc2cccnc12
CC(C)(C)OC(=O)N[C@H](Cc1ccc(Cl)cc1)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)n1c(CNC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)nc2cccnc12
CC(C)(C)OC(=O)N[C@H](Cc1cc(F)ccc1Cl)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1cccc(F)c1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1cccc(F)c1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)CC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1c(F)ccc(F)c1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)Cn1c(CNC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)nc2cccnc12
CC(C)(C)C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
C[C@H](c1ccccc1)n1c(CNC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)nc2cccnc12
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1CC1CC1
CC(C)(C)OC(=O)N[C@H](Cc1c(F)cccc1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
FC(F)(F)c1ccccc1C[C@@H](NC(=O)C1(CC1)C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
C[C@@H](c1ccccc1)n1c(CNC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)nc2cccnc12
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1OC(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccc(F)cc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1cc(F)ccc1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
Fc1ccc(F)c(C[C@@H](NC(=O)C2(CC2)C(F)(F)F)C(=O)NCc2nc3cccnc3n2C2(CC2)c2ccccc2)c1F
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1c(F)cccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
FC(F)(F)c1ccccc1C[C@@H](NC(=O)c1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
FC(F)(F)c1ccccc1C[C@@H](NC(=O)c1ccccc1)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC1(CC1)C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
Fc1cccc(F)c1C[C@@H](NC(=O)C1(CC1)C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
FC(F)(F)Oc1ccccc1C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1c(F)cccc1Cl)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC1(CC1)C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1cccc(Cl)c1)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C(C)(C)C
Cn1c(CNC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)nc2cccnc12
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1CC(F)(F)F
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
FC(F)(F)Oc1ccccc1C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1Cl)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1CC(F)(F)C(F)(F)F
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2ncccc2[nH]1
CC(n1c(CNC(=O)[C@@H](Cc2ccccc2C(F)(F)F)NC(=O)OC(C)(C)C)nc2cccnc12)C(F)(F)F
FC(F)(F)C1(CC1)C(=O)N[C@H](Cc1ccccc1Cl)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
Nc1cncc(Nc2ccc(Oc3ccc(OC(F)(F)F)cc3)cc2)n1
Cc1cc(Oc2ccc(Cl)cc2)ccc1Nc1nccc(N)n1
Nc1ncnc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
CNc1ncnc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
Clc1ccc(Oc2ccc(Nc3ncncn3)cc2)cc1
Nc1ccnc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
Nc1cc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)ncn1
Nc1nccc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
Nc1cc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)ccn1
Nc1cccc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
Nc1cncc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)c1
Nc1ccnc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)c1
Nc1cc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)cnn1
Nc1cnnc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)c1
Nc1cncc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
Nc1nc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)ns1
Nc1nnc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)s1
Nc1ccnc(Oc2ccc(Oc3ccc(Cl)cc3)cc2)n1
Nc1ccnc(Nc2ccc(Nc3ccc(Cl)cc3)cc2)n1
CN(c1ccc(Cl)cc1)c1ccc(Nc2nccc(N)n2)cc1
Cc1cc(Nc2nccc(N)n2)ccc1Oc1ccc(Cl)cc1
Nc1ccnc(Nc2ccc(Oc3cccc(Cl)c3)cc2)n1
Nc1ccnc(Nc2ccc(Oc3ccccc3Cl)cc2)n1
Nc1ccnc(Nc2ccc(Oc3ccc(F)cc3)cc2)n1
Cc1ccc(Oc2ccc(Nc3nccc(N)n3)cc2)cc1
Nc1ccnc(Nc2ccc(Oc3ccc(cc3)C3CC3)cc2)n1
Nc1ccnc(Nc2ccc(Oc3ccc(cc3)-c3ccccc3)cc2)n1
Nc1ccnc(Nc2ccc(Oc3ccc(cc3)C#N)cc2)n1
CS(=O)(=O)c1ccc(Oc2ccc(Nc3nccc(N)n3)cc2)cc1
NC(=O)c1ccc(Oc2ccc(Nc3nccc(N)n3)cc2)cc1
Nc1ccnc(Nc2ccc(Oc3ccncc3)cc2)n1
CN(C)c1ccc(Oc2ccc(Nc3nccc(N)n3)cc2)cc1
Nc1ccnc(Nc2ccc(Oc3ccc(OC(F)(F)F)cc3)cc2)n1
Nc1nsc(Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
Nc1ccnc(Nc2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)n1
Nc1cncc(Nc2ccc(Oc3ccccc3)cc2)n1
Nc1cncc(Nc2ccc(Oc3ccc(F)cc3)cc2)n1
Cc1ccc(Oc2ccc(Nc3cncc(N)n3)cc2)cc1
Nc1cncc(Nc2ccc(Oc3ccc(cc3)C3CC3)cc2)n1
Nc1cncc(Nc2ccc(Oc3ccc(cc3)C#N)cc2)n1
Nc1cncc(Nc2ccc(Oc3ccc(cc3)C(F)(F)F)cc2)n1
Cc1c(C)c2c(OC3CCN(Cc4cscn4)CC3)ncnc2n1Cc1ccccc1
Fc1cccnc1CN1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cnccn1
Fc1ccccc1Cn1ccc2c(OC3CCN(Cc4ccccn4)CC3)ncnc12
Fc1cccc(Cn2ccc3c(OC4CCN(Cc5ccccn5)CC4)ncnc23)c1F
Fc1c(Cl)cccc1Cn1ccc2c(OC3CCN(Cc4ccccn4)CC3)ncnc12
Fc1c(Cn2ccc3c(OC4CCN(Cc5ccccn5)CC4)ncnc23)cccc1C(F)(F)F
FC(F)(F)c1nc(OC2CCN(Cc3cscn3)CC2)c2ccn(Cc3ccccc3)c2n1
FC(F)(F)c1ccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)cc1
Cc1cccnc1CN1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12
C(N1CCC(C1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cscn1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1ccccn1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cccnc1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1ccncc1
Cc1cccc(CN2CCC(CC2)Oc2ncnc3n(Cc4ccccc4)ccc23)n1
Cc1ccc(CN2CCC(CC2)Oc2ncnc3n(Cc4ccccc4)ccc23)nc1
Cc1ccnc(CN2CCC(CC2)Oc2ncnc3n(Cc4ccccc4)ccc23)c1
Fc1cccc(CN2CCC(CC2)Oc2ncnc3n(Cc4ccccc4)ccc23)n1
Fc1ccc(CN2CCC(CC2)Oc2ncnc3n(Cc4ccccc4)ccc23)nc1
Fc1cn(Cc2ccccc2)c2ncnc(OC3CCN(Cc4cscn4)CC3)c12
Clc1cn(Cc2ccccc2)c2ncnc(OC3CCN(Cc4cscn4)CC3)c12
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cscn1
Cc1nc(OC2CCN(Cc3cscn3)CC2)c2ccn(Cc3ccccc3)c2n1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ncc12)c1cscn1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)cnc12)c1cscn1
CC1(C)CN(Cc2ccccc2)c2ncnc(OC3CCN(Cc4cscn4)CC3)c12
CC1(C)C(=O)N(Cc2ccccc2)c2ncnc(OC3CCN(Cc4cscn4)CC3)c12
C(N1CCC(CC1)Oc1ncnc2n(ccc12)-c1ccccc1)c1cscn1
C(Cn1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12)c1ccccc1
C(C1CCCCC1)n1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12
Fc1ccccc1Cn1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12
Fc1cccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)c1
Fc1ccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)cc1
Clc1ccccc1Cn1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12
Clc1cccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)c1
Clc1ccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)cc1
Cc1ccccc1Cn1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12
Cc1cccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)c1
Cc1ccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)cc1
FC(F)(F)c1ccccc1Cn1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12
FC(F)(F)c1cccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)c1
Fc1cccc(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)c1F
Fc1c(Cl)cccc1Cn1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12
Fc1c(Cn2ccc3c(OC4CCN(Cc5cscn5)CC4)ncnc23)cccc1C(F)(F)F
Fc1cccc(F)c1Cn1ccc2c(OC3CCN(Cc4cscn4)CC3)ncnc12
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1ccccc1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cocn1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cnc[nH]1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1ccn[nH]1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cn[nH]c1
Cn1cc(CN2CCC(CC2)Oc2ncnc3n(Cc4ccccc4)ccc23)cn1
Cn1ccnc1CN1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12
Cc1nc(CN2CCC(CC2)Oc2ncnc3n(Cc4ccccc4)ccc23)cs1
C(N1CCC(CC1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1nccs1
C(N1CCC(CC1)Nc1ncnc2n(Cc3ccccc3)ccc12)c1cscn1
C(N1CC(C1)Oc1ncnc2n(Cc3ccccc3)ccc12)c1cscn1
Cc1cn(Cc2ccccc2)c2ncnc(OC3CCN(Cc4cscn4)CC3)c12
CN1CCN(CC1)c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OC(F)(F)F)cc1 |r|
CCCCOc1ccc(cc1)C(=O)N[C@@H]1COc2cccc(N3CCN(C)CC3)c2C1 |r|
CN1CCN(CC1)c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCCC(F)(F)F)nc1 |r|
CN1CCN(CC1)c1cccc2OC[C@H](Cc12)NC(=O)c1nn(nc1C)-c1ccccc1 |r|
CN1CCN(CC1)c1cccc2OC[C@H](Cc12)NC(=O)c1nn(nc1C)-c1ccc(C)cc1C |r|
FC(F)(F)Oc1ccc(cc1)C(=O)N[C@@H]1COc2cccc(c2C1)-c1ccccn1 |r|
FC(F)(F)Oc1ccc(cc1)C(=O)N[C@@H]1COc2cccc(c2C1)-c1cccnc1 |r|
FC(F)(F)Oc1ccc(cc1)C(=O)N[C@@H]1COc2cccc(c2C1)-c1ccncc1 |r|
FC(F)(F)COc1ccc(cn1)C(=O)N[C@@H]1COc2cccc(-c3ccncc3)c2C1 |r|
OCc1ccc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
OCc1cc(ccn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
OCc1ccc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCCOCC(F)(F)F)nc1 |r|
CC(O)c1ccc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCCOCC(F)(F)F)nc1 |r|
Cc1nn(nc1C(=O)N[C@@H]1COc2cccc(-c3ccncc3)c2C1)-c1ccccc1 |r|
COCCn1nc(C)c(n1)C(=O)N[C@@H]1COc2cccc(-c3ccncc3)c2C1 |r|
COCCn1nc(C)c(n1)C(=O)N[C@@H]1COc2cccc(-c3cccnc3)c2C1 |r|
CC(C)Cn1nc(C)c(n1)C(=O)N[C@@H]1COc2cccc(-c3cccnc3)c2C1 |r|
COc1ncc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
COc1ncc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCCC(F)(F)F)nc1 |r|
COc1ncc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(COCC(F)(F)F)nc1 |r|
Cc1ncc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
COc1cnc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
Cc1cnc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(COCC(F)(F)F)nc1 |r|
COc1cnc(cn1)-c1cccc2OC[C@@H](Cc12)NC(=O)c1ccc(COCC(F)(F)F)nc1 |r|
COc1cnc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(COCC(F)(F)F)nc1 |r|
FC(F)(F)COc1ccc(cn1)C(=O)N[C@@H]1COc2cccc(-c3cccnc3)c2C1 |r|
CN1CCN(CC1)c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
COc1ncc(cc1F)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
Cc1cc(cnc1CO)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCCOCC(F)(F)F)nc1 |r|
FC(F)(F)CCOc1ccc(cn1)C(=O)N[C@@H]1COc2cccc(-c3cncnc3)c2C1 |r|
Cc1cnc(cn1)-c1cccc2OC[C@H](Cc12)NC(=O)c1ccc(OCC(F)(F)F)nc1 |r|
COc1ncc(cn1)-c1cccnc1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cccnc1C(F)(F)CNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cccnc1C(C)CNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cc(C)cnc1CCNC(=O)c1ccc(COCC(F)(F)F)nc1
COc1ncc(cn1)-c1ccc(C)nc1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1cnc(cn1)-c1cccc(F)c1C(F)(F)CNC(=O)c1ccc(COCC(F)(F)F)nc1
COc1cnc(cn1)-c1ccccc1C(F)(F)CNC(=O)c1ccc(COCC(F)(F)F)nc1
Cc1cnc(cn1)-c1c(F)ccc(F)c1CCNC(=O)c1ccc(COCC(F)(F)F)nc1
COc1cnc(cn1)-c1c(OC)ccc(F)c1CCNC(=O)c1ccc(COCC(F)(F)F)nc1
COc1cnc(cn1)-c1ccc(Cl)cc1CCNC(=O)c1ccc(COCC(F)(F)F)nc1
COc1ncc(cn1)-c1ccccc1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cccc(OC(F)F)c1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1ccccc1C(F)(F)CNC(=O)c1ccc(COCC(F)(F)F)nc1
COc1ncc(cn1)-c1c(C)ccc(F)c1CCNC(=O)c1ccc(OCC(F)(F)F)nc1
COc1cnc(cn1)-c1ccccc1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1c(C)ccc(F)c1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1cnc(cn1)-c1c(F)ccc(F)c1CCNC(=O)c1ccc(COCC(F)(F)F)nc1
COc1cnc(cn1)-c1c(C)ccc(F)c1CCNC(=O)c1ccc(COCC(F)(F)F)nc1
Cc1ncc(cn1)-c1ccccc1CCNC(=O)c1cnc(OCCOCC(F)(F)F)c(C)c1
Cc1ncc(cn1)-c1ccccc1CCNC(=O)c1ccc(nc1)C(=O)NCCCC(F)(F)F
Cc1ncc(cn1)-c1ccccc1CCNC(=O)c1ccc(CNCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cccc(C)c1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
Cc1ncc(cn1)-c1ccccc1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
OCc1ccc(cn1)-c1ccccc1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
Cc1ncc(cn1)-c1ccccc1CCNC(=O)c1ccc(COCC(F)(F)F)nc1
Cc1ncc(cn1)-c1ccccc1CCNC(=O)c1ccc(OCCOCC(F)(F)F)nc1
FC(F)Oc1cnc(cn1)-c1ccccc1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
FC(F)(F)CCOc1ccc(cn1)C(=O)NCCc1ccccc1-c1cccnc1
COc1ccc(CCNC(=O)c2ccc(OCCC(F)(F)F)nc2)c(c1)-c1cnc(OC)nc1
COc1ncc(cn1)-c1cccc(C#N)c1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cccc(Cl)c1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cccc(OC)c1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
COc1ncc(cn1)-c1cccc(F)c1CCNC(=O)c1ccc(OCCC(F)(F)F)nc1
CC(=O)N[C@@H](Cc1cnc[nH]1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1 |r|
Fc1ccc(Oc2ccc(cc2)-c2cccc(NC(=O)[C@H](Cc3cnc[nH]3)NC(=O)C3CC3)n2)cc1 |r|
C(NC(Cc1ccccc1)c1ccccc1)C1CC11CCN(CC1)c1ccccc1
C(Nc1ccccc1N1CCCCC1)C1CC11CCN(Cc2ccccc2)CC1
CN(C)c1cccc2c(cccc12)C(=O)NC1CC11CCN(CC1)c1ccccc1
Fc1ccc(C(=O)NC2CC22CCN(CC2)c2ccccc2)c2ccccc12
CN(C)c1ccc(C(=O)NC2CC22CCN(CC2)c2cc(F)cc(F)c2)c2ccccc12
Fc1cnc(CCN2C(C(=O)NCc3ccc(F)c(c3)C(F)(F)F)c3ccccc3C2=O)nc1
Fc1cnc(CCN2C(C(=O)NCc3cccc(OC(F)(F)F)c3)c3ccccc3C2=O)nc1
Fc1cccc2C(N(CCc3ccccn3)C(=O)c12)C(=O)NCc1ccc(OC(F)(F)F)cc1
Oc1cccc2C(=O)N(CCc3ccccn3)C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c12
FC(F)(F)Oc1ccc(CNC(=O)C2N(C3CCC(F)(F)CC3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(C3CCOCC3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cc1
COc1cccc2C(=O)N(CCc3ccccn3)C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c12
Cc1cccc2C(=O)N(CCc3ccccn3)C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c12
Fc1cccc2C(=O)N(CCc3ccccn3)C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c12
CC1(N(CCc2ccccn2)C(=O)c2ccccc12)C(=O)NCc1ccc(OC(F)(F)F)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCc3cnccn3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCc3ncccn3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CC(F)(F)c3ccccn3)C(=O)c3ccccc23)cc1
CC(C)(Cc1ccccn1)N1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCOc3ccccn3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCCc3ccccn3)C(=O)c3ccccc23)cc1
Cc1cccc(CCN2C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c3ccccc3C2=O)n1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCC#N)C(=O)c3ccccc23)cc1
CC(CC#N)N1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O
FC(F)(F)CCN1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O
FC(F)(F)Oc1ccc(CNC(=O)C2N(C3CC(F)(F)C3)C(=O)c3ccccc23)cc1
CC(C)(C)OC(=O)N1CC(C1)N1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O
CC(C)(C)OC(=O)N1CCC(CC1)N1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O
FC(F)(F)Oc1ccc(CNC(=O)C2N([C@H]3CC[C@@H](CC3)C#N)C(=O)c3ccccc23)cc1 |r,wU:15.14,wD:18.21,(34.65,-34.73,;33.14,-35.05,;32.67,-36.52,;34.23,-36.13,;32.11,-33.91,;30.6,-34.23,;30.13,-35.7,;28.62,-36.02,;27.6,-34.87,;26.09,-35.19,;25.62,-36.66,;24.11,-36.98,;23.08,-35.83,;23.64,-38.44,;24.55,-39.7,;26.09,-39.69,;26.85,-38.36,;28.39,-38.36,;29.16,-39.7,;28.38,-41.03,;26.85,-41.03,;30.7,-39.7,;32.24,-39.71,;23.64,-40.95,;24.11,-42.41,;22.16,-40.47,;20.83,-41.24,;19.49,-40.47,;19.5,-38.93,;20.82,-38.16,;22.16,-38.92,;28.06,-33.41,;29.56,-33.09,)|
FC(F)(F)Oc1ccc(CNC(=O)C2N(C[C@@H]3CCCO3)C(=O)c3ccccc23)cc1 |r|
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCN3CCOCC3)C(=O)c3ccccc23)cc1
FC(F)(F)COc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cn1
FC(F)Oc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cn1
CC(NC(=O)C1N(CCc2ccccn2)C(=O)c2ccccc12)c1ccc(OCC(F)(F)F)cc1
FC(F)(F)COc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1cccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)c1
FC(F)(F)c1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cc1
Cc1ccc(NC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cc1C
Oc1cccc2C(N(CCc3ncc(F)cn3)C(=O)c12)C(=O)NCc1ccc(OC(F)(F)F)cc1
Fc1cnc(CCN2C(C(=O)NCc3ccc(F)c(OC(F)(F)F)c3)c3ccccc3C2=O)nc1
Oc1cccc2C(N(CCc3ccccn3)C(=O)c12)C(=O)NCc1ccc(OC(F)(F)F)cc1
COc1cccc2C(N(CCc3ccccn3)C(=O)c12)C(=O)NCc1ccc(OC(F)(F)F)cc1
Fc1cnc(CCN2C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c3ccccc3C2=O)nc1
CC(C)(CN1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O)c1ccccn1
CC(Cc1ccccn1)N1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O
FC(F)(F)Oc1ccc(CNC(=O)C2N(Cc3ccc(cn3)C(F)(F)F)C(=O)c3ccccc23)cc1
Fc1ccc(CCN2C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c3ccccc3C2=O)nc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCc3ccncc3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCc3cccnc3)C(=O)c3ccccc23)cc1
FC(F)(F)COCCN1C(C(=O)NCc2ccc(OC(F)(F)F)cc2)c2ccccc2C1=O
FC(F)(F)Oc1ccc(CNC(=O)C2N(CC3CC(F)(F)C3)C(=O)c3ccccc23)cc1
FC(F)(F)Oc1ccc(CNC(=O)C2N(CCC3CCOCC3)C(=O)c3ccccc23)cc1
FC(F)(F)CCOc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cn1
FC(F)(F)Cc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cc1
COc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cc1
Brc1ccccc1CNC(=O)C1N(CCc2ccccn2)C(=O)c2ccccc12
Brc1cccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)c1
Brc1ccc(CNC(=O)C2N(CCc3ccccn3)C(=O)c3ccccc23)cc1
Cc1onc(c1CC(=O)NCc1cccc(OCCOCC(F)(F)F)n1)-c1c(C)cccc1C |(5.05,-11.78,;3.92,-12.83,;2.41,-12.53,;1.67,-13.88,;2.72,-15.01,;4.12,-14.35,;5.46,-15.1,;6.78,-14.31,;6.76,-12.77,;8.13,-15.05,;9.45,-14.26,;10.8,-15.01,;12.1,-14.21,;13.45,-14.95,;13.48,-16.5,;12.16,-17.29,;12.17,-18.85,;13.52,-19.61,;14.84,-18.82,;16.18,-19.58,;17.51,-18.8,;18.85,-19.55,;20.18,-18.77,;18.87,-21.09,;20.18,-20.32,;10.81,-16.54,;2.42,-16.52,;3.59,-17.51,;5.04,-17,;3.3,-19.02,;1.84,-19.53,;.68,-18.52,;.97,-17.01,;-.19,-16,)|
Cc1onc(c1CC(=O)NCc1ccc(cc1)-n1cccn1)-c1c(Cl)cccc1Cl |(6.37,-16.57,;5.25,-17.62,;3.73,-17.32,;2.99,-18.67,;4.04,-19.8,;5.44,-19.14,;6.79,-19.89,;8.11,-19.1,;8.08,-17.56,;9.45,-19.84,;10.77,-19.05,;12.12,-19.8,;12.14,-21.34,;13.48,-22.08,;14.8,-21.29,;14.77,-19.74,;13.42,-19,;16.15,-22.03,;16.35,-23.56,;17.86,-23.85,;18.61,-22.5,;17.55,-21.38,;3.75,-21.31,;4.91,-22.3,;6.36,-21.79,;4.62,-23.81,;3.16,-24.32,;2,-23.31,;2.29,-21.8,;1.13,-20.79,)|
Cc1onc(c1CC(=O)NCc1ccc(OCC(F)(F)F)nc1)-c1c(Cl)cccc1Cl |(18.94,3.99,;18.04,2.74,;16.5,2.73,;16.03,1.27,;17.27,.36,;18.52,1.28,;19.98,.81,;21.3,1.6,;21.28,3.14,;22.65,.85,;23.97,1.65,;25.32,.9,;26.62,1.7,;27.97,.96,;28,-.59,;29.35,-1.34,;30.67,-.54,;32.02,-1.29,;32.05,-2.83,;33.34,-.49,;33.34,-2.05,;26.68,-1.38,;25.33,-.64,;17.28,-1.18,;15.95,-1.95,;14.62,-1.18,;15.95,-3.5,;17.28,-4.27,;18.62,-3.5,;18.61,-1.95,;19.94,-1.17,)|
CC(C)Oc1ccc(CNC(=O)Cc2c(C)onc2-c2c(Cl)cccc2Cl)cn1 |(9.43,-.5,;8.08,.24,;8.05,1.78,;6.76,-.55,;5.42,.19,;5.38,1.74,;4.04,2.48,;2.73,1.69,;1.38,2.43,;.06,1.64,;-1.28,2.38,;-1.31,3.92,;-2.6,1.59,;-4.07,2.06,;-4.55,3.52,;-3.65,4.77,;-6.09,3.52,;-6.56,2.05,;-5.31,1.14,;-5.31,-.4,;-6.64,-1.17,;-7.97,-.4,;-6.64,-2.71,;-5.3,-3.48,;-3.97,-2.71,;-3.97,-1.16,;-2.64,-.38,;2.75,.15,;4.09,-.6,)|
CC(C)Oc1ccc(CNC(=O)Nc2c(C)onc2-c2c(Cl)cncc2Cl)cn1 |(9.77,-47,;8.42,-46.25,;8.4,-44.71,;7.11,-47.05,;5.76,-46.3,;5.73,-44.75,;4.38,-44.01,;3.07,-44.81,;1.73,-44.06,;.41,-44.86,;-.94,-44.11,;-.97,-42.57,;-2.26,-44.9,;-3.73,-44.43,;-4.21,-42.97,;-3.31,-41.72,;-5.75,-42.98,;-6.22,-44.44,;-4.97,-45.35,;-4.97,-46.89,;-6.29,-47.66,;-7.63,-46.89,;-6.3,-49.21,;-4.96,-49.98,;-3.63,-49.21,;-3.63,-47.66,;-2.3,-46.88,;3.09,-46.35,;4.44,-47.09,)|
Cc1onc(c1NC(=O)NCc1ccc(cc1)-n1cccn1)-c1c(C)cccc1C |(18.44,-27.81,;17.54,-29.06,;16,-29.06,;15.53,-30.53,;16.78,-31.44,;18.02,-30.52,;19.49,-30.99,;20.81,-30.2,;20.78,-28.66,;22.15,-30.94,;23.47,-30.15,;24.82,-30.9,;24.84,-32.43,;26.18,-33.18,;27.5,-32.39,;27.47,-30.84,;26.13,-30.1,;28.85,-33.13,;29.05,-34.66,;30.56,-34.95,;31.31,-33.6,;30.26,-32.48,;16.78,-32.98,;15.45,-33.75,;14.12,-32.98,;15.45,-35.29,;16.78,-36.06,;18.12,-35.29,;18.12,-33.74,;19.45,-32.97,)|
CC(C)Oc1ccc(CNC(=O)Nc2c(C)onc2-c2c(C)cccc2C)cn1 |(32.67,-21.53,;31.32,-20.79,;31.28,-19.25,;30,-21.58,;28.66,-20.84,;28.62,-19.29,;27.28,-18.55,;25.97,-19.35,;24.62,-18.6,;23.3,-19.39,;21.96,-18.65,;21.93,-17.11,;20.64,-19.44,;19.17,-18.97,;18.69,-17.51,;19.59,-16.26,;17.15,-17.51,;16.68,-18.98,;17.93,-19.89,;17.93,-21.43,;16.6,-22.2,;15.27,-21.43,;16.6,-23.74,;17.94,-24.51,;19.27,-23.74,;19.27,-22.19,;20.6,-21.42,;25.99,-20.88,;27.33,-21.63,)|
CN(C(=O)NCc1ccc(OC2CCOCC2)nc1)c1c(C)onc1-c1c(C)cccc1C |(-1.81,-21.92,;-2.57,-20.59,;-1.25,-19.8,;-1.28,-18.26,;.1,-20.54,;1.42,-19.75,;2.76,-20.5,;4.07,-19.7,;5.41,-20.44,;5.45,-21.99,;6.79,-22.73,;8.11,-21.94,;9.46,-22.69,;10.77,-21.9,;10.75,-20.36,;9.4,-19.61,;8.08,-20.4,;4.12,-22.78,;2.78,-22.04,;-4.04,-20.12,;-4.52,-18.66,;-3.62,-17.41,;-6.06,-18.66,;-6.53,-20.13,;-5.28,-21.04,;-5.28,-22.58,;-6.61,-23.35,;-7.94,-22.58,;-6.61,-24.89,;-5.27,-25.66,;-3.94,-24.89,;-3.94,-23.34,;-2.61,-22.57,)|
CN(C(=O)NCc1ccc(OC2CCOCC2)nc1)c1c(C)onc1-c1ccccc1Cl
Cc1onc(c1NC(=O)NCc1c(F)cccc1Cl)-c1c(C)cccc1C |(12.41,5.36,;11.51,4.11,;9.97,4.1,;9.5,2.64,;10.75,1.73,;11.99,2.64,;13.46,2.17,;14.78,2.97,;14.75,4.51,;16.13,2.22,;17.45,3.02,;18.79,2.27,;18.81,.73,;17.49,-.06,;20.15,-.02,;21.48,.78,;21.44,2.33,;20.1,3.06,;20.06,4.6,;10.75,.19,;9.42,-.58,;8.09,.19,;9.42,-2.13,;10.76,-2.9,;12.09,-2.13,;12.09,-.58,;13.42,.2,)|
Cc1onc(c1NC(=O)OCc1c(F)cccc1Cl)-c1c(C)cccc1C |(33.16,-37.18,;32.26,-38.43,;30.72,-38.43,;30.24,-39.9,;31.49,-40.81,;32.74,-39.89,;34.2,-40.36,;35.52,-39.57,;35.49,-38.03,;36.87,-40.31,;38.19,-39.52,;39.54,-40.27,;39.55,-41.81,;38.23,-42.6,;40.9,-42.55,;42.22,-41.76,;42.19,-40.21,;40.84,-39.47,;40.81,-37.93,;31.5,-42.35,;30.17,-43.12,;28.83,-42.35,;30.17,-44.66,;31.5,-45.44,;32.84,-44.66,;32.83,-43.11,;34.16,-42.34,)|
Cc1onc(c1NC(=O)OCc1c(F)cccc1Cl)-c1c(F)cccc1Cl |(13.99,-37.25,;13.09,-38.5,;11.55,-38.5,;11.08,-39.97,;12.33,-40.88,;13.57,-39.96,;15.04,-40.43,;16.36,-39.64,;16.33,-38.1,;17.7,-40.38,;19.02,-39.59,;20.37,-40.34,;20.39,-41.88,;19.07,-42.67,;21.73,-42.62,;23.06,-41.83,;23.02,-40.28,;21.68,-39.54,;21.64,-38,;12.33,-42.42,;11,-43.19,;9.67,-42.42,;11,-44.73,;12.34,-45.51,;13.67,-44.73,;13.67,-43.18,;15,-42.41,)|
Fc1cccc(Cl)c1COC(=O)Nc1conc1-c1c(Cl)cccc1Cl |(-.29,-41.73,;1.04,-40.94,;2.38,-41.69,;3.7,-40.9,;3.67,-39.35,;2.33,-38.61,;2.29,-37.07,;1.02,-39.4,;-.33,-38.66,;-1.65,-39.45,;-2.99,-38.71,;-3.02,-37.17,;-4.31,-39.5,;-5.78,-39.03,;-6.26,-37.57,;-7.8,-37.57,;-8.27,-39.04,;-7.02,-39.95,;-7.02,-41.49,;-8.35,-42.26,;-9.68,-41.49,;-8.35,-43.8,;-7.02,-44.57,;-5.68,-43.8,;-5.68,-42.25,;-4.35,-41.47,)|
COCc1onc(c1NC(=O)OCc1ccccc1Cl)-c1c(Cl)cccc1Cl |(30.29,-24.05,;29.38,-25.3,;30.01,-26.7,;29.11,-27.95,;27.57,-27.96,;27.1,-29.42,;28.35,-30.33,;29.59,-29.42,;31.06,-29.89,;32.38,-29.09,;32.35,-27.55,;33.73,-29.84,;35.05,-29.04,;36.39,-29.79,;36.41,-31.33,;37.76,-32.08,;39.08,-31.28,;39.05,-29.73,;37.7,-29,;37.66,-27.46,;28.35,-31.87,;27.03,-32.64,;25.69,-31.87,;27.02,-34.19,;28.36,-34.96,;29.69,-34.19,;29.69,-32.64,;31.02,-31.86,)|
CN(C(=O)OCc1c(F)cccc1Cl)c1c(C)onc1-c1c(Cl)cccc1Cl |(-4.22,-30.23,;-4.98,-28.91,;-3.66,-28.11,;-3.69,-26.57,;-2.32,-28.86,;-1,-28.06,;.35,-28.81,;.37,-30.35,;-.95,-31.14,;1.71,-31.1,;3.04,-30.3,;3,-28.75,;1.66,-28.02,;1.62,-26.48,;-6.45,-28.44,;-6.93,-26.97,;-6.03,-25.72,;-8.47,-26.98,;-8.94,-28.44,;-7.69,-29.35,;-7.69,-30.89,;-9.02,-31.66,;-10.35,-30.89,;-9.02,-33.21,;-7.68,-33.98,;-6.35,-33.21,;-6.35,-31.66,;-5.02,-30.88,)|
CC(C)Oc1ccc(COC(=O)N(C)c2c(C)onc2-c2c(Cl)cccc2Cl)cn1 |(48.65,-19.56,;47.31,-18.81,;47.28,-17.27,;45.99,-19.61,;44.64,-18.86,;44.61,-17.31,;43.26,-16.57,;41.95,-17.37,;40.61,-16.62,;39.29,-17.42,;37.94,-16.67,;37.91,-15.13,;36.62,-17.46,;37.38,-18.79,;35.15,-16.99,;34.67,-15.53,;35.58,-14.28,;33.13,-15.54,;32.66,-17,;33.91,-17.91,;33.92,-19.45,;32.59,-20.22,;31.25,-19.45,;32.58,-21.77,;33.92,-22.54,;35.26,-21.77,;35.25,-20.22,;36.58,-19.44,;41.97,-18.91,;43.32,-19.65,)|
Cc1onc(c1NC(=O)OCc1ccc(OC2CCCC2)nc1)-c1c(Cl)cccc1Cl |(15.59,-15.68,;14.69,-16.93,;13.15,-16.94,;12.67,-18.4,;13.92,-19.31,;15.17,-18.39,;16.63,-18.86,;17.95,-18.07,;17.92,-16.53,;19.3,-18.82,;20.62,-18.02,;21.97,-18.77,;23.27,-17.97,;24.62,-18.71,;24.65,-20.26,;26,-21.01,;27.32,-20.21,;28.78,-20.7,;29.69,-19.46,;28.8,-18.2,;27.33,-18.67,;23.33,-21.05,;21.98,-20.31,;13.93,-20.85,;12.6,-21.62,;11.26,-20.85,;12.6,-23.17,;13.93,-23.94,;15.27,-23.17,;15.26,-21.62,;16.59,-20.84,)|
CC(C)Oc1ccc(COC(=O)Nc2c(C)onc2-c2c(Cl)cccc2Cl)cn1 |(7.49,-20.61,;6.15,-19.87,;6.12,-18.33,;4.83,-20.66,;3.48,-19.92,;3.45,-18.37,;2.1,-17.63,;.79,-18.43,;-.55,-17.68,;-1.87,-18.47,;-3.22,-17.73,;-3.25,-16.19,;-4.54,-18.52,;-6.01,-18.05,;-6.49,-16.59,;-5.58,-15.34,;-8.03,-16.59,;-8.5,-18.06,;-7.25,-18.97,;-7.24,-20.51,;-8.57,-21.28,;-9.91,-20.51,;-8.58,-22.82,;-7.24,-23.6,;-5.9,-22.82,;-5.91,-21.27,;-4.58,-20.5,;.81,-19.97,;2.16,-20.71,)|
Cc1onc(c1NC(=O)OCc1cc(Cl)ccc1Cl)-c1c(Cl)cccc1Cl |(-5.13,-5.07,;-6.03,-6.32,;-7.57,-6.33,;-8.04,-7.79,;-6.79,-8.7,;-5.55,-7.79,;-4.08,-8.26,;-2.76,-7.46,;-2.79,-5.92,;-1.41,-8.21,;-.09,-7.41,;1.25,-8.16,;1.27,-9.7,;2.62,-10.45,;2.64,-11.99,;3.94,-9.65,;3.91,-8.1,;2.56,-7.37,;2.52,-5.83,;-6.79,-10.24,;-8.11,-11.01,;-9.45,-10.24,;-8.12,-12.56,;-6.78,-13.33,;-5.45,-12.56,;-5.45,-11.01,;-4.12,-10.23,)|
Cc1onc(c1NC(=O)OCc1ccccc1Cl)-c1c(Cl)cccc1Cl |(15.73,5.12,;14.83,3.87,;13.29,3.87,;12.82,2.4,;14.07,1.49,;15.31,2.41,;16.78,1.94,;18.1,2.73,;18.07,4.27,;19.45,1.99,;20.77,2.78,;22.11,2.04,;22.13,.5,;23.48,-.25,;24.8,.54,;24.77,2.09,;23.42,2.83,;23.38,4.37,;14.07,-.05,;12.75,-.82,;11.41,-.05,;12.74,-2.36,;14.08,-3.13,;15.41,-2.36,;15.41,-.81,;16.74,-.03,)|
Cc1onc(c1NC(=O)OCc1c(F)cccc1Cl)-c1c(Cl)cccc1Cl |(-4.41,5.18,;-5.31,3.94,;-6.85,3.93,;-7.32,2.47,;-6.08,1.56,;-4.83,2.47,;-3.36,2,;-2.04,2.8,;-2.07,4.34,;-.7,2.05,;.62,2.84,;1.97,2.1,;1.99,.56,;.66,-.23,;3.33,-.19,;4.65,.61,;4.62,2.15,;3.27,2.89,;3.24,4.43,;-6.07,.02,;-7.4,-.75,;-8.73,.02,;-7.4,-2.3,;-6.07,-3.07,;-4.73,-2.3,;-4.74,-.75,;-3.4,.03,)|
CN(C(=O)NCc1ccc(OC2CCOCC2)nc1)c1c(C)onc1-c1c(Cl)cccc1Cl |(-2.67,-10.41,;-3.43,-9.09,;-2.11,-8.29,;-2.13,-6.75,;-.76,-9.04,;.56,-8.25,;1.91,-8.99,;3.21,-8.2,;4.56,-8.94,;4.59,-10.48,;5.94,-11.23,;7.26,-10.43,;8.6,-11.18,;9.92,-10.39,;9.89,-8.85,;8.55,-8.1,;7.22,-8.9,;3.27,-11.28,;1.92,-10.53,;-4.89,-8.62,;-5.37,-7.15,;-4.47,-5.91,;-6.91,-7.16,;-7.39,-8.63,;-6.14,-9.53,;-6.13,-11.07,;-7.46,-11.85,;-8.8,-11.08,;-7.46,-13.39,;-6.13,-14.16,;-4.79,-13.39,;-4.8,-11.84,;-3.47,-11.06,)|
Cc1onc(c1CC(=O)NCc1ccc(OCC(F)(F)F)nc1)-c1c(C)cccc1C |(6.37,-16.57,;5.25,-17.62,;3.73,-17.32,;2.99,-18.67,;4.04,-19.8,;5.44,-19.14,;6.79,-19.89,;8.11,-19.1,;8.08,-17.56,;9.45,-19.84,;10.77,-19.05,;12.12,-19.8,;13.42,-19,;14.77,-19.74,;14.8,-21.29,;16.15,-22.03,;16.18,-23.57,;17.53,-24.32,;17.56,-25.86,;18.85,-23.52,;18.85,-25.08,;13.48,-22.08,;12.14,-21.34,;3.75,-21.31,;4.91,-22.3,;6.36,-21.79,;4.62,-23.81,;3.16,-24.32,;2,-23.31,;2.29,-21.8,;1.13,-20.79,)|
Cc1onc(c1NC(=O)NCc1ccc(cc1)-n1cccn1)-c1c(Cl)cccc1Cl |(-3.96,-28.77,;-4.86,-30.01,;-6.4,-30.02,;-6.87,-31.48,;-5.62,-32.39,;-4.38,-31.48,;-2.91,-31.95,;-1.59,-31.15,;-1.62,-29.61,;-.25,-31.9,;1.07,-31.11,;2.42,-31.85,;2.44,-33.39,;3.78,-34.14,;5.1,-33.34,;5.07,-31.8,;3.73,-31.06,;6.45,-34.09,;6.65,-35.62,;8.16,-35.91,;8.91,-34.56,;7.86,-33.43,;-5.62,-33.93,;-6.95,-34.7,;-8.28,-33.93,;-6.95,-36.25,;-5.62,-37.02,;-4.28,-36.25,;-4.28,-34.7,;-2.95,-33.92,)|
Cc1onc(c1NC(=O)NCc1c(F)cccc1Cl)-c1c(Cl)cccc1Cl |(-5.13,4.9,;-6.03,3.65,;-7.57,3.64,;-8.04,2.18,;-6.79,1.27,;-5.55,2.19,;-4.08,1.72,;-2.76,2.51,;-2.79,4.05,;-1.41,1.76,;-.09,2.56,;1.25,1.81,;1.27,.27,;-.05,-.52,;2.62,-.47,;3.94,.32,;3.91,1.87,;2.56,2.61,;2.52,4.15,;-6.79,-.27,;-8.11,-1.04,;-9.45,-.27,;-8.12,-2.59,;-6.78,-3.36,;-5.45,-2.59,;-5.45,-1.04,;-4.12,-.26,)|
CCc1onc(c1NC(=O)OCc1c(F)cccc1Cl)-c1c(Cl)cccc1Cl |(12.19,-25.21,;12.82,-26.62,;11.92,-27.87,;10.38,-27.87,;9.9,-29.34,;11.15,-30.25,;12.4,-29.33,;13.86,-29.8,;15.18,-29.01,;15.16,-27.47,;16.53,-29.75,;17.85,-28.96,;19.2,-29.71,;19.21,-31.24,;17.89,-32.03,;20.56,-31.99,;21.88,-31.2,;21.85,-29.65,;20.5,-28.91,;20.47,-27.37,;11.16,-31.79,;9.83,-32.56,;8.49,-31.79,;9.83,-34.1,;11.16,-34.87,;12.5,-34.1,;12.49,-32.55,;13.82,-31.78,)|
CN(C)c1cccc(COC(=O)Nc2c(C)onc2-c2c(Cl)cccc2Cl)c1 |(27.14,-8,;25.79,-7.26,;25.76,-5.72,;24.48,-8.06,;24.51,-9.61,;23.19,-10.4,;21.84,-9.65,;21.83,-8.11,;20.48,-7.37,;19.16,-8.16,;17.81,-7.42,;17.78,-5.88,;16.49,-8.21,;15.03,-7.74,;14.55,-6.28,;15.45,-5.03,;13.01,-6.28,;12.53,-7.75,;13.78,-8.66,;13.79,-10.2,;12.46,-10.97,;11.12,-10.2,;12.46,-12.51,;13.79,-13.28,;15.13,-12.51,;15.12,-10.96,;16.45,-10.18,;23.13,-7.32,)|
NC(=O)C(c1ccccc1)(c1ccc(F)cc1)c1ccc(F)cc1
CC(C)(C)C(=O)ON[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCc2ccccc2N(CC(F)(F)F)C1=O |r|
FC(F)(F)Oc1cccc(c1)C(=O)NCc1noc(n1)-c1n(CCn2ccnc2)nc2ccccc12
O=C(NCc1noc(n1)-c1nn(CCn2ccnc2)c2ccccc12)c1ccccc1
Fc1ccc(cc1)[C@@H]1CC(=O)NC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
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[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](C)NC(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](C)NC(=O)[C@]1([H])CSSC[C@]3([H])NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@]4([H])CCCN4C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]([H])(CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc4ccccc4)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N1)NC(=O)[C@]([H])(CSSC[C@H](NC(=O)[C@H](Cc1c[nH]c4ccccc14)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@]([H])(NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC3=O)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC2=O)C(C)C |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
CN1CCN(c2ccc(cc2)C(F)(F)F)c2ccc(cc2C1)-c1cccc(n1)C(N)=O
CC(=O)N1CCN(c2ccc(cc2)C(F)(F)F)c2ccc(cc2C1)-c1cccc(n1)C(N)=O
NC(=O)CN1CCN(c2ccc(cc2)C(F)(F)F)c2ccc(cc2C1)-c1cccc(n1)[C@H](O)CO |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2N(CCN(CC3CC3)Cc2c1)c1ccc(cc1)C(F)(F)F |r|
NC(=O)N1CCN(c2ccc(cc2)C(F)(F)F)c2ccc(cc2C1)-c1cccc(n1)[C@H](O)CO |r|
CC(=O)N1CCN(c2ccc(cc2)C(F)(F)F)c2ccc(cc2C1)-c1cccc(n1)[C@H](O)CO |r|
CS(=O)(=O)N1CCN(c2ccc(cc2)C(F)(F)F)c2ccc(cc2C1)-c1cccc(n1)[C@H](O)CO |r|
CNC(=O)CN1CCN(c2ccc(cc2)C(F)(F)F)c2ccc(cc2C1)-c1cccc(n1)[C@H](O)CO |r|
NC(=O)c1cccc(n1)-c1ccc2N(CCNCc2c1)c1ccc(cc1)C(F)(F)F
OC[C@@H](O)c1cccc(n1)-c1ccc2N(CCN(Cc3ncc[nH]3)Cc2c1)c1ccc(cc1)C(F)(F)F |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2N(CCN(CC#N)Cc2c1)c1ccc(cc1)C(F)(F)F |r|
NC(=O)c1cccc(n1)-c1ccc2N(CCOCc2c1)c1ccc(cc1)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc2N(CCCOc2c1)c1ccc(cc1)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc2N(CCCCc2c1)c1ccc(cc1)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc2N(CCCc2c1)c1ccc(cc1)C(F)(F)F
NC(=O)c1cccc(n1)-c1ccc2N(CCc2c1)c1ccc(cc1)C(F)(F)F
CN1Cc2cc(ccc2Oc2ccc(cc12)-c1cccc(n1)[C@H](O)CO)C(F)(F)F |r|
CN1Cc2cc(ccc2Oc2ccc(cc12)C(F)(F)F)-c1cccc(n1)[C@H](O)CO |r|
CN1c2ccc(cc2CCc2cc(ccc12)C(F)(F)F)-c1cccc(n1)[C@H](O)CO |r|
CC(=O)N1c2ccc(Cl)cc2CCc2cc(ccc12)-c1cccc(n1)C(N)=O
NC(=O)c1cccc(n1)-c1ccc2Nc3ccc(Cl)cc3CCc2c1
CN1Cc2cc(ccc2Oc2ccc(cc12)C(F)(F)F)-c1cccc(n1)[C@H](O)[C@@H](O)C(N)=O |r|
NC(=O)CN1Cc2cc(ccc2Oc2ccc(cc12)C(F)(F)F)-c1cccc(n1)[C@H](O)CO |r|
OC[C@@H](O)c1cccc(n1)-c1ccc2Oc3ccc(cc3NCc2c1)C(F)(F)F |r|
CCN1c2ccc(Cl)cc2CCc2cc(ccc12)-c1cccc(n1)C(N)=O
CN1c2ccc(Cl)cc2CCc2cc(ccc12)-c1cccc(n1)C(N)=O
CNC(=O)c1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
COc1ccc(Cl)c(c1)-c1ccc(NC(=O)c2ccnn2C)nc1N
Cc1nocc1C(=O)Nc1ccc(c(N)n1)-c1ccccc1OC(F)(F)F
CNC(=O)c1cnc(N)c(c1)-c1cc(Cl)cc(Cl)c1Cl
CC(=O)Nc1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
Nc1nnc(c(N)n1)-c1cccc(Cl)c1Cl
COc1ccc(cc1N(C)C)C(=O)N1CCC2(CC1)Nc1cc(OC(F)(F)F)ccc1-n1cccc21
COc1ccc(cc1N(C)C)C(=O)N1CCC2(CC1)Nc1cc(OC(F)F)ccc1-n1cccc21
COc1ccc(cc1N(C)C)C(=O)N1CCC2(CC1)Nc1cc(ccc1-n1cccc21)C(F)(F)F
COCCOc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc(OC)c(c3)N(C)C)c3cccn-23)c1
COc1cc2NC3(CCN(CC3)C(=O)c3ccc(OC)c(c3)N(C)C)c3cccn3-c2cc1F
COc1ccc-2c(N[C@@]3(CCN(C[C@@H]3C)C(=O)c3ccc(OC)c(c3)N(C)C)c3cccn-23)c1 |r|
COc1ccc-2c(NC3(CN(C3)C(=O)c3ccc4ncccc4c3)c3cccn-23)c1
COc1ccc-2c(NC3(CCCN(CC3)C(=O)c3ccc(OC)c(c3)N(C)C)c3cccn-23)c1
COc1ccc-2c(NC3(CC4CN(CC4C3)C(=O)c3ccc(OC)c(c3)N(C)C)c3cccn-23)c1
COc1ccc-2c(NC3(CCC(CC3)NC(=O)c3ccc(OC)c(c3)N(C)C)c3cccn-23)c1 |(2.7,-10.77,;4.03,-9.99,;5.36,-10.76,;5.36,-12.31,;6.7,-13.08,;8.03,-12.3,;8.03,-10.76,;9.36,-9.98,;10.7,-10.76,;12.03,-11.53,;13.36,-10.76,;13.36,-9.23,;12.03,-8.46,;10.7,-9.22,;14.7,-8.46,;14.7,-6.92,;13.37,-6.15,;16.04,-6.16,;16.04,-4.62,;17.37,-3.85,;18.71,-4.63,;20.04,-3.86,;21.37,-4.63,;18.7,-6.17,;17.37,-6.93,;20.03,-6.94,;20.03,-8.48,;21.37,-6.18,;10.7,-12.31,;11.84,-13.35,;11.21,-14.76,;9.67,-14.59,;9.36,-13.08,;6.69,-9.99,)|
COc1ccc-2c(N[C@]3(CCN([C@H](C)C3)C(=O)c3ccc(OC)c(c3)N(C)C)c3cccn-23)c1 |r|
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc(OC)c(c3)N3CCCC3)c3cccn-23)c1
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc4OCCN(C)c4c3)c3cccn-23)c1
CCCCc1nc2cc(ccc2o1)C(=O)N1CCC2(CC1)Nc1cc(OC)ccc1-n1cccc21
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc4ncccc4c3)c3cccn-23)c1
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3cccc4ncccc34)c3cccn-23)c1
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc4ccccc4n3)c3cccn-23)c1
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc4cccnc4c3)c3cccn-23)c1
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc4n(C)ccc4c3)c3cccn-23)c1
COc1ccc-2c(NC3(CCN(CC3)C(=O)c3ccc4n(C)ncc4c3)c3cccn-23)c1
CC(C)COc1ccc(C)cc1-c1cccc([C@@H]2CC[C@]3(CCN(C)C3=O)N2)c1F |r|
CN1CC[C@]2(CC[C@H](N2)c2nc(C)cc(n2)-c2ccc(cc2)C(F)(F)F)C1=O |r|
CN1CC[C@]2(CC[C@H](N2)c2cc(ccn2)-c2cccc(OC(F)(F)F)c2)C1=O |r|
FC(F)C(F)(F)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N2CCC2)cc1Cl
CCCOc1ncccc1-c1cc(ccc1Oc1ccc(Cl)cc1)C(=O)NS(C)(=O)=O
Fc1cc(Oc2ccc(cc2-c2ccnn2C2CNC2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1nncs1
Fc1cc(ccc1Cl)[C@@H]1CCNC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1 |r|
c1ccc(cc1)C(c2ccccc2)C(=O)Nc3ccc(cc3)S(=O)(=O)Nc4nccs4
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CS)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC(=O)[C@H](CS)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CS)NC(=O)[C@H](CS)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(N)=O)NC(=O)[C@H](CS)NC(=O)CNC(=O)[C@H](CCCCN)NC(=O)CNC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CS)NC(=O)[C@@H](N)CCC(O)=O)C(C)C)C(N)=O |r|
[H][C@@]12CSSC[C@]3([H])NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC(=O)[C@H](Cc4cnc[nH]4)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]([H])(CSSC[C@H](N)C(=O)N1)NC(=O)[C@H](Cc1c[nH]c4ccccc14)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@]([H])(CSSC[C@H](NC3=O)C(O)=O)NC(=O)[C@H](CC(N)=O)NC2=O |r|
COc1cc(ccc1COCC(O)CN1CCC(CC1)C(=O)Nc1ccccc1)C(F)(F)F
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)C(=O)Nc1ccccc1
OC(COc1cccc(c1)C(=O)c1ccccc1)CN1CCC(CC1)N1Cc2ccccc2C1=O
OC(COc1ccc(cc1)C(=O)c1ccccc1)CN1CCC(CC1)N1Cc2ccccc2C1=O
OC(COc1ccccc1)CN1CCC(CC1)N1Cc2ccccc2C1=O
COc1ccccc1OCC(O)CN1CCC(CC1)N1Cc2ccccc2C1=O
COc1cccc(OCC(O)CN2CCC(CC2)N2Cc3ccccc3C2=O)c1
COc1ccc(OCC(O)CN2CCC(CC2)N2Cc3ccccc3C2=O)cc1
OC(COc1ccccc1C(F)(F)F)CN1CCC(CC1)N1Cc2ccccc2C1=O
OC(COc1cccc(c1)C(F)(F)F)CN1CCC(CC1)N1Cc2ccccc2C1=O
OC(COc1ccc(cc1)C(F)(F)F)CN1CCC(CC1)N1Cc2ccccc2C1=O
COc1cc(ccc1OCC(O)CN1CCC(CC1)N1Cc2ccccc2C1=O)C(F)(F)F
OC(COCc1ccc(cc1)C(F)(F)F)CN1CCC(CC1)N1Cc2ccccc2C1=O
COc1cc(ccc1COCC(O)CN1CCC(CC1)N1Cc2ccccc2C1=O)C(F)(F)F
OC(COc1ccc(cc1)C(F)(F)F)CN1CCC(CC1)NC(=O)c1ccccc1
OC(COc1ccc(cc1)C(F)(F)F)CN1CCC(CC1)C(=O)Nc1ccccc1
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCN(CC1)c1cccc2NC(=O)COc12
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)c1cccc2NC(=O)COc12
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCN(CC1)c1cccc2NC(=O)CCc12
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)c1cccc2NC(=O)CCc12
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCN(CC1)c1cccc2[nH]c(=O)oc12
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)N1C(=O)COc2ccccc12
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)n1c2ccccc2oc1=O
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)N1C(=O)Cc2ccccc12
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)N1Cc2ccccc2C1=O
OC(COc1ccccc1C(=O)c1ccccc1)CN1CCC(CC1)NC(=O)c1ccccc1
Clc1cc(cnc1OCC1CCCC1)N1C(=O)C2(CC2)c2cc3c(NS(=O)(=O)C4CC4)noc3cc12
CC(C)COc1ncc(cc1Cl)N1C(=O)C2(CC2)c2cc3c(NS(C)(=O)=O)noc3cc12
CC1(COc2ncc(cc2Cl)N2C(=O)C3(CC3)c3cc4c(NS(=O)(=O)C5CC5)noc4cc23)CC1
CC(C)COc1ncc(cc1Cl)-c1cccc2cc3c(NS(=O)(=O)C4CC4)noc3cc12
CC(C)COc1ncc(cc1Cl)-c1cncc2cc3c(NS(C)(=O)=O)noc3cc12
CC(C)COc1ncc(cc1Cl)-c1nn(C)c2cc3c(NS(=O)(=O)C4CC4)noc3cc12
FC(F)(F)c1ccc(O[C@@H]2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C1=CCNCC1 |r,t:34|
CC[C@@H]1C[C@@H](Oc2ccc(cc2-c2ccnn2C)C(F)(F)F)c2ccc(cc2O1)S(=O)(=O)Nc1nccs1 |r|
Fc1ccc(nc1)-c1cc(ccc1O[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Cn1nccc1-c1cc(ccc1O[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F |r|
Cn1nccc1-c1cc(ccc1C1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(C2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C1(F)CNC1
FC(F)(F)c1ccc(C2CCOc3cc(ccc23)S(=O)(=O)Nc2nncs2)c(c1)C1=CCNCC1 |t:33|
FC(F)(F)c1ccc(C2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(c1)C1=CCNCC1 |t:33|
FC(F)(F)c1ccc(C2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C1=CCNCC1 |t:33|
FC(F)(F)c1ccc(C2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(Cl)c1
FC(F)(F)c1ccc(C2CCOc3cc(ccc23)S(=O)(=O)Nc2ncns2)c(Cl)c1
CC1(C)CC(c2ccc(cc2O1)S(=O)(=O)Nc1nccs1)c1ccc(cc1C1(F)CNC1)C(F)(F)F
CC1(C)CC(c2ccc(cc2O1)S(=O)(=O)Nc1ncns1)c1ccc(cc1C1=CCNCC1)C(F)(F)F |t:31|
CC1(C)CC(c2ccc(cc2O1)S(=O)(=O)Nc1nccs1)c1ccc(cc1C1=CCNCC1)C(F)(F)F |t:31|
[H][C@@]12CCCN1C(=O)[C@@]([H])(NC(=O)[C@]1([H])CSSC[C@]3([H])NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]([H])(CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc4ccccc4)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N1)NC(=O)[C@]([H])(CSSC[C@H](NC(=O)[C@H](Cc1c[nH]c4ccccc14)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@]([H])(NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC3=O)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC2=O)C(C)C)[C@@H](C)CC |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCCCN)C(N)=O |r|
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCCN)C(N)=O |r|
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[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@H](Cc2ccccc2)NC3=O)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
Nc1noc2ccc(CCOc3cc(F)c(cc3F)S(=O)(=O)Nc3ncns3)cc12
Nc1noc2ccc(cc12)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)NCc1ncccn1
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1cscn1)C(F)(F)F
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1cncs1)C(F)(F)F
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ccccn1)C(F)(F)F
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F
FC(F)(F)c1ccc(c(c1)C1=CCNCC1)-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1 |t:11|
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncccn1)C(F)(F)F
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cccc(OC(F)(F)F)c1 |(30.59,-17,;30.6,-15.46,;31.94,-14.69,;33.27,-15.45,;34.61,-14.68,;34.6,-13.13,;35.93,-12.34,;33.26,-12.37,;31.94,-13.15,;30.6,-12.38,;30.59,-10.85,;31.92,-10.09,;31.92,-8.55,;30.59,-7.77,;29.25,-8.55,;29.25,-10.09,;27.93,-10.86,;27.93,-12.39,;29.27,-13.15,;29.27,-14.7,;30.58,-6.22,;29.04,-6.22,;29.81,-4.89,;31.92,-5.45,;31.92,-3.91,;30.6,-3.14,;30.59,-1.6,;31.94,-.83,;33.27,-1.6,;33.27,-3.14,;35.94,-15.43,;35.95,-16.98,;37.29,-17.74,;38.62,-16.96,;38.61,-15.41,;39.93,-14.63,;39.92,-13.09,;39.9,-11.68,;41.15,-12.05,;38.65,-12.07,;37.27,-14.66,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(cnc1OC)C(F)(F)F |(16.14,-22.44,;16.15,-20.9,;17.49,-20.13,;18.82,-20.89,;20.17,-20.12,;20.15,-18.57,;21.48,-17.78,;18.81,-17.81,;17.49,-18.59,;16.15,-17.82,;16.14,-16.29,;17.47,-15.53,;17.47,-13.99,;16.14,-13.21,;14.81,-13.99,;14.81,-15.53,;13.49,-16.3,;13.49,-17.83,;14.82,-18.6,;14.82,-20.14,;16.13,-11.66,;15.37,-10.32,;14.59,-11.66,;17.47,-10.9,;17.48,-9.35,;16.23,-8.44,;16.71,-6.98,;18.25,-6.98,;18.73,-8.45,;21.5,-20.88,;22.83,-20.1,;24.17,-20.85,;24.18,-22.41,;22.85,-23.19,;21.51,-22.42,;20.18,-23.19,;18.85,-22.43,;25.49,-20.07,;26.69,-19.36,;26.99,-20.62,;25.73,-18.48,)|
COc1cc(ccc1C)-c1cc(OC)c(cc1F)-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(25.5,-13.09,;25.51,-14.64,;24.19,-15.42,;22.85,-14.66,;21.53,-15.44,;21.54,-16.98,;22.87,-17.74,;24.21,-16.97,;25.55,-17.73,;20.19,-14.68,;18.86,-15.46,;17.52,-14.69,;16.19,-15.46,;16.18,-17,;17.53,-13.15,;18.85,-12.37,;20.18,-13.13,;21.51,-12.35,;16.19,-12.39,;16.18,-10.86,;17.51,-10.1,;17.51,-8.56,;16.18,-7.78,;14.85,-8.56,;14.85,-10.1,;13.53,-10.86,;13.53,-12.4,;14.86,-13.16,;14.86,-14.7,;16.17,-6.24,;14.63,-6.23,;15.4,-4.9,;17.51,-5.46,;17.51,-3.92,;16.26,-3.01,;16.74,-1.55,;18.28,-1.55,;18.75,-3.02,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(F)c(F)c1 |(31.76,-38.71,;31.77,-37.17,;33.1,-36.4,;34.44,-37.16,;35.77,-36.39,;35.76,-34.84,;37.09,-34.06,;34.42,-34.08,;33.1,-34.86,;31.77,-34.09,;31.75,-32.57,;33.08,-31.8,;33.08,-30.26,;31.75,-29.48,;30.42,-30.26,;30.42,-31.8,;29.11,-32.57,;29.11,-34.1,;30.44,-34.86,;30.44,-36.41,;31.75,-27.94,;30.21,-27.93,;30.98,-26.6,;33.09,-27.17,;33.09,-25.63,;31.76,-24.86,;31.76,-23.32,;33.1,-22.55,;34.44,-23.32,;34.43,-24.86,;37.11,-37.14,;37.11,-38.69,;38.45,-39.45,;39.79,-38.67,;41.13,-39.43,;39.77,-37.12,;41.1,-36.34,;38.43,-36.37,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(Cl)c(c1)C#N |(16.12,-22.75,;16.13,-21.21,;17.46,-20.44,;18.8,-21.2,;20.14,-20.43,;20.12,-18.88,;21.45,-18.1,;18.78,-18.12,;17.46,-18.91,;16.13,-18.14,;16.12,-16.61,;17.44,-15.85,;17.44,-14.31,;16.12,-13.53,;14.79,-14.31,;14.79,-15.85,;13.47,-16.61,;13.47,-18.14,;14.8,-18.91,;14.8,-20.45,;16.11,-11.99,;15.35,-10.65,;14.57,-11.98,;17.45,-11.22,;17.45,-9.68,;16.2,-8.77,;16.69,-7.31,;18.23,-7.31,;18.7,-8.78,;21.47,-21.18,;21.48,-22.73,;22.81,-23.49,;24.14,-22.71,;25.47,-23.47,;24.13,-21.16,;22.79,-20.41,;25.44,-20.38,;26.76,-19.61,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1cc(Cl)cc(OC(F)(F)F)c1 |(5.02,-34.69,;5.04,-33.16,;6.37,-32.38,;7.71,-33.15,;9.04,-32.37,;9.03,-30.82,;10.36,-30.04,;7.69,-30.06,;6.37,-30.84,;5.03,-30.08,;5.02,-28.55,;6.35,-27.79,;6.35,-26.25,;5.02,-25.47,;3.69,-26.25,;3.69,-27.79,;2.37,-28.55,;2.37,-30.09,;3.7,-30.85,;3.71,-32.39,;5.01,-23.93,;3.47,-23.92,;4.25,-22.59,;6.36,-23.15,;6.36,-21.61,;5.03,-20.85,;5.03,-19.31,;6.37,-18.53,;7.7,-19.31,;7.7,-20.85,;10.38,-33.13,;11.7,-32.35,;13.04,-33.11,;14.37,-32.32,;13.05,-34.66,;11.72,-35.44,;11.73,-36.98,;10.4,-37.75,;9.18,-38.46,;8.88,-37.19,;10.14,-39.34,;10.38,-34.67,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cc(F)cc(Cl)c1 |(19.99,-18.29,;20,-16.75,;21.33,-15.98,;22.67,-16.74,;24,-15.97,;23.99,-14.42,;25.32,-13.64,;22.65,-13.66,;21.33,-14.44,;20,-13.67,;19.98,-12.15,;21.32,-11.38,;21.32,-9.84,;19.98,-9.06,;18.65,-9.84,;18.65,-11.38,;17.34,-12.15,;17.34,-13.68,;18.67,-14.44,;18.67,-15.99,;19.98,-7.52,;18.44,-7.51,;19.21,-6.18,;21.32,-6.75,;21.32,-5.21,;20.07,-4.3,;20.55,-2.84,;22.09,-2.84,;22.57,-4.31,;25.34,-16.72,;25.35,-18.27,;26.68,-19.03,;26.69,-20.57,;28.02,-18.25,;28,-16.7,;29.33,-15.92,;26.66,-15.95,)|
COc1cc(Cl)cc(c1)-c1cc(OC)c(cc1F)-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(23.71,-39.73,;25.04,-38.95,;25.03,-37.41,;26.36,-36.63,;26.35,-35.08,;27.68,-34.3,;25.01,-34.33,;23.69,-35.1,;23.69,-36.65,;22.35,-34.35,;21.02,-35.12,;19.68,-34.36,;18.35,-35.13,;18.33,-36.67,;19.68,-32.82,;21,-32.04,;22.34,-32.8,;23.67,-32.02,;18.34,-32.05,;18.33,-30.53,;19.66,-29.76,;19.66,-28.22,;18.33,-27.44,;17,-28.22,;17,-29.76,;15.68,-30.53,;15.68,-32.06,;17.01,-32.82,;17.02,-34.37,;18.33,-25.9,;16.78,-25.89,;17.56,-24.56,;19.67,-25.13,;19.67,-23.59,;18.42,-22.68,;18.9,-21.22,;20.44,-21.22,;20.91,-22.69,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(F)c(c1)C(F)(F)F |(48.06,-16.66,;48.07,-15.12,;49.4,-14.35,;50.74,-15.11,;52.07,-14.34,;52.06,-12.79,;53.39,-12.01,;50.72,-12.03,;49.41,-12.81,;48.07,-12.05,;48.06,-10.52,;49.39,-9.75,;49.39,-8.21,;48.06,-7.43,;46.72,-8.21,;46.72,-9.75,;45.41,-10.52,;45.41,-12.05,;46.74,-12.82,;46.74,-14.36,;48.05,-5.89,;46.51,-5.89,;47.28,-4.55,;49.39,-5.12,;49.39,-3.58,;48.06,-2.81,;48.06,-1.28,;49.4,-.5,;50.74,-1.28,;50.73,-2.82,;53.41,-15.09,;53.42,-16.64,;54.75,-17.4,;56.09,-16.62,;57.43,-17.38,;56.07,-15.07,;54.73,-14.32,;57.4,-14.29,;58.61,-13.57,;58.91,-14.84,;57.65,-12.69,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1cccnn1)-c1ccc(Cl)c(C)c1 |(44.6,-39.11,;44.62,-37.57,;45.95,-36.8,;47.29,-37.56,;48.62,-36.79,;48.61,-35.24,;49.94,-34.45,;47.27,-34.48,;45.95,-35.26,;44.62,-34.49,;44.6,-32.96,;45.93,-32.2,;45.93,-30.66,;44.6,-29.88,;43.27,-30.66,;43.27,-32.2,;41.95,-32.97,;41.95,-34.5,;43.29,-35.26,;43.29,-36.81,;44.6,-28.34,;43.06,-28.33,;43.83,-27,;45.94,-27.57,;45.94,-26.03,;44.61,-25.26,;44.61,-23.72,;45.95,-22.95,;47.29,-23.72,;47.28,-25.26,;49.96,-37.54,;49.96,-39.09,;51.3,-39.85,;52.63,-39.07,;53.97,-39.83,;52.62,-37.52,;53.95,-36.74,;51.28,-36.77,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ncccn1)-c1cc(F)cc(Cl)c1 |(18.57,-37.88,;18.59,-36.35,;19.92,-35.58,;21.26,-36.34,;22.59,-35.56,;22.58,-34.01,;23.91,-33.23,;21.24,-33.26,;19.92,-34.04,;18.58,-33.27,;18.57,-31.74,;19.9,-30.98,;19.9,-29.44,;18.57,-28.66,;17.24,-29.44,;17.24,-30.98,;15.92,-31.75,;15.92,-33.28,;17.25,-34.04,;17.26,-35.58,;18.56,-27.12,;17.02,-27.11,;17.8,-25.78,;19.91,-26.35,;19.91,-24.81,;21.25,-24.04,;21.25,-22.5,;19.92,-21.73,;18.58,-22.5,;18.58,-24.04,;23.93,-36.32,;23.93,-37.86,;25.27,-38.63,;25.28,-40.17,;26.6,-37.85,;26.59,-36.3,;27.92,-35.52,;25.25,-35.54,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(OC(F)F)c1 |(33.63,-18.23,;33.64,-16.7,;34.97,-15.92,;36.31,-16.69,;37.64,-15.91,;37.63,-14.36,;38.96,-13.58,;36.3,-13.6,;34.98,-14.39,;33.64,-13.62,;33.62,-12.09,;34.96,-11.33,;34.96,-9.79,;33.62,-9.01,;32.29,-9.79,;32.29,-11.33,;30.98,-12.09,;30.98,-13.63,;32.31,-14.39,;32.31,-15.93,;33.62,-7.47,;32.08,-7.46,;32.85,-6.13,;34.96,-6.7,;34.96,-5.15,;33.71,-4.25,;34.19,-2.78,;35.73,-2.79,;36.21,-4.25,;38.98,-16.67,;38.99,-18.21,;40.32,-18.98,;41.66,-18.2,;41.64,-16.65,;42.97,-15.86,;44.31,-16.62,;45.64,-15.84,;44.33,-18.16,;40.3,-15.89,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(c1)C(F)(F)F |(4.06,-19.22,;4.08,-17.68,;5.41,-16.91,;6.75,-17.68,;8.08,-16.9,;8.07,-15.35,;9.4,-14.57,;6.73,-14.59,;5.41,-15.37,;4.07,-14.61,;4.06,-13.08,;5.39,-12.32,;5.39,-10.77,;4.06,-10,;2.73,-10.77,;2.73,-12.32,;1.41,-13.08,;1.41,-14.61,;2.74,-15.38,;2.75,-16.92,;4.06,-8.45,;2.51,-8.45,;3.29,-7.12,;5.4,-7.68,;5.4,-6.14,;4.15,-5.24,;4.63,-3.77,;6.17,-3.78,;6.64,-5.24,;9.42,-17.66,;9.42,-19.2,;10.76,-19.96,;12.09,-19.18,;12.08,-17.64,;10.74,-16.88,;13.41,-16.85,;14.62,-16.14,;14.92,-17.41,;13.65,-15.26,)|
COc1cc(OC)cc(c1)-c1cc(OC)c(cc1F)-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1 |(41.3,-31.89,;41.32,-33.43,;39.99,-34.21,;40.01,-35.76,;38.68,-36.54,;38.68,-38.08,;40.02,-38.84,;37.34,-35.78,;37.33,-34.24,;38.66,-33.46,;36,-33.48,;34.66,-34.26,;33.33,-33.49,;31.99,-34.26,;31.98,-35.8,;33.33,-31.95,;34.65,-31.17,;35.98,-31.93,;37.31,-31.15,;31.99,-31.19,;31.98,-29.66,;33.31,-28.9,;33.31,-27.35,;31.98,-26.58,;30.65,-27.35,;30.65,-28.9,;29.33,-29.66,;29.33,-31.19,;30.66,-31.96,;30.66,-33.5,;31.97,-25.03,;30.43,-25.03,;31.21,-23.7,;33.31,-24.26,;33.32,-22.72,;32.07,-21.82,;32.54,-20.35,;34.09,-20.36,;34.56,-21.82,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(F)c1 |(49.18,-17.82,;49.2,-16.28,;50.53,-15.51,;51.87,-16.27,;53.2,-15.5,;53.19,-13.95,;54.52,-13.17,;51.85,-13.19,;50.53,-13.97,;49.19,-13.21,;49.18,-11.68,;50.51,-10.91,;50.51,-9.37,;49.18,-8.59,;47.85,-9.37,;47.85,-10.91,;46.53,-11.68,;46.53,-13.21,;47.86,-13.98,;47.87,-15.52,;49.17,-7.05,;47.63,-7.04,;48.41,-5.71,;50.52,-6.28,;50.52,-4.74,;49.27,-3.84,;49.75,-2.37,;51.29,-2.37,;51.76,-3.84,;54.53,-16.25,;54.54,-17.8,;55.88,-18.56,;57.21,-17.78,;58.55,-18.54,;57.2,-16.23,;58.52,-15.45,;55.86,-15.48,)|
COc1cc(c(F)cc1-n1c2CCN(Cc2ccc1=O)S(=O)(=O)Nc1nccs1)-c1ccc(Cl)c(C)c1 |(3.61,-16.51,;3.63,-14.97,;4.96,-14.2,;6.3,-14.97,;7.63,-14.19,;7.62,-12.64,;8.95,-11.86,;6.28,-11.88,;4.96,-12.66,;3.62,-11.9,;3.61,-10.37,;4.94,-9.61,;4.94,-8.06,;3.61,-7.29,;2.28,-8.06,;2.28,-9.61,;.96,-10.37,;.96,-11.9,;2.29,-12.67,;2.3,-14.21,;3.6,-5.74,;2.06,-5.74,;2.84,-4.41,;4.95,-4.97,;4.95,-3.43,;3.69,-2.52,;4.17,-1.06,;5.71,-1.06,;6.19,-2.53,;8.96,-14.95,;8.97,-16.49,;10.31,-17.25,;11.64,-16.47,;12.98,-17.24,;11.63,-14.92,;12.95,-14.14,;10.29,-14.17,)|
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(Cl)c2cc(OCc3ccc4ccccc4c3)ccc12
Cc1cccc(c1)-c1ccc2n(nc(Cl)c2c1)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(Cl)c2cc(ccc12)-c1cc(F)ccc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(Cl)c2cc(ccc12)-c1cc(F)c(F)c(F)c1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(Cl)c2cc(ccc12)-c1ccc(Cl)c(F)c1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(Cl)c2cc(ccc12)-c1ccc(OC(F)(F)F)cc1
Cc1ccccc1-c1ccc2n(nc(F)c2c1)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(F)c2cc(ccc12)-c1cccc(Cl)c1
COc1cccc(c1)-c1ccc2n(nc(F)c2c1)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1ncc2cc(ccc12)-c1cccc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1ncc2cc(ccc12)-c1ccc(Cl)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1cc(Cl)c2cc(cnc12)-c1ccc(F)cc1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1cc(Cl)c2cc(cnc12)-c1ccc(F)cc1Cl
Cc1cc(F)ccc1-c1cnc2n(cc(Cl)c2c1)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1cc(F)c2cc(cnc12)-c1cccc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1cc(F)c2cc(cnc12)-c1cccc(Cl)c1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(Cl)c2cc(OCc3ccc(F)cc3)ccc12
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(Cl)c2cc(ccc12)-c1cccc(Cl)c1F
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1nc(F)c2cc(ccc12)-c1cccc(F)c1
Cc1cccc(c1)-c1ccc2n(nc(F)c2c1)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1cc(Cl)c2cc(cnc12)-c1ccc(cc1)C(F)(F)F
CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1cc(F)c2cc(cnc12)-c1ccc(cc1)C(F)(F)F
Fc1cc(c(F)cc1OCC1(CCNCC1)c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1
N[C@H]1CC[C@@](CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccc(Cl)cc1 |r,wU:4.4,1.0,(66.64,-7.74,;66.69,-6.2,;65.39,-5.39,;65.44,-3.85,;66.79,-3.14,;67.56,-1.81,;69.1,-1.82,;69.86,-3.15,;71.4,-3.16,;72.17,-1.84,;73.7,-1.84,;74.47,-.51,;74.47,-3.18,;73.69,-4.51,;72.16,-4.5,;71.38,-5.83,;76.01,-3.18,;76.42,-1.69,;77.5,-2.8,;76.77,-4.52,;78.31,-4.53,;79.22,-3.29,;80.68,-3.77,;80.67,-5.31,;79.21,-5.78,;68.1,-3.93,;68.05,-5.47,;65.69,-2.04,;66.1,-.53,;65,.58,;63.49,.17,;62.41,1.26,;63.09,-1.34,;64.19,-2.44,)|
N[C@H]1CC[C@](CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccc(Cl)cc1 |r,wU:1.0,wD:4.4,(6.2,-22.18,;6.25,-20.64,;4.94,-19.82,;4.99,-18.29,;6.34,-17.57,;7.12,-16.25,;8.66,-16.25,;9.42,-17.59,;10.96,-17.6,;11.72,-16.28,;13.26,-16.28,;14.03,-14.95,;14.03,-17.62,;13.25,-18.95,;11.71,-18.94,;10.93,-20.27,;15.57,-17.62,;15.98,-16.13,;17.06,-17.23,;16.33,-18.96,;17.87,-18.97,;18.78,-17.73,;20.24,-18.21,;20.23,-19.74,;18.77,-20.21,;7.66,-18.37,;7.61,-19.91,;5.24,-16.47,;5.65,-14.97,;4.56,-13.87,;3.05,-14.27,;1.96,-13.18,;2.65,-15.78,;3.75,-16.88,)|
N[C@H]1CC[C@@](CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1 |r,wU:4.4,1.0,(27.38,-21.24,;27.43,-19.7,;26.12,-18.89,;26.17,-17.36,;27.52,-16.64,;28.3,-15.31,;29.84,-15.32,;30.6,-16.66,;32.14,-16.66,;32.9,-15.34,;34.44,-15.34,;35.21,-14.01,;35.21,-16.69,;34.43,-18.01,;32.89,-18.01,;32.11,-19.33,;36.74,-16.69,;37.16,-15.2,;38.24,-16.3,;37.51,-18.03,;39.05,-18.03,;39.95,-16.79,;41.42,-17.27,;41.41,-18.81,;39.94,-19.28,;28.84,-17.43,;28.79,-18.98,;26.42,-15.54,;26.83,-14.03,;25.74,-12.93,;24.23,-13.33,;23.83,-14.85,;24.93,-15.94,)|
CN1CCCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1
CN1C(C)(C)CC(CC1(C)C)Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1nccs1
Fc1cc(c(F)cc1OCC[C@]1(CC[C@@H](CC1)NC1CC1)c1ccccc1)S(=O)(=O)Nc1ncns1 |r,wU:14.18,wD:11.11,(32.57,-20.69,;33.35,-19.36,;34.89,-19.37,;35.67,-18.04,;34.9,-16.7,;35.67,-15.37,;33.36,-16.7,;32.6,-18.02,;31.06,-18.01,;30.3,-16.68,;28.76,-16.67,;27.98,-18,;26.63,-18.72,;26.58,-20.25,;27.89,-21.06,;29.24,-20.34,;29.3,-18.79,;27.83,-22.6,;26.49,-23.32,;24.96,-23.27,;25.68,-24.62,;26.88,-16.89,;25.38,-17.3,;24.27,-16.2,;24.68,-14.69,;26.19,-14.29,;27.29,-15.39,;37.21,-18.04,;38.71,-17.66,;37.62,-16.55,;37.98,-19.38,;39.52,-19.39,;40.42,-18.15,;41.89,-18.63,;41.88,-20.17,;40.41,-20.64,)|
C[C@@]1(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)CC[C@H](N)CC1 |r,wU:1.1,24.26,(59.23,-38.27,;60.33,-39.38,;61.11,-38.05,;62.65,-38.05,;63.41,-39.39,;64.95,-39.4,;65.72,-38.08,;67.25,-38.08,;68.03,-36.75,;68.03,-39.42,;67.25,-40.75,;65.71,-40.74,;64.93,-42.07,;69.56,-39.42,;69.98,-37.93,;71.06,-39.04,;70.33,-40.76,;71.87,-40.77,;72.78,-39.53,;74.24,-40.01,;74.24,-41.55,;72.77,-42.02,;58.98,-40.09,;58.93,-41.63,;60.24,-42.44,;60.19,-43.98,;61.6,-41.72,;61.65,-40.17,)|
ON1CCC[C@H](CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1 |r|
N[C@H]1CC[C@](CCOc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1 |r,wU:1.0,wD:4.4,(3.92,-32.53,;3.97,-31,;2.67,-30.18,;2.72,-28.65,;4.07,-27.93,;4.84,-26.6,;6.38,-26.61,;7.14,-27.95,;8.68,-27.95,;9.45,-26.63,;10.98,-26.64,;11.75,-25.31,;11.75,-27.98,;10.97,-29.31,;9.44,-29.3,;8.66,-30.62,;13.29,-27.98,;13.7,-26.49,;14.79,-27.59,;14.05,-29.32,;15.59,-29.32,;16.5,-28.08,;17.96,-28.56,;17.96,-30.1,;16.49,-30.57,;5.38,-28.73,;5.33,-30.27,;2.97,-26.83,;3.38,-25.33,;2.28,-24.22,;.77,-24.63,;.37,-26.14,;1.47,-27.23,)|
CC(=O)N1CCCC(CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1
CN[C@H]1CC[C@@](CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1 |r,wU:5.5,2.1,(27.81,-33.45,;26.5,-32.64,;26.55,-31.1,;25.25,-30.29,;25.3,-28.76,;26.65,-28.04,;27.42,-26.71,;28.96,-26.72,;29.72,-28.06,;31.26,-28.06,;32.03,-26.74,;33.56,-26.74,;34.33,-25.41,;34.33,-28.09,;33.55,-29.41,;32.02,-29.41,;31.24,-30.73,;35.87,-28.09,;36.28,-26.6,;37.37,-27.7,;36.63,-29.43,;38.17,-29.43,;39.08,-28.19,;40.54,-28.67,;40.54,-30.21,;39.07,-30.68,;27.96,-28.83,;27.91,-30.38,;25.55,-26.94,;25.96,-25.43,;24.86,-24.33,;23.35,-24.73,;22.95,-26.25,;24.05,-27.34,)|
N[C@H]1CC[C@@](CCOc2cc(F)c(cc2Cl)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1 |r,wU:4.4,1.0,(70.59,-20.09,;70.64,-18.56,;69.33,-17.74,;69.38,-16.21,;70.73,-15.49,;71.51,-14.16,;73.05,-14.17,;73.81,-15.51,;75.35,-15.52,;76.11,-14.19,;77.65,-14.2,;78.42,-12.87,;78.42,-15.54,;77.64,-16.87,;76.1,-16.86,;75.32,-18.18,;79.96,-15.54,;80.37,-14.05,;81.45,-15.15,;80.72,-16.88,;82.26,-16.88,;83.17,-15.64,;84.63,-16.12,;84.62,-17.66,;83.16,-18.13,;72.05,-16.29,;72,-17.83,;69.63,-14.39,;70.04,-12.89,;68.95,-11.79,;67.44,-12.19,;67.04,-13.7,;68.14,-14.79,)|
N[C@H]1CC[C@](CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)(CC1)c1ccccc1 |r,wU:1.0,wD:4.4,(42.57,-44.7,;42.62,-43.17,;41.32,-42.35,;41.37,-40.82,;42.72,-40.1,;43.49,-38.77,;45.03,-38.78,;45.8,-40.12,;47.33,-40.12,;48.1,-38.8,;49.63,-38.81,;50.4,-37.47,;50.4,-40.15,;49.63,-41.48,;48.09,-41.47,;47.31,-42.79,;51.94,-40.15,;52.35,-38.66,;53.44,-39.76,;52.71,-41.49,;54.25,-41.49,;55.15,-40.25,;56.62,-40.73,;56.61,-42.27,;55.14,-42.74,;44.03,-40.9,;43.98,-42.44,;41.62,-39,;42.03,-37.49,;40.93,-36.39,;39.42,-36.79,;39.02,-38.31,;40.12,-39.4,)|
C[C@]1(CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)CC[C@H](N)CC1 |r,wU:24.26,wD:1.1,(76.43,-36.87,;77.53,-37.98,;78.31,-36.65,;79.85,-36.65,;80.61,-37.99,;82.15,-38,;82.91,-36.68,;84.45,-36.68,;85.22,-35.35,;85.22,-38.02,;84.44,-39.35,;82.91,-39.34,;82.12,-40.67,;86.76,-38.02,;87.17,-36.53,;88.26,-37.64,;87.53,-39.36,;89.07,-39.37,;89.98,-38.13,;91.44,-38.61,;91.43,-40.15,;89.97,-40.62,;76.18,-38.69,;76.13,-40.23,;77.44,-41.04,;77.38,-42.58,;78.8,-40.32,;78.85,-38.77,)|
Fc1cc(NC[C@H]2CCCNC2)c(Cl)cc1S(=O)(=O)Nc1nccs1 |r|
Fc1cc(c(F)cc1OCC[C@@]1(CC[C@@H](CC1)NC1CC1)c1ccccc1)S(=O)(=O)Nc1ncns1 |r,wU:14.18,11.11,(31.13,-18.84,;31.91,-17.51,;33.45,-17.52,;34.23,-16.19,;33.46,-14.85,;34.23,-13.52,;31.92,-14.85,;31.16,-16.17,;29.62,-16.16,;28.85,-14.82,;27.31,-14.82,;26.54,-16.15,;25.18,-16.86,;25.14,-18.4,;26.44,-19.21,;27.8,-18.49,;27.85,-16.94,;26.39,-20.75,;25.04,-21.47,;23.52,-21.43,;24.24,-22.77,;25.44,-15.04,;23.94,-15.45,;22.84,-14.35,;23.24,-12.84,;24.75,-12.44,;25.85,-13.54,;35.77,-16.19,;36.18,-14.7,;37.26,-15.81,;36.53,-17.53,;38.07,-17.54,;38.98,-16.3,;40.44,-16.78,;40.44,-18.32,;38.97,-18.79,)|
N[C@H]1CC[C@](CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1 |r,wU:1.0,wD:4.4,(47.92,-19.6,;47.97,-18.07,;46.67,-17.25,;46.72,-15.72,;48.07,-15,;48.84,-13.67,;50.38,-13.68,;51.15,-15.02,;52.68,-15.03,;53.45,-13.71,;54.98,-13.71,;55.75,-12.38,;55.75,-15.05,;54.98,-16.38,;53.44,-16.37,;52.66,-17.69,;57.29,-15.05,;57.7,-13.56,;58.79,-14.66,;58.06,-16.39,;59.59,-16.39,;60.5,-15.15,;61.96,-15.63,;61.96,-17.17,;60.49,-17.64,;49.38,-15.8,;49.33,-17.34,;46.97,-13.9,;47.38,-12.4,;46.28,-11.3,;44.78,-11.7,;44.37,-13.21,;45.47,-14.3,)|
ON1CCC[C@@H](CNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)C1 |r|
CN[C@H]1CC[C@](CCOc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)(CC1)c1ccccc1 |r,wU:2.1,wD:5.5,(49.31,-32.69,;48,-31.88,;48.05,-30.34,;46.75,-29.52,;46.8,-27.99,;48.15,-27.28,;48.93,-25.95,;50.46,-25.96,;51.23,-27.29,;52.76,-27.3,;53.53,-25.98,;55.06,-25.98,;55.83,-24.65,;55.83,-27.32,;55.06,-28.65,;53.52,-28.64,;52.74,-29.97,;57.37,-27.32,;57.78,-25.83,;58.87,-26.94,;58.14,-28.66,;59.67,-28.67,;60.58,-27.43,;62.04,-27.91,;62.04,-29.45,;60.57,-29.92,;49.46,-28.07,;49.41,-29.61,;47.05,-26.17,;47.46,-24.67,;46.36,-23.57,;44.86,-23.97,;44.45,-25.48,;45.56,-26.58,)|
N[C@H]1CC[C@@](CCNc2cc(F)c(cc2Cl)S(=O)(=O)Nc2nccs2)(CC1)c1ccccc1 |r,wU:4.4,1.0,(22.89,-44.29,;22.94,-42.75,;21.64,-41.94,;21.69,-40.41,;23.04,-39.69,;23.82,-38.36,;25.35,-38.37,;26.12,-39.7,;27.66,-39.71,;28.42,-38.39,;29.95,-38.39,;30.73,-37.06,;30.73,-39.73,;29.95,-41.06,;28.41,-41.06,;27.63,-42.38,;32.26,-39.74,;32.68,-38.25,;33.76,-39.35,;33.03,-41.08,;34.57,-41.08,;35.48,-39.84,;36.94,-40.32,;36.93,-41.86,;35.47,-42.33,;24.36,-40.48,;24.3,-42.03,;21.94,-38.59,;22.35,-37.08,;21.25,-35.98,;19.75,-36.38,;19.34,-37.89,;20.44,-38.99,)|
COc1cc(c(F)cc1-c1nccc2cc(ccc12)S(=O)(=O)Nc1ccon1)-c1cccc(C)c1
COc1cc(c(C)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(F)c(C)c1 |(45.59,-10.99,;44.26,-11.77,;44.27,-13.31,;45.6,-14.07,;45.61,-15.62,;44.28,-16.39,;44.29,-17.93,;42.95,-15.63,;42.94,-14.09,;41.61,-13.33,;41.6,-11.78,;42.92,-11.01,;42.92,-9.48,;41.58,-8.72,;40.26,-9.49,;40.27,-11.01,;38.94,-11.78,;38.94,-13.33,;40.27,-14.1,;40.27,-15.64,;41.57,-7.17,;40.08,-6.77,;41.17,-5.68,;42.9,-6.4,;42.9,-4.86,;41.65,-3.96,;42.13,-2.49,;43.67,-2.49,;44.15,-3.96,;46.95,-16.38,;46.96,-17.92,;48.29,-18.69,;49.62,-17.91,;50.96,-18.67,;49.61,-16.36,;50.94,-15.58,;48.27,-15.61,)|
COc1cc(c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1ccc(C#N)c(F)c1 |(11.87,-30.75,;10.54,-31.53,;10.55,-33.07,;11.89,-33.83,;11.9,-35.38,;10.57,-36.15,;10.57,-37.7,;9.23,-35.39,;9.23,-33.85,;7.89,-33.09,;7.88,-31.54,;9.21,-30.77,;9.2,-29.24,;7.87,-28.47,;6.55,-29.24,;6.55,-30.77,;5.22,-31.54,;5.22,-33.09,;6.55,-33.86,;6.55,-35.4,;7.85,-26.93,;6.36,-26.52,;7.46,-25.43,;9.19,-26.15,;9.18,-24.61,;7.93,-23.72,;8.4,-22.25,;9.94,-22.24,;10.42,-23.7,;13.24,-36.14,;13.24,-37.69,;14.58,-38.45,;15.91,-37.67,;17.25,-38.43,;18.59,-39.19,;15.9,-36.12,;17.23,-35.34,;14.56,-35.37,)|