Affinity DataIC50: 130nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of strand -transfer (ST) activity in the presence of Mn2+More data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:The compound was tested in vitro for inhibition of HIV-1 replicationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of 3'-processing (TC) in the presence of Mn2+ in vitro More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of strand -transfer (ST) activity in the presence of Mn2+More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of strand -transfer (ST) activity in the presence of Mn2+More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of 3'-processing (TC) in the presence of Mn2+ in vitro More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of strand -transfer (ST) activity in the presence of Mn2+More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 3.14E+3nMAssay Description:Inhibition of 3'-processing (TC) in the presence of Mn2+ in vitro More data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Tested in vitro against strand -transfer (ST) activity in the presence of Mg2+ as the cationic cofactorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of strand -transfer (ST) activity in the presence of Mn2+More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of HIV-1 integrase, under 1 uM for the 3''-preprocessingMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of strand -transfer (ST) activity in the presence of Mn2+More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of 3'-processing (TC) in the presence of Mn2+ in vitro More data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Tested for inhibition of HIV-1 integrase, under 1 uM for the strand transferMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:The compound was tested in vitro for inhibition of HIV-1 replicationMore data for this Ligand-Target Pair