1984 SMILES Strings for WD repeat-containing protein 5

Compound Name
SMILES String
COc1cccc(c1)C(=O)N(CC1CC1)C1CCc2ccc(cc12)-c1cn2CCCc2n1
Cc1ccc(cc1C(F)(F)F)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
COc1cc(ccc1C)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
CCOc1cccc(c1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
COc1cc(C)cc(c1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
Clc1ccc(CC(=O)NC2CCc3ccc(cc23)-c2cn3CCCc3n2)cc1Cl
CC(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
CCC(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
FC(F)(F)CC(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
CC(C)C(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1
Clc1ccc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)cc1Cl |r|
COc1cc(ccc1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
CC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
COc1cc(ccc1C)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Fc1cc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)ccc1Cl |r|
CCC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
CC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1 |r|
CCC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1 |r|
COc1ccc(cn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Clc1cc(ccn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Cc1cnc(Cl)c(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Cc1cc(cc(=O)[nH]1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Cc1cc(Cl)nc(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Cc1cc(ccn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Cc1ccc(cc1O)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
COc1cncc(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
CC(=O)Nc1cc(ccc1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Cc1ccc(C(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)c(Cl)n1 |r|
COc1cc(cc(OC)c1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
Fc1cnccc1C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
O=C(N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1)c1ccc(=O)[nH]c1 |r|
Fc1cncc(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1 |r|
COc1cc(ccc1C)C(=O)N[C@@H]1CCN(C(C)=O)c2ccc(cc12)-c1cn2CCCc2n1 |r|
Fc1ccc(c(Cl)c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NC(C1CC1)C1CC1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2Cl)cc(OC)c1 |t:14|
Clc1cc(Cl)cc(CNC(=O)c2cc(Cl)cc(Cn3ccnc3)c2)c1
COc1cc(CNC(=O)c2cc(Cl)cc(Cn3ccnc3)c2)cc(OC)c1
Cc1ccc(CNC(=O)c2cc(Cl)cc(Cn3ccnc3)c2)cc1Cl
COc1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1
COC(=O)CC(NC(=O)c1cc(Cl)cc(Cn2ccnc2)c1)c1cccc(Cl)c1
Cc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(OC3CCCC3)c2)ccc1Cl
Fc1ccc(c(Cl)c1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1ccccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2cccnc2)cc1Cl
Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccco2)cc1Cl
COc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(Oc3ccccc3)c2)cc(OC)c1
Cc1ccncc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1ccc(Cl)c(c1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1cc(ccn1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
FC(F)(F)c1ccccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccncc2Cl)cc1Cl
Cc1nc(F)ccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Fc1ccc(-c2cc(Cn3ccnc3)cc(c2)C(=O)NCc2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F
COc1cncc(c1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cnccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccoc2C)cc(OC)c1
Cn1nccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
CC(NC(=O)c1cc(Cn2ccnc2)cc(c1)-c1ccc(F)nc1C)C1CCCCC1
Cc1nc(F)ccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NC(C1CC1)C1CC1
Cc1nccn1Cc1cc(cc(c1)-c1ccc(F)cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1
Fc1ccc(c(Cl)c1)-c1cc(Cn2ccnc2C(F)(F)F)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)N2CCCC2)cc1Cl
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccnc2)cc(c1)-c1ccc(F)nc1C)C1CC1
Fc1ccc(c(Cl)c1)-c1cc(Cn2ccnc2)cc(n1)C(=O)NCc1cc(Cl)cc(Cl)c1
CC(C)(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)C1CC1
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)C1CC1
Cc1cccc(CNC(=O)c2cc(Cn3ccnc3)cc(n2)-c2ccc(F)cc2Cl)n1
CCC(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)C1CC1
Cc1cc(C)cc(CNC(=O)c2cc(Cn3ccnc3)cc(n2)-c2ccc(F)cc2Cl)c1
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl
CC(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)c1ccccn1
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1ccc(F)cc1C |t:21|
COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cc1OC |t:15|
Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)ccc1Cl |t:13|
Cc1cc(C)cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)c1 |t:16|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1ccc(F)nc1C |t:21|
COc1cc(CN(C)C(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1 |t:15|
Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1ccc(F)nc1C)C1CC1 |t:17|
Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NC(C1CC1)C1CC1 |t:14|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)c1 |t:16|
Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:13|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)cc(OC)c1 |t:14|
COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)cc1Cl |t:15|
COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cc1OC |t:15|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(F)cc(Cl)c1 |t:13|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)ccc1Cl |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)ccc1Cl |t:14|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)c1 |t:16|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cnccc1C |t:21|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)c1 |t:16|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)ccn1 |t:13|
COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cc1Cl |t:15|
Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(F)cc(Cl)c1 |t:13|
Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cnccc1C)C1CC1 |t:17|
Cc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cn1 |t:14|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)cn1 |t:13|
Cc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)cn1 |t:14|
Cc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)n1 |t:15|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(F)c(C)c2)cc(OC)c1 |t:14|
Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(F)c(C)c2)ccc1Cl |t:13|
Cc1cccc(Oc2cc(CNC3=NCCN3)cc(c2)C(=O)NCc2ccc(Cl)c(Cl)c2)c1 |t:12|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)C(F)(F)F |t:21|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(OC)c(Cl)c2)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(F)c(Cl)c2)cc(OC)c1 |t:14|
Cc1cnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cn1 |t:14|
Cc1ncc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cn1 |t:14|
Cc1cnc(F)c(c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)ccn1 |t:14|
Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cc(C)cnc1F)C1CC1 |t:17|
CN(C)C(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cc(C)cnc1F |t:10|
Cc1cc(cc(C)n1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1 |t:14|
Cc1cnc(F)c(c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1 |t:14|
CN1CC(=O)N=C1NCc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1 |c:5|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NC(=O)CN2C)cc(c1)-c1ccc(F)nc1C |t:21|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(ccc2OC)C(C)C)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(cnc2OC)C(F)(F)F)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2C(F)(F)F)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(F)cnc2OC)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2OC)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)c(F)cc2OC)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)c(F)cc2C)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)c1 |t:16|
CC(NC(=O)c1cc(CNC2=NCCC2)cc(c1)-c1ccc(F)nc1C)c1cc(C)c(Cl)cn1 |t:10|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCC2)cc(c1)-c1ccc(F)nc1C |t:21|
COc1cc(CN(C)C(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1 |t:15|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccnc(C)c2)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cccn2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)cc2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccncc2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cc(C)c(F)cc2C)cc(OC)c1 |t:14|
Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cccc(CO)c2)ccc1Cl |t:13|
Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)cc2C)ccc1Cl |t:13|
Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)c(CO)c2)ccc1Cl |t:13|
Cc1cc(c(C)cc1F)-c1cc(CNC2=NCCC2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1 |t:15|
Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cccnc2C(F)(F)F)ccc1Cl |t:13|
Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)cc2C(F)(F)F)ccc1Cl |t:13|
COc1cc(F)c(C)cc1-c1cc(CNC2=NCCC2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1 |t:16|
COc1cc(F)ccc1-c1cc(CNC2=NCCC2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1 |t:15|
CN1CC(=O)N=C1NCc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(C)c1 |c:5|
Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:14|
Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(F)c1 |t:14|
Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)ccc1Cl |t:13|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(n1)-c1ccc(F)nc1C |t:21|
Cc1cnc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)cn1 |t:14|
Cc1cnc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)nc1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)ccn1 |t:14|
Cc1ncc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)cn1 |t:14|
Cc1ccncc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:13|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:13|
COc1ncc(C)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:15|
Cc1cnccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:13|
Cc1cc(C)nc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)n1 |t:16|
COc1ncc(Cl)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:15|
COc1ccc(C)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:15|
CCOc1ncc(C)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:16|
Fc1ccc(-c2cc(CNC3=NCCC3)cc(n2)C(=O)NCc2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F |t:10|
Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)C1CC1 |t:17|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)nc(c2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1 |t:14|
C[C@H](NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(C)c1 |r,t:10|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F |t:21|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C(F)(F)F)c1 |t:16|
Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C)C1CC1 |t:17|
CC(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1cc(C)c(Cl)cn1 |t:10|
C[C@H](NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F |r,t:10|
Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(=O)[nH]c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)cc(OC)c1
Cc1cc(ccn1)-c1cc(CNC(N)=N)cc(c1)C(=O)NCc1cc(F)cc(Cl)c1
COc1ccc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)cc1Cl
COc1ccnc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)c1
Cc1cc(ccn1)-c1cc(CNC(N)=N)cc(c1)C(=O)NCc1ccc(Cl)cn1
Cc1ccc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)cn1
CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2CC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2CCC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)CC2CC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2CCOC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2(C)CC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CC1(CCCC1)NC(=O)c1cc(Cn2ccnc2)cc(c1)-c1ccc(F)cc1Cl
Cc1nc(F)ccc1-c1cc(Cn2ccnc2C2CC2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(CN(C)C(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1
FC(F)(F)c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(OC3CCC3)c2)cc1Cl
Cc1nccn1Cc1cc(OC2CCC2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1nccn1Cc1cc(cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1)N1CCOCC1
COc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccc(=O)[nH]c2)cc(OC)c1
COc1ccnc(CNC(=O)c2cc(C)c(OC)c(Cn3ccnc3C)c2)c1
Cc1cncn1Cc1cc(nc(c1)-c1cccc(CO)c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1nccn1Cc1cc(nc(c1)-c1ccc(F)cc1C)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1cccc(CO)c1
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)cc1OC
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)nc1C
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1cc(ccc1OC)C(F)(F)F
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)c(c1)C(N)=O
COc1ncccc1-c1cc(Cn2ccnc2C)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)c(CO)c1
Cc1nccn1Cc1cc(nc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(F)ccc1-c1cc(Cn2ccnc2C)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1nccn1Cc1cc(nc(c1)-c1ccncc1C)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1nccn1Cc1cc(nc(c1)-c1ccc(F)c(c1)C(N)=O)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2N)-c2ccc(F)cc2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2N)-c2ccc(F)cc2C)cc(OC)c1 |t:14|
CNc1c(cc(CNC2=NCCC2)cc1-c1ccc(F)cc1C)C(=O)N(C)Cc1cc(OC)cc(OC)c1 |t:8|
CNc1c(cc(CNC2=NCCN2)cc1-c1ccc(F)cc1C)C(=O)N(C)Cc1cc(OC)cc(OC)c1 |t:8|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2NC(C)=O)-c2ccc(F)cc2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2NC(C)=O)-c2ccc(F)cc2C)cc(OC)c1 |t:14|
Clc1cc(Cl)cc(CNC(=O)c2cccc(CNC3=NCCN3)c2)c1 |t:18|
CC(C)N(Cc1cccc(Cl)c1)C(=O)c1cccc(CNC2=NCCN2)c1 |t:22|
Clc1ccc(CNC(=O)c2cccc(CNC3=NCCN3)c2)cc1Cl |t:16|
Cc1cc(CNC(=O)c2cccc(CNC3=NCCN3)c2)ccc1Cl |t:15|
CC(NC(=O)c1cccc(CNC2=NCCN2)c1)c1cccc(Cl)c1 |t:12|
Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:10|
Cc1cc(C)cc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)c1 |t:19|
Clc1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:6|
Clc1cc(Cl)cc(CNC(=O)c2cc(Cl)cc(CNC3=NCCN3)c2)c1 |t:19|
Cc1ccc(CNC(=O)c2cc(Cl)cc(CNC3=NCCN3)c2)cc1Cl |t:17|
Cc1cc(C)cc(CNC(=O)c2cc(Cl)cc(CNC3=NCCN3)c2)c1 |t:19|
CC(NC(=O)c1cc(Cl)cc(CNC2=NCCN2)c1)c1cccc(Cl)c1 |t:13|
COc1cc(CNC(=O)c2ccc(Cl)c(CNC3=NCCN3)c2)cc(OC)c1 |t:17|
Clc1cc(Cl)cc(CNC(=O)c2ccc(Cl)c(CNC3=NCCN3)c2)c1 |t:19|
COc1cc(cc(c1)OC)CNC(=O)c2ccc(c(c2)CNC3=NCCN3)F
Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1cc(Cl)ccn1 |t:10|
Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1cc(Cl)cc(Cl)c1 |t:10|
COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(F)c(CNC2=NCCN2)c1 |t:24|
COc1ccc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)cc1OC |t:18|
Cc1ccnc(c1)C(NC(=O)c1ccc(F)c(CNC2=NCCN2)c1)C1CC1 |t:20|
COc1cc(CNC(=O)c2cccc(CNC3=NCCN3)c2F)cc(OC)c1 |t:16|
COc1ccnc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)c1 |t:19|
Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)cn1 |t:10|
COc1cc(CN(C)C(=O)c2ccc(F)c(CNC3=NCCN3)c2)cc(OC)c1 |t:18|
COc1cccc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)n1 |t:19|
COc1ccc(cc1Cl)C(=O)NCc1ccc(F)c(CNC2=NCCN2)c1 |t:22|
COc1cc(CNC(=O)c2ccc(OC)c(CNC3=NCCN3)c2)cc(OC)c1 |t:18|
COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:11|
Cc1ccnc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)c1 |t:18|
COc1cc(OC)cc(c1)C(=O)NCc1cc(F)c(F)c(CNC2=NCCN2)c1 |t:24|
Cc1cc(C)cc(CNC(=O)c2cc(F)c(F)c(CNC3=NCCN3)c2)c1 |t:20|
COc1ccc(CNC(=O)c2cc(F)c(F)c(CNC3=NCCN3)c2)cc1Cl |t:19|
Fc1cc(cc(CNC2=NCCN2)c1F)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:8|
COc1ccnc(CNC(=O)c2cc(F)c(F)c(CNC3=NCCN3)c2)c1 |t:20|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(F)c(F)c(CNC2=NCCN2)c1 |t:25|
Fc1ccc(CNC2=NCCN2)cc1C(=O)NCc1ccc(Cl)c(Cl)c1 |t:7|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)ccc2F)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2ccc(OC)c(CNC3=NCCN3)c2)ccc1Cl |t:18|
COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1cc(Cl)ccn1 |t:11|
COc1ccnc(CNC(=O)c2ccc(OC)c(CNC3=NCCN3)c2)c1 |t:20|
COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(F)c1 |t:11|
COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(C)c1 |t:11|
COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(OC)c(CNC2=NCCN2)c1 |t:25|
COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)cn1 |t:11|
Cc1cc(C)nc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)n1 |t:19|
Cc1cnc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)cn1 |t:17|
Cc1cc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)ccc1Cl |t:16|
Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)c(F)cc1F)C1CC1 |t:17|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)c(F)cc1F |t:21|
CCOc1ccc(cc1CNC1=NCCN1)C(=O)NC(C1CC1)c1cc(C)ccn1 |t:12|
CCOc1ccc(cc1CNC1=NCCN1)C(=O)NC(C)c1cc(OC)cc(OC)c1 |t:12|
COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(OC(C)C)c(CNC2=NCCN2)c1 |t:27|
CC(C)Oc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:13|
Fc1ccc(c(Cl)c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:14|
Cc1cc(C)cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2Cl)c1 |t:16|
Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2Cl)ccc1Cl |t:13|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1 |t:14|
Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cc(OC)c1 |t:14|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:13|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)cc(Cl)c1 |t:13|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1 |t:13|
Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)cc(Cl)c1 |t:13|
Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)ccc1Cl |t:13|
Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cccc(F)n1 |t:13|
Cc1cc(C)cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)c1 |t:16|
Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NC(C1CC1)C1CC1 |t:13|
Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cccc(F)n1 |t:13|
Cc1cc(cnc1F)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:14|
COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)cnc2F)cc1OC |t:15|
COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)cnc2F)cc(OC)c1 |t:14|
Cc1cc(cc(C)n1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)ccn1 |t:14|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2C)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(OC)ccc2OC)c1 |t:16|
COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(Cl)ccc2OC)c1 |t:16|
COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(OC(C)C)c(CNC2=NCCC2)c1 |t:27|
CC(C)Oc1ccc(cc1CNC1=NCCC1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:13|
Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)ccc1Cl |t:13|
Fc1ccc(c(F)n1)-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:14|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)ccn1 |t:21|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCC2)ccn1 |t:21|
Cc1cc(F)ccc1-c1cc(CNC2=NCCC2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1 |t:14|
Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C)ccc1Cl |t:13|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C)cc(OC)c1 |t:14|
COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1 |t:14|
CC(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1cc(Cl)c(C)cn1 |t:10|
COc1cc(OC)cc(c1)C(C)NC(=O)c1ccnc(CNC2=NCCN2)c1 |t:23|
COc1cc(OC)cc(c1)C(C)NC(=O)c1ccnc(CNC2=NCCC2)c1 |t:23|
Cc1nc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1ccccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
COc1ncc(C)cc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1
COc1ccnc(c1)[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1 |r|
COc1cc(c(F)cn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)nc1C)C1CC1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncnc2CCCCc12)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1 |r|
Cc1cc(F)ccc1-c1cc(Cn2ccoc2=N)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cc(C)cnc2OC)c1
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncnc2CCCCc12)C1CC1
Cn1ccn(Cc2cc(C(=O)NC3(CCC3)c3cccc(Br)c3)c(F)c(c2)-c2ccc(F)cc2C(F)(F)F)c1=N
CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncnc2CCCCc12)C1CC1
Cn1ccn(Cc2cc(cc(c2)-c2ncc(F)cc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c1=N |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cn(nc1C(F)(F)F)C1CCCC1)C1CC1 |r|
Cc1cc(F)ccc1-c1cc(Cn2cc[nH]c2=N)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1 |r|
Cc1cc(ccc1Cl)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnc(C)c1)C1CC1
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1
Cn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(F)c2)c1=N |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccncc2C)c1
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C(F)(F)F)ccc1Cl
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1 |r|
COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cc(C)ccc2OC)c1
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C(F)(F)F)C1CC1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C(=C)C(F)(F)F)C1CC1 |r|
Fc1cnc(-c2cc(CN3CCOC3=N)cc(c2)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccn1C)C1CC1
CC(C)n1nccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnn1C)C1CC1
CC(C)n1nccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@H](C1CC1)c1cc(C)ccn1 |r|
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1 |r|
COc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1
Cn1ccn(Cc2cc(nc(c2)-c2ccc(F)cc2C(F)(F)F)C(=O)NC(CC(O)=O)c2ccc(Cl)c(Cl)c2)c1=N
CC(c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1)C(F)(F)F |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1 |r|
COc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCC1CCOCC1
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cnccc1C)C1CC1
COC(=O)CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(Cl)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCC1CCCO1
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccncc2C)ccc1Cl
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C(F)(F)F)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCC1CCOC1
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccnn2C)ccc1Cl
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2F)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1
Cc1cc(CNC(=O)c2cc(Cn3cc[nH]c3=N)cc(c2)-c2cccn2C)ccc1Cl
COC(=O)CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(Cl)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccccc1C)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1
COc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2F)-c2ccc(F)cc2C(F)(F)F)ccc1Cl
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1
Cn1cccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1[nH]c(=O)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
CN1CCN(Cc2cc(cc(c2)-c2cn(C)nc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C1=N |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1
Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cnc(F)cc1C)C1CC1 |r|
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
C[C@H]1CN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C(=N)O1 |r|
COc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
CCn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c1=N |r|
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
C[C@@H]1CN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C(=N)O1 |r|
COc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCCC1)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1 |r|
Cc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
CCn1ccn(Cc2cc(cc(c2)-c2ccc(F)cc2C)C(=O)NCc2cc(OC)cc(OC)c2)c1=N
COc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cn1ccn(Cc2cc(cc(c2)-c2ccnn2C)C(=O)NCc2ccc(Cl)c(Cl)c2)c1=N
COc1cc(CNC(=O)c2cc(Cn3ccn(C4CC4)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCCC1)C1CC1 |r|
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1ccc2[nH]ncc2c1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnn1C(C)C)C1CC1
CCOc1c(cc(Cn2ccn(C)c2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C)c1ccc(F)c(C)c1 |r|
Fc1ccc(c(Cl)c1)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(F)c1 |r|
Cc1cc(F)cc(F)c1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1cccnc1C(F)(F)F)C1CC1 |r|
CCOc1c(cc(Cn2ccn(C)c2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCOc1c(cc(CN2CCOC2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C)c1ccc(F)c(C)c1 |r|
C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(C)c1 |r|
Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1 |r|
Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
CCOc1c(cc(CN2CCOC2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(C)c1 |r|
CC(=O)\N=c1/n(C)ccn1Cc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCOc1c(cc(Cn2ccoc2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F |r|
CCOC(=O)\N=c1/n(C)ccn1Cc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1
COc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cncnc1C(F)(F)F)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1 |r|
COc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)ccc3[nH]ncc23)ccc1Cl
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(F)c(Cl)c1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCN(C)C2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccsc3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1
COc1cc(CN(C)C(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)ccc3[nH]ncc23)cc(OC)c1
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCN(C)C2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1 |r|
COc1cc(CNC(=O)c2cc(CN3CCSC3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)ccc3[nH]ncc23)cc(OC)c1
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(cc1)C(F)(F)F |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1(CC1)C(F)(F)F)C1CC1 |r|
FC(F)Oc1cc(F)ccc1-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
CN1C(=O)CN(Cc2cc(cc(c2)-c2ccc(F)nc2C)C(=O)NCc2ccc(Cl)c(Cl)c2)C1=N
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1OC(F)F)C1CC1 |r|
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1(CC1)C(F)(F)F)C1CC1 |r|
Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C)C1CC1
Cn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)cn2)c1=N |r|
CN1CCN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(Cl)c2)C1=N |r|
FC(F)(F)c1ncccc1-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)ncn1
Cn1ccn(Cc2cc(CN[C@H]3CCc4cc(F)ccc34)cc(c2)-c2cccnc2C(F)(F)F)c1=N |r|
Cc1cccc(c1)C1(CCC1)NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1ncccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)C1CC1
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ncc(F)cn1 |r|
COc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1ncccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cncnc1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCC[C@@H]1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cn(nc1C(F)(F)F)C1CCCC1)C1CC1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)ccn1
Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCC[C@H]1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCSC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(C)nc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)n1
COc1cc(CNC(=O)c2cc(Cn3ccn(CC4CC4)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1
Cc1nccn1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1 |r|
COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)c1
CCn1cc(c(C)n1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Fc1cnc(-c2cc(CN3CCSC3=N)cc(c2)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F |r|
Cc1ncccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ncc(Cl)cn1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1OCC(F)(F)F)C1CC1 |r|
C[C@@H]1CCCN1c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Fc1ccc(cc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C(F)(F)F |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnc2CCCc12)C1CC1 |r|
C[C@@H]1COCCN1c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1 |r|
Cc1n[nH]c2cccc(-c3cc(Cn4ccn(C)c4=N)cc(c3)C(=O)NCc3ccc(Cl)c(C)c3)c12
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(-c3ccccc3)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Fc1ccc(c(Cl)c1)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1c(C)ccc2[nH]ncc12)C1CC1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(CC3CC3)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccoc3=N)cc(c2)-c2ccc(F)cc2Cl)cc(OC)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccsc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
COc1cc(CN(C)C(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccnc(C)c2)cc(OC)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1CC1)C1CC1 |r|
C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(C)c1 |r|
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)C1CC1
CN(Cc1ccc(Cl)c(Cl)c1)C(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cnc(F)nc1C
Cc1cc(ccc1F)[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)C(F)(F)F |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1
Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1nc(C)cc(C)n1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)C1CC1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(F)c1 |r|
Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ncc(Cl)cn1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F |r|
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccsc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2F)cc(OC)c1
CN1CCN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C1=N |r|
C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(Cl)c(C)c1 |r|
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2F)ccc1Cl
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(OC(F)(F)F)c2)cc(OC)c1
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1
COc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccsc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)C1CC1
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(OC)c1 |r|
CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)c1cc(C)c(Cl)cn1
Cn1ccn(Cc2cc(OC(F)(F)F)cc(c2)C(=O)N[C@@H](CC(O)=O)c2cccc(c2)C(F)(F)F)c1=N |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1
COc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C)ccc1Cl
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(OC(F)(F)F)c2)ccc1Cl
COc1cc(CNC(=O)c2cc(Cn3ccoc3=N)cc(c2)-c2ncc(F)cc2C)cc(OC)c1
Cc1nc(F)ccc1-c1cc(CN2CCCC2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)Nc1nc2ccccc2s1
Cn1ccn(Cc2cc(C(=O)N[C@@H](CC(O)=O)c3cccc(c3)C(F)(F)F)c(F)c(c2)-c2ccc(F)cc2C(F)(F)F)c1=N |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncc(F)cc1C)C1CC1
Cc1cc(c(C)cc1F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)c1ccc(Cl)c(Cl)c1 |r|
Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncc(F)cc1C)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2C)ccc1Cl
Cn1ccn(Cc2cc(cc(c2)-c2ccc(F)cc2OC(F)F)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c1=N |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
FC(F)Oc1cc(F)ccc1-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)C1CC1 |r|
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1
COc1cc(CNC(=O)c2cc(CN3CCN(C)C3=N)cc(c2)-c2ccc(F)cc2C(N)=O)cc(OC)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2OC(F)F)cc(OC)c1
Cn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c1=N |r|
COc1cc(CNC(=O)c2cc(Cn3ccoc3=N)cc(c2)-c2cccnc2C(F)(F)F)cc(OC)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1 |r|
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1
CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1 |r|
FC(F)(F)c1ncccc1-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(F)ccc1-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(F)cc1
COc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2C)cc(OC)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1 |r|
Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)C1CC1 |r|
Fc1ccc(cc1Cl)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1 |r|
Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ncc(F)cc2C)cc(OC)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1 |r|
COc1cc(OC)cc(c1)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccccc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C)C1CC1
Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c(=N)o1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C)C1CC1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCc1cn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c(=N)o1 |r|
Cc1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c(=N)c1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ncc(F)cc2C)ccc1Cl
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1coc(=N)n1Cc1cc(cc(c1)-c1cccnc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(F)c2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccccc2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1 |r|
CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
COc1cc(CNC(=O)c2cc(CN3CCOC3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1
CCOc1c(cc(Cn2ccccc2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cn(nc1C(F)(F)F)C1CCCC1)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cncnc1C(F)(F)F)C1CC1 |r|
CCOc1c(cc(Cn2cccc(F)c2=N)cc1C1=CN(C)NC1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r,t:20|
COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1
CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCc1coc(=N)n1Cc1cc(cc(c1)-c1cccnc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
CCOc1c(cc(Cn2cc(F)ccc2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1CCC1)C1CC1 |r|
C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(F)c(Cl)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(F)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C(F)(F)F)ccc1Cl
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1ccc(F)c(C)n1
C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(cc1)C(F)(F)F |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(F)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1
Cn1ccn(Cc2cc(cc(c2)-c2cccc3OC(F)(F)Oc23)C(=O)NCc2ccc(Cl)c(Cl)c2)c1=N
Cc1cc(ccc1F)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccccc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cnc(F)cc2C)cc(OC)c1
COc1cccc(n1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)n1
C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(F)cc1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cc(F)ccc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cnc(F)cc2C)ccc1Cl
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1OC(F)F)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cc(F)ccc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(=O)[nH]c2C)ccc1Cl
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1cccnc1C(F)(F)F)c1ccc(F)c(C)n1 |r|
C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ncc(F)cn1 |r|
COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c[nH]c(=O)cc2C)cc(OC)c1
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)nc1C(F)(F)F)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1OCC(F)(F)F)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)C1CC1
Cc1cc(=O)[nH]cc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)n1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)C1CC1)C1CC1 |r|
COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C)c1
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c[nH]c(=O)cc2C)ccc1Cl
Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1 |r|
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(n1)C(=O)NCc1ncc(Cl)cn1
Cn1ccn(Cc2cc(cc(c2)-c2ccc(F)cc2C(F)(F)F)C(=O)NC(CC(O)=O)c2ccc(Cl)c(Cl)c2)c1=N
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OCC2CC2)c1)C1CC1 |r|
FC(F)Oc1cc(F)ccc1-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(n1)C(=O)NCc1ccc(Cl)c(F)c1
CCC(=O)CNC(=O)CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(Cl)c1
CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C)c1ccc(F)c(C)c1 |r|
Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F |r|
COc1cc(CNC(=O)CC(NC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C(F)(F)F)c2ccc(Cl)c(Cl)c2)cc(OC)c1
CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cc(OC)cc(OC)c1
Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(n1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)ccc1F
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(OCC3CC3)c2)cc(OC)c1
FC(F)Oc1cc(F)ccc1-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cc(F)c(F)c(F)c1
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)C1CC1 |r|
FC(F)(F)c1ncccc1-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cnn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1 |r|
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(F)cc1
CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1 |r|
Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1
Cn1ccn(Cc2cc(cc(c2)-c2ccccc2C(F)(F)F)C(=O)NCc2ccc(Cl)c(Cl)c2)c1=N
C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OCC2CC2)c1)c1ccc(F)c(C)c1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1 |r|
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)nc(c2)-c2ccc(F)cc2C)cc(OC)c1
Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1 |r|
Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OCC2CC2)c1)C1CC1 |r|
Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1 |r|
COc1ccnc(CNC(=O)c2ccc(F)c(Cn3ccn(C)c3=N)c2)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCC(F)CC2)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCC(F)CC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1Cl
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1Cl)C(=O)NC1CCCCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1
C[C@H]1CN(Cc2ccc(F)c(c2)-c2ccc(N3CCN(C)CC3)c(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c2)C[C@@H](C)O1 |r|
COCOc1cc(F)c(cc1C(=O)NC(C)(C)CC(C)(C)C)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(N)=O)c(O)cc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OC(F)(F)F)ccc1F
CC(C)COc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(=O)[nH]n1)-c1cc(CN2CCOCC2)ccc1F
COc1cccc(c1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
COC(=O)c1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OCC2CC2)ncc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CNC2CCCCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1ccc(OC2CCOCC2)nc1F
CCOc1cc(c(nn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOCC2)ccc1F)C(F)(F)F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OCC2CC2)c(F)cc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1F)N1CCCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccccc1F
CC1CN(CCN1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F |r|
C[C@H]1CN(C)CCN1c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OC2CCOCC2)ncc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CNC2CCCC2)cc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CNC2CCCCC2)cc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC(C)(C)C)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)cc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(N2CCOCC2)c1F
CN(C)Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(c1)C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cnc(OCC[Si](C)(C)C)cc1C(F)(F)F)-c1cc(CNC2CCC(F)(F)CC2)ccc1F
CN(Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)C1COC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)N1CCOCC1 |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(O)cc(F)c1F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(CN2CCOCC2)ccc1F
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OCC2CC2)ncc1F |r|
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(C=O)ccc1F)C(F)(F)F
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCC(CC2)N2CCOCC2)ccc1F)C(F)(F)F
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CC[C@H](C2)C(C)C)ccc1F)C(F)(F)F |r|
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCN(CC2)C(C)=O)ccc1F)C(F)(F)F
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCC(F)CC2)ccc1F)C(F)(F)F
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2C3CC2COC3)ccc1F)C(F)(F)F
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCC(C2)S(C)(=O)=O)ccc1F)C(F)(F)F
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN(C)[C@H]2CCOC2)ccc1F)C(F)(F)F |r|
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOC(C)(C)C2)ccc1F)C(F)(F)F
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)cnc1F |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)cnc1F
CCN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CCN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F
CN1CCN(CC1COC(=O)C(C)(C)C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1CO)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCN(CC3CC3)CC2)ccc1F
CN(Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)C1CCCCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCN(Cc3ccc(F)cc3)CC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CC[C@@H](O)C2)ccc1F |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCC(CC2)N2CCOCC2)ccc1F
CN(C)[C@@H]1CCN(Cc2ccc(F)c(c2)-c2ccc(N3CCN(C)CC3)c(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c2)C1 |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCNCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2C3CC2COC3)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CC[C@H](C2)S(C)(=O)=O)ccc1F |r|
CN(Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)[C@H]1CCOC1 |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOC(C)(C)C2)ccc1F
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c(F)ccc(C#N)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)c(F)cc1F |r|
CN1CCN(CC1=O)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1
CC1CN(CCN1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)c(CNC2CCCCC2)c1F |r|
CN1CCN(CC1)c1ncc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ncc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F
CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCCN(CC1)c1ccc(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CNC(=O)c1ccc(F)c(c1)-c1ccc(N2C[C@H](C)N(C)[C@H](C)C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1 |r|
CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F
CN1CCCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CC1 |r|
CN1CC2CN(CC2C1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F
Cc1cc(cc(C)c1F)C(=O)Nc1cc(ccc1N1CCN(CC(F)(F)F)CC1)-c1cc(CN2CCOCC2)ccc1F
C[C@H]1CN(CCN1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncccc1F |r|
Fc1ccc(CN2CCOCC2)cc1-c1ccc(N2CCN(CC(F)(F)F)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1
CN1CCN(CC1)c1c(F)cc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(c(F)c1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CC2CN(CC2C1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(F)cc2[nH]cnc12)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1nc2ccccc2[nH]1)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(=O)[nH]c1)-c1cc(CN2CCOCC2)ccc1F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cnc(NC(C)=O)cc1C)-c1cc(CN2CCOCC2)ccc1F
COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCN(CC3CC3)CC2)ccc1F)C(F)(F)F
CNc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOCC2)ccc1F)C(F)(F)F
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cnc(N)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F
CN(C1CCCCC1)C(=O)c1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)N(C)C1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)c(CN(C)C2COC2)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN(C)C2COC2)c(F)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c(F)ccc(CNC2CCCCC2)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c(F)cc(CNC2CCCCC2)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1F)C(N)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1F)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(N)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F |r|
CC1CN(CC(C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(ncc1F)N1CCOCC1 |r|
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cccc(CN2CCOCC2)c1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCOc2c1
C[C@@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCCC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NC2CC2)nc1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NC2CCCCC2)nc1
CCOc1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)CC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(C)nc1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC2CCCCC2)nc1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(O)nc1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)C#N
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(OCC(F)(F)F)nc1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncnc1
COc1ncc(c(OC)n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)CC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1
CN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCOCC1 |t:31|
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCNCC1 |t:31|
CN1CCN(CC1)c1cc(F)ccc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(C)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)ccc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cnc(NC(C)=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCOCC1 |r|
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(C)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccnc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccncc1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CN(C)[C@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1 |r|
CN(C)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)CC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)nc1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CNC2CCCC2)c1
CC1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(c1)N1CCOCC1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(CN2CCOCC2)c1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(CNC2CCOCC2)c1
CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(CNC2CCOC2)c1
C[C@@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1 |r|
CN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1
CN1CCN(CC1)c1cc(Cl)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1
COc1cc(N2C[C@H](C)N(C)[C@H](C)C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1 |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1)C(F)(F)F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(C)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCOc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC(C)=O)nc1 |r|
COc1cc(=O)[nH]cc1C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OCC2CC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccccc1CNC1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(Cl)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCCCOc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCCOc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2N(C)CCOc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NC(C)=O)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccccc1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccccc1)-c1cnc(nc1)N1CCOCC1 |r|
COc1cc(ccc1F)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1n[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccccc1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccco1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cccnc1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(Cl)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(Cl)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(c1)N1CCOCC1 |r|
COCCOc1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(c1)N1CCOCC1 |r|
COc1ccccc1C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1Cl)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)ccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
COc1cccc(c1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
COCCOc1ccc(cc1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
CC(C)COc1ncc(cc1Cl)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)c(Cl)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCOCC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCNCC1 |r,t:33|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(Cl)c(O)c(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(OCc2ccccc2)c(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)C |r|
COc1cc(cnc1OC)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc2OCOc12)-c1cnc(nc1)N1CCOCC1 |r|
COc1ccc(cc1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)cc(c1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccccc1Cl)-c1cnc(nc1)N1CCOCC1 |r|
COc1cccc(C(=O)Nc2cc(c(F)cc2N2C[C@H](C)N(C)[C@H](C)C2)-c2cnc(nc2)N2CCOCC2)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(F)c1)-c1cnc(nc1)N1CCOCC1 |r|
COc1ccc(cc1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)cc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(NC(C)=O)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1nn(C)c2ccccc12)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1nn(C)c2ccccc12)-c1ccc(cc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN(C)C2COC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCC(F)CC2)c1 |r|
Fc1cc(N2CCN3CCOCC3C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1 |w:12.13|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cnn(C)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cnn(C)c1)-c1ccc(cc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(O)c(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(OCC2CC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(c1)N(C)C)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cocn1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCOCC1 |r|
CC(C)Oc1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(C#N)c(C)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(c1)C#N |r|
COc1cc(cc(n1)C(F)(F)F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
COc1cc(cc(C)n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
COc1ncc(cc1C(F)(F)F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
COc1cc(C#N)c(cn1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c(Cl)cccc1Cl)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N(C)C |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC(C)(C)C |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(F)(F)F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC(F)(F)F)cc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccccc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(Cl)cc1 |r|
COc1ccc(CN2CCC(=CC2)c2cc(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c(cc2F)N2C[C@H](C)N(C)[C@H](C)C2)cc1 |r,c:10|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnnc(C)c1 |r|
CC(C)CN1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:7|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC2CC2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CCC(F)(F)F)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccc(F)cc2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2cccnc2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccsc2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(OCC2CC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(O)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)cc(F)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2nccs2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2cnc(C)o2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2cnn(C)c2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccc(cc2)N2CCOCC2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccc(cc2)N2CCN(C)CC2)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC2CCOCC2)CC1 |r,t:33|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1ccc(cc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N2CCOCC2)c(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N2CCOCC2)c(C)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2NCCc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C(F)(F)F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C(=O)NC(C)(C)C |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)cc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn[nH]c1)-c1ccc(cc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(C)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C(N)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cncc(c1)C(F)(F)F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1nc(C)cs1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1csc(CN(C)C)n1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1n[nH]cc1Cl)-c1cnc(nc1)N1CCOCC1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cncnc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1scnc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(ccc1F)C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
COc1cc(F)cc(c1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1ccc(cc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccn(C)n1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc[nH]n1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1csc(C)n1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cnc(C)s1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC(C)=O)nc1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)C#N |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1sc(C)nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCCN(C)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(Cl)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccnc1OC1CCCCC1 |r|
COc1ccc(CC(=O)N2CCC(=CC2)c2cc(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c(cc2F)N2C[C@H](C)N(C)[C@H](C)C2)cc1 |r,c:12|
COCCOc1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1sccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)c(F)c(Cl)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1Cl)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN(C)C2COC2)c1 |r|
CCOc1cncc(c1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(NC(C)=O)nc1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)C#N |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N(C)C |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N(C)C)c(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N(C)C)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N2CCOCC2)c(Cl)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2OCCOc2c1 |r|
CN1CCN(CC1(C)C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccnc(c1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)cc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(F)c1F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1Cl)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C1CCCC1 |r,t:33|
COc1ccc(cc1)C(C)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:14|
CCC(C)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:7|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C1COC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CCNCC1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(O)nc1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1 |r|
CC(C)Oc1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2OCCOc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C1CCN(C)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)C(C)(C)C |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CCN(CC1)C(=O)C(C)(C)C |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncccn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)S(C)(=O)=O |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1ccc(OCC2CC2)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1Cl)-c1ccc(OCC2CC2)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(C)=O |r,t:33|
CCOC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:8|
CC(C)COC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:10|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)CC(C)(C)C |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CCN(CC1)C(=O)CC(C)(C)C |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)nc1 |r|
CN(C)C1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(Cl)c1)-c1cnc(nc1)N1CCOCC1 |r|
COc1cc(Cl)cc(c1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(Cl)c1F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(cc1C)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccccn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(C)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
COc1cc(ncn1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(Cl)cn1 |r,t:33|
CCOC(=O)c1ccnc(n1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:15|
CNC1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(O)cc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(O)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c(O)cnc2ccccc12)-c1cnc(nc1)N1CCOCC1 |r|
CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)N(C)C |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)N1CCCC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)N1CCN(C)CC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)Oc1ccccc1 |r,t:33|
C[C@H]1CC(C[C@@H](C)O1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(O)cc(F)c1F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OCC2CCC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OCC(C)(C)C)c1 |r|
CCN(CC)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(F)c1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)c(F)c(F)c1)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c(F)cccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCN(C)CC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCN(C)CC1 |r|
CCCN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)CN(C)C |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C(=O)CCC(O)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC(C)(C)C |r,t:34|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(OCC2CC2)nc1 |r|
CCn1cc(C(=O)Nc2cc(c(F)cc2N2C[C@H](C)N(C)[C@H](C)C2)-c2cnc(nc2)N2CCOCC2)c(cc1=O)C(F)(F)F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCN(C)CC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1Cl)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CC(C)(C)OC(C)(C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CC(C)(C)OC(C)(C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc([nH]n1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC(C)(C)C |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC(C)(C)C |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2C(=O)OC(C)(C)C |r,t:33,TLB:13:30:37:33.34|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC(C)(C)C |r,t:34|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC(C)(C)C |r,t:34|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2C(=O)OC(C)(C)C |r,t:34,TLB:13:31:38:34.35|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCNC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCNC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2 |r,t:33,TLB:13:30:37:33.34|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncccn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncccn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2c1ncccn1 |r,t:33,TLB:13:30:37:33.34|
C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CNC(=NC1)N1CCOCC1 |r,c:36|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CCN(C)[C@@H]1CN(C[C@H]1F)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CC(C)[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
CC(C)[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1C2CCC1CC2 |r|
C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)[C@H]1CCOC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)[C@H]1CCOC1 |r|
C[C@H]1CN(C[C@@H](C)N1)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
COc1cc(ncn1)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
COc1cnc(nc1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(F)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1nc(C)cc(C)n1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(C=O)cn1 |r,t:33|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)C1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)C1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)N(C)C |r,t:33|
CCOC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:8|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)N1CCCC1 |r,t:33|
COc1cnc(nc1)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(C)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(F)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N(C)C |r|
C[C@H]1CN(C[C@@H](C)N1C)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nn1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncccn1 |r,t:34|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)N1CCN(Cc2ccc(F)cc2)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)N1CCN(CC1)c1ncccn1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CO)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)S(C)(=O)=O |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCCN(C)CC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(cn1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CN(C)C)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CN2CCOCC2)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CN2CCN(C)CC2)cn1 |r,t:33|
CC(C)COC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:10|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(C=O)cn1 |r,t:33|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(OCC2CC2)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CO)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CN(C)C)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CN2CCOCC2)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CN2CCN(C)CC2)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CC[C@H](C1)N(C)C |r|
CCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1C[C@H](C)O[C@H](C)C1 |r|
CCN(CC)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CC(C)N(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CC[C@H](C1)N(C)C |r|
CCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1C[C@H](C)O[C@H](C)C1 |r|
CCN(CC)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
COc1cnc(nc1)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:11|
COc1cc(ncn1)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:11|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(C)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(F)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)N1CCCC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)c1cnccn1 |r,t:33|
CC(C)COC(=O)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:9|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(C=O)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnn(C)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C#N |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C1CC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C1CC1 |r|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(CN(C)C)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(CN2CCOCC2)cn1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(CN2CCN(C)CC2)cn1 |r,t:33|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
Fc1cc(N2C[C@@H]3CCN[C@@H]3C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1 |r|
CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC1(C)CCC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC1(C)CCC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC1(C)CCC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(n1)N1CCOCC1 |r|
C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
CCCN1CC[C@H]2CN(C[C@@H]12)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CN1CC[C@H]2CN(C[C@@H]12)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1 |r|
C[C@H]1CN(CC[N+]1(C)C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)NCC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N(C)CC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)NC1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N(C)C1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N1CCN(C)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC1(C)COC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC1(C)COC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC1(C)COC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)s1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccs1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccsc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(CN2CCOCC2)c1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)c(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)NCC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)N(C)CC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)NC1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)N(C)C1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)N1CCN(C)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(N)c(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccc(nn1)C1CC1 |r,t:33|
CCc1ccc(nn1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
COc1cc(c(cn1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1)C(F)(F)F |r|
C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc(N)c(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CCN1CC[C@H]2CN(C[C@@H]12)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NCC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)CC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NC1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)C1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCN(C)CC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(cc1)N1CCNCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCNCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NCC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)CC1CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NC1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)C1CCCCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCN(C)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(NC2CCCCC2)n1 |r|
CNc1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)N(C)C |r|
CNC1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(OCC2CC2)nc1 |r|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCNCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCNCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(F)c(c1)C(N)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C(C)(C)C |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCN(CC2CC2)CC1 |r|
Fc1cc(N2CCN(CC2)C2CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c[nH]c(=O)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(NC(=O)OCc2ccccc2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(=O)n(C)c1 |r|
COc1ccc(cc1)C(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:14|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2NC(=O)Cc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccn(C)c(=O)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(=O)n(C)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)C1CCCCC1 |r,t:33|
COCCCN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)c1cnccn1 |r,t:33|
COCCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)S(C)(=O)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NS(C)(=O)=O)nc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(cn1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)S(C)(=O)=O |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)S(C)(=O)=O |r,t:33|
CN(CC1CC1)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CN(CC1CC1)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(cn1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(F)c(c1)C(N)=O |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1 |r|
C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(F)c(c1)C(N)=O |r|
CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
CNC(=O)c1cc(ccc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nccc(n1)N1CCOCC1 |r|
CC(C)OC(=O)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:8|
CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:9|
CC(C)OC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:9|
CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
CNC(=O)c1cc(ccc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
CNC(=O)c1cc(ccc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOC[C@@H]1C |r|
C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(F)n1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)C(F)(F)F |r|
C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cc(C)c(F)c(C)c2)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)N1CCCC1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(s1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(s1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(s1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1csc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(s1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1csc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(s1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)N1CCCC1 |r,t:31|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1(C)CCC1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1(C)CCC1 |r,t:31|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(C(N)=O)c(F)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1CC(F)(F)C1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1CC(F)(F)C1 |r,t:31|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1cnc(nc1)C#N |r,t:31|
C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1nc(cs1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncco1 |r,t:33|
COc1cnc(nc1)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ncc(C=O)cn1 |r,t:32|
COc1cc(ncn1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:12|
CCOC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:8|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)c1ncccn1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(C=O)cn1 |r,t:32|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)C(=O)OC1(C)CCC1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1 |r|
CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(F)c(C(N)=O)c(F)c1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(F)c(C(N)=O)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(N)=O)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(F)c(C(N)=O)c(F)c1 |r|
C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cccc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1 |r|
CC(C)OC(=O)N1CCC=C(CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:9|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2n(C)cnc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2ncn(C)c2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc2scnc12 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2scnc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2ncsc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2n(C)cnc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2ncn(C)c2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cccc2scnc12 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2scnc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2ncsc2c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ncc(s1)C#N |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ncc(s1)C#N |r,t:31|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)c1ncc(s1)C#N |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)c1ncc(s1)C#N |r,t:31|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(s1)C#N |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(s1)C#N |r,t:32|
C[C@@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OC2CCOCC2)n1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(s1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(CC1)C(=O)OC1(C)CCC1 |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(CC1)c1ncc(s1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ccnc(n1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)C(=O)OC1CC(F)(F)C1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)C(=O)OC1CC(F)(F)C1 |r,t:31|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)C(=O)OC1CC(F)(F)C1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)C(=O)OC1CC(F)(F)C1 |r,t:31|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC1CC(F)(F)C1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC1CC(F)(F)C1 |r,t:32|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ccnc(n1)C#N |r,t:31|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccnc(n1)C#N |r,t:33|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)NC2CCCCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)NC2CCCCC2(C)C)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)NCC2CC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(CN2CCOCC2)n1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnn(CCN2CCOCC2)c1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnn(CCN2CCOCC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnn(CCN2CCOCC2)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnn(CCN2CCOCC2)c1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cccc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)F)-c1cnc(nc1)N1CCOCC1 |r|
CC(C)OC(=O)N1CCC=C(CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:9|
CC(C)OC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r,c:9|
CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r,c:9|
CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r,c:9|
CC(C)OC(=O)N1CCC(=CC1)c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r,c:9|
CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r,c:9|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(CC1)C(=O)OC1(C)CCC1 |r,t:32|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(CC1)C(=O)OC1CC(F)(F)C1 |r,t:32|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(CC1)c1ncc(s1)C#N |r,t:32|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC2CCCCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)N(C)CC2CC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC2CCC(F)(F)CC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NCC2CC2)c(F)c1 |r|
C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)c1ccnc(n1)C#N |r,t:31|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1nc(CN2CCOCC2)cs1 |r|
C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCNCC1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(C(=O)NC2CCCCC2(C)C)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ncc(CN2CCOCC2)s1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1csc(CN2CCOCC2)n1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(CN2CCOCC2)cs1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(CN2CCOCC2)s1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N(C)C2CCCCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N(C)C2CCCC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N[C@@H]2CCOC2)c(F)c1 |r|
C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N(C)C2COC2)c(F)c1 |r|
CN1CCN(CC1)c2ccc(cc2NC(=O)c3ccccc3Cl)[N+](=O)[O-]
CC(=O)Nc1ccc(cc1)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(ccc1OC(C)C)-c1cn2CCCc2n1
COc1cc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)ccc1C |r|
Cc1cncc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1
Cc1cccc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1
O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1ccncc1
COc1cccc(c1)C(=O)NCc1cc(ccc1OC(C)C)-c1cn2CCCc2n1
C1Cc2nc(cn2C1)-c1ccccc1
Cc1ccc(OCC(N)=N)cc1
Oc1ccc(cc1)-c1cn2CCSc2n1
CCOc1ccc(cc1)-c1cn2ccccc2n1
C1Cc2nc(cn2C1)-c1ccc(cc1)-c1ccccc1
C(Oc1ccc(cc1)-c1cn2CCCc2n1)c1ccccc1
Fc1cccc(c1F)-c1ccc(cc1)-c1cn2CCCc2n1
C1Cc2nc(cn2C1)-c1ccc2OCOc2c1
COc1cccc(c1)-c1cn2CCCc2n1
CC(=O)Nc1cccc(c1)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1
COc1ccc(cc1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1
O=C(Cc1ccccc1)NCc1cccc(c1)-c1cn2CCCc2n1
COc1cc(C)cc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1
O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1ccccn1
COc1cccc(c1)C(=O)N(C)Cc1cccc(c1)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)N(Cc1cccc(c1)-c1cn2CCCc2n1)C(C)C
COc1cccc(c1)C(=O)N(CC1CCC1)Cc1cccc(c1)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(OC)cc(c1)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(ccc1OC)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)NCc1cc(ccc1N(C)C)-c1cn2CCCc2n1
CN(C)c1ccc(cc1CNC(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1
CC(C)Oc1ccc(cc1CNC(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1
CC(C)Oc1ccc(cc1CN(CC1CC1)C(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1
Clc1ccc(CC(=O)NCc2cc(ccc2OC2CCC2)-c2cn3CCCc3n2)cc1Cl
NC(=N)COc1cccc(Cl)c1
CC(C)Oc1cccc(c1)-c1cn2CCCc2n1
CCC(C)Oc1ccc(cc1)-c1cn2CCCc2n1
O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1ccccc1
COc1cccc(c1)C(=O)N(CC1CC1)Cc1cccc(c1)-c1cn2CCCc2n1
COc1cccc(c1)C(=O)NCc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1
COc1cc(ccc1C)C(=O)N(CC1CC1)Cc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1
NC(=N)c1ccc(cc1)-c1ccccc1
COc1ccc(cc1)-c1cn2CCCc2n1
CN1CCc2cc(ccc12)-c1cn2CCCc2n1
O=C(NCc1cccc(c1)-c1cn2CCCc2n1)C1CCCCC1
Clc1ccc(CC(=O)NCc2cccc(c2)-c2cn3CCCc3n2)cc1Cl
O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1cccnc1
COc1cc(ccn1)C(=O)N(CC1CC1)Cc1cccc(c1)-c1cn2CCCc2n1
CCOc1ccc(cc1CN(CC1CC1)C(=O)c1cccc(OC)c1)-c1cn2CCCc2n1
Clc1ccc(CC(=O)NCc2cc(ccc2N2CCOCC2)-c2cn3CCCc3n2)cc1Cl
Clc1ccc(CC(=O)N(CC2CC2)Cc2cc(ccc2OC2CCC2)-c2cn3CCCc3n2)cc1Cl
CC(C)Oc1ccc(cc1)-c1cn2CCCc2n1
COc1cc(ccc1C)C(=O)NCc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1
COc1cc(ccc1C)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1
COc1ccc(cc1OC)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1
Cn1c(c(C2N(CC(O)=O)C(=O)c3ccccc23)c2ccccc12)-c1ccc(F)cc1
OC(=O)c1cc(NS(=O)(=O)c2ccc(Cl)cc2)cc(c1)C(O)=O
OC(=O)COc1ccc(Br)cc1C1C2=C(CCCC2=O)NC2=C1C(=O)CCC2 |c:23,t:14|
CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(Cl)cc1)c1ccc(Cl)cc1 |r|
CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 |r|
CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccccc1)c1ccccc1 |r|
CN1C2=C(C(C3=C1CCCC3=O)c1cc(Br)cc(Br)c1OCC(O)=O)C(=O)CCC2 |c:2,5|
CN1C2=C(C(C3=C1CCCC3=O)c1cc(Cl)ccc1OCC(O)=O)C(=O)CCC2 |c:2,5|
OC(=O)c1cccc(NS(=O)(=O)c2ccc(Cl)c3ccccc23)c1
CCCCOc1ccc(cc1C)S(=O)(=O)Nc1cccc(c1)C(O)=O
CCCCOc1ccc(cc1C)S(=O)(=O)Nc1ccc(cc1)C(O)=O
CN1C2=C(C(C3=C1CCCC3=O)c1cc(Br)ccc1OCC(O)=O)C(=O)CCC2 |c:2,5|
Cc1c(Cl)ccc(c1Cl)S(=O)(=O)Nc1cccc(c1)C(O)=O
CC[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@](C)(CCCCNC(=O)[C@H](NC1=O)c1ccccc1)NC(=O)C(C)C |r|
COc1cccc(c1)-c1[nH]c2ccccc2c1C1N(CC(O)=O)C(=O)c2ccccc12
COc1ccc(cc1C(C)(C)C)S(=O)(=O)Nc1ccc(cc1)C(O)=O
CCCCOc1ccc(cc1C)S(=O)(=O)Nc1ccccc1C(O)=O
OC(=O)c1ccc(NS(=O)(=O)c2cc(C(=O)Nc3ccccc3)c(Cl)cc2Cl)cc1
CCN1C2=C(C(C3=C1CCCC3=O)c1cc(Br)ccc1OCC(O)=O)C(=O)CCC2 |c:3,6|
Cc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)ccc1Cl
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cccc(OC(F)(F)F)c1
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccccc1
Cc1cccc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)c1
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cccc(Cl)c1
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1
Cc1cc(C)cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)c1
Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cc(Cl)cc(Cl)c1
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C5CC5)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(CN4CCSC4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(CN4CCCC4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4cnn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cccc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)c1
COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)ccc1F
Cc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)ccc1F
COc1cc(CN2CCc3c(cc(CNC(=N)C4CC4)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)ccc1Cl
COc1cc(CN2CCc3c(cc(Cn4ccoc4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1ccc(Br)cc1S(=O)(=O)Nc1cc(Cl)cc(c1O)S(C)(=O)=O
OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O
OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F
CNC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O
CNC(=O)c1cc(cc(c1O)NS(=O)(=O)c2cc(cc(c2O)Cl)Br)C3(CCC3)C#N
CS(=O)(=O)c1cc(cc(c1)S(F)(F)(F)(F)F)NS(=O)(=O)c2cc(ccc2O)Br
COc1ccc(Br)cc1S(=O)(=O)Nc1cc(ccc1O)C(C)(C)C
OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1
OC(=O)c1cc(OC(F)(F)F)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCCCC1)C#N
CCOc1cc(ccc1F)S(=O)(=O)Nc1ccccc1C(O)=O
CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)C1(CCC1)C#N
CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O
COc1ccc(cc1S(=O)(=O)Nc2cc(ccc2O)Cl)Br
Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1CC1
COc1ccc(Cl)cc1S(=O)(=O)Nc1cc(Cl)ccc1O
COc1ccc(Br)cc1S(=O)(=O)Nc1ccccc1O
Oc1ccc(Cl)cc1NS(=O)(=O)c1cc(Br)ccc1O
Oc1ccc(OC(F)(F)F)cc1NS(=O)(=O)c1cc(Br)ccc1O
Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)S(F)(F)(F)(F)F
Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CC1)C(F)(F)F
c1cc(c(cc1C2(CCC2)C#N)NS(=O)(=O)c3cc(ccc3O)Br)O
Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCCCC1)C#N
OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1CC1
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1CC1
OC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(C2CC2)c1F
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F
OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)C1(CCC1)C#N
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCCCC1)C#N
CNC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)ccc2O)cc(C2CC2)c1F
CNC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(C2CC2)c1F
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F
CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)C1(CCC1)C#N
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCCCC1)C#N
COCCNc1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N
CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1
CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)S(F)(F)(F)(F)F
CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)C1(CCC1)C#N
CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N
CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N
CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)S(F)(F)(F)(F)F
CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N
COc1ccccc1S(=O)(=O)Nc1cc(Cl)ccc1O
OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(OC(F)(F)F)c1
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F
CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2OC)c1O)C1(CCC1)C#N
COc1ccc(I)cc1S(=O)(=O)Nc1cc(Cl)ccc1O
Oc1ccc(Cl)cc1NS(=O)(=O)c1cccc(Br)c1
COc1ccc(Br)cc1S(=O)(=O)Nc1cc(ccc1O)-c1ccccc1
Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CC1)C#N
Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCCC1)C#N
OC(=O)c1cc(OC(F)(F)F)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O
CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F
Oc1ccc(Br)cc1S(=O)(=O)Nc1cc(cc(Nc2nc[nH]n2)c1O)C1(CCC1)C#N
CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1
CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)S(F)(F)(F)(F)F
COc1ccc(cc1S(=O)(=O)Nc2cc(cc(c2O)C(=O)O)Cl)Br
c1cc(c(cc1Br)S(=O)(=O)Nc2cc(c(c(c2O)C(=O)O)F)C3CC3)O
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N
CNC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCCCC1)C#N
COc1ccc(Br)cc1S(=O)(=O)Nc1ccc(Cl)cc1O
CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N
CCOc1ccc(c(C)c1C)S(=O)(=O)Nc1ccccc1C(O)=O
OC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)S(F)(F)(F)(F)F
CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O
OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CCCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)-c1ccccc1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)-c1ccccc1C(F)(F)F
CC(C)CCn1cnc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C(C1CC1)C1CC1
CC(C)n1cnc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CCC1
c1c(cc(c(c1S(=O)(=O)Nc2cn(cn2)C3CCCC3)O)Cl)Br
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CCNC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CC2)cn1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CCC2)cn1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CCCC2)cn1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CCCO2)cn1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C(=O)C1CCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C(=O)C1CCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1ncn(n1)C1CCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cc([nH]n1)C1CCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1ccn(n1)C1CCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cnn(c1)C1CCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cnc(s1)C1CCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1nc2ccccc2s1
Cc1nc(cn1C2CCCC2)NS(=O)(=O)c3cc(cc(c3O)Cl)Br
CCc1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1
CCOC(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1
OC(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1
CNC(=O)c1nc(cn1C2CCCC2)NS(=O)(=O)c3cc(cc(c3O)Cl)Br
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(C2CCCC2)c(n1)C(=O)N1CCC(CC1)C1CCCN1
COCCN1CCN(CC1)C(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1
Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(C2CCCC2)c(n1)C(=O)N1CC2(CNC2)C1
CS(=O)(=O)c1nc(cn1C2CCCC2)NS(=O)(=O)c3cc(cc(c3O)Cl)Br
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)C1CCOCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCN
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCCN)cc1
CN1CCC(CC1)C(=O)NCC#Cc1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)C1CCC(O)CC1 |(17.19,-25.43,;17.21,-23.89,;18.55,-23.13,;18.56,-21.59,;17.23,-20.81,;15.9,-21.57,;15.88,-23.11,;17.25,-19.27,;15.92,-18.49,;15.94,-16.95,;17.28,-16.19,;18.61,-16.97,;18.6,-18.51,;19.92,-19.3,;21.26,-18.54,;21.28,-17,;22.59,-19.32,;22.57,-20.86,;23.9,-21.64,;23.88,-23.18,;25.24,-20.88,;26.57,-21.66,;25.25,-19.34,;26.6,-18.58,;23.93,-18.56,;23.94,-17.02,;17.29,-14.65,;17.31,-13.11,;17.33,-11.57,;18.67,-10.81,;18.68,-9.27,;20.02,-8.51,;17.36,-8.49,;17.37,-6.95,;16.04,-6.17,;14.7,-6.93,;13.37,-6.14,;14.68,-8.47,;16.01,-9.25,)|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)CC1CCOCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)CCCCO
CC(C)C(N)C(=O)NCC#Cc1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN(C)C(=O)c1ccc(cc1)C(=O)NCC#Cc1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)c1ccc(cc1)C(=O)N1CCOCC1
COC(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(O)=O
CN(C)C(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)N1CCOCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NC1CCOCC1
CN1CCC(CC1)NC(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NCCCN1CCOCC1
CN1CCN(CC1)C(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NCCN1CCOCC1
COC(=O)c1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(cc1)C(=O)N1CCOCC1
CN1CCC(CC1)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CCOCC2)cc1
CN(C)C(=O)c1ccc(cc1)-c1cc(Nc2ncnc(Cl)c2N)c(cc1F)N1CCN(C)CC1
c1cc2c(cc1C(=O)O)ncn2C3CCCCC3
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)OC(C)(C)C
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCc1ccc(CC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)cc1 |r|
COc1ccc(cc1CNC(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOc2ccc(cc2CNC(=O)Cc2ccc(Cl)c(Cl)c2)-c2cn3CCCc3n2)C(C)(C)C)cc1 |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCc1ccc(CNc2ccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
CN1CCN(CC1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)c1ccc(cc1)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
CC[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](CCCCNC(=O)[C@H](NC1=O)c1ccccc1)NC(=O)C(C)C |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(cc1)C(=O)NCCCN
CN(C(=O)c1cc(N)c(F)c(C)c1Cl)c1cc(ccc1N1CCN(C)CC1)C(=O)Oc1ccccc1
[H][C@]12CS[C@@H](CCCCC(=O)NCCCCCC(=O)Nc3ccc(cc3)-c3ccc(N4CCN(C)CC4)c(NC(=O)c4cc(N)c(F)c(C)c4Cl)c3)[C@@]1([H])NC(=O)N2 |r|
[H]/N=C(\NC)/NCCC[C@H]1C(=O)N[C@H](C(=O)N[C@@H](C(=O)NCC[C@@](C(=O)N1)(C)NC(=O)C(C)C)c2ccccc2)CC
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3OC)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3O)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cccnc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cccnc3OC)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cc(C)cnc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cccnc3C(F)(F)F)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccncc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cc(C)ncc3C)C2=O)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2conc2C)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2cn(C)nc2C)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2c(C)nn(C)c2C)cc(OC)c1 |(-7.99,2,;-6.65,1.23,;-6.65,-.31,;-5.32,-1.07,;-5.32,-2.62,;-3.98,-3.39,;-2.65,-2.62,;-2.65,-1.08,;-1.32,-.31,;.02,-1.08,;1.35,-.31,;2.67,-1.08,;2.67,-2.61,;4,-3.38,;5.34,-2.61,;5.5,-1.08,;7,-.76,;7.77,-2.09,;9.31,-2.09,;6.74,-3.24,;7.14,-4.73,;1.35,-3.38,;.02,-2.62,;-1.32,-3.39,;-1.32,-4.93,;1.35,1.23,;2.59,2.13,;4.08,1.73,;2.12,3.6,;.58,3.6,;-.19,4.93,;.1,2.13,;-1.39,1.73,;-6.65,-3.39,;-7.98,-2.62,;-9.31,-3.39,;-9.31,-4.93,;-7.98,-1.08,)|
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2cc(C)nn2C)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc2C(=O)N(Cc3cc(OC)cc(OC)c3)CCc12
COc1cc(CN2CCc3c(cc(Cn4ccnc4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4cccn4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4cccc4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4cnnc4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
CCc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3cc(OC)cc(OC)c3)C(=O)c2c1
COc1cc(CN2CCc3c(cc(Cn4ccnc4C(C)C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccnc4C4CC4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
COc1cc(CN2CCc3c(cc(Cn4ccnc4C(F)F)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1
Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3ccccn3)C(=O)c2c1
Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3cccc(C)n3)C(=O)c2c1
Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3cc(C)ccn3)C(=O)c2c1
Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3ncccc3C)C(=O)c2c1
Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3ccnc(C)c3)C(=O)c2c1
COc1ccnc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)c1
CCc1ccnc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(Cc3cc(OC)ccn3)CCc12
CCc1ccnc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(CC)nc2C(F)(F)F)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@@H](C)c1cc(OC)ccn1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@H](C)c1cc(OC)ccn1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@H](C1CC1)c1cc(OC)ccn1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@@H](C1CC1)c1cc(C)ccn1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CCc12)[C@H](C)c1cc(OC)ccn1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CCc12)[C@@H](C1CC1)c1cc(OC)ccn1 |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CCc12)[C@H](C1CC1)c1cc(OC)ccn1 |r|
Clc1ccc(OCCCNC2=NCCN2)c(Cl)c1 |t:10|
CC(C)C[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](C)NC(=O)[C@@H](N)CS)[C@@H](C)O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CS)C(O)=O |r|
NCCCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](N)CS)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CS)C(O)=O |r|
C[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CS)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CS)C(O)=O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CS)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CS)C(O)=O |r|
CC(C)C[C@H](NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](N)CS)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CS)C(O)=O |r|
CC(C)C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CS)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CS)C(O)=O |r|
CC(C)[C@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCC(O)=O)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC(=O)CNC(=O)[C@@H](N)CS)C(=O)N[C@@H](CS)C(O)=O |r|
CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CSCc2ccc(CSC[C@H](NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](CC(N)=O)NC1=O)C(O)=O)cc2 |r|
CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CSC\C=C/CSC[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CC(N)=O)NC1=O)C(O)=O |r,c:27|
CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CSCc2cccc(CSC[C@H](NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](CC(N)=O)NC1=O)C(O)=O)n2 |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)CO)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C(C)C)C(O)=O |r|
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCc1c(F)cc(cc1F)-c1cccc(c1)S(F)(=O)=O
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CNC(=O)c1ccc(F)c(c1)-c1ccc(N2C[C@H](C)N(C)[C@H](C)C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)C(C)(C)C)c1ccc(cc1)-c1scnc1C |r|
COc1cc(CN2Cc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cc(CN2CCCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1
COc1cc(CN2COc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cc(Cn2cnc3c(cc(Cn4ccn(C)c4=N)cc3c2=O)-c2ccc(F)cc2C)cc(OC)c1
COc1cc(CN2CNc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1
COc1cc(CN2CCOc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1
COc1cc(CN2CC(=O)Nc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1
COc1cc(CN2CCNc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2c1OCCN([C@@H](C1CC1)c1cc(OC)ccn1)C2=O |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CNc12)[C@@H](C1CC1)c1cc(OC)ccn1 |r|
COc1cnc2cccc(N3CCc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1
CCc1cc(OC)c2nccc(N3CCc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1
COc1cnc2cccc(N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1
CCc1cc(OC)c2nccc(N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1
CCc1cc(OC)c2nccc(N3COc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1
COc1ccc2CCCC(N3CCOc4c(cc(Cn5ccnc5C)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2c1OCCN([C@H]1CCOc3ccc(OC)cc13)C2=O |r|
CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2c1OCCN([C@H]1CCOc3ccc(OC)cc13)C2=O |r|
COc1cnc2CCC[C@H](N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1 |r|
CCc1cnc2CCC[C@H](N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1 |r|
CCc1cc(C(=O)NC)c2nccc(N3CCc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1
CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)c1ccc(c(c1)C(O)=O)-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)COCCOCCNC(=S)Nc1ccc(c(c1)C(O)=O)-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(=O)N[C@H]1CC(=O)NCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)C(C)C)C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(O)=O)C(N)=O |wU:35.35,17.17,4.4,97.105,93.108,110.115,wD:26.26,8.8,2.2,82.86,89.92,117.122,(7.98,8.47,;7.98,6.93,;9.31,6.16,;10.65,6.93,;9.31,4.62,;7.98,3.85,;6.64,4.62,;6.64,6.16,;5.31,3.85,;5.31,2.31,;6.64,1.54,;6.64,0,;5.31,-.77,;7.98,-.77,;3.98,4.62,;2.64,3.85,;2.64,2.31,;1.31,4.62,;1.31,6.16,;2.64,6.93,;2.64,8.47,;1.31,9.24,;3.98,9.24,;-.02,3.85,;-1.36,4.62,;-1.36,6.16,;-2.69,3.85,;-2.69,2.31,;-1.36,1.54,;-1.36,0,;-2.69,-.77,;-.02,-.77,;-4.02,4.62,;-5.36,3.85,;-5.36,2.31,;-6.69,4.62,;-6.69,6.16,;-5.36,6.93,;-4.02,6.16,;-5.36,8.47,;-8.03,3.85,;-9.36,4.62,;-9.36,6.16,;-10.69,3.85,;-12.03,4.62,;-13.36,3.85,;-14.7,4.62,;-16.03,3.85,;-17.36,4.62,;-18.7,3.85,;-20.03,4.62,;-21.37,3.85,;-21.37,2.31,;-22.7,4.62,;-22.7,6.16,;-24.02,6.95,;-24,8.49,;-22.65,9.24,;-21.33,8.45,;-21.35,6.91,;-19.79,8.45,;-19.02,7.12,;-19.02,9.79,;-22.65,10.78,;-23.98,11.55,;-25.32,10.78,;-26.65,11.55,;-26.65,13.09,;-27.99,13.86,;-25.32,13.86,;-23.98,13.09,;-22.65,13.86,;-21.32,13.09,;-19.98,13.86,;-18.65,13.09,;-17.31,13.86,;-18.65,11.55,;-19.98,10.78,;-21.32,11.55,;10.65,3.85,;10.65,2.31,;11.98,4.62,;13.31,3.85,;13.31,2.31,;14.65,1.54,;15.98,2.31,;17.31,-3.08,;18.65,-2.31,;19.98,-3.08,;21.32,-2.31,;21.32,-.77,;19.98,0,;18.65,-.77,;19.98,1.54,;18.65,2.31,;18.65,3.85,;19.98,4.62,;17.31,4.62,;15.98,3.85,;14.65,4.62,;14.65,6.16,;17.31,6.16,;15.98,6.93,;18.65,6.93,;21.31,2.31,;21.31,3.85,;22.65,1.54,;22.65,-3.08,;23.98,-2.31,;22.65,-4.62,;23.98,-5.39,;25.32,-4.62,;25.32,-3.08,;26.65,-5.39,;23.98,-6.93,;22.65,-7.7,;25.32,-7.7,;25.32,-9.24,;23.99,-10.01,;23.99,-11.55,;22.65,-12.32,;21.32,-11.55,;22.65,-13.86,;26.65,-10.01,;26.65,-11.55,;27.99,-9.24,)|
CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(C)=O)C(=O)N[C@H]1CC(=O)NCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)C(C)C)C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(O)=O)C(N)=O |r|
CC(=O)NCC(=O)N[C@H](CO)C(=O)N[C@H](C)C(=O)N[C@H](CCCNC(=N)N)C(=O)N[C@H](C)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](C(=O)N[C@H](Cc1c[nH]cn1)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](CCCNC(=N)N)C(=O)N[C@H](CCCCN)C(=O)N[C@H](CO)C(N)=O)C(C)C
[#6]-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6])-[#7]-[#6](-[#6])=O)-[#6](-[#7])=O |r|
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2nn(C)cc12
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
CCNC(=O)C[C@@H]1N=C(c2ccc(Cl)cc2)c2cc(OC)ccc2-n2c(C)nnc12 |r,t:7|
CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O |r,wU:31.32,47.48,18.19,4.4,80.80,wD:52.55,8.15,36.44,69.69,22.28,89.89,(27.37,4.47,;27.37,2.95,;28.73,2.16,;26.02,2.16,;26.02,.64,;24.71,-.17,;23.37,.6,;23.37,2.12,;22.04,-.16,;22.04,-1.73,;23.37,-2.49,;24.77,-1.9,;25.79,-3.05,;25.01,-4.38,;23.51,-4.02,;20.72,.63,;19.39,-.15,;19.39,-1.72,;18.04,.63,;16.7,-.14,;15.35,.6,;15.35,2.12,;14.04,-.17,;14.04,-1.73,;15.35,-2.5,;15.35,-4.06,;14.01,-4.83,;16.68,-4.82,;12.71,.62,;11.39,-.17,;11.39,-1.74,;10.04,.6,;10.04,2.13,;8.7,-.16,;7.35,.59,;7.35,2.12,;6.03,-.17,;6.03,-1.73,;7.35,-2.5,;7.35,-4.07,;8.7,-4.81,;8.69,-6.35,;7.34,-7.14,;10,-7.07,;4.71,.63,;3.39,-.16,;3.39,-1.73,;2.04,.62,;2.04,2.14,;.68,-.11,;-.67,.62,;-.67,2.15,;-2,-.14,;-2,-1.7,;-.66,-2.46,;-3.29,.69,;-4.58,-.16,;-4.58,-1.7,;-5.93,.62,;-7.26,-.15,;-8.59,.62,;-9.92,-.15,;-8.59,2.16,;18.04,2.15,;19.39,2.94,;16.71,2.92,;27.37,-.15,;27.37,-1.71,;28.7,.63,;30.03,-.15,;30.03,-1.72,;31.35,-2.49,;31.35,-4.05,;32.69,-4.81,;32.66,-6.35,;31.32,-7.15,;34.02,-7.12,;31.35,.61,;31.35,2.14,;32.69,-.15,;34.03,.63,;34.03,2.15,;35.38,2.94,;35.38,4.46,;36.73,5.24,;36.75,6.77,;35.38,-.16,;35.38,-1.72,;36.71,.61,;38.05,-.16,;38.05,-1.72,;39.37,-2.48,;39.37,.6,;40.73,-.17,;39.37,2.13,)|
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[#6]-[#6@@H](-[#8])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6](-[#7])=O)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7](-[#6])-[#6])-[#7](-[#6])-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6])-[#7])-[#6@@H](-[#6])-[#8])-[#6](=O)-[#7]-[#6@@H](-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#8])-[#6](-[#7])=O |r|
CC(C)C[C@H](NC(=O)[C@H](CC1=CN=CN1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCC(=O)NCC(=O)NCC(=O)N[C@@H](CCCCNC(=O)C1=C(C=CC=C1C1=C2C=CC(=O)C=C2OC2=C1C=CC(O)=C2)C(O)=O)C(N)=O |r,c:12,118,120,123,125,129,133,136,139,t:10,116|
CC(C)C[C@H](NC(=O)[C@H](CC1=CN=CN1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)C1=C(C=CC=C1C1=C2C=CC(=O)C=C2OC2=C1C=CC(O)=C2)C(O)=O)C(N)=O |r,c:12,122,124,127,129,133,137,140,143,t:10,120|
CC(C)C[C@H](NC(=O)[C@H](CC1=CN=CN1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)C1=C(C=CC=C1C1=C2C=CC(=O)C=C2OC2=C1C=CC(O)=C2)C(O)=O)C(N)=O |r,c:12,112,114,117,119,123,127,130,133,t:10,110|
CC(C)C[C@H](NC(=O)[C@H](CC1=CN=CN1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)C1=C(C=CC=C1C1=C2C=CC(=O)C=C2OC2=C1C=CC(O)=C2)C(O)=O)C(N)=O |r,c:12,114,116,119,121,125,129,132,135,t:10,112|
CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O |r,wU:31.32,47.49,4.4,67.67,18.19,wD:22.28,56.56,36.44,76.76,8.15,(20.76,2.59,;20.76,1.08,;22.11,.3,;19.42,.3,;19.42,-1.22,;18.1,-2.03,;16.76,-1.27,;16.76,.25,;15.45,-2.03,;15.45,-3.58,;16.76,-4.34,;18.16,-3.75,;19.17,-4.89,;18.4,-6.21,;16.9,-5.87,;14.12,-1.26,;12.79,-2.02,;12.79,-3.58,;11.44,-1.25,;10.11,-2.02,;8.76,-1.28,;8.76,.24,;7.45,-2.04,;7.45,-3.6,;8.76,-4.36,;8.76,-5.91,;7.44,-6.63,;10.07,-6.66,;6.14,-1.22,;4.83,-2.02,;4.83,-3.58,;3.48,-1.25,;3.48,.27,;2.14,-2.01,;.77,-1.31,;.77,.21,;-.55,-2.06,;-.55,-3.61,;.77,-4.37,;.77,-5.93,;2.14,-6.63,;2.08,-8.17,;.76,-8.87,;3.41,-8.88,;-1.86,-1.27,;-3.19,-2.04,;-3.19,-3.57,;-4.53,-1.26,;-4.53,.28,;-5.85,-2.03,;11.44,.26,;12.79,1.04,;10.13,1.02,;20.76,-2,;20.76,-3.55,;22.09,-1.22,;23.43,-1.98,;23.43,-3.54,;24.74,-4.3,;24.74,-5.85,;26.07,-6.63,;26.06,-8.17,;24.71,-8.95,;27.36,-8.93,;24.74,-1.23,;24.74,.29,;26.07,-2,;27.4,-1.22,;27.4,.3,;28.74,1.08,;28.74,2.59,;30.09,3.37,;30.12,4.88,;28.74,-2,;28.74,-3.55,;30.08,-1.24,;31.42,-2.01,;31.42,-3.56,;32.73,-4.32,;32.73,-1.26,;34.07,-2.03,;32.73,.26,)|
[#6]-[#6@H](-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6])-[#6](-[#7])=O |r|
[#6]-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6])-[#7]-[#6]=O)-[#6](-[#7])=O |r|
[#6]-[#6@H](-[#7]-[#6](-[#6])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7](-[#6])-[#6@@H](-[#6])-[#6](-[#7])=O |r|
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)cc1)[N+]([O-])=O
COc1cccc(c1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(O)c1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1Cl)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(C)=O)[N+]([O-])=O
CN(C)CCN(C)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
NC1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
NC1CCN(C1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
[O-][N+](=O)c1ccc(N2CCNCC2)c(NC(=O)c2ccccc2Cl)c1
CN(C)C1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
CCN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
[O-][N+](=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccccc2Cl)c1
[O-][N+](=O)c1ccc(N2CCOCC2)c(NC(=O)c2ccccc2Cl)c1
CN1CCCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
CC1CN(CCN1C)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O
[O-][N+](=O)c1ccc(F)c(NC(=O)c2ccccc2Cl)c1
c1ccc2c(c1)ccc(c2c3c4ccccc4ccc3C(=O)O)C(=O)O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)-c1ccncc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)-c1ccco1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)C1CC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)C(O)=O
CN1CCN(CC1)c1ccc(N)cc1NC(=O)c1ccccc1Cl
CN1CCN(CC1)c1ccc(Br)cc1NC(=O)c1ccccc1Cl
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)C(F)(F)F
COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccccc2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccco1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccnc1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)Cc1ccccc1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc2ncccc12)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc2ccccc12)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)C1CCCCC1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1)[N+]([O-])=O
Cc1c(ccc(c1Cl)C(=O)Nc2cc(ccc2N3CCN(CC3)C)N(=O)=O)F
COc1cc(ccc1F)C(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)cc1Cl)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnn(CCN2CCOCC2)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1)-c1cnc2ccccc2c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)cc(C)c1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c(F)c(C)c(F)c(C)c1F)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCCc2c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2ccccc2c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2[nH]ccc2c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC(C)=O)nc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N)nc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccncc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)[N+]([O-])=O
CN1CCN(CC1)c1ccc(N)cc1NC(=O)c1ccc(F)c(C)c1Cl
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1cccc(c1)C(O)=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)C(O)=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)C#N
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccccc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(F)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1cncnc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(N)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)-c1ccccc1
CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)C(O)=O
CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccncc1
CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)[N+]([O-])=O
CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(N)cc1
CN1CCN(CC1)c1ccc(cc1NS(=O)(=O)c1ccc(F)cc1)[N+]([O-])=O
COc1ccc(cc1)S(=O)(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O
COc1ccc(cc1OC)S(=O)(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O
COc1cc(OC)c(c(OC)c1)S(=O)(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1C(=O)Nc1ccc(F)c(C)c1Cl)[N+]([O-])=O
COc1cccc(NC(=O)c2cc(ccc2N2CCN(C)CC2)[N+]([O-])=O)c1
CN1CCN(CC1)c1ccc(cc1C(=O)Nc1ccc(F)cc1F)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1C(=O)Nc1ccccc1Cl)[N+]([O-])=O
CCOC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(c2)[N+]([O-])=O)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)C(=O)Oc1ccccc1
COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(c(F)c(C)c2Cl)[N+]([O-])=O)c1
COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CCOC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(C)c2Cl)c1
CC(C)OC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(c2)[N+]([O-])=O)c1
CC(C)OC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(N)c2)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)C(=O)Oc1ccccc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)C(=O)Oc1ccccc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)C(=O)OC1CCCCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C(=O)OC1CCCCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)C(O)=O
CN1CCN(CC1)c2ccc(cc2NC(=O)c3cccc(c3)OC)C(=O)OC
COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(N)c2)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)C(=O)OC1CCCCC1
COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(c2)[N+]([O-])=O)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)C(O)=O
COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(C)c2Cl)c1
CC(C)OC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)C(=O)OC1CCCCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)C(=O)OC1CCCCC1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)C(=O)Oc1ccccc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C(=O)Oc1ccccc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CCNCC2)cc1
CC(N)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)c2ccccc2)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(c1)[N+]([O-])=O)-c1ccc(cc1)[N+]([O-])=O
COC(=O)c1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(c(F)c(C)c2Cl)[N+]([O-])=O)c1
Cc1c(F)ccc(C(=O)Nc2cc(ccc2NCCN)[N+]([O-])=O)c1Cl
CCCC(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)-c1ccncc1
Cc1c(F)ccc(C(=O)Nc2cc(ccc2N2CCN(CC2)c2ccc(F)cc2)[N+]([O-])=O)c1Cl
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)-c1ccncc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccncc1
CC(C)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(NC(C)=O)c(F)c(C)c1Cl)-c1ccc(cc1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(N)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCCNC(=O)OC(C)(C)C)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C(C)(C)NC(=O)OC(C)(C)C)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCNC(=O)OC(C)(C)C)cc1
CC(NC(=O)OC(C)(C)C)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CNC(=O)OC(C)(C)C)cc1
CCC(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(C)=O)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)-c1ccncc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)-c1ccc(N)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(NC(C)=O)c(F)c(C)c1Cl)-c1ccncc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(NC(C)=O)c(F)c(C)c1Cl)-c1ccc(N)cc1
COc1ccc(cc1)N1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)[N+]([O-])=O
Cc1c(F)ccc(C(=O)Nc2cc(ccc2N2CCN(Cc3ccccc3)CC2)[N+]([O-])=O)c1Cl
Cc1c(F)ccc(C(=O)Nc2cc(ccc2NCCN2CCCC2)[N+]([O-])=O)c1Cl
CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)-c1ccc(cc1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C(C)(C)N)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)-c1ccc(cc1)[N+]([O-])=O
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CC2)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCN)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CN)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CCCCC2)cc1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccccc1
Cc1c(F)ccc(C(=O)Nc2cc(ccc2NCCCn2ccnc2)[N+]([O-])=O)c1Cl
CC(C)CC(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1
CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(N)c1)-c1ccc(N)cc1
Cc1c(F)ccc(C(=O)Nc2cc(ccc2N2CCN(CC2)c2ccccn2)[N+]([O-])=O)c1Cl