TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Tested for binding affinity against alpha-2 adrenergic receptor in rat brain using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Tested for binding affinity against alpha-2 adrenergic receptor in rat brain using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-2 adrenergic receptor of bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Tested for binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-CGP- 26505 as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards beta-2 receptor of bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Tested for binding affinity against beta-2 adrenergic receptor in bovine lung using [3H]DHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards beta-2 receptor of bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Tested for binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-CGP- 26505 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Tested for binding affinity against alpha-1 adrenergic receptor in rat brain using [3H]-Prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+3nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.24E+3nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.28E+3nMAssay Description:Tested for binding affinity against alpha-2 adrenergic receptor in rat brain using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 1.48E+3nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.49E+3nMAssay Description:Tested for binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-CGP- 26505 as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.57E+3nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.78E+3nMAssay Description:Tested for binding affinity against alpha-2 adrenergic receptor in rat brain using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.98E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.45E+3nMAssay Description:Tested for binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-CGP- 26505 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.12E+3nMAssay Description:Tested for binding affinity against alpha-2 adrenergic receptor in rat brain using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.58E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.80E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Tested for binding affinity against beta-2 adrenergic receptor in bovine lung using [3H]DHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to D2 receptorMore data for this Ligand-Target Pair