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Found 374 with Last Name = 'town' and Initial = 'c'
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318541(Ac-ARAEVHLRKS-NH2 | CHEMBL1086450)
Affinity DataKi:  3nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318527(Ac-ART-NH2 | CHEMBL1085865)
Affinity DataKi:  20nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318542(CHEMBL1086451 | H2N-SARAEVHLRKS-NH2)
Affinity DataKi:  20nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318544(Ac-ARAEVHL-NH2 | CHEMBL1086453)
Affinity DataKi:  30nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318547(Ac-ARAE-NH2 | CHEMBL1085604)
Affinity DataKi:  80nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318545(Ac-ARAEVH-NH2 | CHEMBL1086454)
Affinity DataKi:  90nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318548(Ac-ARA-NH2 | CHEMBL1086455)
Affinity DataKi:  120nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318521(Ac-ARA-CONHMe | CHEMBL1084621)
Affinity DataKi:  150nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318546(Ac-ARAEV-NH2 | CHEMBL1086531)
Affinity DataKi:  160nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318539(Ac-GSARAEVHLRKS-NH2 | CHEMBL1086448)
Affinity DataKi:  160nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318540(Ac-SARAEVHLRKS-NH2 | CHEMBL1086449)
Affinity DataKi:  200nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318523(Ac-ARA-COOCH3 | CHEMBL1084623)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318537(CHEMBL1086083 | CHO-ARA-NH2)
Affinity DataKi:  3.20E+3nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318543(Ac-RAEVHLRKS-NH2 | CHEMBL1086452)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318522(Ac-ARA-CONMe2 | CHEMBL1084622)
Affinity DataKi:  6.50E+3nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318535(CHEMBL1086456 | H2N-ARAEVHLRKS-NH2)
Affinity DataKi:  7.30E+3nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318529(CHEMBL1082285 | H2N-ARTK(Me2)QTARKS-NH2)
Affinity DataKi:  9.00E+3nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318528(CHEMBL1082284 | H2N-ARTK(Me)QTARKS-NH2)
Affinity DataKi:  1.50E+4nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318524(CHEMBL1082281 | H2N-ARTKQTARKS-NH2)
Affinity DataKi:  1.51E+4nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318530(CHEMBL1082286 | H2N-ARTK(Me3)QTARKS-NH2)
Affinity DataKi:  1.56E+4nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318549(Ac-AR-NH2 | CHEMBL1085605)
Affinity DataKi:  2.70E+4nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318526(CHEMBL1085864 | H2N-ART-NH2)
Affinity DataKi:  2.73E+4nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318536(CHEMBL1085606 | H2N-ARA-NH2)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318538(Ac-AR-(N-Me)A-NH2 | CHEMBL1084620)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318534((7S,24S,27S,30S,33S,36S,39S,42S)-36-((1H-imidazol-...)
Affinity DataIC50:  1nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells after 24 hrs by optimized fluorescent polarization based saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318525(Ac-ARTKQTARKS-NH2 | CHEMBL1082282)
Affinity DataIC50:  6nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190017((4R,5R)-4-(2-fluorophenyl)-5-((S)-hydroxy(5-phenyl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318533((7S,24S,27S,30S,33S,36S,39S,42S)-36-((1H-imidazol-...)
Affinity DataIC50:  14nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells after 24 hrs by optimized fluorescent polarization based saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318541(Ac-ARAEVHLRKS-NH2 | CHEMBL1086450)
Affinity DataIC50:  20nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190020(4-(5-((S)-hydroxy((2R,3R)-1-methyl-5-oxo-3-phenylp...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataIC50:  30nMAssay Description:Activity at human PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190010((4R,5R)-4-(2-fluorophenyl)-5-((S)-hydroxy(5-(pyrid...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190010((4R,5R)-4-(2-fluorophenyl)-5-((S)-hydroxy(5-(pyrid...)
Affinity DataIC50:  30nMAssay Description:Inhibition of estradiol to estrone conversion in MG63 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190030((4R,5R)-5-((S)-hydroxy(5-(phenylsulfonyl)thiophen-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataIC50:  49nMAssay Description:Activity at human PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataIC50:  56nMAssay Description:Activity at human PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190015((4R,5R)-4-(2-fluorophenyl)-5-((S)-(5-(4-fluorophen...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190004((4R,5R)-4-(2-fluorophenyl)-5-((S)-(5-(4-fluorophen...)
Affinity DataIC50:  60nMAssay Description:Inhibition of estradiol to estrone conversion in MG63 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190004((4R,5R)-4-(2-fluorophenyl)-5-((S)-(5-(4-fluorophen...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190004((4R,5R)-4-(2-fluorophenyl)-5-((S)-(5-(4-fluorophen...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190031((4R,5R)-5-((S)-hydroxy(5-(morpholinosulfonyl)thiop...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318527(Ac-ART-NH2 | CHEMBL1085865)
Affinity DataIC50:  80nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318542(CHEMBL1086451 | H2N-SARAEVHLRKS-NH2)
Affinity DataIC50:  80nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190011((4R,5R)-5-((S)-hydroxy(5-(pyridin-3-yl)thiophen-2-...)
Affinity DataIC50:  90nMAssay Description:Inhibition of estradiol to estrone conversion in MG63 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190006((4R,5R)-5-((S)-(5-(4-fluorophenyl)thiophen-2-yl)(h...)
Affinity DataIC50:  100nMAssay Description:Inhibition of estradiol to estrone conversion in MG63 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190009((4R,5R)-5-((S)-hydroxy(5-phenylthiophen-2-yl)methy...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190035((4R,5R)-5-((S)-(5-(4-fluorophenyl)thiophen-2-yl)(h...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190028((4R,5R)-5-((S)-(5-(2-fluorophenyl)thiophen-2-yl)(h...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190006((4R,5R)-5-((S)-(5-(4-fluorophenyl)thiophen-2-yl)(h...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50190006((4R,5R)-5-((S)-(5-(4-fluorophenyl)thiophen-2-yl)(h...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human recombinant 17beta-HSD2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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