Compile Data Set for Download or QSAR
maximum 50k data
Found 63 with Last Name = 'scotese' and Initial = 'a'
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429069(CHEMBL2335736)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429068(CHEMBL2335740)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429069(CHEMBL2335736)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429067(CHEMBL2335737)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  10nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429067(CHEMBL2335737)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429068(CHEMBL2335740)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(CHEMBL153469 | N-Hydroxy-3-(4-methoxy-benzenesulfo...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  30nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429065(CHEMBL2331599)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  50nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  50nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  60nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152197(2-[3-(5-Aminomethyl-2,4-dimethyl-benzylamino)-5-ch...)
Affinity DataKi:  93nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429066(CHEMBL2335741)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429065(CHEMBL2331599)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152198(2-[3-(4-Amino-cyclohexylamino)-5-chloro-6-methyl-2...)
Affinity DataKi:  138nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM16127(2,2 -methanediylbis(1H-benzimidazole-6-carboximida...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429064(CHEMBL2335738)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  200nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429066(CHEMBL2335741)
Affinity DataKi:  244nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152202(2-[3-(4-Amino-benzylamino)-5-chloro-6-methyl-2-oxo...)
Affinity DataKi:  245nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429064(CHEMBL2335738)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152200(CHEMBL183528 | N-(3-Aminomethyl-phenyl)-2-{5-chlor...)
Affinity DataKi:  290nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(CHEMBL153469 | N-Hydroxy-3-(4-methoxy-benzenesulfo...)
Affinity DataKi:  300nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152205(2-[3-(3-Aminomethyl-benzylamino)-5-chloro-6-methyl...)
Affinity DataKi:  390nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152206(CHEMBL187587 | N-(3-Aminomethyl-phenyl)-2-{5-chlor...)
Affinity DataKi:  426nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  500nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152196(CHEMBL184815 | N-(3-Aminomethyl-phenyl)-2-{5-chlor...)
Affinity DataKi:  518nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152193(CHEMBL187649 | N-(3-Aminomethyl-phenyl)-2-{3-[(6-a...)
Affinity DataKi:  580nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  600nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  600nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152203(2-[3-(4-Aminomethyl-benzylamino)-5-chloro-6-methyl...)
Affinity DataKi:  615nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  700nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152194(2-[3-(2-Amino-benzylamino)-5-chloro-6-methyl-2-oxo...)
Affinity DataKi:  875nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152204(CHEMBL360210 | N-(3-Aminomethyl-phenyl)-2-[5-chlor...)
Affinity DataKi:  970nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(CHEMBL153469 | N-Hydroxy-3-(4-methoxy-benzenesulfo...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152195(CHEMBL187168 | N-(3-Aminomethyl-phenyl)-2-[3-(4-be...)
Affinity DataKi:  1.24E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152199(CHEMBL183942 | N-(3-Aminomethyl-phenyl)-2-(5-chlor...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152201(CHEMBL187651 | N-(3-Aminomethyl-phenyl)-2-[5-chlor...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429063(CHEMBL2335739)
Affinity DataKi:  3.34E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 63 total ) | Next | Last >>
Jump to: