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  • 6BH2: linked kdm5a jmj domain bound to the inhibitor (r)-n-(1-(3-isopropyl- 1h-pyrazole-5-carbonyl)pyrrolidin-3-yl)cyclopropanecarboxamide (compound n54) (10.1021/ACS.JMEDCHEM.8B00261 )
  • 6EK6: crystal structure of kdm5b in complex with s49195a.
  • 5V9T: crystal structure of selective pyrrolidine amide kdm5a inhibitor n- {(3r)-1-[3-(propan-2-yl)-1h-pyrazole-5-carbonyl]pyrrolidin-3- yl}cyclopropanecarboxamide (compound 48) (10.1016/J.BMCL.2017.05.016 )