780 SMILES Strings for Tryptophan 5-hydroxylase 1

Compound Name
SMILES String
COc1ccc(cc1OC)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc2ccccc2c1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(CN2CCOCC2)nc1Cl)c1cccnc1F
COc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(CN3CCOCC3)cc2Cl)c(F)c1
COc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(CN3CCOCC3)nc2Cl)c(F)c1
COc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(nc2Cl)C(=O)NC2CC2)c(F)c1
COc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(NS(C)(=O)=O)nc2Cl)c(F)c1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(CN2CCOCC2)nc1Cl)c1ccc(Cl)cc1F
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)N1CCOCC1)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1ccc(Cl)cc1F
CCc1ncccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(Cl)cc1F
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(Cl)cc1F)C(F)F
CN(C)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
COC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C#N)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(I)nc1Cl)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(N)=O)c1ccc(Cl)cc1F
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C#N)c1ccc(Cl)cc1F
CCn1nc(cc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(Cl)cc1F)C(=O)OC
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cnc(nc1Cl)C(F)(F)F)c1ccc(Cl)cc1F
CN(CC(F)(F)F)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(Cl)cc1F
CN(C)c1ncc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
COC1(C)CN(C1)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CN(C)C1(CC1)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cnc(C)nc1C)c1ccc(Cl)cc1F
CN(C1CC1)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)-c1ncco1)c1ccc(Cl)cc1F
CN(c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1)S(C)(=O)=O
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCCS1(=O)=O)c1ccc(Cl)cc1F
CN(C)S(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(Cl)cc1F
CNS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1C1CC1)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)C1(CC1)Oc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1C1CC1)C(=O)NC1CC1)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)C(C)(C)Oc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(Cl)cc1F
CN(C)C(=O)c1ccc(OC2(CC2)C(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CN(C)C(=O)c1ccc(OC(C)(C)C(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)S(C)(=O)=O)c1ccc(Cl)cc1F
CNS(=O)(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CN(C)S(=O)(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cccc2n(C)ccc12)c1ccc(Cl)cc1F
COc1ccc2c(OCC(=O)N3CCc4nc5sc(C)nn5c4C3c3ccc(Cl)cc3F)cc(C)nc2c1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccnc2c(C)c(Cl)ccc12)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccnc2c(F)ccc(F)c12)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)N1CCOCC1)c1c(C)noc1C
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1c(C)noc1C
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(F)cc1F)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(F)cc1Cl)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(C)nc1C)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1)C(F)(F)F)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cccnc1F)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cccnc1C)c1ccc(cc1F)C1CC1
CCc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(cc1F)C1CC1
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(cc1F)C1CC1
CCc1ncccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(F)cc1C)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cccnc1Cl)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1)S(N)(=O)=O)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cccnc1C(F)(F)F)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1C)S(N)(=O)=O)c1ccc(cc1F)C1CC1
CN(C)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(cc2F)C2CC2)c(C)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1C)N1CCCC1)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1ccc(cc1F)C1CC1
CCc1nc(C)ccc1OC1(CC1)C(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc[n+]([O-])c1Cl)c1ccc(cc1F)C1CC1
CCc1c(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(cc2F)C2CC2)ccc(C)[n+]1[O-]
COC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(cc2F)C2CC2)c(Cl)n1
CN(C)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(cc2F)C2CC2)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C#N)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(F)(F)F)c1ccc(cc1F)C1CC1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(cc2F)C2CC2)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cnc(C)nc1C)c1ccc(cc1F)C1CC1
CN(C1CC1)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(cc2F)C2CC2)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)-c1ncco1)c1ccc(cc1F)C1CC1
CCc1ncccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1cnc(s1)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1cnc(s1)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cccnc1Cl)c1cnc(s1)N1CCOCC1
CN(C)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cnc(s2)N2CCOCC2)c(Cl)n1
CN(C)Cc1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CCc1ncccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1cc(CN(C)C)cs1
CN(C)Cc1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(Cl)cc1C
CN(C)Cc1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N(C)C
CN(C)Cc1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N(C)CC(F)(F)F
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1cnc(nc1)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)N1CCOCC1)c1cnc(nc1)C1CC1
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1cnc(nc1C)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)N1CCOCC1)c1cnc(nc1C)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(Cl)cc1C)c1nc(no1)-c1ccccc1
CCc1ncccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1nc(no1)-c1ccccc1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1nc(no1)-c1ccccc1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1coc(n1)-c1ccccc1
CCc1ncccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1coc(n1)-c1ccccc1
CC(=O)Nc1ccc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1ncc(cc1F)C1CC1
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ncc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(F)(F)F)c1ncc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C#N)c1ncc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1F)N1CCOCC1)c1ncc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cc(F)c(I)nc1Cl)c1ncc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cc(F)cnc1Cl)c1ncc(cc1F)C1CC1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(cc2F)C2CC2)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1cc(F)c(nc1Cl)N1CCOCC1)c1ncc(cc1F)C1CC1
CN(CC(F)(F)F)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(cc2F)C2CC2)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1c(Cl)nc(N2CCOCC2)c(F)c1F)c1ncc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1c(F)cc(nc1Cl)N1CCOCC1)c1ncc(cc1F)C1CC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ncc(cc1F)C1CC1
CN(C)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cnc(OC(F)F)cc2C)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1cnc(OC(F)F)cc1C
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1cnc(OC(F)F)cc1C
CN(C)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)nc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1C)S(N)(=O)=O)c1ccc(Cl)nc1F
CNc1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)nc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(F)(F)F)c1ccc(Cl)nc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C#N)c1ccc(Cl)nc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C#N)c1ccc(Cl)nc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C(F)(F)F)c1ccc(Cl)nc1F
CN(C)Cc1csc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CN(C)C(=O)c1csc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1cc(cs1)C(C)(C)O
COC(=O)c1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1sccc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1C)S(N)(=O)=O)c1sccc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(F)(F)F)c1sccc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1sccc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C(F)(F)F)c1sccc1F
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2sccc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(CN)cc1Cl)c1sccc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1)c1sccc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(=O)(=O)C2CC2)nc1Cl)c1sccc1F
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2sccc2F)c(Cl)n1
CN(C)c1ncc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2sccc2F)c(Cl)n1
CCn1nc(cc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1sccc1F)C(=O)OC
CCn1nc(cc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1sccc1F)C(=O)N(C)C
CCN(CC)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3[C@@H]2c2sccc2F)c(Cl)n1
Cc1nn2c3[C@@H](N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)-c1ncco1)c1sccc1F
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(F)(F)F
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C#N
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1cccnc1Cl
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C#N
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2sc(cc2F)C(=O)N(C)C)c(Cl)n1
CN(C)C(=O)c1cc(F)c(s1)[C@@H]1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(F)(F)F
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(N)=O
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C#N
CNC(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1cc(F)cnc1Cl
COC(=O)c1ccc(o1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CCOC(=O)c1csc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CCOC(=O)c1csc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(F)(F)F
CCOC(=O)c1csc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
COC(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
COC(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
COC(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(=O)(=O)C2CC2)nc1Cl
COC(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1
CCOC(=O)c1coc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CCOC(=O)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CCOC(=O)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
CCOC(=O)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C#N
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C(F)(F)F)c1ncc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1ncc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C#N)c1ncc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C#N)c1ncc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(F)(F)F)c1ncc(C)cc1F
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(C)cc2F)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(C)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ncc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(=O)(=O)C2CC2)nc1Cl)c1ncc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)cc1Cl)c1ncc(C)cc1F
COC1(C)CN(C1)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3[C@@H]2c2ncc(C)cc2F)c(Cl)n1
CN(C)C1(CC1)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3[C@@H]2c2ncc(C)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)-c1ncco1)c1ncc(C)cc1F
CN(C1CC1)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(C)cc2F)c(Cl)n1
CN(c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3[C@@H]2c2ncc(C)cc2F)c(Cl)n1)S(C)(=O)=O
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2[C@@H]1c1ncc(C)cc1F
Cc1nn2c3[C@@H](N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCCS1(=O)=O)c1ncc(C)cc1F
CCc1nc(Cl)ncc1OCC(=O)N1CCc2nc3sc(C)nn3c2[C@@H]1c1ncc(C)cc1F
CCc1nc(NS(C)(=O)=O)ncc1OCC(=O)N1CCc2nc3sc(C)nn3c2[C@@H]1c1ncc(C)cc1F
COc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2[C@@H]1c1ncc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1scnc1C
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C#N)c1scnc1C
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C(F)(F)F)c1scnc1C
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(F)(F)F)c1scnc1C
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3[C@@H]2c2scnc2C)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1ncc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1)c1ncc(Cl)cc1F
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(N)=O)c1ncc(Cl)cc1F
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ncc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)cc1Cl)c1ncc(Cl)cc1F
CN(C)C(=O)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CN(C)C(=O)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CN(C)C(=O)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1ncccc1F
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncccc2F)c(Cl)n1
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncccc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ncccc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1cncs1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cncs2)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1cncs1
CNC(=O)c1ccc(o1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CNC(=O)c1ccc(o1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CCNC(=O)Nc1nc(cs1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
COC1(COC1)c1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)-c1ncco1)c1ccc(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(C)cc1F
CN(C1CC1)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(C)cc2F)c(Cl)n1
Cc1nn2c3[C@@H](N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(C)cc1F
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(OC(F)F)cc2F)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(F)cc2F)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(cc2F)C(F)(F)F)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cc(F)ccc2F)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cccc(Cl)c2F)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cnc(C)s2)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cnc(s2)-c2ccccc2)c(Cl)n1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(C)c(F)c2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(C)c(F)c1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCCS1(=O)=O)c1ccc(C)c(F)c1F
CCc1nc(Cl)ncc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(C)c(F)c1F
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1ccc(C)c(F)c1F
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cccc(F)c2F)c(Cl)n1
CCN(CC)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
COC1(COC1)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nc(C)c(o1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(nc2Cl)N2CCOCC2)c(C)o1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2sc(C)nc2C)c(Cl)n1
Cc1nc(C)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
Cc1nc(C)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)-c1ncco1
CN(C1CC1)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2sc(C)nc2C)c(Cl)n1
Cc1nc(C)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCCS1(=O)=O
CN(c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2sc(C)nc2C)c(Cl)n1)S(C)(=O)=O
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1sc(C)nc1C
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2[C@@H]1c1sc(C)nc1C)N1CCCS1(=O)=O
CCc1nc(NS(C)(=O)=O)ncc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1sc(C)nc1C
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1sccc1F)C(=O)NC1CC1
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1sccc1F
CCc1nc(C)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
CC(C)c1nc(C)c(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(C)nn3c2C1c1cc(F)c(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1cc(F)c(C)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ncc(F)cc1C
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1sc(nc1C)C(F)(F)F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(OC(F)(F)F)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(=O)NC1CC1)c1ccc(OC(F)(F)F)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(CN)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(=O)NC1CC1)c1ccc(CN)cc1F
COC(=O)c1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(NS(C)(=O)=O)nc2Cl)c(F)c1
COC(=O)c1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(nc2Cl)C(=O)NC2CC2)c(F)c1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(cc1F)C(C)(C)O
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(=O)NC1CC1)c1ccc(cc1F)C(C)(C)O
COC(C)(C)c1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(nc2Cl)C(=O)NC2CC2)c(F)c1
COC(C)(C)c1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(NS(C)(=O)=O)nc2Cl)c(F)c1
COCc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(NS(C)(=O)=O)nc2Cl)c(F)c1
COCc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(nc2Cl)C(=O)NC2CC2)c(F)c1
COCCOc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(nc2Cl)C(=O)NC2CC2)c(F)c1
COCCOc1ccc(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(NS(C)(=O)=O)nc2Cl)c(F)c1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1csc(c1)C1OCCO1
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4scnn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Fc1cc(Cl)ccc1C1N(CCc2nc3scnn3c12)C(=O)COc1ccc(cc1Cl)C#N
Fc1cc(Cl)ccc1C1N(CCc2nc3scnn3c12)C(=O)COc1ccc(nc1Cl)-c1ncco1
CCc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(Cl)cc1F
CCc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C#N)c1ccc(Cl)cc1F
CCc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)-c1ncco1)c1ccc(Cl)cc1F
CCc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCN(C)CC1)c1ccc(Cl)cc1F
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sc(nn4c3C2c2ccc(Cl)cc2F)C2CC2)c(Cl)n1
Fc1cc(Cl)ccc1C1N(CCc2nc3sc(nn3c12)C1CC1)C(=O)COc1ccc(cc1Cl)C#N
Fc1cc(Cl)ccc1C1N(CCc2nc3sc(nn3c12)C1CC1)C(=O)COc1ccc(nc1Cl)-c1ncco1
CN1CCN(CC1)c1ccc(OCC(=O)N2CCc3nc4sc(nn4c3C2c2ccc(Cl)cc2F)C2CC2)c(Cl)n1
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sc(nn4c3C2c2ccc(Cl)cc2F)C(F)(F)F)c(Cl)n1
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1ccc(Cl)cc1F)C(F)(F)F
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1ccc(Cl)cc1F)C(F)(F)F)N1CCCS1(=O)=O
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(nn3c2[C@@H]1c1ccc(Cl)cc1F)C(F)(F)F)N1CCCS1(=O)=O
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1ncc(C)cc1F)C(F)(F)F)N1CCCS1(=O)=O
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1ncc(C)cc1F)C(F)(F)F
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1ccc(C)cc1F)C(F)(F)F
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1sc(C)nc1C)C(F)(F)F)N1CCCS1(=O)=O
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1sc(C)nc1C)C(F)(F)F
COc1ccc(cc1OC)C1N(CCc2nc3sccn3c12)C(=O)COc1ccc2ccccc2c1
COc1ccc(cc1OC)C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(CN2CCOCC2)cc1Cl
COc1ccc(cc1OC)C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(Cl)cc1Cl
Fc1ncccc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(CN2CCOCC2)cc1Cl
Fc1ncccc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccccc1C(F)(F)F
Cc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2cccnc2F)cc1
Cc1ccccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cccnc1F
Cc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cccnc1F
Cn1nc(OCC(=O)N2CCc3nc4sccn4c3C2c2cccnc2F)c(c1Cl)C(F)(F)F
Fc1ncccc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(CN2CCOCC2)nc1Cl
COc1ccc(C2N(CCc3nc4sccn4c23)C(=O)COc2ccc(CN3CCOCC3)cc2Cl)c(F)c1
COc1ccc(C2N(CCc3nc4sccn4c23)C(=O)COc2ccc(CN3CCOCC3)nc2Cl)c(F)c1
COc1ccc(C2N(CCc3nc4sccn4c23)C(=O)COc2ccc3ccncc3c2)c(F)c1
CCc1cc(F)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(OC)cc1F
CCc1cc(F)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(Cl)cc1F
Fc1cc(Cl)ccc1[C@@H]1C2N3C=CSC3=NC2=CCN1C(=O)COc1ccc(cc1Cl)N1CCOCC1 |c:12,16,19|
Cc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(Cl)cc1F
Fc1cc(Cl)ccc1C1N(CCc2nc3sccn3c12)C(=O)COc1cccnc1Cl
Fc1cc(Cl)ccc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(CN2CCOCC2)nc1Cl
Fc1cc(Cl)ccc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CCc1ncccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(Cl)cc1F
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1c(C)noc1C
Cc1noc(C)c1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(Cl)cc1Cl
Cc1noc(C)c1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
Cc1noc(C)c1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(Cl)cc1C
CCc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1c(C)noc1C
Fc1cc(ccc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1)C1CC1
Fc1cc(cnc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(nc1Cl)C(F)(F)F)C1CC1
Fc1cc(cnc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(nc1Cl)C#N)C1CC1
Fc1ccsc1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(NS(=O)(=O)C2CC2)nc1Cl
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2sccc2F)c(Cl)n1
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2sccc2F)c(Cl)n1
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2sccc2F)c(Cl)n1
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2sccc2F)c(Cl)c1
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(NS(C)(=O)=O)cc1Cl
CN(C)C(=O)c1cc(F)c(s1)C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
Cc1ccc(C2N(CCc3nc4sccn4c23)C(=O)COc2ccc(Cl)cc2C)c(F)c1
CCc1ncccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(C)cc1F
Cc1ccc(C2N(CCc3nc4sccn4c23)C(=O)COc2cccnc2Cl)c(F)c1
CCc1cc(F)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(C)cc1F
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(cc1F)C(F)(F)F
Cc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2nc3ccccc3s2)cc1
Cc1ccccc1OCC(=O)N1CCc2nc3sccn3c2C1c1nc2ccccc2s1
Clc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2nc3ccccc3s2)c(Cl)c1
Cc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1nc2ccccc2s1
FC(F)(F)c1cccc(OCC(=O)N2CCc3nc4sccn4c3C2c2nc3ccccc3s2)c1Cl
Clc1ncccc1OCC(=O)N1CCc2nc3sccn3c2C1c1nc2ccccc2s1
Cn1nc(OCC(=O)N2CCc3nc4sccn4c3C2c2nc3ccccc3s2)c(Cl)c1C(F)(F)F
Clc1nc(CN2CCOCC2)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1nc2ccccc2s1
O=C(COc1ccc2ccncc2c1)N1CCc2nc3sccn3c2C1c1nc2ccccc2s1
FC(F)(F)c1cccc(OCC(=O)N2CCc3nc4sccn4c3C2c2cnn(c2)-c2ccccc2)c1Cl
Clc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2cnn(c2)-c2ccccc2)c(Cl)c1
Cc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2cnn(c2)-c2ccccc2)cc1
Cc1ccccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cnn(c1)-c1ccccc1
Clc1cc(CN2CCOCC2)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cnn(c1)-c1ccccc1
Clc1nc(CN2CCOCC2)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cnn(c1)-c1ccccc1
Cc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cnn(c1)-c1ccccc1
FC(F)(F)c1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2cnn(c2)-c2ccccc2)c(Cl)c1
CCc1ncccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cnn(c1)-c1ccccc1
Clc1ccc(OCC(=O)N2CCc3nc4sccn4c3C2c2cc3cccnc3s2)c(Cl)c1
Cc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cc2cccnc2s1
Clc1ncccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cc2cccnc2s1
Clc1nc(CN2CCOCC2)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1cc2cccnc2s1
Cc1ccc(Cl)c(OCC(=O)N2CCc3nc4sccn4c3C2c2cc3cccnc3s2)c1
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1c(C)nn(C)c1C
Cc1nn(C)c(C)c1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
Cc1nn(C)c(C)c1C1N(CCc2nc3sccn3c12)C(=O)COc1ccc(Cl)cc1C
CCc1cc(Cl)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1c(C)nn(C)c1C
CCc1ncccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(cc1F)C(F)F
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(cc1F)C(F)F
FC(F)c1ccc(C2N(CCc3nc4sccn4c23)C(=O)COc2cccnc2Cl)c(F)c1
CCc1nc(C)ccc1OCC(=O)N1CCc2nc3sccn3c2C1c1ccc(nc1C)C(F)(F)F
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sc(CF)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1ccc(Cl)cc1F
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1ccc(Cl)cc1F)N1CCCS1(=O)=O
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1ncc(C)cc1F)N1CCCS1(=O)=O
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1ncc(C)cc1F
Cc1ccc(C2N(CCc3nc4sc(CF)nn4c23)C(=O)COc2ccc(NS(C)(=O)=O)nc2Cl)c(F)c1
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1ccc(C)cc1F
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1sc(C)nc1C)C(=O)NC1CC1
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1sc(C)nc1C
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(CF)nn3c2C1c1sc(C)nc1C)N1CCCS1(=O)=O
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sc(nn4c3C2c2ccc(Cl)cc2F)C(F)F)c(Cl)n1
CCc1nc(NS(C)(=O)=O)ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1ccc(Cl)cc1F)C(F)F
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1ccc(Cl)cc1F)C(F)F)N1CCCS1(=O)=O
CS(=O)(=O)Nc1ccc(OCC(=O)N2CCc3nc4sc(nn4c3[C@@H]2c2ccc(Cl)cc2F)C(F)F)c(Cl)n1
Cc1ccc(C2N(CCc3nc4sc(nn4c23)C(F)F)C(=O)COc2ccc(NS(C)(=O)=O)nc2Cl)c(F)c1
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1sc(C)nc1C)C(F)F)C(=O)NC1CC1
CCc1nc(ccc1OCC(=O)N1CCc2nc3sc(nn3c2C1c1sc(C)nc1C)C(F)F)N1CCCS1(=O)=O
COC(=O)CCS(=O)(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)S(N)(=O)=O)c1ccc(Cl)cc1F
CN(CCO)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
COCCN(C)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CC1CCC(C)N1c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(=O)(=O)C2CC2)nc1Cl)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCCC1=O)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1)c1ccc(Cl)cc1F
C[C@H]1C[C@H](C)CN(C1)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(N)nc1Cl)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(=O)NCC#N)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(=O)NO)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C(N)=O)c1ccc(Cl)cc1F
CNc1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C1CC1)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)N1CC(F)(F)C1)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(=O)(=O)C2CC2)cc1Cl)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCC(F)(F)CC1)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CC2CC1CO2)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(cc1Cl)C1CC1)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCNCC1=O)c1ccc(Cl)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCC(F)(F)C1)c1ccc(Cl)cc1F
CONC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ccc(Cl)cc2F)c(Cl)n1
CN(C)C(=O)c1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CN(C)C(=O)c1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1
CN(C)C(=O)c1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
CN(C)C(=O)c1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
CN(C)C(=O)c1csc(c1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cc(cs2)C(=O)N(C)C)c(Cl)n1
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N(C)C
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(F)(F)F
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1cc(F)cnc1Cl
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1cccnc1Cl
CN(C)c1ncc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1
CN(C)C(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2cnc(s2)N(C)C)c(Cl)n1
CN(C)Cc1ccc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CNC(=O)c1ccc(OCC(=O)N2CCc3nc4sc(C)nn4c3C2c2ncc(s2)C(=O)N(C)C)c(Cl)n1
CN(C)C(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CC(F)(F)C1
CN(C)C(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl
CN(C)C(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CN(C)C(=O)c1cnc(s1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1csc(c1)C(O)=O
CN(C)C(=O)c1ccc(o1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)C(=O)N(C)C
CN(C)C(=O)c1ccc(o1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CN(C)C(=O)c1coc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
CNC(=O)c1csc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(cc1Cl)C(F)(F)F
CNC(=O)c1csc(n1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1csc(CO)c1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1cc(cs1)C(O)=O
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1nc(cs1)C(N)=O
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1cnc(s1)N1CC(F)(F)C1
CCNc1nn(C)c(C2N(CCc3nc4sc(C)nn4c23)C(=O)COc2ccc(nc2Cl)N2CCOCC2)c1C
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1nc(N)sc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1cc(cs1)-c1nn[nH]n1
CN(C)Cc1cc(cs1)C1N(CCc2nc3sc(C)nn3c12)C(=O)COc1ccc(nc1Cl)N1CCOCC1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)N1CCOCC1)c1sc(cc1F)-c1nnn[nH]1
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(nc1Cl)C(=O)NC1CC1)c1ccc(OCCO)cc1F
Cc1nn2c3C(N(CCc3nc2s1)C(=O)COc1ccc(NS(C)(=O)=O)nc1Cl)c1ccc(OCCO)cc1F
CCCn1c2nc(Cc3nc4ccc(O)cc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCCN1c2c(n(c(n2)Cc3[nH]c4cc5c(cc4n3)OCO5)Cc6ccccc6)C(=O)NC1=O
CCCn1c2nc(Cc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3nc4cc5OCOc5cc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Oc1ccc2nc(Cc3nc4n(C5CC5)c(=O)[nH]c(=O)c4n3Cc3ccccc3)[nH]c2c1
CCN1c2c(n(c(n2)Cc3[nH]c4ccccc4n3)Cc5ccccc5)C(=O)NC1=O
O=c1[nH]c(=O)c2n(Cc3ccccc3)c(Cc3nc4cc5OCOc5cc4[nH]3)nc2n1C1CC1
CCCn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
COc1cccc(c1)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)-c1ccc(CC(N)C(O)=O)cc1)C(F)(F)F |r|
CCn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
c1ccc(cc1)Cn2c(nc3c2C(=O)NC(=O)N3C4CC4)Cc5[nH]c6ccccc6n5
COc1ccc2nc(Cc3nc4n(C5CC5)c(=O)[nH]c(=O)c4n3Cc3ccccc3)[nH]c2c1
CCn1c2nc(Cc3nc4ccc(cc4[nH]3)-c3cc[nH]n3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3nc4cc(F)c(cc4[nH]3)N(C)C)n(Cc3ccccc3)c2c(=O)[nH]c1=O
O=c1[nH]c(=O)c2n(Cc3ccccc3)c(Cc3nc4cc(ccc4[nH]3)N3CCOCC3)nc2n1C1CC1
CCn1c2nc(Cc3nc4ccccc4[nH]3)n(Cc3ccc(F)cc3)c2c(=O)[nH]c1=O
OCCOc1ccc2nc(Cc3nc4n(C5CC5)c(=O)[nH]c(=O)c4n3Cc3ccccc3)[nH]c2c1
COC(=O)c1ccc2nc(Cc3nc4n(C5CC5)c(=O)[nH]c(=O)c4n3Cc3ccccc3)[nH]c2c1
Fc1ccc2nc(Cc3nc4n(C5CC5)c(=O)[nH]c(=O)c4n3Cc3ccccc3)[nH]c2c1
CCn1c2nc(Cc3nc4cc(F)c(cc4[nH]3)N3CCOCC3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Cc3nc4cc(NC(=O)CC[C@H](N)C(O)=O)ccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O |r|
O=c1[nH]c(=O)c2n(Cc3ccccc3)c(Cc3nc4cc(ccc4[nH]3)N3CCNCC3)nc2n1C1CC1
Cn1c2nc(Sc3nc4cc(NC(=O)CC[C@H](N)C(O)=O)ccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O |r|
CC(=O)Nc1ccc2nc(Cc3nc4n(C)c(=O)[nH]c(=O)c4n3Cc3ccccc3)[nH]c2c1
Cn1c2nc(Cc3nc4ccc(Br)cc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
O=c1[nH]c(=O)c2n(Cc3ccccc3)c(Cc3nc4ccc(cc4[nH]3)C#N)nc2n1C1CC1
Cn1c2nc(Cc3nc4cc(ccc4[nH]3)N3CCOCC3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Cc3nc4ccc(N)cc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4cc(N)ccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Cc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
COc1ccc2[nH]c(Sc3nc4n(C)c(=O)[nH]c(=O)c4n3Cc3ccccc3)nc2c1
Cn1c2nc(Sc3nc4cc(NC(=O)C[C@H](N)C(O)=O)ccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O |r|
Cn1c2nc(Cc3nc4ccc(cc4[nH]3)N3CCC(CC3)C(O)=O)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4cc(NCC(O)=O)ccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cc1ccc2[nH]c(Sc3nc4n(C)c(=O)[nH]c(=O)c4n3Cc3cncs3)nc2c1
Cc1ccc2[nH]c(Sc3nc4n(C)c(=O)[nH]c(=O)c4n3Cc3ccccc3)nc2c1
CCn1c2nc(Cc3nc4ncccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3nccs3)c2c(=O)[nH]c1=O
CC(=O)Nc1ccc(Cn2c(Sc3nc4ccccc4[nH]3)nc3n(C)c(=O)[nH]c(=O)c23)cc1
Cn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3cnco3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3ccc(N)cc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3ccc(cc3)N3CCOCC3)c2c(=O)[nH]c1=O
CN1CCN(CC1)c1ccc2nc(Cc3nc4n(C)c(=O)[nH]c(=O)c4n3Cc3ccccc3)[nH]c2c1
CCn1c(Sc2nc3n(C)c(=O)[nH]c(=O)c3n2Cc2ccccc2)nc2ccccc12
Cn1c2nc(Sc3nc4cc(Cl)c(Cl)cc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4cc(ccc4[nH]3)S(O)(=O)=O)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4ccc(cc4[nH]3)C(O)=O)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4ccccc4s3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cn1c2nc(Sc3nc4cccnc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
Cc1nnc(Cn2c(Sc3nc4ccccc4[nH]3)nc3n(C)c(=O)[nH]c(=O)c23)o1
Cn1c2nc(Sc3nc4ccccc4[nH]3)n(Cc3ccco3)c2c(=O)[nH]c1=O
Cc1ccc2[nH]c(Sc3nc4n(C)c(=O)[nH]c(=O)c4n3Cc3ccco3)nc2c1
Cn1c2nc(Nc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Nc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCCn1c2nc(Nc3nc4ccccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCN1c2c(n(c(n2)Cc3cn4c(n3)CCCC4)Cc5ccccc5)C(=O)NC1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)-c3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)C(=O)OC)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc4OCOc4c3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)C(O)=O)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)-c3ccn(C)n3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)-c3noc(C)n3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)-c3ncccn3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)-c3nccs3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)-c3ccc(cn3)C(F)(F)F)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)-c3nc(C)no3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4nc(C)sc4n3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccsc4n3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccsc4n3)n(Cc3ccc(cc3)-c3ccn(C)n3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(C)sc4n3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(C)sc4n3)n(Cc3ccc(cc3)-c3ccn(C)n3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)-c3ccn(C)n3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(CC(=O)OC)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(Cl)sc4n3)n(Cc3ccc(cc3)-c3ccn(C)n3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(Cl)sc4n3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
O=c1[nH]c(=O)c2n(Cc3ccccc3)c(Cc3cn4ccccc4n3)nc2n1C1CC1
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(CCO)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(CC(O)=O)cc3)c2c(=O)[nH]c1=O
CCCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(C)sc4n3)n(Cc3ccc(F)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(C)sc4n3)n(Cc3ccc(OC)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(Cl)sc4n3)n(Cc3ccc(NC(C)=O)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(Cl)sc4n3)n(Cc3ccc(cc3)-n3cncn3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(C)sc4n3)n(Cc3ccc(NC(C)=O)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)-n3cncn3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(C)sc4n3)n(Cc3ccc(cc3)N3CCCC3=O)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)-n3ccnc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4cc(Cl)sc4n3)n(Cc3ccc(cc3)N3CC(F)(F)C3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(NC(C)=O)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)N3CCCC3=O)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)N3CC(F)(F)C3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)N3CC(C3)OC)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4CCCCc4n3)n(Cc3ccc(cc3)-c3noc(C)n3)c2c(=O)[nH]c1=O
CCOC(=O)[C@@H](N)Cc1ccc(cc1)-c1cc(O[C@H](c2ccc(Cl)cc2-n2ccc(C)n2)C(F)(F)F)nc(N)n1
COc1cccc(c1)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)-c1ccc(C[C@H](N)C(O)=O)cc1)C(F)(F)F
N[C@@H](Cc1ccc(cc1)-c1cc(OC(c2ccc(cc2)-c2cccc(F)c2)C(F)(F)F)nc(N)n1)C(O)=O |r|
CCn1c2nc(Cc3cn4ccccc4n3)n(Cc3ccc(cc3)-c3ccc(cn3)C(F)(F)F)c2c(=O)[nH]c1=O
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)-c1ccc(CC(N)C(O)=O)cc1)C(F)(F)F |r|
NC(Cc1ccc(cc1)-c1cc(O[C@H](c2ccc(cc2)-c2cccc(F)c2)C(F)(F)F)nc(N)n1)C(O)=O |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1ncnc2c(csc12)-c1ccc(C[C@H](N)C(O)=O)cc1)C(F)(F)F |r|
COc1cccc(c1)-c1ccc(Cn2ccc3c(nc(N)nc23)-c2ccc(C[C@H](N)C(O)=O)cc2)cc1 |r|
CCOC(=O)[C@@H](N)Cc1ccc(cc1)-c1csc2c(O[C@H](c3ccc(Cl)cc3-n3ccc(C)n3)C(F)(F)F)ncnc12 |r|
COc1cccc(c1)-c1ccc(Cn2ccc3c(ncnc23)-c2ccc(C[C@H](N)C(O)=O)cc2)cc1 |r|
N[C@@H](Cc1ccc(cc1)-c1csc2c(O[C@H](c3ccc(Cl)cc3-c3cccc(F)c3)C(F)(F)F)ncnc12)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1csc2c(OC(c3ccc(Cl)cc3-c3ccccc3)C(F)(F)F)ncnc12)C(O)=O |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1ncnc2c(csc12)C1=CCC(C[C@H](N)C(O)=O)CC1)C(F)(F)F |r,t:28|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)C1=CCC(C[C@H](N)C(O)=O)CC1)C(F)(F)F |r,t:25|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(C)n1)C1=CCC(C[C@H](N)C(O)=O)CC1)C(F)(F)F |r,t:25|
COc1cccc(c1)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)C1=CCC(C[C@H](N)C(O)=O)CC1)C(F)(F)F |r,t:26|
N[C@@H](Cc1ccc(cc1)-c1csc2c(OC(c3ccc(Cl)cc3-c3ccc(F)cc3)C(F)(F)F)ncnc12)C(O)=O |r|
N[C@@H](CC1CCC(=CC1)c1cc(OC(c2ccc(Cl)cc2-c2ccccc2)C(F)(F)F)nc(N)n1)C(O)=O |r,c:6|
N[C@@H](CC1CCC(=CC1)c1cc(O[C@H](c2ccc(Cl)cc2C2=CCCOC2)C(F)(F)F)nc(N)n1)C(O)=O |r,c:6,t:23|
N[C@@H](Cc1ccc(cc1)-c1csc2c(O[C@H](c3ccc(Cl)cc3C3=CCCOC3)C(F)(F)F)ncnc12)C(O)=O |r,t:25|
N[C@@H](CC1CCC(=CC1)c1cc(O[C@H](c2ccc(Cl)cc2C2=CCC(F)(F)CC2)C(F)(F)F)nc(N)n1)C(O)=O |r,c:6,t:23|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)C1=CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r,t:25|
Nc1nc(O[C@H](c2ccc(Cl)cc2C2=CCOCC2)C(F)(F)F)cc(n1)C1=CCC2(CNC(C2)C(O)=O)CC1 |r,t:14,29|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1ncnc2c(csc12)C1=CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r,t:28|
N[C@@H](CC1CCC(=CC1)c1cc(O[C@H](c2ccc(Cl)cc2C2=CCOCC2)C(F)(F)F)nc(N)n1)C(O)=O |r,c:6,t:23|
COc1cccc(c1)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)C1=CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r,t:26|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1nc(N)nc2c(csc12)-c1ccc(C[C@H](N)C(O)=O)cc1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2C2=CCCOC2)C(F)(F)F)cc(n1)C1=CCC2(CNC(C2)C(O)=O)CC1 |r,t:14,29|
N[C@@H](Cc1ccc(Cl)cc1)C(O)=O |r|
COc1ccc(cc1)-c1nc(no1)-c1ccc(C[C@H](N)C(O)=O)cc1
COc1ccc(cc1OC)-c1nc(no1)-c1ccc(C[C@H](N)C(O)=O)cc1
N[C@@H](Cc1ccc(cc1)-c1noc(n1)-c1ccc(F)cc1)C(O)=O
COc1ccc(cc1-c1ccccc1)-c1nc(no1)-c1ccc(C[C@H](N)C(O)=O)cc1
COc1ccc(cc1)-c1cc(ccc1OC)-c1nc(no1)-c1ccc(C[C@H](N)C(O)=O)cc1
COc1ccc(cc1-c1ccc(O)cc1)-c1nc(no1)-c1ccc(C[C@H](N)C(O)=O)cc1
CCOC(=O)[C@@H](N)Cc1ccc(cc1)-c1noc(n1)-c1ccc(OC)c(c1)-c1ccc(O)cc1
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)-c1ccc(C[C@H](N)C(O)=O)cc1)C(F)(F)F |r|
COc1ccc(cc1-c1cccc(O)c1)-c1nc(no1)-c1ccc(C[C@H](N)C(O)=O)cc1
COc1ccc(cc1-c1ccccc1O)-c1nc(no1)-c1ccc(C[C@H](N)C(O)=O)cc1
CN1CCN(CC1)c1ccc2[nH]c(Cc3nc4n(C)c(=O)[nH]c(=O)c4n3Cc3ccccc3)nc2c1
CCCn1c2nc(Cc3nc4cc(O)ccc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCOc1ccc2[nH]c(Cc3nc4n(CC)c(=O)[nH]c(=O)c4n3Cc3ccccc3)nc2c1
CCn1c2nc(Cc3nc4cc(N(C)C)c(F)cc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3nc4cc(N5CCOCC5)c(F)cc4[nH]3)n(Cc3ccccc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccsc4n3)n(CC(=O)c3ccc(OC)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccsc4n3)n(CC(=O)c3ccc(N)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccsc4n3)n(CC(=O)c3ccc(O)cc3)c2c(=O)[nH]c1=O
CCn1c2nc(Cc3cn4ccsc4n3)n(CC(=O)c3ccc(CO)cc3)c2c(=O)[nH]c1=O
CCN1c2c(n(c(n2)Cc3cn4cc(sc4n3)C)CC5COC5)C(=O)NC1=O
N[C@@H](Cc1ccc(cc1)-c1cnc(NCC2CCCCC2)cn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cc(OC(c2sccc2-c2ccco2)C(F)(F)F)nc(N)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cc(OC(c2ccccc2-n2ccc(n2)C(F)(F)F)C(F)(F)F)nc(N)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cc(OC(c2ccccc2-c2ccco2)C(F)(F)F)nc(N)n1)C(O)=O |r|
Cc1cccc(c1)-c1ccccc1C(Oc1cc(nc(N)n1)-c1ccc(C[C@H](N)C(O)=O)cc1)C(F)(F)F |r|
N[C@@H](Cc1ccc(cc1)-c1cc(OC(c2ccc3ccccc3c2)C(F)(F)F)nc(N)n1)C(O)=O |r|
C[C@@H](Oc1cc(nc(N)n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
C[C@@H](Nc1cc(nc(N)n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
CCn1c2ccccc2c2cc(CNc3ccc(nc3)-c3ccc(C[C@H](N)C(O)=O)cc3)ccc12 |r|
COc1ccc(CNc2ccc(nn2)-c2ccc(C[C@H](N)C(O)=O)cc2)cc1OC1CCCC1 |r|
COc1ccc(CNc2ccc(cc2)-c2ccc(C[C@H](N)C(O)=O)cc2)cc1OC1CCCC1 |r|
C[C@@H](Nc1nc(N)nc(n1)-c1ccc(cc1)C(N)CC(O)=O)c1ccc2ccccc2c1 |r|
C[C@@H](Nc1nc(N)nc(n1)-c1ccc(CC(C)(N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2ccc3ccccc3c2)n1)C(O)=O |r|
C[C@@H](Nc1nc(N)nc(n1)-c1ccn(C[C@H](N)C(O)=O)n1)c1ccc2ccccc2c1 |r|
C[C@@H](Nc1nc(N)nc(n1)N1CCC(C[C@H](N)C(O)=O)CC1)c1ccc2ccccc2c1 |r|
C[C@@H](Nc1nc(N)nc(n1)-c1ccc(CC(N)C(O)=O)nc1)c1ccc2ccccc2c1 |r|
C[C@@H](Nc1nc(N)nc(n1)-c1cccc(CC(N)C(O)=O)c1)c1ccc2ccccc2c1 |r|
C[C@@H](Nc1nc(N)nc(n1)-c1ccc(CC(N)C(O)=O)c(F)c1)c1ccc2ccccc2c1 |r|
C[C@H](c1ccc2ccccc2c1)Nc3nc(nc(n3)N)c4ccc(cc4)C[C@@H](C(=O)O)N
Cc1ccccc1c2ccccc2CNc3cnc(cn3)c4ccc(cc4)C[C@@H](C(=O)O)N
N[C@@H](Cc1ccc(cc1)-c1cnc(NCc2ccc(cc2)-c2ccccc2)cn1)C(O)=O |r|
COc1ccc(CNc2cnc(cn2)-c2ccc(C[C@H](N)C(O)=O)cc2)cc1OC |r|
CCn1c2ccccc2c2cc(CNc3cnc(cn3)-c3ccc(C[C@H](N)C(O)=O)cc3)ccc12 |r|
COc1ccc(CNc2cnc(cn2)-c2ccc(C[C@H](N)C(O)=O)cc2)c(OC2CCCC2)c1 |r|
N[C@@H](Cc1ccc(cc1)-c1cnc(NCc2ccc3ccccc3c2)cn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cnc(NCC2CCc3ccccc3C2)cn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cnc(NCc2cnc3ccccc3c2)cn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cnc(NCc2ccccn2)cn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cnc(NCc2ccc(cc2)C#N)cn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1cnc(NCc2ccoc2)cn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCC2CCCCC2)n1)C(O)=O |r|
Cc1ccc(CNc2nc(N)nc(n2)-c2ccc(C[C@H](N)C(O)=O)cc2)cc1C |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2ccc(cc2)C(F)(F)F)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2ccccc2)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2ccc(cc2)-c2ccccc2)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2ccccc2-c2ccccc2)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2cccc(c2)-c2ccccc2)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2ccc(Oc3ccccc3)cc2)n1)C(O)=O |r|
Cc1ccc(cc1)-c1ccc(CNc2nc(N)nc(n2)-c2ccc(C[C@H](N)C(O)=O)cc2)cc1 |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NCc2ccc(cc2)-c2ccc(cc2)C(F)(F)F)n1)C(O)=O |r|
CC(Nc1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc(cc1)-c1ccccc1 |r|
CC(Nc1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)C12CC3CC(CC(C3)C1)C2 |r,TLB:1:22:25:29.27.28,THB:27:26:23:29.28.30,27:28:25.26.31:23,30:28:25:31.22.23,30:22:25:29.27.28|
C[C@H](Nc1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
CC(C)(Nc1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(OC(c2ccc3ccccc3c2)C(F)(F)F)n1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)-c1nc(N)nc(NC(c2ccc3ccccc3c2)C(F)(F)F)n1)C(O)=O |r|
C[C@@H](N(C)c1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
CCC(Nc1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
CC(C)CC(Nc1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
CC(C)C(Nc1nc(N)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
N[C@@H](Cc1ccc(cc1)-c1nc(NCc2ccc3ccccc3c2)nc(n1)N1CCOCC1)C(O)=O |r|
CNc1nc(N[C@H](C)c2ccc3ccccc3c2)nc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1 |r|
CC(Nc1ncnc(n1)-c1ccc(C[C@H](N)C(O)=O)cc1)c1ccc2ccccc2c1 |r|
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(=O)NCC(=O)OCC)[C@@]1(C)Cc1nc3ccccc3nc1C2(C)C |r,t:9|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCN(C[C@H](N)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CC2CCC(C1)N2C[C@H](N)C(O)=O)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCCN(C[C@H](N)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CC2CCC(C1)C2NCC(O)=O)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CC2CCC1CN2C[C@H](N)C(O)=O)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1C2CCC1CN(C[C@H](N)C(O)=O)C2)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CCNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC(CC1)C(N)CC(O)=O)C(F)(F)F |r|
CC1CN(CC(C)C1NCC(O)=O)c1cc(O[C@H](c2ccc(Cl)cc2-n2ccc(C)n2)C(F)(F)F)nc(N)n1 |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)-c1ccc(NS(C)(=O)=O)cc1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC(C)(CC1)NCC(O)=O)C(F)(F)F |r|
CN1CC2(C[C@H]1C(O)=O)CCN(CC2)c1cc(O[C@H](c2ccc(Cl)cc2-n2ccc(C)n2)C(F)(F)F)nc(N)n1 |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(Oc2ccccc2)n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1ccnc(c1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(O)n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1nc(N)nc(n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(N)nc(n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cnc(cn1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cnnc(c1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cncc(n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC(CC1)NCC(O)=O)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)[C@@H]1CCN(C[C@H](N)C(O)=O)C1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC(CCC(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1C2CC1CN(C[C@H](N)C(O)=O)C2)C(F)(F)F |r,THB:17:22:34.26.27:24|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC(CNCC(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CCC(N2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CC2CC(C1)N2C[C@H](N)C(O)=O)C(F)(F)F |r,THB:29:28:22.23.27:25|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC(CC1)Nc1nn[nH]n1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CNC(C2)C(O)=O)C1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)C#CC[C@H](N)C(O)=O)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CC2(C1)CNC(C2)C(O)=O)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(C)n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1ccn(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(NC2CCCCC2)n1)N1CCC2(CNC(C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1cn(cn1)-c1ccccc1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1-n1cncn1)C(O)=O |r|
Cc1ccn(n1)-c1ccccc1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1-n1cccn1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1-n1nccn1)C(O)=O |r|
CN\C(NCc1ccccc1-c1ccccc1)=N/C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
CN(Cc1ccccc1-c1ccccc1)C(\N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)Nc1ccccc1-c1ccccc1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCCCc1ccccc1-c1ccccc1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCCc1ccccc1-c1ccccc1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccc(cc1)-c1ccccc1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1cccc(c1)-c1ccccc1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1-c1ccccc1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1)C(O)=O |r|
[#7]-[#6@@H](-[#6]-c1ccc(cc1)-[#6](=O)\[#7]=[#6](\[#7])-[#7])-[#6](-[#8])=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(OC2CCCCC2)cccc1N1CCCCC1)C(O)=O |r|
CC(C)Oc1cccc(N2CCCCC2)c1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2ccccc2)cccc1N1CCCCC1)C(O)=O |r|
COc1ccc(Oc2cccc(N3CCCCC3)c2CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2ccccc2Cl)cccc1N1CCCCC1)C(O)=O |r|
Cc1ccc(Oc2cccc(N3CCCCC3)c2CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2cccc(c2)C(F)(F)F)cccc1N1CCCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2ccc(Cl)cc2)cccc1N1CCCCC1)C(O)=O |r|
Cc1ccccc1Oc1cccc(N2CCCCC2)c1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2ccccc2C(F)(F)F)cccc1N1CCCCC1)C(O)=O |r|
COc1ccccc1Oc1cccc(N2CCCCC2)c1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
Cc1cccc(Oc2cccc(N3CCCCC3)c2CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2cccc(Cl)c2)cccc1N1CCCCC1)C(O)=O |r|
COc1cccc(Oc2cccc(N3CCCCC3)c2CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2ccc(cc2)C(F)(F)F)cccc1N1CCCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccc(Cl)cc1N1CCCCC1)C(O)=O |r|
Cc1ccc(CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c(c1)N1CCCCC1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1cccc(Cl)c1N1CCCCC1)C(O)=O |r|
COc1ccc(CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c(c1)N1CCCCC1 |r|
Cc1cccc(CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c1N1CCCCC1 |r|
COc1cccc(CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c1N1CCCCC1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(cccc1-c1ccccc1)N1CCCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Cl)cccc1N1CCCCC1)C(O)=O |r|
Cc1ccc(N2CCCCC2)c(CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c1 |r|
COc1ccc(N2CCCCC2)c(CN\C(N)=N\C(=O)c2ccc(C[C@H](N)C(O)=O)cc2)c1 |r|
COc1cccc(N2CCCCC2)c1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1cc(Cl)ccc1N1CCCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1cc(ccc1N1CCCCC1)-c1ccccc1)C(O)=O |r|
Cc1cccc(N2CCCCC2)c1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(cccc1C(F)(F)F)N1CCCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1cc(ccc1N1CCCCC1)-c1nccs1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCOCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCC(O)CC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCSCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCC(CC1)c1ccccc1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CC2CC2C1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCC(Cc2ccccc2)CC1)C(O)=O |r|
COC1CCN(CC1)c1ccccc1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
CC1CC(C)CN(C1)c1ccccc1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
CC1CCCN(C1)c1ccccc1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
CC1CCCCN1c1ccccc1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CC2CCC1C2)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCC1)C(O)=O |r|
CCN(CC)c1ccccc1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
CCOc1cccc(N2CCCCC2)c1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(OC2CCC2)cccc1N1CCCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCCCC1)C(O)=O |r|
Cc1cccc(N2CCCCCC2)c1CN\C(N)=N\C(=O)c1ccc(C[C@H](N)C(O)=O)cc1 |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1ccccc1N1CCCCCC1)C(O)=O |r|
N[C@@H](Cc1ccc(cc1)C(=O)\N=C(/N)NCc1c(Oc2ccccc2)cccc1N1CCCCCC1)C(O)=O |r|
Nc1nc(O[C@H](c2ccc(cc2)-c2ccc3[nH]ncc3c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Cc1ccn(n1)-c1cc(ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F)-c1ccc(Cl)c(Cl)c1 |r|
Cc1ccn(n1)-c1cc(ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F)-c1ccc(C)c(C)c1 |r|
c1ccc(cc1)c2cc(ccc2[C@H](C(F)(F)F)Oc3cc(nc(n3)N)N4CCC5(CC4)C[C@H](NC5)C(=O)O)Cl
Nc1nc(O[C@H](c2ccc(Cl)cc2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
CS(=O)(=O)c1ccc(cc1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
CCOc1ccc(cc1Cl)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1cccc(n1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cccnc2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Cc1cc(ccc1Cl)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2ccc(Cl)cc2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
CS(=O)(=O)Nc1cccc(c1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2ccc(F)c(F)c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cc(F)cc(Cl)c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cccc(F)c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cccc(Cl)c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Cc1cccc(c1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
CC(C)(C)c1cccc(c1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cccc(c2)C(F)(F)F)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
COc1cccc(c1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Nc1nc(O[C@H](c2ccc(cc2)-c2ccc3cnccc3c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
CSc1ccc2cc(ccc2n1)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Cn1ncc2cc(ccc12)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1nn(C)c2cc(ccc12)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Cc1n(C)nc2cc(ccc12)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(cc2)-c2ccc3ncc(F)cc3c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
COc1ccc(cc1)-c1ccc([C@@H](Oc2cc(nc(N)n2)N2CCC3(CN[C@@H](C3)C(O)=O)CC2)C(F)(F)F)c(c1)-n1ccc(C)n1 |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2ccc(cc2)S(N)(=O)=O)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cccc(c2)N2CCCC2=O)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
CN(C)S(=O)(=O)c1cccc(c1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
NC(=O)c1cccc(c1)-c1cc(Cl)ccc1[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cccc(c2)C#N)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
Nc1nc(O[C@H](c2ccc(Cl)cc2-c2cc(F)cc(F)c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
CS(=O)(=O)c1cccc(c1)c2cc(ccc2[C@H](C(F)(F)F)Oc3cc(nc(n3)N)N4CCC5(CC4)C[C@H](NC5)C(=O)O)Cl
Nc1nc(O[C@H](c2ccc(cc2)-c2ccc3NC(=O)CCc3c2)C(F)(F)F)cc(n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1 |r|
CN1CCc2cc(ccc2C1=O)-c1ccc(cc1)[C@@H](Oc1cc(nc(N)n1)N1CCC2(CN[C@@H](C2)C(O)=O)CC1)C(F)(F)F |r|