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Found 3364 with Last Name = 'das' and Initial = 'b'
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Indian Institute Of Technology (B.H.U.)

Curated by ChEMBL
LigandPNGBDBM50246967(CHEMBL4080228 | US10570121, Example 81)
Affinity DataKi: <0.100nMAssay Description:Inhibition of EZH2 Y641N mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50499869(CHEMBL3742140)
Affinity DataKi:  0.145nMAssay Description:Displacement of [3H]Spiroperidol from cloned rat dopamine D3 receptor expressed in HEK293 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Long Island University

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to DPP-4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  0.447nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Indian Institute Of Technology (B.H.U.)

Curated by ChEMBL
LigandPNGBDBM50156024(CHEMBL3780852)
Affinity DataKi:  0.800nMAssay Description:Binding affinity towards human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Indian Institute Of Technology (B.H.U.)

Curated by ChEMBL
LigandPNGBDBM50272462(CHEMBL525528 | N-(Adamant-1-yl)-7-fluoro-4-oxo-1-p...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity towards human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  0.850nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50499868(CHEMBL3740286)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]Spiroperidol from cloned rat dopamine D3 receptor expressed in HEK293 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Indian Institute Of Technology (B.H.U.)

Curated by ChEMBL
LigandPNGBDBM50193709(CHEMBL3911017)
Affinity DataKi:  1.20nMAssay Description:Inhibition of EZH2 Y641N mutant (unknown origin)More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50499867(CHEMBL3740041)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]Spiroperidol from cloned rat dopamine D3 receptor expressed in HEK293 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  1.29nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50610253(CHEMBL5283620)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  1.35nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50610247(CHEMBL5276671)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  1.95nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610247(CHEMBL5276671)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50115277((2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphtha...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50115277((2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphtha...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Spiroperidol from cloned rat dopamine D3 receptor expressed in HEK293 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50610250(CHEMBL5267221)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314073(3-(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-ox...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of p38alpha kinaseMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50610248(CHEMBL5274131)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50499871(CHEMBL3740760)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]Spiroperidol from cloned rat dopamine D3 receptor expressed in HEK293 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50610249(CHEMBL5282690)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610249(CHEMBL5282690)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319849(CHEMBL1083921 | N-((2-chloro-1-(2-chloro-4,6-dimet...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319896(CHEMBL1084999 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610250(CHEMBL5267221)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Long Island University

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataKi:  5nMAssay Description:Binding affinity to FAP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319906(CHEMBL1083933 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50610251(CHEMBL5272529)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319893(CHEMBL1083952 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319869(CHEMBL1086504 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50346920(CHEMBL1795686)
Affinity DataKi:  6nMAssay Description:Inhibition of p38beta kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319890(CHEMBL1082696 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50610252(CHEMBL5266134)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610251(CHEMBL5272529)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50314008(CHEMBL1087165 | N-(cyclopropylmethyl)-2,2,2-triflu...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]Tyr-o-CRF from human CRFR1 expressed in human IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319903(CHEMBL1082302 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610253(CHEMBL5283620)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50499876(CHEMBL3740829)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]Spiroperidol from cloned rat dopamine D3 receptor expressed in HEK293 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319905(CHEMBL1083319 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319907(CHEMBL1086468 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319882(CHEMBL1082338 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319902(CHEMBL1083935 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610248(CHEMBL5274131)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50499874(CHEMBL3740143)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Spiroperidol from cloned rat dopamine D3 receptor expressed in HEK293 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50319889(CHEMBL1086594 | N-((2-chloro-1-mesityl-6-(trifluor...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I] Tyr-o-CRF from human CRF[125I]receptor expressed in human IMR-3[125I]cells after 100 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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